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Harry Heaney - Related publications

Affiliations: 
Organic Chemistry Loughborough University, Loughborough, England, United Kingdom 
Area:
heterocyclic chemistry
Website:
http://www.lboro.ac.uk/departments/chemistry/staff/professor-harry-heaney.html
NOTE: We are testing a new system for identifying relevant work based on semantic analysis that identifies similarities between recently published papers and the current author's publications. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches.
50 most relevant papers in past 60 days:
Year Citation  Score
2021 Zhou Y, Zhao P, Wang LS, Yu XX, Huang C, Wu YD, Wu AX. Direct C-C Bond Cleavage of 1,3-Dicarbonyl Compounds as a Single-Carbon Synthon: Synthesis of 2-Aryl-4-quinolinecarboxylates. Organic Letters. PMID 34346696 DOI: 10.1021/acs.orglett.1c02267   
2021 Ren J, Du FH, Jia MC, Hu ZN, Chen Z, Zhang C. Ring Expansion Fluorination of Unactivated Cyclopropanes Mediated by a New Monofluoroiodane(III) Reagent. Angewandte Chemie (International Ed. in English). PMID 34523779 DOI: 10.1002/anie.202108589   
2021 Chen X, Zhang G, Zeng R. Dehydrogenative Aza-[4 + 2] Cycloaddition of Amines with 1,3-Dienes via Dual Catalysis. Organic Letters. PMID 34459616 DOI: 10.1021/acs.orglett.1c02558   
2021 Thirupataiah B, Reddy GS, Mounika G, Kumar JS, Hossain KA, Mudgal J, Mathew JE, Shenoy GG, Rajadurai M, Parsa KVL, Pal M. Pd-catalysed general access to 7-membered N/O-heterocyclic compounds as potential agents against inflammation. Chemical Communications (Cambridge, England). PMID 34515287 DOI: 10.1039/d1cc04140a   
2021 O'Hagan D, Clark J, Neyyappadath RM, Yu C, Slawin AMZ, Cordes DB. Janus all-cis 2,3,4,5,6-pentafluorocyclohexyl building blocks applied to medicinal chemistry and bioactives discovery chemistry'. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 34486192 DOI: 10.1002/chem.202102819   
2021 Matheau-Raven D, Dixon DJ. General α-Amino 1,3,4-Oxadiazole Synthesis via Late-Stage Reductive Functionalization of Tertiary Amides and Lactams*. Angewandte Chemie (International Ed. in English). PMID 34191400 DOI: 10.1002/anie.202107536   
2021 Song ZL, Wang R, Luo J, Zheng C, Gao L, Zhang H. O2-Assisted Four-component Reaction of Vinyl Magnesium Bromide with Chiral N-tert-Butanesulfinyl Imines To Form syn-1, 3-Amino Alcohols. Angewandte Chemie (International Ed. in English). PMID 34523225 DOI: 10.1002/anie.202109566   
2021 Nakagawa Y, Yamaguchi K, Hosokawa S. Iodide-Mediated [3 + 2]-Cycloaddition Reaction with -Tosylaziridines and α,β-Unsaturated Ketones. The Journal of Organic Chemistry. 86: 7787-7796. PMID 34032429 DOI: 10.1021/acs.joc.1c00532   
2021 Wang J, Yu J, Chen J, Jiang Y, Xiao T. Doyle-Kirmse reaction using 3,3-difluoroallyl sulfide and -sulfonyl-1,2,3-triazole: an efficient access to -difluoroallylated multifunctional quaternary carbon. Organic & Biomolecular Chemistry. PMID 34338276 DOI: 10.1039/d1ob01129d   
2021 Mao ZY, Nie XD, Feng YM, Si CM, Wei BG, Lin GQ. Cu(OTf) catalyzed Ugi-type reaction of ,-acetals with isocyanides for the synthesis of pyrrolidinyl and piperidinyl 2-carboxamides. Chemical Communications (Cambridge, England). 57: 9248-9251. PMID 34519320 DOI: 10.1039/d1cc03113a   
2021 Dai M, Wang YC, Cui C. Flow Chemistry-Enabled Divergent and Enantioselective Total Syntheses of Massarinolin A, Purpurolides B, D, E, 2,3-Deoxypurpurolide C, and Structural Revision of Massarinolin A. Angewandte Chemie (International Ed. in English). PMID 34405497 DOI: 10.1002/anie.202109625   
2021 Utecht-Jarzyńska G, Nagła K, Mlostoń G, Heimgartner H, Palusiak M, Jasiński M. A straightforward conversion of 1,4-quinones into polycyclic pyrazoles via [3 + 2]-cycloaddition with fluorinated nitrile imines. Beilstein Journal of Organic Chemistry. 17: 1509-1517. PMID 34285722 DOI: 10.3762/bjoc.17.108   
2021 Liu Y, Qi X, Wu XF. Palladium-Catalyzed Reductive Aminocarbonylation of Benzylammonium Triflates with -Nitrobenzaldehydes for the Synthesis of 3-Arylquinolin-2(1)-ones. The Journal of Organic Chemistry. PMID 34542996 DOI: 10.1021/acs.joc.1c01984   
2021 Zhao H, Shen P, Sun D, Zhai H, Zhao Y. Transition-Metal-Free [3+2] Dehydration Cycloaddition of Donor-Acceptor Cyclopropanes With 2-Naphthols. Frontiers in Chemistry. 9: 711257. PMID 34336794 DOI: 10.3389/fchem.2021.711257   
2021 Wu W, Wen S, Zhang X, Lin Q, Weng Z. Silver-Catalyzed Regioselective Synthesis of Highly Substituted 2-Trifluoromethyl Pyrroles. Organic Letters. PMID 34339203 DOI: 10.1021/acs.orglett.1c02136   
2021 An J, Intano J, Richard A, Kim T, Gascón JA, Howell AR. Easily accessible non-aromatic heterocycles with handles: 4-bromo-2,3-dihydrofurans from 1,2-dibromohomoallylic alcohols. Chemical Science. 12: 10347-10353. PMID 34377420 DOI: 10.1039/d1sc01013a   
2021 Hou BL, Wong JJ, Lv N, Wang YQ, Houk KN, Li CC. Facile generation of bridged medium-sized polycyclic systems by rhodium-catalysed intramolecular (3+2) dipolar cycloadditions. Nature Communications. 12: 5239. PMID 34475378 DOI: 10.1038/s41467-021-25513-7   
2021 Das J, Das SK. Trifluoroethanol-promoted ring-opening cyclization of 4-(2-oxiranylmethoxy)indoles: access to 4,5-fused indoles. Organic & Biomolecular Chemistry. PMID 34286792 DOI: 10.1039/d1ob01030a   
2021 Lodhi R, Prakash M, Samanta S. Diastereoselective desymmetrization reactions of prochiral -quinamines with cyclopropenes generated : access to fused hydroindol-5-one scaffolds. Organic & Biomolecular Chemistry. PMID 34369544 DOI: 10.1039/d1ob01322j   
2021 Huang C, Shi F, Cui Y, Li C, Lin J, Liu Q, Qin A, Wang H, Wu G, Wu P, Xiao J, Xu H, Yuan Y, Zhai Y, Zheng WF, et al. A palladium-catalyzed approach to allenic aromatic ethers and first total synthesis of terricollene A. Chemical Science. 12: 9347-9351. PMID 34349905 DOI: 10.1039/d1sc01896e   
2021 Wang X, Shao Y, Zhang S, Lu T, Du D. N-Heterocyclic Carbene-Catalyzed Formal [3+3] Annulation of Alkynyl Acylazoliums for the Synthesis of Benzofuro[3,2-]pyridin-2-ones. The Journal of Organic Chemistry. PMID 34328328 DOI: 10.1021/acs.joc.1c01230   
2021 Jiang LL, Hu SJ, Xu Q, Zheng H, Wei WT. Radical Cyclization of 1,n-Enynes and 1,n-Dienes for the Synthesis of 2-Pyrrolidones. Chemistry, An Asian Journal. PMID 34423568 DOI: 10.1002/asia.202100829   
2021 Drusgala M, Frühwirt P, Glotz G, Hogrefe K, Torvisco A, Fischer R, Wilkening HMR, Kelterer AM, Gescheidt G, Haas M. Isolable Geminal Bisgermenolates: A New Synthon in Organo-metallic Chemistry. Angewandte Chemie (International Ed. in English). PMID 34464492 DOI: 10.1002/anie.202111636   
2021 Li W, Wang Y, Qi H, Shi R, Li J, Chen S, Xu XM, Wang WL. Diverse privileged -polycyclic skeletons accessed from a metal-free cascade cyclization reaction. Organic & Biomolecular Chemistry. PMID 34476428 DOI: 10.1039/d1ob01206a   
2021 Wang T, Tang Z, Luo H, Tian Y, Xu M, Lu Q, Li B. Access to ()-β-Substituted Enamides from 1-H-1,2,3-Triazoles. Organic Letters. PMID 34346679 DOI: 10.1021/acs.orglett.1c02087   
2021 Vartanova AE, Levina II, Rybakov VB, Ivanova OA, Trushkov IV. Donor-Acceptor Cyclopropane Ring Opening with 6-Amino-1,3-dimethyluracil and Its Use in Pyrimido[4,5-]azepines Synthesis. The Journal of Organic Chemistry. PMID 34382810 DOI: 10.1021/acs.joc.1c01064   
2021 Liu J, Zhou Y, Zhu J, Yu ZX. Synthesizing Molecules with Linear Tricyclic 5/5/5 and 6/5/5 Skeletons via [5 + 2 + 1]/Ene Strategy. Organic Letters. PMID 34533313 DOI: 10.1021/acs.orglett.1c02766   
2021 Vuong W, Vederas JC. Improved Synthesis of a Cyclic Glutamine Analogue Used in Antiviral Agents Targeting 3C and 3CL Proteases Including SARS-CoV-2 M. The Journal of Organic Chemistry. PMID 34459196 DOI: 10.1021/acs.joc.1c01299   
2021 Zheng H, Wang K, De Angelis L, Arman HD, Doyle MP. Brønsted Acid Catalyzed Oxocarbenium-Olefin Metathesis/Rearrangements of 1-Isochromene Acetals with Vinyl Diazo Compounds. Journal of the American Chemical Society. PMID 34510888 DOI: 10.1021/jacs.1c07271   
2021 Sun SY, Raju S, Vedarethinam G, Chen PL, Chuang SC. TfOH-promoted Classical Nazarov-type Cyclization of Benzofulvenes: Synthesis of Polycyclic 5,10'-spiro[benzo[]phenanthridine-5,6'-dibenzopentalenes]. Organic Letters. PMID 34355911 DOI: 10.1021/acs.orglett.1c01809   
2021 Wang Q, Zha M, Zhou F, Chen X, Wang B, Liu G, Qian L. CBr Mediated [4 + 1] Dehydrocyclization for the Synthesis of Functionalized Imidazo[1,5-a]heterocycles from Pyridin-2-ylmethanamines and Aldehydes. Acs Omega. 6: 20303-20308. PMID 34395978 DOI: 10.1021/acsomega.1c02181   
2021 Chen ZD, Xu WK, Guo JM, Chen L, Wei BG, Si CM, Lin GQ. A One-Pot Approach to 2-Substituted-2-(Dimethoxyphosphoryl)-Pyrrolidines from Substituted -Butyl 4-Oxobutylcarbamates and Trimethyl Phosphite. The Journal of Organic Chemistry. 86: 11442-11455. PMID 34479405 DOI: 10.1021/acs.joc.1c00935   
2021 Chiku K, Yoshida M, Ono H, Kitaoka M. Generation of 3-deoxypentulose by the isomerization and β-elimination of 4-O-substituted glucose and fructose. Carbohydrate Research. 508: 108402. PMID 34303026 DOI: 10.1016/j.carres.2021.108402   
2021 Tokuyama H. Construction of N-Heterocycles Fused with a Highly Substituted Benzene Ring by a Benzyne-Mediated Cyclization/Functionalization Cascade Reaction and Its Application to the Total Synthesis of Marine Natural Products. Chemical & Pharmaceutical Bulletin. 69: 707-716. PMID 34334514 DOI: 10.1248/cpb.c21-00389   
2021 Gummidi L, Kerru N, Ebenezer O, Awolade P, Sanni O, Islam MS, Singh P. Multicomponent reaction for the synthesis of new 1,3,4-thiadiazole-thiazolidine-4-one molecular hybrids as promising antidiabetic agents through α-glucosidase and α-amylase inhibition. Bioorganic Chemistry. 115: 105210. PMID 34332231 DOI: 10.1016/j.bioorg.2021.105210   
2021 Martin JS, Mackenzie CJ, Gilbert IH. Synthesis of a Series of Diaminoindoles. The Journal of Organic Chemistry. PMID 34351743 DOI: 10.1021/acs.joc.1c00652   
2021 Tarigopula C, Manojveer S, Balamurugan R. Synthesis of Highly Substituted Biaryls by the Construction of a Benzene Ring via Formed Acetals. The Journal of Organic Chemistry. 86: 11871-11883. PMID 34425048 DOI: 10.1021/acs.joc.1c01277   
2021 Gazizov AS, Smolobochkin AV, Kuznetsova EA, Abdullaeva DS, Burilov AR, Pudovik MA, Voloshina AD, Syakaev VV, Lyubina AP, Amerhanova SK, Voronina JK. The Highly Regioselective Synthesis of Novel Imidazolidin-2-Ones via the Intramolecular Cyclization/Electrophilic Substitution of Urea Derivatives and the Evaluation of Their Anticancer Activity. Molecules (Basel, Switzerland). 26. PMID 34361587 DOI: 10.3390/molecules26154432   
2021 Wang W, Bao ZP, Qi X, Wu XF. Nickel-Catalyzed One-Pot Carbonylative Synthesis of 2-Mono- and 2,3-Disubstituted Thiochromenones from 2-Bromobenzenesulfonyl Chlorides and Alkynes. Organic Letters. PMID 34370477 DOI: 10.1021/acs.orglett.1c02442   
2021 Straathof NJW, Magnus CB, Zhuravlev F, Jensen AI. Novel Bifunctional [16]aneS-Derived Chelators for Soft Radiometals. Molecules (Basel, Switzerland). 26. PMID 34361752 DOI: 10.3390/molecules26154603   
2021 Piovan L, Souza JPA, Bandeira PT, Menezes LRA, Bespalhok MB, Scariot DB, Garcia FP, Giese SOK, Hughes DL, Nakamura CV, Barison A, Oliveira ARM, Campos RB. Synthesis, Mechanism Elucidation and Biological Insights of Tellurium(IV)-containing Heterocycles. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 34406689 DOI: 10.1002/chem.202102287   
2021 Apostol TV, Marutescu LG, Draghici C, Socea LI, Olaru OT, Nitulescu GM, Pahontu EM, Saramet G, Enache-Preoteasa C, Barbuceanu SF. Synthesis and Biological Evaluation of New -Acyl-α-amino Ketones and 1,3-Oxazoles Derivatives. Molecules (Basel, Switzerland). 26. PMID 34443608 DOI: 10.3390/molecules26165019   
2021 Wang K, Guan HR, Ren WL, Yang HT, Miao CB. Copper-Catalyzed Cascade Annulation of Malonate-Tethered -Acyl Oximes with Cyclic 1,3-Dicarbonyl Compounds for the Synthesis of Spiro-Pentacyclic Derivatives. The Journal of Organic Chemistry. PMID 34369761 DOI: 10.1021/acs.joc.1c01122   
2021 Wang Z, Yue G, Ji X, Song H, Yan P, Zhao J, Jia X. Tandem Michael Addition-Cyclization of Nitroalkenes with 1,3-Dicarbonyl Compounds Accompanied by Removal of Nitro Group. The Journal of Organic Chemistry. PMID 34494850 DOI: 10.1021/acs.joc.1c01586   
2021 Zheng D, Jana K, Alasmary FA, Daniliuc CG, Studer A. Transition-Metal-Free Intramolecular Radical Aminoboration of Unactivated Alkenes. Organic Letters. PMID 34542297 DOI: 10.1021/acs.orglett.1c03024   
2021 Wen S, Tian Q, Chen Y, Zhang Y, Cheng G. Annulation of CF-Imidoyl Sulfoxonium Ylides with 1,3-Dicarbonyl Compounds: Access to 1,2,3-Trisubstituted 5-Trifluoromethylpyrroles. Organic Letters. PMID 34543038 DOI: 10.1021/acs.orglett.1c02598   
2021 Zhu M, Huang XL, Sun S, Zheng C, You SL. Visible-Light-Induced Dearomatization of Indoles/Pyrroles with Vinylcyclopropanes: Expedient Synthesis of Structurally Diverse Polycyclic Indolines/Pyrrolines. Journal of the American Chemical Society. PMID 34398603 DOI: 10.1021/jacs.1c07082   
2021 Usachev SA, Nigamatova DI, Mysik DK, Naumov NA, Obydennov DL, Sosnovskikh VY. 2-Aryl-6-Polyfluoroalkyl-4-Pyrones as Promising R-Building-Blocks: Synthesis and Application for Construction of Fluorinated Azaheterocycles. Molecules (Basel, Switzerland). 26. PMID 34361567 DOI: 10.3390/molecules26154415   
2021 Vartanova AE, Plodukhin AY, Ratmanova NK, Andreev IA, Anisimov MN, Gudimchuk NB, Rybakov VB, Levina II, Ivanova OA, Trushkov IV, Alabugin IV. Expanding Stereoelectronic Limits of - Cyclizations: Synthesis of Benz[]azepines from Donor-Acceptor Cyclopropanes. Journal of the American Chemical Society. PMID 34406759 DOI: 10.1021/jacs.1c07088   
2021 Zhang K, Tran C, Alami M, Hamze A, Provot O. Synthesis and Biological Activities of Pyrazino[1,2-]indole and Pyrazino[1,2-]indol-1-one Derivatives. Pharmaceuticals (Basel, Switzerland). 14. PMID 34451876 DOI: 10.3390/ph14080779