David J. Austin, Ph.D. - Publications

Affiliations: 
chemistry Yale University, New Haven, CT 
Website:
http://www.fenwick.com/professionals/Pages/davidaustin.aspx

59 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2010 Koenig SG, Loewe RS, Austin DJ. ChemInform Abstract: An Improved Synthesis of (4S)-4,5-O-Isopropylidenepent-(2Z)-enoate. Cheminform. 33: no-no. DOI: 10.1002/chin.200239204  0.635
2010 PADWA A, AUSTIN DJ, PRICE AT, WEINGARTEN MD. ChemInform Abstract: Intramolecular Cycloaddition Reaction of Isomuenchnones Derived from N- Alkenyl Substituted Diazoimides. Cheminform. 27: no-no. DOI: 10.1002/CHIN.199625055  0.44
2010 PADWA A, AUSTIN DJ, HORNBUCKLE SF. ChemInform Abstract: Ligand-Induced Selectivity in the Rhodium(II)-Catalyzed Reactions of . alpha.-Diazo Carbonyl Compounds. Cheminform. 27: no-no. DOI: 10.1002/CHIN.199620052  0.422
2010 PADWA A, AUSTIN DJ, PRICE AT. ChemInform Abstract: Synthesis of Polyheterocyclic Ring Compounds by the Intramolecular Cycloaddition of N-Alkenyl Substituted Diazoimides. Cheminform. 26: no-no. DOI: 10.1002/CHIN.199515168  0.403
2010 PADWA A, AUSTIN DJ. ChemInform Abstract: Ligand Effects on the Chemoselectivity of Transition Metal Catalyzed Reactions of α-Diazo Carbonyl Compounds Cheminform. 26: no-no. DOI: 10.1002/CHIN.199509287  0.391
2010 PADWA A, AUSTIN DJ, PRICE AT, SEMONES MA, DOYLE MP, PROTOPOPOVA MN, WINCHESTER WR, TRAN A. ChemInform Abstract: Ligand Effects on Dirhodium(II) Carbene Reactivities. Highly Effective Switching Between Competitive Carbenoid Transformations. Cheminform. 25: no-no. DOI: 10.1002/chin.199402062  0.344
2010 HASSNER A, MAURYA R, FRIEDMAN O, GOTTLIEB HE, PADWA A, AUSTIN D. ChemInform Abstract: Stereochemistry. Part 82. On the Conformations of Fused Five-Membered Heterocyclic Rings Derived from the Intramolecular Oxime Olefin Cycloaddition Reaction. Cheminform. 24: no-no. DOI: 10.1002/chin.199350203  0.436
2010 COX GG, MOODY CJ, AUSTIN DJ, PADWA A. ChemInform Abstract: Chemoselectivity of Rhodium Carbenoids. A Comparison of the Selectivity for O-H Insertion Reactions or Carbonyl Ylide Formation versus Aliphatic and Aromatic C-H Insertion and Cyclopropanation. Cheminform. 24: no-no. DOI: 10.1002/chin.199342063  0.4
2010 PADWA A, AUSTIN DJ, GAREAU Y, KASSIR JM, XU SL. ChemInform Abstract: Rearrangement of Alkynyl and Vinyl Carbenoids via the Rhodium(II)- Catalyzed Cyclization Reaction of α-Diazo Ketones. Cheminform. 24: no-no. DOI: 10.1002/CHIN.199335093  0.44
2010 PADWA A, AUSTIN DJ, PRECEDO L, ZHI L. ChemInform Abstract: Cycloaddition Reactions of Pyridinium and Related Azomethine Ylides. Cheminform. 24: no-no. DOI: 10.1002/CHIN.199323089  0.424
2010 PADWA A, AUSTIN DJ, HORNBUCKLE SF, PRICE AT. ChemInform Abstract: Rhodium(II)-Catalyzed Intramolecular Dipolar Cycloaddition Reactions of Carbonyl Ylides. Computational and Empirical Studies of the Regio- and Chemoselective Effect of Catalyst Ligand. Cheminform. 24: no-no. DOI: 10.1002/CHIN.199313087  0.416
2010 FAIRFAX DJ, AUSTIN DJ, XU SL, PADWA A. ChemInform Abstract: Alternatives to α-Diazo Ketones for Tandem Cyclization- Cycloaddition and Carbenoid-Alkyne Metathesis Strategies. Novel Cyclic Enol-Ether Formation via Carbonyl Ylide Rearrangement Reactions. Cheminform. 24: no-no. DOI: 10.1002/CHIN.199310089  0.458
2010 HERTZOG DL, AUSTIN DJ, NADLER WR, PADWA A. ChemInform Abstract: Intramolecular Cycloaddition of Isomuenchnones Derived from the Rhodium(II)-Catalyzed Cyclization of Diazoimides. Cheminform. 24: no-no. DOI: 10.1002/CHIN.199301078  0.429
2010 PADWA A, AUSTIN DJ, ISHIDA M, MULLER CL, MURPHREE SS, YESKE PE. ChemInform Abstract: Tunable Regioselectivity Associated with the Reaction of 2,3-Dihalo-1-( phenylsulfonyl)-1-propenes with Ambident Nucleophilic Reagents. Cheminform. 23: no-no. DOI: 10.1002/CHIN.199230124  0.424
2010 PADWA A, AUSTIN DJ, CHIACCHIO U, KASSIR JM, RESCIFINA A, XU SL. ChemInform Abstract: Rearrangement of o-Alkynyl Substituted α-Diazoacetophenones. Conversion to β-Naphthols via Arylketene Intermediates. Cheminform. 23: no-no. DOI: 10.1002/CHIN.199227099  0.342
2010 PADWA A, AUSTIN DJ, HORNBUCKLE SF, SEMONES MA, DOYLE MP, PROTOPOPOVA MN. ChemInform Abstract: Control of Chemoselectivity in Catalytic Carbenoid Reactions. Dirhodium(II) Ligand Effects on Relative Reactivities. Cheminform. 23: no-no. DOI: 10.1002/chin.199227092  0.413
2010 PADWA A, AUSTIN DJ, XU SL. ChemInform Abstract: Rhodium(II)-Catalyzed Cyclizations of α-Diazo Substituted Alkynes. A New Mode of Reaction. Cheminform. 23: no-no. DOI: 10.1002/CHIN.199219153  0.43
2006 Boehmerle W, Splittgerber U, Lazarus MB, McKenzie KM, Johnston DG, Austin DJ, Ehrlich BE. Paclitaxel induces calcium oscillations via an inositol 1,4,5-trisphosphate receptor and neuronal calcium sensor 1-dependent mechanism. Proceedings of the National Academy of Sciences of the United States of America. 103: 18356-61. PMID 17114292 DOI: 10.1073/Pnas.0607240103  0.704
2005 Videlock EJ, Chung VK, Hall JM, Hines J, Agapakis CM, Austin DJ. Identification of a molecular recognition role for the activation loop phosphotyrosine of the SRC tyrosine kinase. Journal of the American Chemical Society. 127: 1600-1. PMID 15700969 DOI: 10.1021/Ja047957C  0.504
2005 Savizky RM, Austin DJ. Rhodium(II)-Catalyzed 1,3-Dipolar Cycloaddition Reactions Modern Rhodium-Catalyzed Organic Reactions. 433-454. DOI: 10.1002/3527604693.ch19  0.767
2004 Chung R, Yu E, Incarvito CD, Austin DJ. Hypervalent iodine-mediated vicinal syn diazidation: application to the total synthesis of (+/-)-dibromophakellstatin. Organic Letters. 6: 3881-4. PMID 15496054 DOI: 10.1021/Ol0490532  0.617
2004 Lee Y, Yeo H, Liu SH, Jiang Z, Savizky RM, Austin DJ, Cheng YC. Increased anti-P-glycoprotein activity of baicalein by alkylation on the A ring. Journal of Medicinal Chemistry. 47: 5555-66. PMID 15481991 DOI: 10.1021/Jm049949C  0.736
2004 McKenzie KM, Videlock EJ, Splittgerber U, Austin DJ. Simultaneous identification of multiple protein targets by using complementary-DNA phage display and a natural-product-mimetic probe. Angewandte Chemie (International Ed. in English). 43: 4052-5. PMID 15300693 DOI: 10.1002/Anie.200454004  0.719
2003 Liu F, Johnson EF, Austin DJ, Anderson KS. Adenosine-anchored triphosphate subsite probing: distinguishing between HER-2 and HER-4 tyrosine protein kinases. Bioorganic & Medicinal Chemistry Letters. 13: 3587-92. PMID 14505676 DOI: 10.1016/S0960-894X(03)00761-3  0.36
2003 Koenig SG, Miller SM, Leonard KA, Löwe RS, Chen BC, Austin DJ. A transient N-O-linked Pauson-Khand strategy for the synthesis of the deschloro carbocyclic core of the palau'amines and styloguanidines. Organic Letters. 5: 2203-6. PMID 12816409 DOI: 10.1021/Ol0344063  0.737
2003 Koenig SG, Leonard KA, Löwe RS, Austin DJ. Corrigendum to “Synthesis of 3,4-substituted cyclopentenones via an intramolecular Pauson–Khand reaction of NO linked enynes” Tetrahedron Letters. 44: 3995. DOI: 10.1016/S0040-4039(03)00672-5  0.694
2002 Savinov SN, Austin DJ. Diastereofacial solid phase synthesis and self-promoted cleavage of a [2.2.1] bicyclic diversity scaffold. Organic Letters. 4: 1419-22. PMID 11975593 DOI: 10.1021/Ol017264Q  0.701
2002 Savinov SN, Austin DJ. Modular evolution of a chiral auxiliary for the 1,3-dipolar cycloaddition of isomünchnones with vinyl ethers. Organic Letters. 4: 1415-8. PMID 11975592 DOI: 10.1021/Ol017263Y  0.71
2002 Koenig SG, Löwe RS, Austin DJ. An improved synthesis of (4S)-4,5-O-isopropylidenepent- (2Z)-enoate Synthetic Communications. 32: 1379-1383. DOI: 10.1081/Scc-120003634  0.664
2001 Liu F, Austin DJ. A general synthesis of 5'-azido-5'-deoxy-2',3'-O-isopropylidene nucleosides. The Journal of Organic Chemistry. 66: 8643-5. PMID 11735550 DOI: 10.1021/Jo015800M  0.386
2001 Savinov SN, Austin DJ. The cloning of human genes using cDNA phage display and small-molecule chemical probes. Combinatorial Chemistry & High Throughput Screening. 4: 593-7. PMID 11562262 DOI: 10.2174/1386207013330814  0.692
2001 Liu F, Austin DJ. Synthesis of a new class of 5'-functionalized adenosines using a rh(ii)-catalyzed 1,3-dipolar cycloaddition. Organic Letters. 3: 2273-6. PMID 11463294 DOI: 10.1021/Ol015995K  0.446
2001 Sche PP, McKenzie KM, White JD, Austin DJ. Corrigendum to: "Display cloning: functional identification of natural product receptors using cDNA-phage display" [Chemistry & Biology 6 (1999) 707-716]. Chemistry & Biology. 8: 399-400. PMID 11325595 DOI: 10.1016/S1074-5521(01)00012-6  0.715
2001 Liu F, Austin DJ. Synthesis of a new class of 5′-functionalized adenosines using a Rh(II)-catalyzed 1,3-dipolar cycloaddition Organic Letters. 3: 2273-2276. DOI: 10.1021/ol015995k  0.321
2001 Liu F, Austin DJ. Synthesis of 5′-functionalized adenosine: Suppression of cyclonucleoside formation Tetrahedron Letters. 42: 3153-3154. DOI: 10.1016/S0040-4039(01)00395-1  0.451
2000 Koenig SG, Leonard KA, Lowe RS, Austin DJ. Synthesis of 3,4-substituted cyclopentenones via an intramolecular Pauson-Khand reaction of N-O linked enynes Tetrahedron Letters. 41: 9393-9396. DOI: 10.1016/S0040-4039(00)01495-7  0.705
1999 Sche PP, McKenzie KM, White JD, Austin DJ. Display cloning: functional identification of natural product receptors using cDNA-phage display. Chemistry & Biology. 6: 707-16. PMID 10508685 DOI: 10.1016/S1074-5521(00)80018-6  0.725
1999 Savinov SN, Austin DJ. The diastereoselective cycloaddition of vinyl ethers with isomunchnones Chemical Communications. 1813-1814. DOI: 10.1039/A903381E  0.7
1998 Whitehouse DL, Nelson KH, Savinov SN, Löwe RS, Austin DJ. A metathetical cycloaddition-cycloreversion approach to the formation of furan scaffold libraries. Bioorganic & Medicinal Chemistry. 6: 1273-82. PMID 9784868 DOI: 10.1016/S0968-0896(98)00115-1  0.718
1997 Liberles SD, Diver ST, Austin DJ, Schreiber SL. Inducible gene expression and protein translocation using nontoxic ligands identified by a mammalian three-hybrid screen. Proceedings of the National Academy of Sciences of the United States of America. 94: 7825-30. PMID 9223271 DOI: 10.1073/Pnas.94.15.7825  0.747
1997 Whitehouse DL, Savinov SN, Austin DJ. An improved synthesis and selective coupling of a hydroxy based photolabile linker for solid phase organic synthesis Tetrahedron Letters. 38: 7851-7852. DOI: 10.1016/S0040-4039(97)10133-2  0.68
1997 Whitehouse DL, Nelson KH, Savinov SN, Austin DJ. A chemoselective rhodium(II) mediated solid phase 1,3-dipolar cycloaddition and its application to a thermally self-cleaving puran scaffold Tetrahedron Letters. 38: 7139-7142. DOI: 10.1016/S0040-4039(97)01768-1  0.711
1996 Padwa A, Austin DJ, Price AT, Weingarten MD. Studies on the intramolecular cycloaddition reaction of isomünchnones derived from N-alkenyl substituted diazoimides Tetrahedron. 52: 3247-3260. DOI: 10.1016/0040-4020(95)01108-0  0.436
1995 Holsinger LJ, Spencer DM, Austin DJ, Schreiber SL, Crabtree GR. Signal transduction in T lymphocytes using a conditional allele of Sos. Proceedings of the National Academy of Sciences of the United States of America. 92: 9810-4. PMID 7568223 DOI: 10.1073/Pnas.92.21.9810  0.322
1995 Spencer DM, Graef I, Austin DJ, Schreiber SL, Crabtree GR. A general strategy for producing conditional alleles of Src-like tyrosine kinases. Proceedings of the National Academy of Sciences of the United States of America. 92: 9805-9. PMID 7568222 DOI: 10.1073/Pnas.92.21.9805  0.342
1994 Austin DJ, Crabtree GR, Schreiber SL. Proximity versus allostery: the role of regulated protein dimerization in biology. Chemistry & Biology. 1: 131-6. PMID 9383382 DOI: 10.1016/1074-5521(94)90002-7  0.348
1994 Padwa A, Austin DJ, Price AT. Synthesis of polyheterocyclic ring compounds by the intramolecular cycloaddition of N-alkenyl substituted diazoimides Tetrahedron Letters. 35: 7159-7162. DOI: 10.1016/0040-4039(94)85349-5  0.417
1994 Padwa A, Austin DJ. Ligand Effects on the Chemoselectivity of Transition Metal Catalyzed Reactions ofα-Diazo Carbonyl Compounds Angewandte Chemie International Edition in English. 33: 1797-1815. DOI: 10.1002/Anie.199417971  0.419
1993 Hassner A, Maurya R, Friedman O, Gottlieb HE, Padwa A, Austin D. Stereochemistry. 82. Conformation of fused five-membered heterocyclic rings derived from the intramolecular oxime olefin cycloaddition reaction The Journal of Organic Chemistry. 58: 4539-4546. DOI: 10.1021/Jo00069A011  0.367
1993 Padwa A, Austin DJ, Precedo L, Zhi L. Cycloaddition reactions of pyridinium and related azomethine ylides The Journal of Organic Chemistry. 58: 1144-1150. DOI: 10.1021/Jo00057A029  0.453
1993 Padwa A, Austin DJ, Price AT, Semones MA, Doyle MP, Protopopova MN, Winchester WR, Tran A. Ligand effects on dirhodium(II) carbene reactivities. Highly effective switching between competitive carbenoid transformations Journal of the American Chemical Society. 115: 8669-8680. DOI: 10.1021/Ja00072A021  0.405
1993 Padwa A, Austin DJ, Gareau Y, Kassir JM, Xu SL. Rearrangement of alkynyl and vinyl carbenoids via the rhodium(II)-catalyzed cyclization reaction of .alpha.-diazo ketones Journal of the American Chemical Society. 115: 2637-2647. DOI: 10.1021/JA00060A012  0.416
1993 Cox GG, Moody CJ, Austin DJ, Padwa A. Chemoselectivity of rhodium carbenoids. A comparison of the selectivity for OH insertion reactions or carbonyl ylide formation versus aliphatic and aromatic CH insertion and cyclopropanation Tetrahedron. 49: 5109-5126. DOI: 10.1016/S0040-4020(01)81876-7  0.459
1992 Padwa A, Austin DJ, Ishida M, Muller CL, Murphree SS, Yeske PE. Tunable regioselectivity associated with the reaction of 2,3-dihalo-1-(phenylsulfonyl)-1-propenes with ambident nucleophilic reagents The Journal of Organic Chemistry. 57: 1161-1169. DOI: 10.1021/Jo00030A024  0.44
1992 Padwa A, Austin DJ, Hornbuckle SF, Semones MA, Doyle MP, Protopopova MN. Control of chemoselectivity in catalytic carbenoid reactions. Dirhodium(II) ligand effects on relative reactivities Journal of the American Chemical Society. 114: 1874-1876. DOI: 10.1021/Ja00031A048  0.404
1992 Padwa A, Austin DJ, Hornbuckle SF, Price AT. Rhodium (II) catalyzed intramolecular dipolar cycloaddition reactions of carbonyl ylides. Computational and empirical studies of the regio- and chemoselective effect of catalyst ligand Tetrahedron Letters. 33: 6427-6430. DOI: 10.1016/S0040-4039(00)79006-X  0.448
1992 Hertzog DL, Austin DJ, Nadler WR, Padwa A. Intramolecular cycloaddition of isomünchnones derived from the rhodium(II) catalyzed cyclization of diazoimides Tetrahedron Letters. 33: 4731-4734. DOI: 10.1016/S0040-4039(00)61271-6  0.422
1991 Padwa A, Austin DJ, Xu SL. Rhodium (II) catalyzed cyclizations of α-diazo substituted alkynes. A new mode of reaction Tetrahedron Letters. 32: 4103-4106. DOI: 10.1016/S0040-4039(00)79874-1  0.451
1991 Padwa A, Austin DJ, Chiacchio U, Kassir JM, Rescifina A, Xu SL. Rearrangement of o-alkynyl substituted α-diazoacetophenones. Conversion to β-naphthols via arylketene intermediates Tetrahedron Letters. 32: 5923-5926. DOI: 10.1016/S0040-4039(00)79427-5  0.36
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