Year |
Citation |
Score |
2022 |
Liu L, Schuetze R, Gerberich JL, Lopez R, Odutola SO, Tanpure RP, Charlton-Sevcik AK, Tidmore JK, Taylor EA, Kapur P, Hammers H, Trawick ML, Pinney KG, Mason RP. Demonstrating Tumor Vascular Disrupting Activity of the Small-Molecule Dihydronaphthalene Tubulin-Binding Agent OXi6196 as a Potential Therapeutic for Cancer Treatment. Cancers. 14. PMID 36077745 DOI: 10.3390/cancers14174208 |
0.619 |
|
2021 |
Guo Y, Wang H, Gerberich JL, Odutola SO, Charlton-Sevcik AK, Li M, Tanpure RP, Tidmore JK, Trawick ML, Pinney KG, Mason RP, Liu L. Imaging-Guided Evaluation of the Novel Small-Molecule Benzosuberene Tubulin-Binding Agent KGP265 as a Potential Therapeutic Agent for Cancer Treatment. Cancers. 13. PMID 34638255 DOI: 10.3390/cancers13194769 |
0.602 |
|
2016 |
Herdman CA, Strecker TE, Tanpure RP, Chen Z, Winters A, Gerberich J, Liu L, Hamel E, Mason RP, Chaplin DJ, Trawick ML, Pinney KG. Synthesis and Biological Evaluation of Benzocyclooctene-based and Indene-based Anticancer Agents that Function as Inhibitors of Tubulin Polymerization. Medchemcomm. 7: 2418-2427. PMID 28217276 DOI: 10.1039/C6Md00459H |
0.816 |
|
2015 |
Herdman CA, Devkota L, Lin CM, Niu H, Strecker TE, Lopez R, Liu L, George CS, Tanpure RP, Hamel E, Chaplin DJ, Mason RP, Trawick ML, Pinney KG. Structural interrogation of benzosuberene-based inhibitors of tubulin polymerization. Bioorganic & Medicinal Chemistry. PMID 26775540 DOI: 10.1016/J.Bmc.2015.10.012 |
0.757 |
|
2015 |
Tanpure RP, Ren B, Peat TS, Bornaghi LF, Vullo D, Supuran CT, Poulsen SA. Carbonic anhydrase inhibitors with dual-tail moieties to match the hydrophobic and hydrophilic halves of the carbonic anhydrase active site. Journal of Medicinal Chemistry. 58: 1494-501. PMID 25581127 DOI: 10.1021/jm501798g |
0.374 |
|
2014 |
Fisher GM, Tanpure RP, Douchez A, Andrews KT, Poulsen SA. Synthesis and evaluation of antimalarial properties of novel 4-aminoquinoline hybrid compounds. Chemical Biology & Drug Design. 84: 462-72. PMID 24720445 DOI: 10.1111/cbdd.12335 |
0.398 |
|
2013 |
Tanpure RP, George CS, Strecker TE, Devkota L, Tidmore JK, Lin CM, Herdman CA, Macdonough MT, Sriram M, Chaplin DJ, Trawick ML, Pinney KG. Synthesis of structurally diverse benzosuberene analogues and their biological evaluation as anti-cancer agents. Bioorganic & Medicinal Chemistry. 21: 8019-32. PMID 24183586 DOI: 10.1016/J.Bmc.2013.08.035 |
0.665 |
|
2012 |
Tanpure RP, George CS, Sriram M, Strecker TE, Tidmore JK, Hamel E, Charlton-Sevcik AK, Chaplin DJ, Trawick ML, Pinney KG. An Amino-Benzosuberene Analogue That Inhibits Tubulin Assembly and Demonstrates Remarkable Cytotoxicity. Medchemcomm. 3: 720-724. PMID 23772309 DOI: 10.1039/C2Md00318J |
0.721 |
|
2011 |
Tanpure RP, Nguyen BL, Strecker TE, Aguirre S, Sharma S, Chaplin DJ, Siim BG, Hamel E, Lippert JW, Pettit GR, Trawick ML, Pinney KG. Regioselective synthesis of water-soluble monophosphate derivatives of combretastatin A-1. Journal of Natural Products. 74: 1568-74. PMID 21718055 DOI: 10.1021/Np200104T |
0.787 |
|
2010 |
Tanpure RP, Strecker TE, Chaplin DJ, Siim BG, Trawick ML, Pinney KG. Regio- and stereospecific synthesis of mono-beta-d-glucuronic acid derivatives of combretastatin A-1. Journal of Natural Products. 73: 1093-101. PMID 20496923 DOI: 10.1021/Np100108E |
0.689 |
|
2009 |
Tanpure RP, Harkrider AR, Strecker TE, Hamel E, Trawick ML, Pinney KG. Application of the McMurry coupling reaction in the synthesis of tri- and tetra-arylethylene analogues as potential cancer chemotherapeutic agents. Bioorganic & Medicinal Chemistry. 17: 6993-7001. PMID 19733085 DOI: 10.1016/J.Bmc.2009.08.011 |
0.786 |
|
2003 |
Hadimani MB, Hua J, Jonklaas MD, Kessler RJ, Sheng Y, Olivares A, Tanpure RP, Weiser A, Zhang J, Edvardsen K, Kane RR, Pinney KG. Synthesis, in vitro, and in vivo evaluation of phosphate ester derivatives of combretastatin A-4. Bioorganic & Medicinal Chemistry Letters. 13: 1505-8. PMID 12699742 DOI: 10.1016/S0960-894X(03)00206-3 |
0.777 |
|
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