Sitthivut Charoensutthivarakul - Related publications

Affiliations: 
2010-2014 Chemistry University of Liverpool, Liverpool, England, United Kingdom 
 2017-2019 Chemistry University of Cambridge, Cambridge, England, United Kingdom 
Area:
Medicinal Chemistry
NOTE: We are testing a new system for identifying relevant work based on semantic analysis that identifies similarities between recently published papers and the current author's publications. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches.
50 most relevant papers in past 60 days:
Year Citation  Score
2021 Chia W, Gomez-Lorenzo MG, Castellote I, Tong JX, Chandramohanadas R, Thu Chu TT, Shen W, Go ML, de Cozar C, Crespo B, Almela MJ, Neria-Serrano F, Franco V, Gamo FJ, Tan KSW. High-Content Phenotypic Screen of a Focused TCAMS Drug Library Identifies Novel Disruptors of the Malaria Parasite Calcium Dynamics. Acs Chemical Biology. PMID 34609851 DOI: 10.1021/acschembio.1c00512   
2021 González-Bacerio J, Arocha I, Aguado ME, Méndez Y, Marsiccobetre S, Izquierdo M, Rivera DG, Figarella K, Uzcátegui NL. KBE009: A Bestatin-Like Inhibitor of the Acidic M17 Aminopeptidase with In Vitro Anti-Trypanosomal Activity. Life (Basel, Switzerland). 11. PMID 34685408 DOI: 10.3390/life11101037   
2021 Ashton TD, Ngo A, Favuzza P, Bullen HE, Gancheva MR, Romeo O, Parkyn Schneider M, Nguyen N, Steel RWJ, Duffy S, Lowes KN, Sabroux HJ, Avery VM, Boddey JA, Wilson DW, et al. Property activity refinement of 2-anilino 4-amino substituted quinazolines as antimalarials with fast acting asexual parasite activity. Bioorganic Chemistry. 117: 105359. PMID 34689083 DOI: 10.1016/j.bioorg.2021.105359   
2021 Cooper RA, Kirkman L. Can repurposing drugs play a role in malaria control? The Journal of Experimental Medicine. 218. PMID 34807244 DOI: 10.1084/jem.20211512   
2021 Yang B, Wang D, Liu M, Wu X, Yin J, Zhu G. Host cells with transient overexpression of MDR1 as a novel in vitro model for evaluating on-target effect for activity against the epicellular Cryptosporidium parasite. The Journal of Antimicrobial Chemotherapy. PMID 34648615 DOI: 10.1093/jac/dkab369   
2021 Zeng W, Zhao H, Zhao W, Yang Q, Li X, Li X, Duan M, Wang X, Li C, Xiang Z, Chen X, Cui L, Yang Z. Molecular Surveillance and Drug Susceptibilities of Isolates From the China-Myanmar Border. Frontiers in Cellular and Infection Microbiology. 11: 738075. PMID 34790586 DOI: 10.3389/fcimb.2021.738075   
2021 Orlando LMR, Lechuga GC, da Silva Lara L, Ferreira BS, Pereira CN, Silva RC, Dos Santos MS, Pereira MCS. Structural Optimization and Biological Activity of Pyrazole Derivatives: Virtual Computational Analysis, Recovery Assay and 3D Culture Model as Potential Predictive Tools of Effectiveness against . Molecules (Basel, Switzerland). 26. PMID 34771151 DOI: 10.3390/molecules26216742   
2021 Berry A, Menard S, Nsango SE, Abate L, Concordet D, Tchioffo Tsapi M, Iriart X, Awono-Ambéné PH, Roche B, Morlais I. The Rare, the Best: Spread of Antimalarial-Resistant Plasmodium falciparum Parasites by Mosquito Vectors. Microbiology Spectrum. 9: e0085221. PMID 34668767 DOI: 10.1128/Spectrum.00852-21   
2021 Graciano IA, de Carvalho AS, de Carvalho da Silva F, Ferreira VF. 1,2,3-Triazole- and Quinoline-Based Hybrids with Potent Antiplasmodial Activity. Medicinal Chemistry (Shariqah (United Arab Emirates)). PMID 34758718 DOI: 10.2174/1573406418666211110143041   
2021 Temporão A, Sanches-Vaz M, Luís R, Nunes-Cabaço H, Smith TK, Prudêncio M, Figueiredo LM. Excreted Trypanosoma brucei proteins inhibit Plasmodium hepatic infection. Plos Neglected Tropical Diseases. 15: e0009912. PMID 34714824 DOI: 10.1371/journal.pntd.0009912   
2021 Bansal M, Upadhyay C, Poonam, Kumar S, Rathi B. Phthalimide analogs for antimalarial drug discovery. Rsc Medicinal Chemistry. 12: 1854-1867. PMID 34825184 DOI: 10.1039/d1md00244a   
2021 da Cunha AFS, Di C Oliveira YL, Dolabella SS, Scher R, Souto EB, Lopez JA, Jain S. Anti-leishmanial compounds from microbial metabolites: a promising source. Applied Microbiology and Biotechnology. PMID 34625819 DOI: 10.1007/s00253-021-11610-6   
2021 Gupta M, Kumar S, Kumar R, Kumar A, Verma R, Darokar MP, Rout P, Pal A. Inhibition of heme detoxification pathway in malaria parasite by 3-hydroxy-11-keto-β-boswellic acid isolated from Boswellia serrata. Biomedicine & Pharmacotherapy = Biomedecine & Pharmacotherapie. 144: 112302. PMID 34678731 DOI: 10.1016/j.biopha.2021.112302   
2021 Atkinson LE, McCoy CJ, Crooks BA, McKay FM, McVeigh P, McKenzie D, Irvine A, Harrington J, Rosa BA, Mitreva M, Marks NJ, Maule AG, Mousley A. Phylum-Spanning Neuropeptide GPCR Identification and Prioritization: Shaping Drug Target Discovery Pipelines for Nematode Parasite Control. Frontiers in Endocrinology. 12: 718363. PMID 34659113 DOI: 10.3389/fendo.2021.718363   
2021 Hammam E, Sinha A, Baumgarten S, Nardella F, Liang J, Miled S, Bonhomme F, Erdmann D, Arcangioli B, Arimondo PB, Dedon P, Preiser P, Scherf A. Malaria Parasite Stress Tolerance Is Regulated by DNMT2-Mediated tRNA Cytosine Methylation. Mbio. e0255821. PMID 34724812 DOI: 10.1128/mBio.02558-21   
2021 Zhao H, Pi L, Zhao L, Qin Y, Zeng W, Xiang Z, Yang Q, Pan M, Li X, Zou C, Chen X, Zhao W, Lu Y, Wu Y, Duan M, et al. First Detection in West Africa of a Mutation That May Contribute to Artemisinin Resistance . Frontiers in Genetics. 12: 701750. PMID 34691144 DOI: 10.3389/fgene.2021.701750   
2021 Arya R, Dhembla C, Makde RD, Sundd M, Kundu S. An overview of the fatty acid biosynthesis in the protozoan parasite Leishmania and its relevance as a drug target against leishmaniasis. Molecular and Biochemical Parasitology. 246: 111416. PMID 34555376 DOI: 10.1016/j.molbiopara.2021.111416   
2021 Wang S, Ma Y, Wang W, Dai Y, Sun H, Li J, Wang S, Li F. Status and prospect of novel treatment options toward alveolar and cystic echinococcosis. Acta Tropica. 106252. PMID 34808118 DOI: 10.1016/j.actatropica.2021.106252   
2021 Gunnarsson S, Prabakaran S. In silico identification of novel open reading frames in Plasmodium falciparum oocyte and salivary gland sporozoites using proteogenomics framework. Malaria Journal. 20: 71. PMID 33546698 DOI: 10.1186/s12936-021-03598-1   
2021 Penna-Coutinho J, da Silva Araújo M, Campos Aguiar AC, Sá PM, Rios CT, Medeiros JF, Pereira DB, Boechat N, Krettli AU. MEFAS, a hybrid of artesunate-mefloquine active against asexual stages of Plasmodium vivax in field isolates, inhibits malaria transmission. International Journal For Parasitology. Drugs and Drug Resistance. 17: 150-155. PMID 34637981 DOI: 10.1016/j.ijpddr.2021.09.003   
2021 Dassonville-Klimpt A, Schneider J, Damiani C, Tisnerat C, Cohen A, Azas N, Marchivie M, Guillon J, Mullié C, Agnamey P, Totet A, Dormoi J, Taudon N, Pradines B, Sonnet P. Design, synthesis, and characterization of novel aminoalcohol quinolines with strong in vitro antimalarial activity. European Journal of Medicinal Chemistry. 113981. PMID 34782182 DOI: 10.1016/j.ejmech.2021.113981   
2021 Tallant C, Bamborough P, Chung CW, Gamo FJ, Kirkpatrick R, Larminie C, Martín J, Prinjha R, Rioja I, Simola DF, Gabarró R, Calderón F. Expanding Bromodomain Targeting into Neglected Parasitic Diseases. Acs Infectious Diseases. PMID 34612618 DOI: 10.1021/acsinfecdis.1c00387   
2021 Taki AC, Byrne JJ, Jabbar A, Lum KY, Hayes S, Addison RS, Ramage KS, Hofmann A, Ekins MG, Wang T, Chang BCH, Davis RA, Gasser RB. High Throughput Screening of the NatureBank 'Marine Collection' in a Bioassay Identifies Anthelmintic Activity in Extracts from a Range of Sponges from Australian Waters. Molecules (Basel, Switzerland). 26. PMID 34641389 DOI: 10.3390/molecules26195846   
2021 Kumar S, Haile MT, Hoopmann MR, Tran LT, Michaels SA, Morrone SR, Ojo KK, Reynolds LM, Kusebauch U, Vaughan AM, Moritz RL, Kappe SHI, Swearingen KE. Plasmodium falciparum Calcium-Dependent Protein Kinase 4 is Critical for Male Gametogenesis and Transmission to the Mosquito Vector. Mbio. e0257521. PMID 34724830 DOI: 10.1128/mBio.02575-21   
2021 Benítez-Cardoza CG, Brieba LG, Arroyo R, Rojo-Domínguez A, Vique-Sánchez JL. Triosephosphate isomerase as a therapeutic target against trichomoniasis. Molecular and Biochemical Parasitology. 246: 111413. PMID 34537286 DOI: 10.1016/j.molbiopara.2021.111413   
2021 Van Bocxlaer K, Croft SL. Pharmacokinetics and pharmacodynamics in the treatment of cutaneous leishmaniasis - challenges and opportunities. Rsc Medicinal Chemistry. 12: 472-482. PMID 34041488 DOI: 10.1039/d0md00343c   
2021 Clemons B, Barratt J, Lane M, Qvarnstrom Y, Teal AE, Zayas G, Madison-Antenucci S. Assessing an Adaptation of the Universal Parasite Diagnostic Assay for Bloodborne Parasites in a US State Public Health Laboratory. The American Journal of Tropical Medicine and Hygiene. PMID 34749306 DOI: 10.4269/ajtmh.21-0707   
2021 Cygan AM, Jean Beltran PM, Mendoza AG, Branon TC, Ting AY, Carr SA, Boothroyd JC. Proximity-Labeling Reveals Novel Host and Parasite Proteins at the Parasitophorous Vacuole Membrane. Mbio. e0026021. PMID 34749525 DOI: 10.1128/mBio.00260-21   
2021 Luo L, Yang J, Wang C, Wu J, Li Y, Zhang X, Li H, Zhang H, Zhou Y, Lu A, Chen S. Natural products for infectious microbes and diseases: an overview of sources, compounds, and chemical diversities. Science China. Life Sciences. PMID 34705221 DOI: 10.1007/s11427-020-1959-5   
2021 Minassian AM, Themistocleous Y, Silk SE, Barrett JR, Kemp A, Quinkert D, Nielsen CM, Edwards NJ, Rawlinson TA, Ramos Lopez F, Roobsoong W, Ellis KJ, Cho JS, Aunin E, Otto TD, et al. Controlled human malaria infection with a clone of Plasmodium vivax with high quality genome assembly. Jci Insight. PMID 34609964 DOI: 10.1172/jci.insight.152465   
2021 Lee WC, Russell B, Lee B, Chu CS, Phyo AP, Sriprawat K, Lau YL, Nosten F, Rénia L. Plasmodium falciparum rosetting protects schizonts against artemisinin. Ebiomedicine. 73: 103680. PMID 34749300 DOI: 10.1016/j.ebiom.2021.103680   
2021 Duong MC, Pham OKN, Nguyen PT, Nguyen VVC, Nguyen PH. Predictors of treatment failures of plasmodium falciparum malaria in Vietnam: a 4-year single-centre retrospective study. Malaria Journal. 20: 205. PMID 33926479 DOI: 10.1186/s12936-021-03720-3   
2021 da Costa KM, Marques da Fonseca L, Dos Reis JS, Santos MARDC, Previato JO, Mendonça-Previato L, Freire-de-Lima L. -Sialidase as a Potential Vaccine Target Against Chagas Disease. Frontiers in Cellular and Infection Microbiology. 11: 768450. PMID 34765570 DOI: 10.3389/fcimb.2021.768450   
2021 Davis NM, Lissner MM, Richards CL, Chevée V, Gupta AS, Gherardini FC, Schneider DS. Metabolomic Analysis of Diverse Mice Reveals Hepatic Arginase-1 as Source of Plasma Arginase in Plasmodium chabaudi Infection. Mbio. e0242421. PMID 34607466 DOI: 10.1128/mBio.02424-21   
2021 Ong JJY, Russell B, Han JH. Berok Growth Inhibition Assay by Thiol-reactive Probe Based Flow Cytometric Measurement. Bio-Protocol. 11: e4147. PMID 34604452 DOI: 10.21769/BioProtoc.4147   
2021 Mowbray CE, Braillard S, Glossop PA, Whitlock GA, Jacobs RT, Speake J, Pandi B, Nare B, Maes L, Yardley V, Freund Y, Wall RJ, Carvalho S, Bello D, Van den Kerkhof M, et al. DNDI-6148: A Novel Benzoxaborole Preclinical Candidate for the Treatment of Visceral Leishmaniasis. Journal of Medicinal Chemistry. PMID 34711050 DOI: 10.1021/acs.jmedchem.1c01437   
2021 Hunt AG, Howe DK, Brown A, Yeargan M. Transcriptional dynamics in the protozoan parasite Sarcocystis neurona and mammalian host cells after treatment with a specific inhibitor of apicomplexan mRNA polyadenylation. Plos One. 16: e0259109. PMID 34710156 DOI: 10.1371/journal.pone.0259109   
2021 Martins-Duarte ES, Portes JA, da Silva RB, Pires HS, Garden SJ, de Souza W. In vitro activity of N-phenyl-1,10-phenanthroline-2-amines against tachyzoites and bradyzoites of Toxoplasma gondii. Bioorganic & Medicinal Chemistry. 50: 116467. PMID 34666274 DOI: 10.1016/j.bmc.2021.116467   
2021 Elmi T, Hajialiani F, Asadi MR, Sadeghi S, Namazi MJ, Tabatabaie F, Zamani Z. Antimalarial effects of the hydroalcoholic extract of in vitro and in vivo. Journal of Parasitic Diseases : Official Organ of the Indian Society For Parasitology. 45: 1055-1064. PMID 34789989 DOI: 10.1007/s12639-021-01359-0   
2021 Ramírez AM, Tang THT, Suárez ML, Fernández AÁ, García CM, Hisam S, Rubio JM. Assessment of Commercial Real-Time PCR Assays for Detection of Malaria Infection in a Non-Endemic Setting. The American Journal of Tropical Medicine and Hygiene. PMID 34662870 DOI: 10.4269/ajtmh.21-0406   
2021 Beri D, Singh M, Rodriguez M, Yazdanbakhsh K, Lobo CA. Sickle Cell Anemia and Infection. Pathogens (Basel, Switzerland). 10. PMID 34832591 DOI: 10.3390/pathogens10111435   
2021 Yusuf MA, Vatandoost H, Oshaghi MA, Hanafi-Bojd AA, Manu AY, Enayati A, Ado A, Abdullahi AS, Jalo RI, Firdausi A. Biochemical Mechanism of Insecticide Resistance in Malaria Vector, s.l in Nigeria. Iranian Journal of Public Health. 50: 101-110. PMID 34178768 DOI: 10.18502/ijph.v50i1.5076   
2021 Lodoen MB, Smith NC, Soldati-Favre D, Ferguson DJP, van Dooren GG. Nanos gigantium humeris insidentes: old papers informing new research into toxoplasma gondii. International Journal For Parasitology. PMID 34736901 DOI: 10.1016/j.ijpara.2021.10.004   
2021 Singh N, Bhatnagar S. Machine Learning for Prediction of Drug Targets in Microbe Associated Cardiovascular Diseases by Incorporating Host-pathogen Interaction Network Parameters. Molecular Informatics. e2100115. PMID 34676983 DOI: 10.1002/minf.202100115   
2021 Bonam SR, Rénia L, Tadepalli G, Bayry J, Kumar HMS. Malaria Vaccines and Vaccine Adjuvants. Vaccines. 9. PMID 34696180 DOI: 10.3390/vaccines9101072   
2021 Pramasivan S, Ngui R, Jeyaprakasam NK, Liew JWK, Low VL, Mohamed Hassan N, Wan Sulaiman WY, Jaraee R, Abdul Rahman R, Jelip J, Vythilingam I. Spatial distribution of Plasmodium knowlesi cases and their vectors in Johor, Malaysia: in light of human malaria elimination. Malaria Journal. 20: 426. PMID 34715864 DOI: 10.1186/s12936-021-03963-0   
2021 Mantilla BS, Paes-Vieira L, de Almeida Dias F, Calderano SG, Elias MC, Cosentino-Gomes D, Oliveira PL, Meyer-Fernandes JR, Silber AM. Higher expression of proline dehydrogenase altered mitochondrial function and increased Trypanosoma cruzi differentiation in vitro and in the insect vector. The Biochemical Journal. 478: 3891-3903. PMID 34661234 DOI: 10.1042/BCJ20210428   
2021 Mair I, McNeilly TN, Corripio-Miyar Y, Forman R, Else KJ. Embracing nature's complexity: Immunoparasitology in the wild. Seminars in Immunology. 101525. PMID 34785137 DOI: 10.1016/j.smim.2021.101525   
2021 Wichers JS, van Gelder C, Fuchs G, Ruge JM, Pietsch E, Ferreira JL, Safavi S, von Thien H, Burda PC, Mesén-Ramirez P, Spielmann T, Strauss J, Gilberger TW, Bachmann A. Characterization of Apicomplexan Amino Acid Transporters (ApiATs) in the Malaria Parasite Plasmodium falciparum. Msphere. e0074321. PMID 34756057 DOI: 10.1128/mSphere.00743-21   
2021 Stanisic DI, Ho MF, Nevagi R, Cooper E, Walton M, Islam MT, Hussein WM, Skwarczynski M, Toth I, Good MF. Development and Evaluation of a Cryopreserved Whole-Parasite Vaccine in a Rodent Model of Blood-Stage Malaria. Mbio. 12: e0265721. PMID 34663097 DOI: 10.1128/mBio.02657-21