Year |
Citation |
Score |
2020 |
Verhoeven J, Deraet X, Pande V, Sun W, Alonso M, De Proft F, Meerpoel L, Thuring JW, Verniest G. Synthesis and Reactivity of Spirocarbocycles as Scaffolds for Nucleoside Analogues. The Journal of Organic Chemistry. PMID 33196210 DOI: 10.1021/acs.joc.0c01825 |
0.336 |
|
2019 |
Verhoeven J, De Vleeschouwer F, Kong H, Van Hecke K, Pande V, Sun W, Vos A, Wu T, Meerpoel L, Thuring JW, Verniest G. Preparation of 4'-Spirocyclobutyl Nucleoside Analogues as Novel and Versatile Adenosine Scaffolds. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 31609050 DOI: 10.1002/chem.201904574 |
0.322 |
|
2019 |
Hernández-Molina Y, Verniest G, Casals-Hung M, Acevedo-MartÃnez J, Cos P. Synthesis and biological evaluation of benzimidazolyl substituted aloe-emodin derivatives Arkivoc. 2019: 152-162. DOI: 10.24820/Ark.5550190.P010.684 |
0.454 |
|
2018 |
Marien N, Bheemireddy NR, De Vleeschouwer F, Goderis S, Van Hecke K, Verniest G. Metal-free cyclization of o-nitroaryl ynamides and ynamines towards spiropseudoindoxyls. Angewandte Chemie (International Ed. in English). PMID 29570239 DOI: 10.1002/anie.201800340 |
0.345 |
|
2017 |
Verniest G, Marien N, Luo T. Synthesis of Piperidinone and Azepanone Fused Indoles via a Wagner–Meerwein Type 1,2-Amide Migration of 2-Spiropseudoindoxyls Synlett. 28: 934-938. DOI: 10.1055/S-0036-1588138 |
0.312 |
|
2017 |
Marien N, Verniest G. Gold(I)-catalyzed synthesis of dihydrodibenzoquinolizinium salts Advanced Synthesis & Catalysis. 359: 1996-2000. DOI: 10.1002/ADSC.201700126 |
0.364 |
|
2016 |
Verlinden S, Ballet S, Verniest G. Synthesis of Heterocycle-Bridged Peptidic Macrocycles through 1,3-Diyne Transformations European Journal of Organic Chemistry. 2016: 5807-5812. DOI: 10.1002/Ejoc.201601215 |
0.464 |
|
2015 |
Meiresonne T, Verniest G, De Kimpe N, Mangelinckx S. Synthesis of 2-Fluoro-1,4-benzoxazines and 2-Fluoro-1,4-benzoxazepin-5-ones by Exploring the Nucleophilic Vinylic Substitution (S(N)V) Reaction of gem-Difluoroenamides. The Journal of Organic Chemistry. 80: 5111-24. PMID 25901523 DOI: 10.1021/Acs.Joc.5B00507 |
0.756 |
|
2015 |
Marien N, Brigou B, Pinter B, De Proft F, Verniest G. Synthesis of 2-spiropseudoindoxyls via an intramolecular nitroalkyne redox-dipolar cycloaddition cascade. Organic Letters. 17: 270-3. PMID 25545133 DOI: 10.1021/Ol503364W |
0.477 |
|
2015 |
Meiresonne T, Verniest G, De Kimpe N, Mangelinckx S. ChemInform Abstract: Synthesis of 2-Fluoro-1,4-benzoxazines and 2-Fluoro-1,4-benzoxazepin-5-ones by Exploring the Nucleophilic Vinylic Substitution (SNV) Reaction of gem-Difluoroenamides. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201539159 |
0.39 |
|
2014 |
Schurgers B, Brigou B, Urbanczyk-Lipkowska Z, Tourwé D, Ballet S, De Proft F, Van Lommen G, Verniest G. Synthesis of fused 3-aminoazepinones via trapping of a new class of cyclic seven-membered allenamides with furan. Organic Letters. 16: 3712-5. PMID 25007412 DOI: 10.1021/Ol501529Z |
0.516 |
|
2013 |
Kenis S, D'hooghe M, Verniest G, Reybroeck M, Dang Thi TA, Pham The C, Thi Pham T, Törnroos KW, Van Tuyen N, De Kimpe N. Nucleophile-directed selective transformation of cis-1-tosyl-2-tosyloxymethyl-3-(trifluoromethyl)aziridine into aziridines, azetidines, and benzo-fused dithianes, oxathianes, dioxanes, and (thio)morpholines. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 5966-71. PMID 23512331 DOI: 10.1002/Chem.201204485 |
0.733 |
|
2013 |
Moens M, Verniest G, De Schrijver M, ten Holte P, Thuring J, Deroose F, De Kimpe N. ChemInform Abstract: Synthesis of 2-Aryl-3-hydroxymethyl-5,5-difluoropiperidines. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201312129 |
0.401 |
|
2013 |
Piron K, Kenis S, Verniest G, Surmont R, Thuring JW, ten Holte P, Deroose F, De Kimpe N. ChemInform Abstract: Synthesis of gem-Difluorinated 1,6-Naphthyridine-5,7-diones. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201301140 |
0.373 |
|
2013 |
Pace V, Holzer W, Verniest G, Alcántara AR, De Kimpe N. Chemoselective Synthesis ofN-Substituted α-Amino-α′-chloro KetonesviaChloromethylation of Glycine-Derived Weinreb Amides Advanced Synthesis & Catalysis. 355: 919-926. DOI: 10.1002/Adsc.201201043 |
0.521 |
|
2012 |
Kenis S, D'hooghe M, Verniest G, Dang Thi TA, Pham The C, Van Nguyen T, De Kimpe N. Synthesis of 1-alkyl-2-(trifluoromethyl)azetidines and their regiospecific ring opening toward diverse α-(trifluoromethyl)amines via intermediate azetidinium salts. The Journal of Organic Chemistry. 77: 5982-92. PMID 22721444 DOI: 10.1021/Jo300694Y |
0.737 |
|
2012 |
Moens M, Verniest G, De Schrijver M, ten Holte P, Thuring J, Deroose F, De Kimpe N. Synthesis of 2-aryl-3-hydroxymethyl-5,5-difluoropiperidines Tetrahedron. 68: 9284-9288. DOI: 10.1016/J.Tet.2012.08.049 |
0.54 |
|
2012 |
Piron K, Kenis S, Verniest G, Surmont R, Thuring JW, ten Holte P, Deroose F, De Kimpe N. Synthesis of gem-difluorinated 1,6-naphthyridine-5,7-diones Tetrahedron. 68: 6941-6947. DOI: 10.1016/J.Tet.2012.05.122 |
0.475 |
|
2011 |
Kenis S, D'hooghe M, Verniest G, Nguyen VD, Thi TA, Nguyen TV, De Kimpe N. Straightforward synthesis of 1-alkyl-2-(trifluoromethyl)aziridines starting from 1,1,1-trifluoroacetone. Organic & Biomolecular Chemistry. 9: 7217-23. PMID 21874207 DOI: 10.1039/C1Ob05813D |
0.747 |
|
2011 |
Surmont R, Verniest G, De Schrijver M, Thuring JW, ten Holte P, Deroose F, De Kimpe N. Synthesis of 3-amino-4-fluoropyrazoles. The Journal of Organic Chemistry. 76: 4105-11. PMID 21500813 DOI: 10.1021/Jo2000989 |
0.617 |
|
2011 |
Piron K, Verniest G, Hende EV, Kimpe ND. Synthesis of 3-fluoropyrrolidines and 3-fluoroazetidines Arkivoc. 2012. DOI: 10.3998/Ark.5550190.0013.502 |
0.437 |
|
2010 |
Surmont R, Verniest G, De Kimpe N. New synthesis of fluorinated pyrazoles. Organic Letters. 12: 4648-51. PMID 20843014 DOI: 10.1021/Ol1019713 |
0.644 |
|
2010 |
Surmont R, Verniest G, De Kimpe N. Short synthesis of the seed germination inhibitor 3,4,5-trimethyl-2(5H)-furanone. The Journal of Organic Chemistry. 75: 5750-3. PMID 20704450 DOI: 10.1021/Jo1010476 |
0.589 |
|
2010 |
Pace V, Verniest G, Sinisterra JV, Alcántara AR, De Kimpe N. Improved Arndt-Eistert synthesis of alpha-diazoketones requiring minimal diazomethane in the presence of calcium oxide as acid scavenger. The Journal of Organic Chemistry. 75: 5760-3. PMID 20672806 DOI: 10.1021/Jo101105G |
0.57 |
|
2010 |
Surmont R, Verniest G, Thuring JW, Ten Holte P, Deroose F, De Kimpe N. Synthesis of 5-amino- and 5-hydroxy-3,3-difluoropiperidines. Organic & Biomolecular Chemistry. 8: 4514-7. PMID 20668779 DOI: 10.1039/C0Ob00231C |
0.656 |
|
2010 |
Verniest G, Piron K, Van Hende E, Thuring JW, Macdonald G, Deroose F, De Kimpe N. Synthesis of aminomethylated 4-fluoropiperidines and 3-fluoropyrrolidines. Organic & Biomolecular Chemistry. 8: 2509-12. PMID 20407687 DOI: 10.1039/C003380D |
0.661 |
|
2010 |
Surmont R, Verniest G, Thuring JW, Macdonald G, Deroose F, De Kimpe N. Synthesis of 4-substituted 3,3-difluoropiperidines. The Journal of Organic Chemistry. 75: 929-32. PMID 20050617 DOI: 10.1021/Jo902164Z |
0.68 |
|
2010 |
Verniest G, Wang X, De Kimpe N, Padwa A. Heteroaryl cross-coupling as an entry toward the synthesis of lavendamycin analogues: a model study. The Journal of Organic Chemistry. 75: 424-33. PMID 20017470 DOI: 10.1021/Jo902287T |
0.668 |
|
2010 |
Verniest G, England D, De Kimpe N, Padwa A. Synthesis of substituted β-carbolines via gold(III)-catalyzed cycloisomerization of N-propargylamides Tetrahedron. 66: 1496-1502. DOI: 10.1016/J.Tet.2009.10.033 |
0.561 |
|
2010 |
Verniest G, England D, De Kimpe N, Padwa A. ChemInform Abstract: Synthesis of Substituted β-Carbolines via Gold(III)-Catalyzed Cycloisomerization of N-Propargylamides. Cheminform. 41: no-no. DOI: 10.1002/CHIN.201024146 |
0.53 |
|
2010 |
Surmont R, Verniest G, De Groot A, Thuring JW, De Kimpe N. Morpholinosulfur Trifluoride (Morph-DAST)-Mediated Rearrangement in the Fluorination of Cyclic α,α-Dialkoxy Ketones toward 1,2-Dialkoxy-1,2-difluorinated Compounds Advanced Synthesis & Catalysis. 352: 2751-2756. DOI: 10.1002/Adsc.201000466 |
0.389 |
|
2009 |
Surmont R, Verniest G, De Kimpe N. Gold-catalyzed synthesis of 2-aryl-3-fluoropyrroles. Organic Letters. 11: 2920-3. PMID 19507840 DOI: 10.1021/Ol900953N |
0.684 |
|
2009 |
De Sterck B, Van Speybroeck V, Mangelinckx S, Verniest G, De Kimpe N, Waroquier M. Theoretical study on the structural properties of various solvated metalated 3-halo-1-azaallylic anions. The Journal of Physical Chemistry. A. 113: 6375-80. PMID 19425551 DOI: 10.1021/Jp811317Y |
0.7 |
|
2009 |
Colpaert F, Mangelinckx S, Verniest G, De Kimpe N. Asymmetric synthesis of alpha-alkylated N-sulfinyl imidates as new chiral building blocks. The Journal of Organic Chemistry. 74: 3792-7. PMID 19366202 DOI: 10.1021/Jo900046T |
0.759 |
|
2009 |
Van Hende E, Verniest G, Deroose F, Thuring JW, Macdonald G, De Kimpe N. Synthesis of 1-Boc-3-fluoroazetidine-3-carboxylic acid. The Journal of Organic Chemistry. 74: 2250-3. PMID 19216497 DOI: 10.1021/Jo802791R |
0.617 |
|
2009 |
Surmont R, Verniest G, Colpaert F, Macdonald G, Thuring JW, Deroose F, De Kimpe N. New synthesis of 3-fluoropyrroles. The Journal of Organic Chemistry. 74: 1377-80. PMID 19115927 DOI: 10.1021/Jo802272N |
0.631 |
|
2009 |
Declerck R, De Sterck B, Verstraelen T, Verniest G, Mangelinckx S, Jacobs J, De Kimpe N, Waroquier M, Van Speybroeck V. Insight into the solvation and isomerization of 3-halo-1-azaallylic anions from ab initio metadynamics calculations and NMR experiments. Chemistry (Weinheim An Der Bergstrasse, Germany). 15: 580-4. PMID 18991305 DOI: 10.1002/Chem.200800948 |
0.667 |
|
2009 |
De Kimpe N, Surmont R, Verniest G, De Weweire A, Thuring J, Macdonald G, Deroose F. Efficient Synthesis of 3-Alkoxy-4,4-difluoropiperidines Synlett. 2009: 1933-1936. DOI: 10.1055/S-0029-1217533 |
0.476 |
|
2009 |
De Kimpe N, Van Hende E, Verniest G, Thuring J, Macdonald G, Deroose F. Synthesis of 3-Aminomethyl-3-fluoropiperidines Synlett. 2009: 1765-1768. DOI: 10.1055/S-0029-1217360 |
0.557 |
|
2009 |
Surmont R, Verniest G, De Weweire A, Thuring JW, Macdonald G, Deroose F, De Kimpe N. ChemInform Abstract: Efficient Synthesis of 3-Alkoxy-4,4-difluoropiperidines. Cheminform. 40. DOI: 10.1002/CHIN.200950156 |
0.326 |
|
2009 |
Van Hende E, Verniest G, Thuring J, Macdonald G, Deroose F, De Kimpe N. ChemInform Abstract: Synthesis of 3-Aminomethyl-3-fluoropiperidines. Cheminform. 40. DOI: 10.1002/CHIN.200949145 |
0.359 |
|
2008 |
Verniest G, Padwa A. Gold- and silver-mediated cycloisomerizations of N-propargylamides. Organic Letters. 10: 4379-82. PMID 18763788 DOI: 10.1021/Ol801847J |
0.516 |
|
2008 |
Verniest G, Surmont R, Van Hende E, Deweweire A, Deroose F, Thuring JW, De Kimpe N. New entries toward 3,3-difluoropiperidines. The Journal of Organic Chemistry. 73: 5458-61. PMID 18547110 DOI: 10.1021/Jo800768Q |
0.681 |
|
2008 |
Karikomi M, D'hooghe M, Verniest G, De Kimpe N. Regio- and stereocontrolled synthesis of novel 3-sulfonamido-2,3,4,5-tetrahydro-1,5-benzothiazepines from 2-(bromomethyl)- or 2-(sulfonyloxymethyl)aziridines. Organic & Biomolecular Chemistry. 6: 1902-4. PMID 18480901 DOI: 10.1039/B804246M |
0.762 |
|
2008 |
Karikomi M, D'hooghe M, Verniest G, De Kimpe N. ChemInform Abstract: Regio- and Stereocontrolled Synthesis of Novel 3-Sulfonamido-2,3,4,5-tetrahydro-1,5-benzothiazepines from 2-(Bromomethyl)- or 2-(Sulfonyloxymethyl)aziridines. Cheminform. 39. DOI: 10.1002/CHIN.200841173 |
0.393 |
|
2007 |
Verniest G, Colpaert F, Van Hende E, De Kimpe N. Synthesis and reactivity of 1-substituted 2-fluoro- and 2,2-difluoroaziridines. The Journal of Organic Chemistry. 72: 8569-72. PMID 17915923 DOI: 10.1021/Jo071253E |
0.654 |
|
2007 |
Van Hende E, Verniest G, Surmont R, De Kimpe N. Synthesis of 3-substituted 2-fluoro- and 2,2-difluoroaziridines. Organic Letters. 9: 2935-7. PMID 17602490 DOI: 10.1021/Ol071127X |
0.599 |
|
2007 |
Vansteenkiste P, Van Speybroeck V, Verniest G, De Kimpe N, Waroquier M. Four-membered heterocycles with a carbon-heteroatom exocyclic double bond at the 3-position: puckering potential and thermodynamic properties. The Journal of Physical Chemistry. A. 111: 2797-803. PMID 17388369 DOI: 10.1021/Jp068454R |
0.577 |
|
2007 |
Claessens S, Verniest G, Jacobs J, Van Hende E, Habonimana P, Nguyen Van T, Van Puyvelde L, De Kimpe N. A Survey of Synthetic Routes Towards the Pyranonaphthoquinone Antibiotic Pentalongin and Syntheses of the Corresponding Nitrogen Derivatives Cheminform. 38. DOI: 10.1055/S-2007-973888 |
0.372 |
|
2006 |
Verniest G, Van Hende E, Surmont R, De Kimpe N. Direct electrophilic alpha-fluorination of imines: efficient synthesis of mono- and difluoroimines. Organic Letters. 8: 4767-70. PMID 17020298 DOI: 10.1021/Ol061720Z |
0.579 |
|
2006 |
Van Brabandt W, Verniest G, De Smaele D, Duvey G, De Kimpe N. Synthesis of 3-fluoroazetidines. The Journal of Organic Chemistry. 71: 7100-2. PMID 16930075 DOI: 10.1021/Jo061095B |
0.617 |
|
2006 |
Vansteenkiste P, Van Speybroeck V, Verniest G, De Kimpe N, Waroquier M. Applicability of the hindered rotor scheme to the puckering mode in four-membered rings. The Journal of Physical Chemistry. A. 110: 3838-44. PMID 16526670 DOI: 10.1021/Jp056211D |
0.521 |
|
2006 |
Verniest G, Claessens S, De Kimpe N. Stereoselective Reduction of N-(3-Arylcyclobutylidene)amines. Cheminform. 37. DOI: 10.1016/J.Tetlet.2006.03.023 |
0.479 |
|
2006 |
Claessens S, Verniest G, El Hady S, Nguyen Van T, Kesteleyn B, Van Puyvelde L, De Kimpe N. The behaviour of the natural pyranonaphthoquinone pentalongin in alcoholic solvents Tetrahedron. 62: 5152-5158. DOI: 10.1016/J.Tet.2006.03.018 |
0.321 |
|
2005 |
Verniest G, Colpaert J, Törnroos KW, De Kimpe N. New synthesis of semisquaric acid derivatives via chlorinated N-(cyclobutylidene)amines. The Journal of Organic Chemistry. 70: 4549-52. PMID 15903345 DOI: 10.1021/Jo0502044 |
0.676 |
|
2005 |
Verniest G, De Kimpe N. Synthesis of 2(5H)-Furanones via Oxidative Ring Expansion of 4-Hydroxy-2-cyclobutenones. Cheminform. 36. DOI: 10.1055/S-2005-864805 |
0.44 |
|
2005 |
Verniest G, Colpaert J, Törnroos KW, De Kimpe N. New synthesis of semisquaric acid derivatives via chlorinated N-(cyclobutylidene)amines Journal of Organic Chemistry. 70: 4549-4552. DOI: 10.1021/jo0502044 |
0.627 |
|
2005 |
Verniest G, Claessens S, De Kimpe N. Synthesis of chlorinated 2-(aminomethyl)- and 2-(alkoxymethyl)pyrroles Tetrahedron. 61: 4631-4637. DOI: 10.1016/J.TET.2005.02.086 |
0.394 |
|
2005 |
Verniest G, Claessens S, De Kimpe N. Synthesis of Chlorinated 2-(Aminomethyl)- and 2-(Alkoxymethyl)pyrroles. Cheminform. 36. DOI: 10.1016/J.Tet.2005.02.086 |
0.494 |
|
2005 |
Verniest G, Claessens S, Bombeke F, Thienen TV, Kimpe ND. Synthesis of 2-aryl-4-chloropyrroles via ring expansion of 2-aryl-1-chlorocyclopropanecarbaldehydes Tetrahedron. 61: 2879-2887. DOI: 10.1016/J.Tet.2005.01.087 |
0.5 |
|
2005 |
Nguyen Van T, Verniest G, Claessens S, De Kimpe N. Total synthesis of four naturally occurring 2-azaanthraquinone antibiotics, 6-deoxy-8-methylbostrycoidin, 6-deoxybostrycoidin, 7-O-demethyl-6-deoxybostrycoidin and scorpinone Tetrahedron. 61: 2295-2300. DOI: 10.1016/J.Tet.2005.01.035 |
0.365 |
|
2005 |
Verniest G, Claessens S, Bombeke F, Van Thienen T, De Kimpe N. Synthesis of 2-Aryl-4-chloropyrroles via Ring Expansion of 2-Aryl-1-chlorocyclopropanecarbaldehydes. Cheminform. 36. DOI: 10.1002/CHIN.200530095 |
0.398 |
|
2004 |
Verniest G, Boterberg S, Colpaert J, Van Thienen T, Stevens CV, De Kimpe N. Synthesis of 2-Substituted Cyclobutanones as γ-Irradiation Marker Products of Lipid-Containing Foods. Cheminform. 35. DOI: 10.1055/S-2004-825590 |
0.531 |
|
2004 |
Verniest G, Boterberg S, Bombeke F, Stevens CV, De Kimpe N. New Ring Expansion of Cyclobutanones: Synthesis of Pyrrolinones, Pyrrolidines and Pyrroles. Cheminform. 35. DOI: 10.1055/S-2004-822900 |
0.637 |
|
2004 |
Verniest G, De Kimpe N. New Synthesis of 3-Arylpyrroles. Cheminform. 35. DOI: 10.1055/S-2003-42047 |
0.481 |
|
2003 |
Salgado A, Dejaegher Y, Verniest G, Boeykens M, Gauthier C, Lopin C, Tehrani KA, De Kimpe N. Synthesis of 1-Alkyl-2-methylazetidin-3-ones and 1-Alkyl-2-methylazetidin-3-ols. Cheminform. 34. DOI: 10.1016/S0040-4020(03)00241-2 |
0.482 |
|
2003 |
Salgado A, Dejaegher Y, Verniest G, Boeykens M, Gauthier C, Lopin C, Tehrani KA, De Kimpe N. Synthesis of 1-alkyl-2-methylazetidin-3-ones and 1-alkyl-2-methylazetidin-3-ols Tetrahedron. 59: 2231-2239. DOI: 10.1016/S0040-4020(03)00241-2 |
0.443 |
|
2002 |
Verniest G, Bombeke F, Kulinkovich O, De Kimpe N. Stereoselective synthesis of cis-2-aryl- and 2-alkyl-1-chlorocyclopropanecarboxaldehydes Tetrahedron Letters. 43: 599-602. DOI: 10.1016/S0040-4039(01)02228-6 |
0.525 |
|
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