| Year |
Citation |
Score |
| 2019 |
Ghosh AK, Williams JN, Kovela S, Takayama J, Simpson HM, Walters DE, Hattori SI, Aoki M, Mitsuya H. Potent HIV-1 protease inhibitors incorporating squaramide-derived P2 ligands: Design, synthesis, and biological evaluation. Bioorganic & Medicinal Chemistry Letters. PMID 31416666 DOI: 10.1016/J.Bmcl.2019.08.006 |
0.3 |
|
| 2014 |
Ghosh AK, Schiltz GE, Rusere LN, Osswald HL, Walters DE, Amano M, Mitsuya H. Design and synthesis of potent macrocyclic HIV-1 protease inhibitors involving P1-P2 ligands. Organic & Biomolecular Chemistry. 12: 6842-54. PMID 25050776 DOI: 10.1039/C4Ob00738G |
0.302 |
|
| 2012 |
Symersky J, Osowski D, Walters DE, Mueller DM. Oligomycin frames a common drug-binding site in the ATP synthase. Proceedings of the National Academy of Sciences of the United States of America. 109: 13961-5. PMID 22869738 DOI: 10.1073/Pnas.1207912109 |
0.306 |
|
| 2011 |
Ghosh AK, Chapsal BD, Baldridge A, Steffey MP, Walters DE, Koh Y, Amano M, Mitsuya H. Design and synthesis of potent HIV-1 protease inhibitors incorporating hexahydrofuropyranol-derived high affinity P(2) ligands: structure-activity studies and biological evaluation. Journal of Medicinal Chemistry. 54: 622-34. PMID 21194227 DOI: 10.1021/Jm1012787 |
0.315 |
|
| 2010 |
Aluvila S, Kotaria R, Sun J, Mayor JA, Walters DE, Harrison DH, Kaplan RS. The yeast mitochondrial citrate transport protein: molecular determinants of its substrate specificity. The Journal of Biological Chemistry. 285: 27314-26. PMID 20551333 DOI: 10.1074/Jbc.M110.137364 |
0.309 |
|
| 2010 |
Mayor JA, Sun J, Kotaria R, Walters DE, Oh KJ, Kaplan RS. Probing the effect of transport inhibitors on the conformation of the mitochondrial citrate transport protein via a site-directed spin labeling approach. Journal of Bioenergetics and Biomembranes. 42: 99-109. PMID 20354774 DOI: 10.1007/S10863-010-9280-0 |
0.303 |
|
| 2010 |
Ghosh AK, Gemma S, Simoni E, Baldridge A, Walters DE, Ide K, Tojo Y, Koh Y, Amano M, Mitsuya H. Synthesis and biological evaluation of novel allophenylnorstatine-based HIV-1 protease inhibitors incorporating high affinity P2-ligands. Bioorganic & Medicinal Chemistry Letters. 20: 1241-6. PMID 20034787 DOI: 10.1016/J.Bmcl.2009.11.123 |
0.305 |
|
| 2010 |
Aluvila S, Sun J, Harrison DH, Walters DE, Kaplan RS. Inhibitors of the mitochondrial citrate transport protein: validation of the role of substrate binding residues and discovery of the first purely competitive inhibitor. Molecular Pharmacology. 77: 26-34. PMID 19843634 DOI: 10.1124/Mol.109.058750 |
0.323 |
|
| 2008 |
Remani S, Sun J, Kotaria R, Mayor JA, Brownlee JM, Harrison DH, Walters DE, Kaplan RS. The yeast mitochondrial citrate transport protein: identification of the Lysine residues responsible for inhibition mediated by Pyridoxal 5'-phosphate. Journal of Bioenergetics and Biomembranes. 40: 577-85. PMID 19002576 DOI: 10.1007/S10863-008-9187-1 |
0.324 |
|
| 2007 |
Ma C, Remani S, Sun J, Kotaria R, Mayor JA, Walters DE, Kaplan RS. Identification of the substrate binding sites within the yeast mitochondrial citrate transport protein. The Journal of Biological Chemistry. 282: 17210-20. PMID 17400551 DOI: 10.1074/Jbc.M611268200 |
0.318 |
|
| 2006 |
Ghosh AK, Sridhar PR, Leshchenko S, Hussain AK, Li J, Kovalevsky AY, Walters DE, Wedekind JE, Grum-Tokars V, Das D, Koh Y, Maeda K, Gatanaga H, Weber IT, Mitsuya H. Structure-based design of novel HIV-1 protease inhibitors to combat drug resistance. Journal of Medicinal Chemistry. 49: 5252-61. PMID 16913714 DOI: 10.1021/Jm060561M |
0.316 |
|
| 2006 |
Ma C, Remani S, Kotaria R, Mayor JA, Walters DE, Kaplan RS. The mitochondrial citrate transport protein: evidence for a steric interaction between glutamine 182 and leucine 120 and its relationship to the substrate translocation pathway and identification of other mechanistically essential residues. Biochimica Et Biophysica Acta. 1757: 1271-6. PMID 16904062 DOI: 10.1016/J.Bbabio.2006.06.011 |
0.326 |
|
| 2005 |
Ghosh AK, Swanson LM, Cho H, Leshchenko S, Hussain KA, Kay S, Walters DE, Koh Y, Mitsuya H. Structure-based design: synthesis and biological evaluation of a series of novel cycloamide-derived HIV-1 protease inhibitors. Journal of Medicinal Chemistry. 48: 3576-85. PMID 15887965 DOI: 10.1021/Jm050019I |
0.326 |
|
| 2005 |
Ma C, Kotaria R, Mayor JA, Remani S, Walters DE, Kaplan RS. The yeast mitochondrial citrate transport protein: characterization of transmembrane domain III residue involvement in substrate translocation. The Journal of Biological Chemistry. 280: 2331-40. PMID 15498760 DOI: 10.1074/Jbc.M411474200 |
0.323 |
|
| 1981 |
Berman E, Walters DE, Allerhand A. Structure and dynamic behavior of the oligosaccharide side chain of bovine pancreatic ribonuclease B. Application of carbon 13 nuclear magnetic resonance spectroscopy. The Journal of Biological Chemistry. 256: 3853-7. PMID 7217059 |
0.488 |
|
| 1980 |
Walters DE, Allerhand A. Tautomeric states of the histidine residues of bovine pancreatic ribonuclease A. Application of carbon 13 nuclear magnetic resonance spectroscopy. The Journal of Biological Chemistry. 255: 6200-4. PMID 7391017 |
0.476 |
|
| 1979 |
Grunewald GL, Creese MW, Walters DE. APPLICATION OF CNDO/2 CALCULATIONS AND X-RAY CRYSTALLOGRAPHIC ANALYSIS OF THE DESIGN OF CONFORMATIONALLY DEFINED ANALOGS OF METHAMPHETAMINE Acs Symposium Series. 439-487. |
0.47 |
|
| 1978 |
Grunewald GL, Walters DE, Kroboth TR. Synthesis of bridgehead hydroxyl-substituted benzobicyclo[3.2.1]octenes and -octadienes via an acyloin rearrangement in the benzobicyclo[2.2.2]octene ring system Journal of Organic Chemistry. 43: 3478-3481. DOI: 10.1021/Jo00412A012 |
0.477 |
|
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