| Year |
Citation |
Score |
| 2022 |
Aksenov AV, Kirilov NK, Arutiunov NA, Aksenov DA, Kuzminov IK, Aksenov NA, Turner DN, Rogelj S, Kornienko A, Rubin M. Reductive Cleavage of 4'-Spiro[indole-3,5'-isoxazoles] En Route to 2-(1-Indol-3-yl)acetamides with Anticancer Activities. The Journal of Organic Chemistry. PMID 36260110 DOI: 10.1021/acs.joc.2c01627 |
0.308 |
|
| 2022 |
Mathieu V, Superchi S, Masi M, Scafato P, Kornienko A, Evidente A. In Vitro Effects of Fungal Phytotoxins on Cancer Cell Viability: First Insight into Structure Activity Relationship of a Potent Metabolite of Radicinin. Toxins. 14. PMID 36006179 DOI: 10.3390/toxins14080517 |
0.319 |
|
| 2022 |
Goulart Stollmaier J, Thomson J, Endoma-Arias MA, Simionescu R, Vernaza A, Mesa-Diaz N, Smith M, Du L, Kornienko A, Hudlicky T. Conversion of Natural Narciclasine to Its C-1 and C-6 Derivatives and Their Antitumor Activity Evaluation: Some Unusual Chemistry of Narciclasine. Molecules (Basel, Switzerland). 27. PMID 35807391 DOI: 10.3390/molecules27134141 |
0.31 |
|
| 2022 |
Habaz L, Bedard K, Smith M, Du L, Kornienko A, Hudlicky T. Design and Synthesis of C-1 Methoxycarbonyl Derivative of Narciclasine and Its Biological Activity. Molecules (Basel, Switzerland). 27. PMID 35744934 DOI: 10.3390/molecules27123809 |
0.352 |
|
| 2021 |
Ticli V, Zhao Z, Du L, Kornienko A, Hudlicky T. Synthesis and biological evaluation of 10-benzyloxy-Narciclasine. Tetrahedron. 101. PMID 35058668 DOI: 10.1016/j.tet.2021.132505 |
0.344 |
|
| 2021 |
Maslivetc V, Laguera B, Chandra S, Dasari R, Olivier WJ, Smith JA, Bissember AC, Masi M, Evidente A, Mathieu V, Kornienko A. Polygodial and Ophiobolin A Analogues for Covalent Crosslinking of Anticancer Targets. International Journal of Molecular Sciences. 22. PMID 34681916 DOI: 10.3390/ijms222011256 |
0.312 |
|
| 2021 |
Aksenov AV, Arutiunov NA, Kirilov NK, Aksenov DA, Grishin IY, Aksenov NA, Wang H, Du L, Betancourt T, Pelly SC, Kornienko A, Rubin M. [3 + 2]-Annulation of pyridinium ylides with 1-chloro-2-nitrostyrenes unveils a tubulin polymerization inhibitor. Organic & Biomolecular Chemistry. PMID 34387294 DOI: 10.1039/d1ob01141c |
0.342 |
|
| 2020 |
Aksenov NA, Aksenov AV, Kirilov NK, Arutiunov NA, Aksenov DA, Maslivetc V, Zhao Z, Du L, Rubin M, Kornienko A. Nitroalkanes as electrophiles: synthesis of triazole-fused heterocycles with neuroblastoma differentiation activity. Organic & Biomolecular Chemistry. PMID 32813002 DOI: 10.1039/D0Ob01007C |
0.464 |
|
| 2020 |
Turner DN, Edwards L, Kornienko A, Frolova LV, Rogelj S. Synergistic action of substituted indole derivatives and clinically used antibiotics against drug-resistant bacteria. Future Microbiology. PMID 32483987 DOI: 10.2217/Fmb-2019-0094 |
0.324 |
|
| 2020 |
Eyong KO, Ketsemen HL, Zhao Z, Du L, Ingels A, Mathieu V, Kornienko A, Hull KG, Folefoc GN, Baskaran S, Romo D. Antiproliferative activity of naphthoquinones and indane carboxylic acids from lapachol against a panel of human cancer cell lines Medicinal Chemistry Research. 29: 1058-1066. DOI: 10.1007/S00044-020-02545-0 |
0.317 |
|
| 2019 |
van Rixel VH, Ramu V, Auyeung AB, Beztsinna N, Léger DY, Hilt ST, Le Dévédec SE, Yildiz T, Betancourt T, Gildner B, Hudnall TW, Sol V, Liagre B, Kornienko A, Bonnet S. Photo-uncaging of a ruthenium-caged microtubule-targeted rigidin analogue in hypoxic cancer cells and in a xenograft mouse model. Journal of the American Chemical Society. PMID 31625740 DOI: 10.1021/Jacs.9B07225 |
0.398 |
|
| 2019 |
Segat GC, Moreira CG, Santos EC, Heller M, Schwanke RC, Aksenov AV, Aksenov NA, Aksenov DA, Kornienko A, Marcon R, Calixto JB. A new series of acetohydroxamates shows in vitro and in vivo anticancer activity against melanoma. Investigational New Drugs. PMID 31493129 DOI: 10.1007/S10637-019-00849-6 |
0.375 |
|
| 2019 |
Pereira RB, Evdokimov NM, Lefranc F, Valentão P, Kornienko A, Pereira DM, Andrade PB, Gomes ANGM. Marine-Derived Anticancer Agents: Clinical Benefits, Innovative Mechanisms, and New Targets. Marine Drugs. 17. PMID 31159480 DOI: 10.3390/Md17060329 |
0.697 |
|
| 2019 |
Aksenov AV, Aksenov DA, Arutiunov NA, Aksenov NA, Aleksandrova EV, Zhao Z, Du L, Kornienko A, Rubin M. Synthesis of Spiro[indole-3,5'-isoxazoles] with Anticancer Activity via a Formal (4+1)-Spirocyclization of Nitroalkenes to Indoles. The Journal of Organic Chemistry. PMID 31070030 DOI: 10.1021/Acs.Joc.9B00808 |
0.435 |
|
| 2019 |
Turner DN, Just J, Dasari R, Smith JA, Bissember AC, Kornienko A, Rogelj S. Activity of natural and synthetic polygodial derivatives against Trypanosoma cruzi amastigotes, trypomastigotes and epimastigotes. Natural Product Research. 1-4. PMID 31032640 DOI: 10.1080/14786419.2019.1597350 |
0.388 |
|
| 2019 |
Masi M, Dasari R, Evidente A, Mathieu V, Kornienko A. Chemistry and biology of ophiobolin A and its congeners. Bioorganic & Medicinal Chemistry Letters. 29: 859-869. PMID 30765189 DOI: 10.1016/J.Bmcl.2019.02.007 |
0.419 |
|
| 2019 |
Reisenauer K, Tao Y, Ingros A, Philip T, Evidente A, Kornienko A, Romo D, Taube J. Abstract P4-07-10: Epithelial-mesenchymal transition sensitizes breast cancer cells to paraptosis-mediated cell death via the fungus-derived sesterpenoid, Ophiobolin A Cancer Research. 79. DOI: 10.1158/1538-7445.Sabcs18-P4-07-10 |
0.342 |
|
| 2019 |
Masi M, Van slambrouck S, Gunawardana S, van Rensburg M, James P, Mochel J, Heliso P, Albalawi A, Cimmino A, van Otterlo W, Kornienko A, Green I, Evidente A. Alkaloids isolated from Haemanthus humilis Jacq., an indigenous South African Amaryllidaceae: Anticancer activity of coccinine and montanine South African Journal of Botany. 126: 277-281. DOI: 10.1016/J.Sajb.2019.01.036 |
0.339 |
|
| 2018 |
Aksenov NA, Aksenov AV, Kornienko A, De Carvalho A, Mathieu V, Aksenov DA, Ovcharov SN, Griaznov GD, Rubin M. A nitroalkane-based approach to one-pot three-component synthesis of isocryptolepine and its analogs with potent anti-cancer activities. Rsc Advances. 8: 36980-36986. PMID 35558925 DOI: 10.1039/c8ra08155g |
0.316 |
|
| 2018 |
Dasari R, Błauż A, Medellin D, Kassim R, Viera C, Santarosa M, Van der Westhuyzen A, van Otterlo W, Olivas T, Yildiz T, Betancourt T, Shuster CB, Rogelj S, Rychlik B, Hudnall T, ... ... Kornienko A, et al. Microtubule-Targeting 7-Deazahypoxanthines Derived from Marine Alkaloid Rigidins: Exploration of the N3 and N9 Positions and Interaction with Multi-Drug Resistance Proteins. Chemmedchem. PMID 30562414 DOI: 10.1002/Cmdc.201800658 |
0.387 |
|
| 2018 |
Lefranc F, Koutsaviti A, Ioannou E, Kornienko A, Roussis V, Kiss R, Newman D. Algae metabolites: from in vitro growth inhibitory effects to promising anticancer activity. Natural Product Reports. PMID 30556575 DOI: 10.1039/C8Np00057C |
0.388 |
|
| 2018 |
Garcia DG, Gonçalves-de-Albuquerque CF, da Silva CI, Kiss R, Dasari R, Chandra S, Kornienko A, Burth P. "Effect of polygodial and its direct derivatives on the mammalian Na/K-ATPase activity". European Journal of Pharmacology. PMID 29715454 DOI: 10.1016/J.Ejphar.2018.04.031 |
0.371 |
|
| 2018 |
Dasari S, Samy ALPA, Narvekar P, Dontaraju VS, Dasari R, Kornienko A, Munirathinam G. Polygodial analog induces apoptosis in LNCaP prostate cancer cells. European Journal of Pharmacology. PMID 29572068 DOI: 10.1016/J.Ejphar.2018.03.029 |
0.342 |
|
| 2018 |
van der Westhuyzen AE, Frolova LV, Kornienko A, van Otterlo WAL. The Rigidins: Isolation, Bioactivity, and Total Synthesis-Novel Pyrrolo[2,3-d]Pyrimidine Analogues Using Multicomponent Reactions. The Alkaloids. Chemistry and Biology. 79: 191-220. PMID 29455836 DOI: 10.1016/Bs.Alkal.2017.12.003 |
0.517 |
|
| 2018 |
Pellegrino S, Meyer M, Zorbas C, Bouchta SA, Saraf K, Pelly SC, Yusupova G, Evidente A, Mathieu V, Kornienko A, Lafontaine DLJ, Yusupov M. The Amaryllidaceae Alkaloid Haemanthamine Binds the Eukaryotic Ribosome to Repress Cancer Cell Growth. Structure (London, England : 1993). PMID 29429877 DOI: 10.1016/J.Str.2018.01.009 |
0.368 |
|
| 2018 |
Govindaraju K, Ingels A, Hasan MN, Sun D, Mathieu V, Masi M, Evidente A, Kornienko A. Synthetic analogues of the montanine-type alkaloids with activity against apoptosis-resistant cancer cells. Bioorganic & Medicinal Chemistry Letters. PMID 29409754 DOI: 10.1016/J.Bmcl.2018.01.041 |
0.44 |
|
| 2018 |
Govindaraju K, Masi M, Colin M, Mathieu V, Evidente A, Hudnall TW, Kornienko A. Novel Topologically Complex Scaffold Derived from Alkaloid Haemanthamine. Molecules (Basel, Switzerland). 23. PMID 29382096 DOI: 10.3390/Molecules23020255 |
0.401 |
|
| 2018 |
Aksenov NA, Aksenov A, Kornienko A, De Carvalho A, Mathieu V, Aksenov DA, Ovcharov SN, Griaznov GD, Rubin M. A nitroalkane-based approach to one-pot three-component synthesis of isocryptolepine and its analogs with potent anti-cancer activities Rsc Advances. 8: 36980-36986. DOI: 10.1039/C8Ra08155G |
0.427 |
|
| 2017 |
Kornienko A, La Clair JJ. Covalent modification of biological targets with natural products through Paal-Knorr pyrrole formation. Natural Product Reports. PMID 28808718 DOI: 10.1039/C7Np00024C |
0.317 |
|
| 2017 |
Carvalho A, Chu J, Meinguet C, Kiss R, Vandenbussche G, Masereel B, Wouters J, Kornienko A, Pelletier J, Mathieu V. Data in support of a harmine-derived beta-carboline in vitro effects in cancer cells through protein synthesis. Data in Brief. 12: 546-551. PMID 28529967 DOI: 10.1016/J.Dib.2017.05.006 |
0.354 |
|
| 2017 |
Carvalho A, Chu J, Meinguet C, Kiss R, Vandenbussche G, Masereel B, Wouters J, Kornienko A, Pelletier J, Mathieu V. A harmine-derived beta-carboline displays anti-cancer effects in vitro by targeting protein synthesis. European Journal of Pharmacology. PMID 28322844 DOI: 10.1016/J.Ejphar.2017.03.034 |
0.395 |
|
| 2017 |
Aksenov AV, Aksenov DA, Orazova NA, Aksenov NA, Griaznov GD, De Carvalho A, Kiss R, Mathieu V, Kornienko A, Rubin M. One-Pot, Three-Component Assembly of Indoloquinolines: Total Synthesis of Isocryptolepine. The Journal of Organic Chemistry. PMID 28253622 DOI: 10.1021/Acs.Joc.6B03084 |
0.457 |
|
| 2016 |
Ciavatta ML, Lefranc F, Carbone M, Mollo E, Gavagnin M, Betancourt T, Dasari R, Kornienko A, Kiss R. Marine Mollusk-Derived Agents with Antiproliferative Activity as Promising Anticancer Agents to Overcome Chemotherapy Resistance. Medicinal Research Reviews. PMID 27925266 DOI: 10.1002/Med.21423 |
0.418 |
|
| 2016 |
Henry S, Kidner R, Reisenauer MR, Magedov IV, Kiss R, Mathieu V, Lefranc F, Dasari R, Evidente A, Yu X, Ma X, Pertsemlidis A, Cencic R, Pelletier J, Cavazos DA, ... ... Kornienko A, et al. 5,10b-Ethanophenanthridine amaryllidaceae alkaloids inspire the discovery of novel bicyclic ring systems with activity against drug resistant cancer cells. European Journal of Medicinal Chemistry. 120: 313-328. PMID 27218860 DOI: 10.1016/J.Ejmech.2016.05.004 |
0.408 |
|
| 2016 |
Gomes NG, Dasari R, Chandra S, Kiss R, Kornienko A. Marine Invertebrate Metabolites with Anticancer Activities: Solutions to the "Supply Problem". Marine Drugs. 14. PMID 27213412 DOI: 10.3390/Md14050098 |
0.375 |
|
| 2016 |
Panayides JL, Mathieu V, Banuls LM, Apostolellis H, Dahan-Farkas N, Davids H, Harmse L, Rey ME, Green IR, Pelly SC, Kiss R, Kornienko A, van Otterlo WA. Synthesis and in vitro growth inhibitory activity of novel silyl- and trityl-modified nucleosides. Bioorganic & Medicinal Chemistry. PMID 27157005 DOI: 10.1016/J.Bmc.2016.04.036 |
0.378 |
|
| 2016 |
Evdokimov NM, Magedov IV, McBrayer D, Kornienko A. Isatin derivatives with activity against apoptosis-resistant cancer cells. Bioorganic & Medicinal Chemistry Letters. 26: 1558-60. PMID 26883150 DOI: 10.1016/J.Bmcl.2016.02.015 |
0.739 |
|
| 2016 |
Cimmino A, Mathieu V, Masi M, Baroncelli R, Boari A, Pescitelli G, Ferderin M, Lisy R, Evidente M, Tuzi A, Zonno MC, Kornienko A, Kiss R, Evidente A. Higginsianins A and B, Two Diterpenoid α-Pyrones Produced by Colletotrichum higginsianum, with in Vitro Cytostatic Activity. Journal of Natural Products. 79: 116-25. PMID 26697898 DOI: 10.1021/Acs.Jnatprod.5B00779 |
0.34 |
|
| 2016 |
Masi M, Cimmino A, Maddau L, Kornienko A, Tuzi A, Evidente A. Crystal structure and absolute configuration of sphaeropsidin A and its 6- O - p -bromobenzoate Tetrahedron Letters. 57: 4592-4594. DOI: 10.1016/J.Tetlet.2016.08.098 |
0.376 |
|
| 2015 |
Medellin DC, Zhou Q, Scott R, Hill RM, Frail RS, Dasari R, Ontiveros SJ, Pelly SC, van Otterlo WA, Betancourt T, Shuster CB, Hamel E, Bai R, LaBarbera DV, Rogelj S, ... ... Kornienko A, et al. Novel Microtubule-Targeting 7-Deazahypoxanthines Derived from Marine Alkaloid Rigidins with Potent In Vitro and In Vivo Anticancer Activities. Journal of Medicinal Chemistry. PMID 26641132 DOI: 10.1021/Acs.Jmedchem.5B01426 |
0.42 |
|
| 2015 |
Dasari R, De Carvalho A, Medellin DC, Middleton KN, Hague F, Volmar MN, Frolova LV, Rossato MF, De La Chapa JJ, Dybdal-Hargreaves NF, Pillai A, Mathieu V, Rogelj S, Gonzales CB, Calixto JB, ... ... Kornienko A, et al. Synthetic and Biological Studies of Sesquiterpene Polygodial: Activity of 9-Epipolygodial against Drug-Resistant Cancer Cells. Chemmedchem. PMID 26434977 DOI: 10.1002/Cmdc.201500360 |
0.447 |
|
| 2015 |
Dasari R, De Carvalho A, Medellin DC, Middleton KN, Hague F, Volmar MN, Frolova LV, Rossato MF, De La Chapa JJ, Dybdal-Hargreaves NF, Pillai A, Kälin RE, Mathieu V, Rogelj S, Gonzales CB, ... ... Kornienko A, et al. Wittig derivatization of sesquiterpenoid polygodial leads to cytostatic agents with activity against drug resistant cancer cells and capable of pyrrolylation of primary amines. European Journal of Medicinal Chemistry. 103: 226-37. PMID 26360047 DOI: 10.1016/J.Ejmech.2015.08.047 |
0.437 |
|
| 2015 |
Dasari R, Masi M, Lisy R, Ferdérin M, English LR, Cimmino A, Mathieu V, Brenner AJ, Kuhn JG, Whitten ST, Evidente A, Kiss R, Kornienko A. Fungal metabolite ophiobolin A as a promising anti-glioma agent: In vivo evaluation, structure-activity relationship and unique pyrrolylation of primary amines. Bioorganic & Medicinal Chemistry Letters. 25: 4544-8. PMID 26341136 DOI: 10.1016/J.Bmcl.2015.08.066 |
0.393 |
|
| 2015 |
Evidente A, Kornienko A, Lefranc F, Cimmino A, Dasari R, Evidente M, Mathieu V, Kiss R. Sesterterpenoids with Anticancer Activity. Current Medicinal Chemistry. 22: 3502-22. PMID 26295461 DOI: 10.2174/0929867322666150821101047 |
0.34 |
|
| 2015 |
Mathieu V, Chantôme A, Lefranc F, Cimmino A, Miklos W, Paulitschke V, Mohr T, Maddau L, Kornienko A, Berger W, Vandier C, Evidente A, Delpire E, Kiss R. Sphaeropsidin A shows promising activity against drug-resistant cancer cells by targeting regulatory volume increase. Cellular and Molecular Life Sciences : Cmls. PMID 25868554 DOI: 10.1007/S00018-015-1902-6 |
0.362 |
|
| 2015 |
Kornienko A, Evidente A, Vurro M, Mathieu V, Cimmino A, Evidente M, van Otterlo WA, Dasari R, Lefranc F, Kiss R. Toward a Cancer Drug of Fungal Origin. Medicinal Research Reviews. PMID 25850821 DOI: 10.1002/Med.21348 |
0.364 |
|
| 2015 |
Aksenov AV, Smirnov AN, Magedov IV, Reisenauer MR, Aksenov NA, Aksenova IV, Pendleton AL, Nguyen G, Johnston RK, Rubin M, De Carvalho A, Kiss R, Mathieu V, Lefranc F, Correa J, ... ... Kornienko A, et al. Activity of 2-aryl-2-(3-indolyl)acetohydroxamates against drug-resistant cancer cells. Journal of Medicinal Chemistry. 58: 2206-20. PMID 25671501 DOI: 10.1021/Jm501518Y |
0.374 |
|
| 2015 |
Masi M, Frolova LV, Yu X, Mathieu V, Cimmino A, De Carvalho A, Kiss R, Rogelj S, Pertsemlidis A, Kornienko A, Evidente A. Jonquailine, a new pretazettine-type alkaloid isolated from Narcissus jonquilla quail, with activity against drug-resistant cancer. Fitoterapia. 102: 41-8. PMID 25598189 DOI: 10.1016/J.Fitote.2015.01.009 |
0.347 |
|
| 2014 |
Mikhalin AA, Evdokimov NM, Frolova LV, Magedov IV, Kornienko A, Johnston R, Rogelj S, Tartis MS. Lipophilic prodrug conjugates allow facile and rapid synthesis of high-loading capacity liposomes without the need for post-assembly purification. Journal of Liposome Research. 1-29. PMID 25534989 DOI: 10.3109/08982104.2014.992022 |
0.712 |
|
| 2014 |
Evidente A, Kornienko A, Cimmino A, Andolfi A, Lefranc F, Mathieu V, Kiss R. Fungal metabolites with anticancer activity. Natural Product Reports. 31: 617-27. PMID 24651312 DOI: 10.1039/C3Np70078J |
0.4 |
|
| 2014 |
Scott R, Karki M, Reisenauer MR, Rodrigues R, Dasari R, Smith WR, Pelly SC, van Otterlo WA, Shuster CB, Rogelj S, Magedov IV, Frolova LV, Kornienko A. Synthetic and biological studies of tubulin targeting c2-substituted 7-deazahypoxanthines derived from marine alkaloid rigidins. Chemmedchem. 9: 1428-35. PMID 24644272 DOI: 10.1002/Cmdc.201300532 |
0.469 |
|
| 2014 |
Dasari R, Banuls LM, Masi M, Pelly SC, Mathieu V, Green IR, van Otterlo WA, Evidente A, Kiss R, Kornienko A. C1,C2-ether derivatives of the Amaryllidaceae alkaloid lycorine: retention of activity of highly lipophilic analogues against cancer cells. Bioorganic & Medicinal Chemistry Letters. 24: 923-7. PMID 24393582 DOI: 10.1016/J.Bmcl.2013.12.073 |
0.436 |
|
| 2014 |
Rastogi SK, Medellin DC, Kornienko A. C-H functionalization directed by transformable nitrogen heterocycles: synthesis of ortho-oxygenated arylnaphthalenes from arylphthalazines. Organic & Biomolecular Chemistry. 12: 410-3. PMID 24281239 DOI: 10.1039/C3Ob42255K |
0.411 |
|
| 2014 |
Dasari R, Kornienko A. Multicomponent synthesis of the medicinally important pyrrolo[2,3-d] pyrimidine scaffold (minireview) Chemistry of Heterocyclic Compounds. 50: 139-144. DOI: 10.1007/S10593-014-1456-9 |
0.422 |
|
| 2014 |
Dasari R, Kornienko A. MULTICOMPONENT SYNTHESIS OF THE MEDICINALLY IMPORTANT PYRROLO[2,3- d ]PYRIMIDINE SCAFFOLD Chemistry of Heterocyclic Compounds. 160-165. DOI: 10.1007/1294 |
0.433 |
|
| 2013 |
Aksenov AV, Smirnov AN, Aksenov NA, Aksenova IV, Frolova LV, Kornienko A, Magedov IV, Rubin M. Metal-free transannulation reaction of indoles with nitrostyrenes: a simple practical synthesis of 3-substituted 2-quinolones. Chemical Communications (Cambridge, England). 49: 9305-7. PMID 23999797 DOI: 10.1039/C3Cc45696J |
0.351 |
|
| 2013 |
Frolova LV, Magedov IV, Romero AE, Karki M, Otero I, Hayden K, Evdokimov NM, Banuls LM, Rastogi SK, Smith WR, Lu SL, Kiss R, Shuster CB, Hamel E, Betancourt T, ... ... Kornienko A, et al. Exploring natural product chemistry and biology with multicomponent reactions. 5. Discovery of a novel tubulin-targeting scaffold derived from the rigidin family of marine alkaloids. Journal of Medicinal Chemistry. 56: 6886-900. PMID 23927793 DOI: 10.1021/Jm400711T |
0.739 |
|
| 2013 |
Magedov IV, Lefranc F, Frolova LV, Banuls LM, Peretti AS, Rogelj S, Mathieu V, Kiss R, Kornienko A. Antiproliferative activity of 2,3-disubstituted indoles toward apoptosis-resistant cancers cells. Bioorganic & Medicinal Chemistry Letters. 23: 3277-82. PMID 23622980 DOI: 10.1016/J.Bmcl.2013.03.110 |
0.361 |
|
| 2013 |
Bury M, Girault A, Mégalizzi V, Spiegl-Kreinecker S, Mathieu V, Berger W, Evidente A, Kornienko A, Gailly P, Vandier C, Kiss R. Ophiobolin A induces paraptosis-like cell death in human glioblastoma cells by decreasing BKCa channel activity. Cell Death & Disease. 4: e561. PMID 23538442 DOI: 10.1038/Cddis.2013.85 |
0.307 |
|
| 2013 |
Kornienko A, Mathieu V, Rastogi SK, Lefranc F, Kiss R. Therapeutic agents triggering nonapoptotic cancer cell death. Journal of Medicinal Chemistry. 56: 4823-39. PMID 23517069 DOI: 10.1021/Jm400136M |
0.357 |
|
| 2013 |
Van Goietsenoven G, Mathieu V, Lefranc F, Kornienko A, Evidente A, Kiss R. Narciclasine as well as other Amaryllidaceae isocarbostyrils are promising GTP-ase targeting agents against brain cancers. Medicinal Research Reviews. 33: 439-55. PMID 22419031 DOI: 10.1002/Med.21253 |
0.304 |
|
| 2013 |
Masi M, Andolfi A, Mathieu V, Boari A, Cimmino A, Moreno Y Banuls L, Vurro M, Kornienko A, Kiss R, Evidente A. Fischerindoline, a pyrroloindole sesquiterpenoid isolated from Neosartorya pseudofischeri, with in vitro growth inhibitory activity in human cancer cell lines Tetrahedron. 69: 7466-7470. DOI: 10.1016/J.Tet.2013.06.031 |
0.302 |
|
| 2012 |
Vshyvenko S, Scattolon J, Hudlicky T, Romero AE, Kornienko A, Ma D, Tuffley I, Pandey S. Unnatural C-1 homologues of pancratistatin - Synthesis and promising biological activities. Canadian Journal of Chemistry. 90: 932-943. PMID 28017970 DOI: 10.1139/V2012-073 |
0.443 |
|
| 2012 |
Magedov IV, Kornienko A. MULTICOMPONENT REACTIONS IN ALKALOID-BASED DRUG DISCOVERY. Chemistry of Heterocyclic Compounds. 48: 33-38. PMID 27917001 DOI: 10.1007/S10593-012-0965-7 |
0.355 |
|
| 2012 |
Magedov IV, Evdokimov NM, Karki M, Peretti AS, Lima DT, Frolova LV, Reisenauer MR, Romero AE, Tongwa P, Fonari A, Altig J, Rogelj S, Antipin MY, Shuster CB, Kornienko A. Reengineered epipodophyllotoxin. Chemical Communications (Cambridge, England). 48: 10416-8. PMID 22986348 DOI: 10.1039/c2cc35044k |
0.676 |
|
| 2012 |
Magedov IV, Kireev AS, Jenkins AR, Evdokimov NM, Lima DT, Tongwa P, Altig J, Steelant WF, Van slambrouck S, Antipin MY, Kornienko A. Structural simplification of bioactive natural products with multicomponent synthesis. 4. 4H-pyrano-[2,3-b]naphthoquinones with anticancer activity. Bioorganic & Medicinal Chemistry Letters. 22: 5195-8. PMID 22819765 DOI: 10.1016/J.Bmcl.2012.06.073 |
0.744 |
|
| 2012 |
Luchetti G, Johnston R, Mathieu V, Lefranc F, Hayden K, Andolfi A, Lamoral-Theys D, Reisenauer MR, Champion C, Pelly SC, van Otterlo WA, Magedov IV, Kiss R, Evidente A, Rogelj S, ... Kornienko A, et al. Bulbispermine: a crinine-type Amaryllidaceae alkaloid exhibiting cytostatic activity toward apoptosis-resistant glioma cells. Chemmedchem. 7: 815-22. PMID 22389235 DOI: 10.1002/Cmdc.201100608 |
0.416 |
|
| 2012 |
Cimmino A, Evidente A, Mathieu V, Andolfi A, Lefranc F, Kornienko A, Kiss R. Phenazines and cancer. Natural Product Reports. 29: 487-501. PMID 22337153 DOI: 10.1039/C2Np00079B |
0.395 |
|
| 2012 |
Abid O, Khalid M, Hussain MT, Hanif M, Qadeer G, Rama NH, Kornienko A, Khan KM. Synthesis and anti-cancer, anti-metastatic evaluation of some new fluorinated isocoumarins and 3,4-dihydroisocoumarins Journal of Fluorine Chemistry. 135: 240-245. DOI: 10.1016/J.Jfluchem.2011.11.011 |
0.433 |
|
| 2011 |
Frolova LV, Malik I, Uglinskii PY, Rogelj S, Kornienko A, Magedov IV. Multicomponent Synthesis of 2,3-Dihydrochromeno[4,3-d]pyrazolo[3,4-b]pyridine-1,6-diones: A Novel Heterocyclic Scaffold with Antibacterial Activity. Tetrahedron Letters. 52: 6643-6645. PMID 22162894 DOI: 10.1016/J.Tetlet.2011.10.012 |
0.469 |
|
| 2011 |
Evdokimov NM, Kornienko A, Magedov IV. Aryliodine (III) Diacetates as Substrates for Pd-Ag Catalyzed Arylation of Alkenes. Tetrahedron Letters. 52: 4327-4329. PMID 22058576 DOI: 10.1016/J.Tetlet.2011.06.051 |
0.672 |
|
| 2011 |
Evdokimov NM, Lamoral-Theys D, Mathieu V, Andolfi A, Frolova LV, Pelly SC, van Otterlo WA, Magedov IV, Kiss R, Evidente A, Kornienko A. In search of a cytostatic agent derived from the alkaloid lycorine: synthesis and growth inhibitory properties of lycorine derivatives. Bioorganic & Medicinal Chemistry. 19: 7252-61. PMID 22019045 DOI: 10.1016/J.Bmc.2011.09.051 |
0.743 |
|
| 2011 |
Vshyvenko S, Scattolon J, Hudlicky T, Romero AE, Kornienko A. Synthesis of C-1 homologues of pancratistatin and their preliminary biological evaluation. Bioorganic & Medicinal Chemistry Letters. 21: 4750-2. PMID 21757350 DOI: 10.1016/J.Bmcl.2011.06.068 |
0.464 |
|
| 2011 |
Daly S, Hayden K, Malik I, Porch N, Tang H, Rogelj S, Frolova LV, Lepthien K, Kornienko A, Magedov IV. Unprecedented C-2 arylation of indole with diazonium salts: Syntheses of 2,3-disubstituted indoles and their antimicrobial activity. Bioorganic & Medicinal Chemistry Letters. 21: 4720-3. PMID 21752646 DOI: 10.1016/J.Bmcl.2011.06.081 |
0.388 |
|
| 2011 |
Magedov IV, Frolova L, Manpadi M, Bhoga Ud, Tang H, Evdokimov NM, George O, Georgiou KH, Renner S, Getlik M, Kinnibrugh TL, Fernandes MA, Van slambrouck S, Steelant WF, Shuster CB, ... ... Kornienko A, et al. Anticancer properties of an important drug lead podophyllotoxin can be efficiently mimicked by diverse heterocyclic scaffolds accessible via one-step synthesis. Journal of Medicinal Chemistry. 54: 4234-46. PMID 21615090 DOI: 10.1021/Jm200410R |
0.744 |
|
| 2011 |
Evdokimov NM, Van Slambrouck S, Heffeter P, Tu L, Le Calvé B, Lamoral-Theys D, Hooten CJ, Uglinskii PY, Rogelj S, Kiss R, Steelant WF, Berger W, Yang JJ, Bologa CG, Kornienko A, et al. Structural simplification of bioactive natural products with multicomponent synthesis. 3. Fused uracil-containing heterocycles as novel topoisomerase-targeting agents. Journal of Medicinal Chemistry. 54: 2012-21. PMID 21388138 DOI: 10.1021/Jm1009428 |
0.768 |
|
| 2011 |
Frolova LV, Evdokimov NM, Hayden K, Malik I, Rogelj S, Kornienko A, Magedov IV. One-pot multicomponent synthesis of diversely substituted 2-aminopyrroles. A short general synthesis of rigidins A, B, C, and D. Organic Letters. 13: 1118-21. PMID 21268660 DOI: 10.1021/Ol103149B |
0.76 |
|
| 2010 |
Van Goietsenoven G, Andolfi A, Lallemand B, Cimmino A, Lamoral-Theys D, Gras T, Abou-Donia A, Dubois J, Lefranc F, Mathieu V, Kornienko A, Kiss R, Evidente A. Amaryllidaceae alkaloids belonging to different structural subgroups display activity against apoptosis-resistant cancer cells. Journal of Natural Products. 73: 1223-7. PMID 20550100 DOI: 10.1021/Np9008255 |
0.407 |
|
| 2010 |
Lamoral-Theys D, Pottier L, Kerff F, Dufrasne F, Proutière F, Wauthoz N, Neven P, Ingrassia L, Antwerpen PV, Lefranc F, Gelbcke M, Pirotte B, Kraus JL, Nève J, Kornienko A, et al. Simple di- and trivanillates exhibit cytostatic properties toward cancer cells resistant to pro-apoptotic stimuli. Bioorganic & Medicinal Chemistry. 18: 3823-33. PMID 20466556 DOI: 10.1016/J.Bmc.2010.04.047 |
0.422 |
|
| 2010 |
Collins J, Rinner U, Moser M, Hudlicky T, Ghiviriga I, Romero AE, Kornienko A, Ma D, Griffin C, Pandey S. Chemoenzymatic synthesis of Amaryllidaceae constituents and biological evaluation of their C-1 analogues. The next generation synthesis of 7-deoxypancratistatin and trans-dihydrolycoricidine. The Journal of Organic Chemistry. 75: 3069-84. PMID 20373760 DOI: 10.1021/Jo1003136 |
0.465 |
|
| 2010 |
Lamoral-Theys D, Pottier L, Dufrasne F, Nève J, Dubois J, Kornienko A, Kiss R, Ingrassia L. Natural polyphenols that display anticancer properties through inhibition of kinase activity. Current Medicinal Chemistry. 17: 812-25. PMID 20156174 DOI: 10.2174/092986710790712183 |
0.326 |
|
| 2010 |
Lamoral-Theys D, Decaestecker C, Mathieu V, Dubois J, Kornienko A, Kiss R, Evidente A, Pottier L. Lycorine and its derivatives for anticancer drug design. Mini Reviews in Medicinal Chemistry. 10: 41-50. PMID 20105122 DOI: 10.2174/138955710791112604 |
0.362 |
|
| 2009 |
Lamoral-Theys D, Andolfi A, Van Goietsenoven G, Cimmino A, Le Calvé B, Wauthoz N, Mégalizzi V, Gras T, Bruyère C, Dubois J, Mathieu V, Kornienko A, Kiss R, Evidente A. Lycorine, the main phenanthridine Amaryllidaceae alkaloid, exhibits significant antitumor activity in cancer cells that display resistance to proapoptotic stimuli: an investigation of structure-activity relationship and mechanistic insight. Journal of Medicinal Chemistry. 52: 6244-56. PMID 19788245 DOI: 10.1021/Jm901031H |
0.389 |
|
| 2009 |
Manpadi M, Kireev AS, Magedov IV, Altig J, Tongwa P, Antipin MY, Evidente A, van Otterlo WA, Kornienko A. Synthesis of structurally simplified analogues of pancratistatin: truncation of the cyclitol ring. The Journal of Organic Chemistry. 74: 7122-31. PMID 19743883 DOI: 10.1021/Jo901494R |
0.444 |
|
| 2009 |
Evidente A, Kireev AS, Jenkins AR, Romero AE, Steelant WF, Van Slambrouck S, Kornienko A. Biological evaluation of structurally diverse amaryllidaceae alkaloids and their synthetic derivatives: discovery of novel leads for anticancer drug design. Planta Medica. 75: 501-7. PMID 19235683 DOI: 10.1055/S-0029-1185340 |
0.4 |
|
| 2009 |
Evidente A, Kornienko A. Anticancer evaluation of structurally diverse Amaryllidaceae alkaloids and their synthetic derivatives Phytochemistry Reviews. 8: 449-459. DOI: 10.1007/S11101-008-9119-Z |
0.34 |
|
| 2008 |
Luchetti G, Ding K, Kornienko A, d'Alarcao M. Synthesis of Differentially Protected myo- and chiro-Inositols from D-Xylose; Stereoselectivity in Intramolecular SmI(2)-Promoted Pinacol Reactions. Synthesis. 2008: 3148-3154. PMID 20622936 DOI: 10.1055/S-2008-1067259 |
0.729 |
|
| 2008 |
Luchetti G, Ding K, d'Alarcao M, Kornienko A. Enantio- and Diastereodivergent Synthetic Route to Multifarious Cyclitols from D-Xylose via Ring-Closing Metathesis. Synthesis. 2008: 3142-3147. PMID 19802347 DOI: 10.1055/S-2008-1067260 |
0.734 |
|
| 2008 |
Kornienko A, Evidente A. Chemistry, biology, and medicinal potential of narciclasine and its congeners. Chemical Reviews. 108: 1982-2014. PMID 18489166 DOI: 10.1021/Cr078198U |
0.351 |
|
| 2008 |
Sigstedt SC, Hooten CJ, Callewaert MC, Jenkins AR, Romero AE, Pullin MJ, Kornienko A, Lowrey TK, Slambrouck SV, Steelant WF. Evaluation of aqueous extracts of Taraxacum officinale on growth and invasion of breast and prostate cancer cells. International Journal of Oncology. 32: 1085-90. PMID 18425335 DOI: 10.3892/Ijo.32.5.1085 |
0.306 |
|
| 2008 |
Magedov IV, Manpadi M, Ogasawara MA, Dhawan AS, Rogelj S, Van Slambrouck S, Steelant WF, Evdokimov NM, Uglinskii PY, Elias EM, Knee EJ, Tongwa P, Antipin MY, Kornienko A. Structural simplification of bioactive natural products with multicomponent synthesis. 2. antiproliferative and antitubulin activities of pyrano[3,2-c]pyridones and pyrano[3,2-c]quinolones. Journal of Medicinal Chemistry. 51: 2561-70. PMID 18361483 DOI: 10.1021/Jm701499N |
0.749 |
|
| 2008 |
Magedov IV, Luchetti G, Evdokimov NM, Manpadi M, Steelant WF, Van Slambrouck S, Tongwa P, Antipin MY, Kornienko A. Novel three-component synthesis and antiproliferative properties of diversely functionalized pyrrolines. Bioorganic & Medicinal Chemistry Letters. 18: 1392-6. PMID 18221874 DOI: 10.1016/J.Bmcl.2008.01.019 |
0.73 |
|
| 2007 |
Manpadi M, Uglinskii PY, Rastogi SK, Cotter KM, Wong YS, Anderson LA, Ortega AJ, Van Slambrouck S, Steelant WF, Rogelj S, Tongwa P, Antipin MY, Magedov IV, Kornienko A. Three-component synthesis and anticancer evaluation of polycyclic indenopyridines lead to the discovery of a novel indenoheterocycle with potent apoptosis inducing properties. Organic & Biomolecular Chemistry. 5: 3865-72. PMID 18004468 DOI: 10.1039/B713820B |
0.447 |
|
| 2007 |
Magedov IV, Manpadi M, Slambrouck SV, Steelant WF, Rozhkova E, Przheval'skii NM, Rogelj S, Kornienko A. Discovery and investigation of antiproliferative and apoptosis-inducing properties of new heterocyclic podophyllotoxin analogues accessible by a one-step multicomponent synthesis. Journal of Medicinal Chemistry. 50: 5183-92. PMID 17894480 DOI: 10.1021/Jm070528F |
0.473 |
|
| 2007 |
Magedov IV, Manpadi M, Evdokimov NM, Elias EM, Rozhkova E, Ogasawara MA, Bettale JD, Przheval'skii NM, Rogelj S, Kornienko A. Antiproliferative and apoptosis inducing properties of pyrano[3,2-c]pyridones accessible by a one-step multicomponent synthesis. Bioorganic & Medicinal Chemistry Letters. 17: 3872-6. PMID 17512729 DOI: 10.1016/J.Bmcl.2007.05.004 |
0.741 |
|
| 2007 |
Evdokimov NM, Kireev AS, Yakovenko AA, Antipin MY, Magedov IV, Kornienko A. One-step synthesis of heterocyclic privileged medicinal scaffolds by a multicomponent reaction of malononitrile with aldehydes and thiols. The Journal of Organic Chemistry. 72: 3443-53. PMID 17408286 DOI: 10.1021/Jo070114U |
0.745 |
|
| 2007 |
Magedov IV, Manpadi M, Rozhkova E, Przheval'skii NM, Rogelj S, Shors ST, Steelant WF, Van slambrouck S, Kornienko A. Structural simplification of bioactive natural products with multicomponent synthesis: dihydropyridopyrazole analogues of podophyllotoxin. Bioorganic & Medicinal Chemistry Letters. 17: 1381-5. PMID 17188868 DOI: 10.1016/J.Bmcl.2006.11.095 |
0.427 |
|
| 2006 |
Evdokimov NM, Kireev AS, Yakovenko AA, Antipin MY, Magedov IV, Kornienko A. Convenient one-step synthesis of a medicinally relevant benzopyranopyridine system. Tetrahedron Letters. 47: 9309-9312. PMID 23243322 DOI: 10.1016/J.Tetlet.2006.10.110 |
0.73 |
|
| 2006 |
Rastogi SK, Kornienko A. A solution to the stereochemical problems posed by amaryllidaceae constituents using a highly syn-selective arylcuprate conjugate addition to γ-amino and γ-carbamato-α,β-enoates. Tetrahedron, Asymmetry. 17: 3170-3176. PMID 22791936 DOI: 10.1016/J.Tetasy.2006.11.029 |
0.307 |
|
| 2006 |
Kireev AS, Nadein ON, Agustin VJ, Bush NE, Evidente A, Manpadi M, Ogasawara MA, Rastogi SK, Rogelj S, Shors ST, Kornienko A. Synthesis and biological evaluation of aromatic analogues of conduritol F, L-chiro-inositol, and dihydroconduritol F structurally related to the amaryllidaceae anticancer constituents. The Journal of Organic Chemistry. 71: 5694-707. PMID 16839151 DOI: 10.1021/Jo0607562 |
0.404 |
|
| 2006 |
Kireev AS, Manpadi M, Kornienko A. Selectivity guidelines and a reductive elimination-based model for predicting the stereochemical course of conjugate addition reactions of organocuprates to gamma-alkoxy-alpha,beta-enoates. The Journal of Organic Chemistry. 71: 2630-40. PMID 16555814 DOI: 10.1021/Jo052383V |
0.318 |
|
| 2006 |
Evdokimov NM, Magedov IV, Kireev AS, Kornienko A. One-step, three-component synthesis of pyridines and 1,4-dihydropyridines with manifold medicinal utility. Organic Letters. 8: 899-902. PMID 16494469 DOI: 10.1021/Ol052994+ |
0.732 |
|
| 2005 |
Kireev AS, Breithaupt AT, Collins W, Nadein ON, Kornienko A. Enantiodivergent formal synthesis of (+)-and (-)-cyclophellitol from D-xylose based on the latent symmetry concept Journal of Organic Chemistry. 70: 742-745. PMID 15651835 DOI: 10.1021/Jo048459P |
0.46 |
|
| 2005 |
Manpadi M, Kornienko A. Highly anti-selective conjugate addition of arylcuprates to a γ-alkoxy-α,β-enoate. a new method to address stereochemical challenges presented by Amaryllidaceae alkaloids Tetrahedron Letters. 46: 4433-4437. DOI: 10.1016/J.Tetlet.2005.05.006 |
0.329 |
|
| 2004 |
Nadein ON, Kornienko A. An approach to pancratistatins via ring-closing metathesis: efficient synthesis of novel 1-aryl-1-deoxyconduritols F. cv. Organic Letters. 6: 831-4. PMID 14986986 DOI: 10.1021/Ol049942P |
0.434 |
|
| 2003 |
Hanessian S, Kornienko A, Swayze EE. Probing the functional requirements of the L-haba side-chain of amikacin - Synthesis, 16S A-site rRNA binding, and antibacterial activity Tetrahedron. 59: 995-1007. DOI: 10.1016/S0040-4020(02)01625-3 |
0.319 |
|
| 2001 |
Hanessian S, Tremblay M, Kornienko A, Moitessier N. Design, modeling and synthesis of functionalized paromamine analogs Tetrahedron. 57: 3255-3265. DOI: 10.1016/S0040-4020(01)00194-6 |
0.307 |
|
| 1999 |
Kornienko A, d'Alarcao M. Synthesis of cyclitols via ring-closing metathesis Tetrahedron-Asymmetry. 10: 827-829. DOI: 10.1016/S0957-4166(99)00065-8 |
0.737 |
|
| 1998 |
Kornienko A, Marnera G, d'Alarcao M. Synthesis of a jojoba bean disaccharide. Carbohydrate Research. 310: 141-4. PMID 9794077 DOI: 10.1016/S0008-6215(98)00168-2 |
0.722 |
|
| 1998 |
Kornienko A, Turner DI, Jaworek CH, D'Alarcao M. Practical synthesis of a differentially protected myo-inositol Tetrahedron Asymmetry. 9: 2783-2786. DOI: 10.1016/S0957-4166(98)00302-4 |
0.752 |
|
| 1997 |
Kornienko A, d'Alarcao M. Enantiospecific synthesis of a differentially protected L-chiro-inositol from D-xylose Tetrahedron Letters. 38: 6497-6500. DOI: 10.1016/S0040-4039(97)01513-X |
0.734 |
|
| Show low-probability matches. |