| Year |
Citation |
Score |
| 2021 |
Rohde JM, Karavadhi S, Pragani R, Liu L, Fang Y, Zhang W, McIver A, Zheng H, Liu Q, Davis MI, Urban DJ, Lee TD, Cheff DM, Hollingshead M, Henderson MJ, et al. Discovery and Optimization of 2-1λ-Pyridin-2-one Inhibitors of Mutant Isocitrate Dehydrogenase 1 for the Treatment of Cancer. Journal of Medicinal Chemistry. PMID 33822623 DOI: 10.1021/acs.jmedchem.1c00019 |
0.636 |
|
| 2017 |
Urban DJ, Martinez NJ, Davis MI, Brimacombe KR, Cheff DM, Lee TD, Henderson MJ, Titus SA, Pragani R, Rohde JM, Liu L, Fang Y, Karavadhi S, Shah P, Lee OW, ... McIver A, et al. Assessing inhibitors of mutant isocitrate dehydrogenase using a suite of pre-clinical discovery assays. Scientific Reports. 7: 12758. PMID 28986582 DOI: 10.1038/S41598-017-12630-X |
0.761 |
|
| 2016 |
McIver A, Zhang W, Liu Q, Jiang X, Stashko M, Nichols J, Miley M, Norris-Drouin J, Machius M, DeRyckere D, Wood E, Graham D, Earp HS, Kireev D, Frye S, et al. Discovery of Macrocyclic Pyrimidines as MerTK-specific Inhibitors. Chemmedchem. PMID 28032464 DOI: 10.1002/Cmdc.201600589 |
0.749 |
|
| 2016 |
Buchanan MK, Needham CN, Neill NE, White MC, Kelly CB, Mastro-Kishton K, Chauvigne-Hines LM, Goodwin TJ, McIver AL, Bartolotti LJ, Frampton AR, Bourdelais AJ, Varadarajan S. Glycoconjugated Site-selective DNA-Methylating Agent Targeting Glucose Transporters on Glioma Cells. Biochemistry. PMID 28000448 DOI: 10.1021/acs.biochem.6b01075 |
0.744 |
|
| 2013 |
Zhang W, McIver AL, Stashko MA, DeRyckere D, Branchford BR, Hunter D, Kireev D, Miley MJ, Norris-Drouin J, Stewart WM, Lee M, Sather S, Zhou Y, Di Paola JA, Machius M, et al. Discovery of Mer specific tyrosine kinase inhibitors for the treatment and prevention of thrombosis. Journal of Medicinal Chemistry. 56: 9693-700. PMID 24219778 DOI: 10.1021/Jm501217P |
0.756 |
|
| 2012 |
Govan JM, McIver AL, Riggsbee C, Deiters A. Hydrogen peroxide induced activation of gene expression in mammalian cells using boronate estrone derivatives. Angewandte Chemie (International Ed. in English). 51: 9066-70. PMID 22855386 DOI: 10.1002/Anie.201203222 |
0.617 |
|
| 2011 |
Govan JM, McIver AL, Deiters A. Stabilization and photochemical regulation of antisense agents through PEGylation. Bioconjugate Chemistry. 22: 2136-42. PMID 21928851 DOI: 10.1021/Bc200411N |
0.718 |
|
| 2011 |
Dush MK, McIver AL, Parr MA, Young DD, Fisher J, Newman DR, Sannes PL, Hauck ML, Deiters A, Nascone-Yoder N. Heterotaxin: a TGF-β signaling inhibitor identified in a multi-phenotype profiling screen in Xenopus embryos. Chemistry & Biology. 18: 252-63. PMID 21338922 DOI: 10.1016/J.Chembiol.2010.12.008 |
0.724 |
|
| 2010 |
Georgianna WE, Lusic H, McIver AL, Deiters A. Photocleavable polyethylene glycol for the light-regulation of protein function. Bioconjugate Chemistry. 21: 1404-7. PMID 20715846 DOI: 10.1021/Bc100084N |
0.69 |
|
| 2010 |
McIver AL, Deiters A. Tricyclic alkaloid core structures assembled by a cyclotrimerization-coupled intramolecular nucleophilic substitution reaction. Organic Letters. 12: 1288-91. PMID 20178343 DOI: 10.1021/Ol100177U |
0.728 |
|
| 2010 |
Nascone-Yoder NM, Dush M, McIver A, Parr M, Young D, Fisher J, Hauck M, Deiters A. Heterotaxin: A novel TGF-beta signaling inhibitor identified in a multi-phenotype profiling screen in Xenopus embryos Developmental Biology. 344: 526. DOI: 10.1016/J.Ydbio.2010.05.483 |
0.711 |
|
| 2009 |
McIver A, Young DD, Deiters A. ChemInform Abstract: A General Approach to Triphenylenes and Azatriphenylenes: Total Synthesis of Dehydrotylophorine and Tylophorine. Cheminform. 40. DOI: 10.1002/CHIN.200908201 |
0.744 |
|
| 2008 |
McIver A, Young DD, Deiters A. A general approach to triphenylenes and azatriphenylenes: total synthesis of dehydrotylophorine and tylophorine. Chemical Communications (Cambridge, England). 4750-2. PMID 18830481 DOI: 10.1039/B811068A |
0.718 |
|
| Show low-probability matches. |