| Year |
Citation |
Score |
| 2020 |
Pirrone MG, Gysin M, Haldimann K, Hobbie SN, Vasella A, Crich D. Predictive Analysis of the Side Chain Conformation of the Higher Carbon Sugars: Application to the Preorganization of the Aminoglycoside Ring 1 Side Chain for Binding to the Bacterial Ribosomal Decoding A Site. The Journal of Organic Chemistry. PMID 32902280 DOI: 10.1021/Acs.Joc.0C01836 |
0.335 |
|
| 2020 |
Sonousi A, Vasella A, Crich D. Synthesis of a Pseudotrisaccharide Suitable for Synthesis of Ring I Modified 4,5-2-Deoxystreptamine Type Aminoglycoside Antibiotics. The Journal of Organic Chemistry. PMID 32336094 DOI: 10.1021/Acs.Joc.0C00743 |
0.416 |
|
| 2020 |
Pirrone MG, Matsushita T, Vasella A, Crich D. Stereospecific synthesis of methyl 2-amino-2,4-dideoxy-6S-deuterio-α-D-xylo-hexopyranoside and methyl 2-amino-2,4-dideoxy-6S-deuterio-4-propyl-α-d-glucopyranoside: Side chain conformation of the novel aminoglycoside antibiotic propylamycin. Carbohydrate Research. 491: 107984. PMID 32217361 DOI: 10.1016/J.Carres.2020.107984 |
0.435 |
|
| 2019 |
Quirke JCK, Rajasekaran P, Sarpe VA, Sonousi A, Osinnii I, Gysin M, Haldimann K, Fang QJ, Shcherbakov D, Hobbie SN, Sha SH, Schacht J, Vasella A, Böttger EC, Crich D. Apralogs: Apramycin 5-O-Glycosides and Ethers with Improved Antibacterial Activity and Ribosomal Selectivity and Reduced Susceptibility to the Aminoacyltranserferase (3)-IV Resistance Determinant. Journal of the American Chemical Society. PMID 31790244 DOI: 10.1021/Jacs.9B11601 |
0.323 |
|
| 2019 |
Sati GC, Sarpe VA, Furukawa T, Mondal S, Mantovani M, Hobbie SN, Vasella A, Böttger EC, Crich D. Modification at the 2'-Position of the 4,5-Series of 2-Deoxystreptamine Aminoglycoside Antibiotics to Resist Aminoglycoside Modifying Enzymes and Increase Ribosomal Target Selectivity. Acs Infectious Diseases. PMID 31436080 DOI: 10.1021/Acsinfecdis.9B00128 |
0.318 |
|
| 2019 |
Sonousi A, Shcherbakov D, Vasella A, Böttger EC, Crich D. Synthesis, ribosomal selectivity, and antibacterial activity of netilmicin 4'-derivatives. Medchemcomm. 10: 946-950. PMID 31303992 DOI: 10.1039/C9Md00153K |
0.407 |
|
| 2019 |
Sarpe VA, Pirrone MG, Haldimann K, Hobbie SN, Vasella A, Crich D. Synthesis of saccharocin from apramycin and evaluation of its ribosomal selectivity. Medchemcomm. 10: 554-558. PMID 31057735 DOI: 10.1039/C9Md00093C |
0.356 |
|
| 2018 |
Sonousi A, Sarpe VA, Brilkova M, Schacht J, Vasella A, Böttger EC, Crich D. Effects of the 1-N-(4-Amino-2S-hydroxybutyryl) and 6'-N-(2-Hydroxyethyl) Substituents on Ribosomal Selectivity, Cochleotoxicity and Antibacterial Activity in the Sisomicin Class of Aminoglycoside Antibiotics. Acs Infectious Diseases. PMID 29708331 DOI: 10.1021/Acsinfecdis.8B00052 |
0.333 |
|
| 2017 |
Mandhapati AR, Yang G, Kato T, Shcherbakov D, Hobbie SN, Vasella A, Böttger EC, Crich D. Structure-Based Design and Synthesis of Apramycin-Paromomycin Analogues. Importance of the Configuration at the 6'-Position and Differences Between the 6'-Amino and Hydroxy Series. Journal of the American Chemical Society. PMID 28892368 DOI: 10.1021/Jacs.7B07754 |
0.363 |
|
| 2017 |
Kato T, Vasella A, Crich D. Stereospecific synthesis of methyl 2-amino-2-deoxy-(6S)-deuterio-α,β-d-glucopyranoside and methyl 2,6-diamino-2,6-dideoxy-(6R)-deuterio-α,β-d-glucopyranoside: Side chain conformations of the 2-amino-2-deoxy and 2,6-diamino-2,6-dideoxyglucopyranosides. Carbohydrate Research. 448: 10-17. PMID 28554123 DOI: 10.1016/J.Carres.2017.05.015 |
0.374 |
|
| 2017 |
Sati GC, Scherbakov D, Hobbie SN, Vasella A, Böttger EC, Crich D. N6', N6''' and O4' Modifications to Neomycin Affect Ribosomal Selectivity Without Compromising Antibacterial Activity. Acs Infectious Diseases. PMID 28343384 DOI: 10.1021/Acsinfecdis.6B00214 |
0.334 |
|
| 2015 |
Kato T, Yang G, Teo Y, Juskeviciene R, Perez-Fernandez D, Shinde HM, Salian S, Bernet B, Vasella A, Böttger EC, Crich D. Synthesis and Antiribosomal Activities of 4'-O-, 6'-O-, 4″-O-, 4',6'-O- and 4″,6″-O-Derivatives in the Kanamycin Series Indicate Differing Target Selectivity Patterns between the 4,5- and 4,6-Series of Disubstituted 2-Deoxystreptamine Aminoglycoside Antibiotics. Acs Infectious Diseases. 1: 479-486. PMID 27623314 DOI: 10.1021/Acsinfecdis.5B00069 |
0.301 |
|
| 2015 |
Matsushita T, Chen W, Juskeviciene R, Teo Y, Shcherbakov D, Vasella A, Böttger EC, Crich D. Influence of 4'-O-Glycoside Constitution and Configuration on Ribosomal Selectivity of Paromomycin. Journal of the American Chemical Society. 137: 7706-17. PMID 26024064 DOI: 10.1021/Jacs.5B02248 |
0.321 |
|
| 2015 |
Mandhapati AR, Kato T, Matsushita T, Ksebati B, Vasella A, Böttger EC, Crich D. Fluorine-decoupled carbon spectroscopy for the determination of configuration at fully substituted, trifluoromethyl- and perfluoroalkyl-bearing carbons: comparison with 19F-1H heteronuclear Overhauser effect spectroscopy. The Journal of Organic Chemistry. 80: 1754-63. PMID 25561269 DOI: 10.1021/Jo502677A |
0.311 |
|
| 2014 |
Mandhapati ARe, Shcherbakov D, Duscha S, Vasella A, Böttger EC, Crich D. Importance of the 6'-hydroxy group and its configuration for apramycin activity Chemmedchem. 9: 2074-2083. PMID 25045149 DOI: 10.1002/Cmdc.201402146 |
0.303 |
|
| 2014 |
Perez-Fernandez D, Shcherbakov D, Matt T, Leong NC, Kudyba I, Duscha S, Boukari H, Patak R, Dubbaka SR, Lang K, Meyer M, Akbergenov R, Freihofer P, Vaddi S, Thommes P, ... ... Vasella A, et al. 4'-O-substitutions determine selectivity of aminoglycoside antibiotics. Nature Communications. 5: 3112. PMID 24473108 DOI: 10.1038/Ncomms4112 |
0.3 |
|
| 2014 |
Chen W, Matsushita T, Shcherbakov D, Boukari H, Vasella A, Böttger EC, Crich D. Synthesis, antiribosomal and antibacterial activity of 4′-O- glycopyranosyl paromomycin aminoglycoside antibiotics Medchemcomm. 5: 1179-1187. DOI: 10.1039/C4Md00119B |
0.314 |
|
| 2014 |
Schulze-Adams M, Bernet B, Touboul D, Egli D, Herdeis L, Vasella A. Oligonucleotide Analogues with Integrated Bases and Backbone. Part 32: Thiomethylene- and Aminomethylene-Linked GG Dinucleosides of the ONIB Type: Formation of Quadruplexes Helvetica Chimica Acta. 97: 1244-1268. DOI: 10.1002/Hlca.201400175 |
0.316 |
|
| 2013 |
Huang MH, Duchek J, Vasella A. Synthesis of a pseudodisaccharide α-C-glycosidically linked to an 8-alkylated guanine. Molecules (Basel, Switzerland). 18: 3906-16. PMID 23549297 DOI: 10.3390/Molecules18043906 |
0.463 |
|
| 2012 |
Salian S, Matt T, Akbergenov R, Harish S, Meyer M, Duscha S, Shcherbakov D, Bernet BB, Vasella A, Westhof E, Böttger EC. Structure-activity relationships among the kanamycin aminoglycosides: role of ring I hydroxyl and amino groups. Antimicrobial Agents and Chemotherapy. 56: 6104-8. PMID 22948879 DOI: 10.1128/Aac.01326-12 |
0.383 |
|
| 2011 |
Peifer M, Vasella A. Autonomously pairing cysteinyl-linked nucleotide analogues with a unique architecture. Journal of the American Chemical Society. 133: 4264-7. PMID 21384899 DOI: 10.1021/Ja200829S |
0.327 |
|
| 2011 |
Duchek J, Huang M, Vasella A. Towards stable di-carba analogues of guanofosfocins Tetrahedron Letters. 52: 2940-2942. DOI: 10.1016/J.Tetlet.2011.02.102 |
0.473 |
|
| 2011 |
De Giacomo F, Peifer M, Rajic Z, Vasella A. Oligonucleotide analogues with integrated bases and Backbone. Part 28 1): Hydrazide- and amide-linked analogues. 2. di-, tetra-, octa-, and decamers: Synthesis and association Helvetica Chimica Acta. 94: 1153-1193. DOI: 10.1002/Hlca.201100124 |
0.41 |
|
| 2011 |
Duchek J, Vasella A. Synthesis of Benzimidazoles by Phosphine-Mediated Reductive Cyclisation of ortho-Nitro-anilides Helvetica Chimica Acta. 94: 977-986. DOI: 10.1002/Hlca.201100123 |
0.353 |
|
| 2011 |
del Carmen Ruiz Ruiz M, Vasella A. The ‘t-Amino Effect’ of ortho-Nitroso Amines. Synthesis of 2,6-Diaminoadenine Derivatives from 6-(Dialkylamino)-5-nitrosopyrimidines Helvetica Chimica Acta. 94: 785-800. DOI: 10.1002/Hlca.201100098 |
0.415 |
|
| 2010 |
Kreße G, Felber H, Ritter A, Ascherl B, Vasella A. Ene reactions with α-chloronitroso compounds: Asymmetric synthesis of N-allylhydroxylamines Recueil Des Travaux Chimiques Des Pays-Bas. 105: 295-298. DOI: 10.1002/Recl.19861050911 |
0.378 |
|
| 2010 |
Bogliotti N, Bernet B, Vasella A. Oligonucleotide Analogues with Integrated Bases and Backbones. Part 23 Helvetica Chimica Acta. 93: 659-667. DOI: 10.1002/Hlca.201300043 |
0.327 |
|
| 2010 |
Collin M, Vasella A. Towards the Synthesis of 1-Deoxy-1-nitropiperidinoses Helvetica Chimica Acta. 93: 2297-2317. DOI: 10.1002/Hlca.201000326 |
0.4 |
|
| 2010 |
Stichler-Bonaparte J, Bernet B, Vasella A. ChemInform Abstract: Oligosaccharide Analogues of Polysaccharides. Part 25. Synthesis of Mono- and Diethynylated Analogues of 2-Acetamido-2-deoxy-D-glucopyranose. Cheminform. 33: no-no. DOI: 10.1002/CHIN.200249174 |
0.337 |
|
| 2010 |
Storz T, Bernet B, Vasella A. ChemInform Abstract: β-Lactams from D-Erythrose-Derived Imines: A Convenient Synthesis of 2,3-Diamino-2,3-dideoxy-D-mannonic Acid Derivatives. Cheminform. 31: no-no. DOI: 10.1002/CHIN.200012238 |
0.309 |
|
| 2010 |
Vasella A, Wenger W, Rajamannar T. ChemInform Abstract: Glycosylidene Carbenes. Part 28. Synthesis of Glycosyl Boranes and Glycosyl Borinates. Cheminform. 31: no-no. DOI: 10.1002/CHIN.200006216 |
0.305 |
|
| 2010 |
WIDAUER C, BERNET B, VASELLA A. ChemInform Abstract: Synthesis of Enantiomerically Pure Carbohydrate-Derived Annulated Cyclopentadienes and of a Ferrocene. Cheminform. 29: no-no. DOI: 10.1002/CHIN.199825210 |
0.339 |
|
| 2010 |
XU J, EGGER A, BERNET B, VASELLA A. ChemInform Abstract: Oligosaccharide Analogues of Polysaccharides. Part 9. Synthesis and Thermolysis of Acetylenosaccharide-Derived 1,2-Dialkynylbenzenes. Cheminform. 28: no-no. DOI: 10.1002/CHIN.199705246 |
0.352 |
|
| 2010 |
CZOLLNER L, BAUDIN G, BERNET B, VASELLA A. ChemInform Abstract: Synthesis of a 1,2-trans-Configurated, Equatorial Glycosylphosphonate Analogue of D-myo-Inositol 1,4,5-Trisphosphate. Cheminform. 24: no-no. DOI: 10.1002/CHIN.199331252 |
0.312 |
|
| 2010 |
MAHMOOD K, VASELLA A, BERNET B. ChemInform Abstract: Deoxy-nitrosugars. Part 17. Synthesis of Ketose-Derived Nucleosides from 1-Deoxy-1-nitroribose. Cheminform. 23: no-no. DOI: 10.1002/CHIN.199205277 |
0.344 |
|
| 2009 |
Mathew T, Billich A, Cavallari M, Bornancin F, Nussbaumer P, De Libero G, Vasella A. Synthesis and evaluation of sphingolipid analogues: modification of the hydroxy group at C(1) of 7-oxasphingosine, and of the hydroxy group at C(1) and the amide group of 7-oxaceramides. Chemistry & Biodiversity. 6: 705-24. PMID 19479849 DOI: 10.1002/Cbdv.200900013 |
0.325 |
|
| 2009 |
Mathew T, Billaud C, Billich A, Cavallari M, Nussbaumer P, De Libero G, Vasella A. Synthesis of 7-aza- and 7-thiasphingosines, and evaluation of their interaction with sphingosine kinases and with T-cells. Chemistry & Biodiversity. 6: 725-38. PMID 19479838 DOI: 10.1002/Cbdv.200900039 |
0.306 |
|
| 2009 |
Steinlin T, Vasella A. Acylation of a 6-(Methylamino)-5-nitrosopyrimidine and 1,3-Dipolar Cycloaddition of an 8-MethylisoxanthopterinN(5)-Oxide. Synthesis ofC(6),N(8)-Disubstituted Isoxanthopterins Helvetica Chimica Acta. 92: 588-606. DOI: 10.1002/Hlca.200900009 |
0.43 |
|
| 2009 |
Rajan R, Mathew T, Buffa R, Bornancin F, Cavallari M, Nussbaumer P, De Libero G, Vasella A. Synthesis and Evaluation ofN-Acetyl-2-amino-2-deoxy-α-D-galactosyl 1-Thio-7-oxaceramide, a New Analogue ofα-D-Galactosyl Ceramide Helvetica Chimica Acta. 92: 918-927. DOI: 10.1002/Hlca.200800454 |
0.393 |
|
| 2009 |
Collin M, Hobbie S, Böttger E, Vasella A. Synthesis and Evaluation ofS- andC(1)-Substituted Analogues of Lincomycin Helvetica Chimica Acta. 92: 230-266. DOI: 10.1002/Hlca.200800343 |
0.372 |
|
| 2008 |
Zhang F, Vasella A. A New Synthesis of Ciliapterin and Dictyopterin. Ene Reactions of (Alkenylamino)-nitroso-pyrimidines Helvetica Chimica Acta. 91: 2351-2360. DOI: 10.1002/Hlca.200890255 |
0.396 |
|
| 2008 |
Steinlin T, Sonati T, Vasella A. Synthesis and Reactivity in [3+2] Cycloadditions of IsoxanthopterinN(5)-Oxides - A New Synthesis of 6-Substituted Pteridinediones Helvetica Chimica Acta. 91: 1879-1887. DOI: 10.1002/Hlca.200890201 |
0.422 |
|
| 2008 |
Collin M, Hobbie S, Böttger E, Vasella A. Synthesis of 1,2,3-Triazole Analogues of Lincomycin Helvetica Chimica Acta. 91: 1838-1848. DOI: 10.1002/Hlca.200890196 |
0.368 |
|
| 2008 |
Pathak R, Perez-Fernandez D, Nandurdikar R, Kalapala S, Böttger E, Vasella A. Synthesis and Evaluation of Paromomycin Derivatives Modified at C(4′) Helvetica Chimica Acta. 91: 1533-1552. DOI: 10.1002/Hlca.200890167 |
0.426 |
|
| 2008 |
Zhang F, Kulesza A, Rani S, Bernet B, Vasella A. 6-(Diazomethyl)-1,3-bis(methoxymethyl)uracil, Synthesis and Transformation into Annulated Pyrimidinediones Helvetica Chimica Acta. 91: 1201-1218. DOI: 10.1002/Hlca.200890132 |
0.385 |
|
| 2008 |
Zhang F, Bernet B, Bonnet V, Dangles O, Sarabia F, Vasella A. 2-Azido-2-deoxycellulose: Synthesis and 1,3-Dipolar Cycloaddition Helvetica Chimica Acta. 91: 608-617. DOI: 10.1002/Hlca.200890064 |
0.348 |
|
| 2008 |
Steinlin T, Vasella A. Diels–Alder Additions, Ene Reactions, and Condensations of 4-(Acylamino)-5-nitrosopyrimidines – Synthesis of 8-Substituted Guanines and of 6-Substituted Pteridinones Helvetica Chimica Acta. 91: 435-450. DOI: 10.1002/Hlca.200890048 |
0.413 |
|
| 2007 |
Zhang F, Vasella A. Regioselective synthesis of 1I,1II,5I,5II,6I,6I,6II,6II-2H8-cellobiose. Carbohydrate Research. 342: 2546-56. PMID 17803982 DOI: 10.1016/J.Carres.2007.07.017 |
0.311 |
|
| 2007 |
Kudyba I, Fernandez DP, Böttger EC, Vasella A. Synthesis of paromomycin derivatives modified at C(5'') to selectively target bacterial rRNA. Carbohydrate Research. 342: 499-519. PMID 17049499 DOI: 10.1016/J.Carres.2006.09.014 |
0.432 |
|
| 2007 |
Zhang X, Bernet B, Vasella A. Oligonucleotide Analogues with Integrated Bases and Backbone. Part 16 Helvetica Chimica Acta. 90: 891-908. DOI: 10.1002/Hlca.201000217 |
0.318 |
|
| 2007 |
Zhang F, Vasella A. Synthesis of Spiropyrimidodiazepines and Spirodiazepinopurines by Tandem Nitroso-ene/Diels–Alder Reactions Helvetica Chimica Acta. 90: 2315-2329. DOI: 10.1002/Hlca.200790238 |
0.373 |
|
| 2007 |
Bernet B, Vasella A. Hydrogen Bonding of Fluorinated Saccharides in Solution: F Acting as H-Bond Acceptor in a Bifurcated H-Bond of 4-Fluorinated Levoglucosans Helvetica Chimica Acta. 90: 1874-1888. DOI: 10.1002/Hlca.200790196 |
0.303 |
|
| 2007 |
Zhang X, Bernet B, Vasella A. Oligonucleotide Analogues with Integrated Bases and Backbone. Part 15 Helvetica Chimica Acta. 90: 864-890. DOI: 10.1002/Hlca.200790090 |
0.316 |
|
| 2007 |
Zhang F, Schweizer W, Xu M, Vasella A. A New Synthesis of Pteridines Substituted with Branched and Linear Alkenyl Groups at C(6). The Nitroso-Ene Reaction of 4-(Alkenoylamino)-5-nitrosopyrimidines Helvetica Chimica Acta. 90: 521-534. DOI: 10.1002/Hlca.200790054 |
0.408 |
|
| 2006 |
Shanmugasundaram B, Debowski AW, Dennis RJ, Davies GJ, Vocadlo DJ, Vasella A. Inhibition of O-GlcNAcase by a gluco-configured nagstatin and a PUGNAc-imidazole hybrid inhibitor. Chemical Communications (Cambridge, England). 4372-4. PMID 17057847 DOI: 10.1039/B612154C |
0.318 |
|
| 2006 |
Vasella A, Storz T. Practical and Efficient Synthesis of a Chiral C5 Building Block, 2-O-Allyl-d-arabinose, from Diacetone-d-glucose Synthesis. 2006: 1461-1464. DOI: 10.1055/S-2006-926418 |
0.401 |
|
| 2006 |
Pabba J, Vasella A. Probing the Interaction of the Hydroxy Group at C(4) of Lactone-Type Inhibitors withβ-Glucosidases andβ-Galactosidases Helvetica Chimica Acta. 89: 2006-2019. DOI: 10.1002/Hlca.200690191 |
0.422 |
|
| 2006 |
Pabba J, Mohal N, Vasella A. Synthesis of Glucuronic, Mannuronic, and Galacturonic Acid-Derived Imidazoles as Inhibitors of Bovine Liverβ-Glucuronidase Helvetica Chimica Acta. 89: 1373-1386. DOI: 10.1002/Hlca.200690137 |
0.423 |
|
| 2006 |
Xu M, Vasella A. A New Synthesis of Pteridines Helvetica Chimica Acta. 89: 1140-1146. DOI: 10.1002/Hlca.200690111 |
0.416 |
|
| 2006 |
Murty K, Xie T, Bernet B, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 26 Helvetica Chimica Acta. 89: 675-730. DOI: 10.1002/Hlca.200690068 |
0.402 |
|
| 2006 |
Pabba J, Rempel BP, Withers SG, Vasella A. Synthesis of glycaro-1,5-lactams and tetrahydrotetrazolopyridine-5- carboxylates: Inhibitors of β-D-glucuronidase and α-L-iduronidase Helvetica Chimica Acta. 89: 635-666. DOI: 10.1002/Hlca.200690066 |
0.392 |
|
| 2006 |
Buser S, Vasella A. Norbornane Mimics of Distortedβ-D-Glucopyranosides – Inhibitors ofβ-D-Glucopyranosidases? Helvetica Chimica Acta. 89: 614-621. DOI: 10.1002/Hlca.200690064 |
0.338 |
|
| 2006 |
Buser S, Vasella A. Synthesis of 2-Azabicyclo[3.2.2]nonane-Derived Monosaccharide Mimics and Their Evaluation as Glycosidase Inhibitors Helvetica Chimica Acta. 89: 416-426. DOI: 10.1002/Hlca.200690042 |
0.341 |
|
| 2005 |
Hrmova M, Streltsov VA, Smith BJ, Vasella A, Varghese JN, Fincher GB. Structural rationale for low-nanomolar binding of transition state mimics to a family GH3 beta-D-glucan glucohydrolase from barley. Biochemistry. 44: 16529-39. PMID 16342944 DOI: 10.1021/Bi0514818 |
0.312 |
|
| 2005 |
Huang CH, Lai WL, Lee MH, Chen CJ, Vasella A, Tsai YC, Liaw SH. Crystal structure of glucooligosaccharide oxidase from Acremonium strictum: a novel flavinylation of 6-S-cysteinyl, 8alpha-N1-histidyl FAD. The Journal of Biological Chemistry. 280: 38831-8. PMID 16154992 DOI: 10.1074/Jbc.M506078200 |
0.344 |
|
| 2005 |
Pabba J, Vasella A. Synthesis of d-gluco-, l-ido-, d-galacto-, and l-altro-configured glycaro-1,5-lactams from tartaric acid Tetrahedron Letters. 46: 3619-3622. DOI: 10.1016/J.Tetlet.2005.03.188 |
0.37 |
|
| 2005 |
Terinek M, Vasella A. Synthesis and evaluation of two mannosamine-derived lactone-type inhibitors of snail β-mannosidase Tetrahedron: Asymmetry. 16: 449-469. DOI: 10.1016/J.Tetasy.2004.11.068 |
0.427 |
|
| 2005 |
Mohal N, Bernet B, Vasella A. Synthesis of a Fusion-Isomeric Cellobionoimidazole and Its Evaluation against thesyn-Protonating Glycosidase Cel7A Helvetica Chimica Acta. 88: 3232-3252. DOI: 10.1002/Hlca.200590260 |
0.436 |
|
| 2005 |
Buser S, Vasella A. 7-Oxanorbornane and Norbornane Mimics of a Distortedβ-D-Mannopyranoside: Synthesis and Evaluation asβ-Mannosidase Inhibitors Helvetica Chimica Acta. 88: 3151-3173. DOI: 10.1002/Hlca.200590255 |
0.391 |
|
| 2005 |
Pathak R, Böttger E, Vasella A. Design and Synthesis of Aminoglycoside Antibiotics to Selectively Target 16S Ribosomal RNA Position 1408 Helvetica Chimica Acta. 88: 2967-2985. DOI: 10.1002/Hlca.200590240 |
0.421 |
|
| 2005 |
Xu M, Miao Z, Bernet B, Vasella A. Functionalised Monocyclic Five- to Seven-Memberedexo-Glycals by Alkynol Cycloisomerisation of Hydroxy Buta-1,3-diynes and 1-Haloalkynols Helvetica Chimica Acta. 88: 2918-2937. DOI: 10.1002/Hlca.200590235 |
0.384 |
|
| 2005 |
Shanmugasundaram B, Vasella A. Synthesis of NewC(2)-Substitutedgluco-Configured Tetrahydroimidazopyridines and Their Evaluation as Glucosidase Inhibitors Helvetica Chimica Acta. 88: 2593-2602. DOI: 10.1002/Hlca.200590199 |
0.357 |
|
| 2005 |
Magdolen P, Vasella A. Monocyclic, Substituted Imidazoles as Glycosidase Inhibitors Helvetica Chimica Acta. 88: 2454-2469. DOI: 10.1002/Hlca.200590182 |
0.308 |
|
| 2005 |
Miao Z, Xu M, Hoffmann B, Bernet B, Vasella A. Functionalised Bicyclicexo-Glycals by Alkynol Cycloisomerisation of Hydroxy 1,3-Diynes and Hydroxy Haloalkynes Helvetica Chimica Acta. 88: 1885-1912. DOI: 10.1002/Hlca.200590145 |
0.404 |
|
| 2005 |
Mohal N, Vasella A. Synthesis of Fusion-Isomeric Imidazopyridines and Their Evaluation as Inhibitors ofsyn- andanti-Protonating Glycosidases Helvetica Chimica Acta. 88: 100-119. DOI: 10.1002/Hlca.200490287 |
0.381 |
|
| 2005 |
Terinek M, Vasella A. Synthesis ofN-Acetylglucosamine-Derived Nagstatin Analogues and Their Evaluation as Glycosidase Inhibitors Helvetica Chimica Acta. 88: 10-22. DOI: 10.1002/Hlca.200490286 |
0.414 |
|
| 2004 |
Rajan R, Wallimann K, Vasella A, Pace D, Genazzani AA, Canonico PL, Condorelli F. Synthesis of 7-oxasphingosine and -ceramide analogues and their evaluation in a model for apoptosis. Chemistry & Biodiversity. 1: 1785-99. PMID 17191816 DOI: 10.1002/Cbdv.200490134 |
0.314 |
|
| 2004 |
Pfister P, Hobbie S, Brüll C, Corti N, Vasella A, Westhof E, Böttger EC. Mutagenesis of 16S rRNA C1409-G1491 base-pair differentiates between 6'OH and 6'NH3+ aminoglycosides. Journal of Molecular Biology. 346: 467-75. PMID 15670597 DOI: 10.1016/J.Jmb.2004.11.073 |
0.3 |
|
| 2004 |
Hrmova M, De Gori R, Smith BJ, Vasella A, Varghese JN, Fincher GB. Three-dimensional structure of the barley beta-D-glucan glucohydrolase in complex with a transition state mimic. The Journal of Biological Chemistry. 279: 4970-80. PMID 14597633 DOI: 10.1074/Jbc.M307188200 |
0.332 |
|
| 2004 |
Vaaje-Kolstad G, Vasella A, Peter MG, Netter C, Houston DR, Westereng B, Synstad B, Eijsink VG, van Aalten DM. Interactions of a family 18 chitinase with the designed inhibitor HM508 and its degradation product, chitobiono-delta-lactone. The Journal of Biological Chemistry. 279: 3612-9. PMID 14597613 DOI: 10.1074/Jbc.M310057200 |
0.315 |
|
| 2004 |
Kulesza A, Frank C, Aebi M, Vasella A. Synthesis of Stable Dolichylphosphomannose Analogues Helvetica Chimica Acta. 87: 3106-3118. DOI: 10.1002/Hlca.200490278 |
0.379 |
|
| 2004 |
Terinek M, Vasella A. Synthesis of Tetrahydropyridoimidazole‐2‐acetates: Effect of Carboxy and Methoxycarbonyl Groups at C(2) on the Inhibition of Some β‐ and α‐Glycosidases Helvetica Chimica Acta. 87: 3035-3049. DOI: 10.1002/Hlca.200490273 |
0.389 |
|
| 2004 |
Eppacher S, Christen M, Vasella A. Synthesis and Incorporation ofC(5?)-Ethynylated Uracil-Derived Phosphoramidites into RNA Helvetica Chimica Acta. 87: 3004-3020. DOI: 10.1002/Hlca.200490271 |
0.33 |
|
| 2004 |
Eppacher S, Bhardwaj PK, Bernet B, Gala JLB, Knöpfel T, Vasella A. Oligonucleosides with a nucleobase-including backbone: Part 12 - Synthesis of mixed ethynylene-linked uridine- and adenosine-derived tetramers Helvetica Chimica Acta. 87: 2969-2986. DOI: 10.1002/Hlca.200490269 |
0.416 |
|
| 2004 |
Kapferer P, Vasella A. Electrophilic Bromination ofN-Acylated Cyclohex-3-en-1-amines: Synthesis of 7-Azanorbornanes Helvetica Chimica Acta. 87: 2764-2789. DOI: 10.1002/Hlca.200490249 |
0.438 |
|
| 2004 |
Böhm M, Vasella A. Probing the Conformational Changes in the Enzymatic Hydrolysis of 2-Acetamido-2-deoxy-β-D-glucopyranosides Helvetica Chimica Acta. 87: 2566-2573. DOI: 10.1002/Hlca.200490229 |
0.395 |
|
| 2004 |
Hu G, Vasella A. Cyclopentanes fromN-Aminoglyconolactams: Reaction Mechanism and Improved Access to Diazocyclopentanones Helvetica Chimica Acta. 87: 2434-2446. DOI: 10.1002/Hlca.200490218 |
0.312 |
|
| 2004 |
Hu G, Vasella A. Synthesis and Oxidation ofN-Aminoglyconolactams: A Synthesis of Mannostatin A Helvetica Chimica Acta. 87: 2405-2433. DOI: 10.1002/Hlca.200490217 |
0.352 |
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| 2004 |
Matthews AJ, Bhardwaj PK, Vasella A. Oligonucleotide analogues with a 'nucleobase-including backbone': Part 10 - Design, synthesis, and association of ether-linked dimers Helvetica Chimica Acta. 87: 2273-2295. DOI: 10.1002/Hlca.200490204 |
0.371 |
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| 2004 |
George TG, Szolcsányi P, Koenig SG, Paterson DE, Isshiki Y, Vasella A. Preparation of an advanced intermediate for the synthesis of stable analogues of guanofosfocin Helvetica Chimica Acta. 87: 1287-1298. DOI: 10.1002/Hlca.200490118 |
0.427 |
|
| 2004 |
Terinek M, Vasella A. Improved Access to Imidazole-phosphonic Acids: Synthesis ofD-manno-Tetrahydroimidazopyridine-2-phosphonates Helvetica Chimica Acta. 87: 719-734. DOI: 10.1002/Hlca.200490067 |
0.435 |
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| 2003 |
Xu M, De Giacomo F, Paterson DE, George TG, Vasella A. An improved procedure for the preparation of 8-substituted guanines. Chemical Communications (Cambridge, England). 1452-3. PMID 12841287 DOI: 10.1039/B302529B |
0.375 |
|
| 2003 |
Hu G, Zimmermann M, Ramana CV, Vasella A. Cyclopentanes from N-amino-glyconolactams. A synthesis of mannostatin A. Chemical Communications (Cambridge, England). 952-3. PMID 12744315 DOI: 10.1039/B301213A |
0.609 |
|
| 2003 |
Matthews AJ, Bhardwaj PK, Vasella A. Oligonucleosides with a nucleobase-including backbone; synthesis and self-association of novel dinucleotide analogues. Chemical Communications (Cambridge, England). 950-1. PMID 12744314 DOI: 10.1039/B300932G |
0.313 |
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| 2003 |
Böhm M, Lorthiois E, Meyyappan M, Vasella A. Isoquinuclidine Mimics ofβ-D-Glucopyranosides: Differences and Similarities in the Mechanism of Action of someβ-D-Glucosidases and aβ-D-Mannosidase Helvetica Chimica Acta. 86: 3818-3835. DOI: 10.1002/Hlca.200390321 |
0.388 |
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| 2003 |
Böhm M, Lorthiois E, Meyyappan M, Vasella A. Synthesis and Evaluation as Glycosidase Inhibitors of Isoquinuclidines Mimicking a Distortedβ-Mannopyranoside Helvetica Chimica Acta. 86: 3787-3817. DOI: 10.1002/Hlca.200390320 |
0.378 |
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| 2003 |
Terinek M, Vasella A. Synthesis ofC(2)-Substitutedmanno-Configured Tetrahydroimidazopyridines and Their Evaluation as Inhibitors of Snailβ-Mannosidase Helvetica Chimica Acta. 86: 3482-3509. DOI: 10.1002/Hlca.200390293 |
0.328 |
|
| 2003 |
Blüchel C, Ramana CV, Vasella A. Synthesis of monosaccharide-derived spirocyclic cyclopropylamines and their evaluation as glycosidase inhibitors Helvetica Chimica Acta. 86: 2998-3036. DOI: 10.1002/Hlca.200390245 |
0.621 |
|
| 2003 |
Mangholz S, Briner K, Bernet B, Vasella A. Glycosylidene Carbenes. Part 32 Helvetica Chimica Acta. 86: 2490-2508. DOI: 10.1002/Hlca.200390202 |
0.309 |
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| 2003 |
Kapferer P, Birault V, Poisson J, Vasella A. Synthesis and Evaluation as Glycosidase Inhibitors of Carbasugar-Derived Spirodiaziridines, Spirodiazirines, and Spiroaziridines Helvetica Chimica Acta. 86: 2210-2227. DOI: 10.1002/Hlca.200390178 |
0.37 |
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| 2003 |
Bernet B, Mangholz S, Briner K, Vasella A. Glycosylidene Carbenes. Part 31 Helvetica Chimica Acta. 86: 1488-1521. DOI: 10.1002/Hlca.200390132 |
0.372 |
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| 2002 |
Koivula A, Ruohonen L, Wohlfahrt G, Reinikainen T, Teeri TT, Piens K, Claeyssens M, Weber M, Vasella A, Becker D, Sinnott ML, Zou JY, Kleywegt GJ, Szardenings M, Ståhlberg J, et al. The active site of cellobiohydrolase Cel6A from Trichoderma reesei: the roles of aspartic acids D221 and D175. Journal of the American Chemical Society. 124: 10015-24. PMID 12188666 DOI: 10.1021/Ja012659Q |
0.323 |
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| 2002 |
von Ballmoos C, Appoldt Y, Brunner J, Granier T, Vasella A, Dimroth P. Membrane topography of the coupling ion binding site in Na+-translocating F1F0 ATP synthase. The Journal of Biological Chemistry. 277: 3504-10. PMID 11719523 DOI: 10.1074/Jbc.M110301200 |
0.303 |
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| 2002 |
Hu G, Vasella A. Regioselective Benzoylation of 6-O-Protected and 4,6-O-Diprotected Hexopyranosides as Promoted by Chiral and Achiral Ditertiary 1,2-Diamines Helvetica Chimica Acta. 85: 4369-4391. DOI: 10.1002/Hlca.200290018 |
0.371 |
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| 2002 |
Bernet B, Bürli R, Xu J, Vasella A. Influence of an Ethynyl or a Buta-1,3-diynyl Group on the Chemical Shifts of Hydroxy Groups of Glucopyranoses Helvetica Chimica Acta. 85: 1800-1811. DOI: 10.1002/1522-2675(200206)85:6<1800::Aid-Hlca1800>3.0.Co;2-S |
0.359 |
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| 2002 |
Remen L, Vasella A. Conformationally Biased Mimics of Mannopyranosylamines: Inhibitors of β-Mannosidases? Helvetica Chimica Acta. 85: 1118. DOI: 10.1002/1522-2675(200204)85:4<1118::Aid-Hlca1118>3.0.Co;2-S |
0.383 |
|
| 2002 |
Bhardwaj P, Vasella A. Oligonucleosides with a Nucleobase-Including Backbone, Part 7 Helvetica Chimica Acta. 85: 699. DOI: 10.1002/1522-2675(200203)85:3<699::Aid-Hlca699>3.0.Co;2-N |
0.337 |
|
| 2002 |
Hoffmann B, Bernet B, Vasella A. Oligosaccharide Analogues of Polysaccharides Helvetica Chimica Acta. 85: 265-287. DOI: 10.1002/1522-2675(200201)85:1<265::Aid-Hlca265>3.0.Co;2-1 |
0.404 |
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| 2001 |
Blüchel C, Linden A, Vasella A. Glycosylidene Carbenes, Part 30, Crystal Structure of a Glucose-DerivedN,N-Unsubstituted Alkoxydiaziridine Helvetica Chimica Acta. 84: 3495-3502. DOI: 10.1002/1522-2675(20011114)84:11<3495::Aid-Hlca3495>3.0.Co;2-N |
0.304 |
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| 2001 |
Stichler-Bonaparte J, Vasella A. Oligosaccharide Analogues of Polysaccharides, Part 23, Synthesis of a Dimeric Acetyleno Cyclodextrin from a Mannopyranose-Derived Dialkyne Helvetica Chimica Acta. 84: 2355-2367. DOI: 10.1002/1522-2675(20010815)84:8<2355::Aid-Hlca2355>3.0.Co;2-X |
0.417 |
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| 2001 |
Hoffmann B, Zanini D, Ripoche I, Bürli R, Vasella A. Oligosaccharide Analogues of Polysaccharides, Part 22, Synthesis of Cyclodextrin Analogues Containing a Buta-1,3-diyne-1,4-diyl or a Butane-1,4-diyl Unit Helvetica Chimica Acta. 84: 1862-1888. DOI: 10.1002/1522-2675(20010613)84:6<1862::Aid-Hlca1862>3.0.Co;2-Z |
0.382 |
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| 2001 |
Czechtizky W, Vasella A. Oligonucleotide Analogues with a Nucleobase-Including Backbone, Part 5, 2′-Deoxy-8-(hydroxymethyl)adenosine- and 2′-Deoxy-6-(hydroxymethyl)uridine-Derived Phosphoramidites: Synthesis and Incorporation into 14-Mer DNA Strands Helvetica Chimica Acta. 84: 594-612. DOI: 10.1002/1522-2675(20010321)84:3<594::Aid-Hlca594>3.0.Co;2-9 |
0.365 |
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| 2000 |
Gunji H, Vasella A. Oligonucleosides with a Nucleobase-Including Backbone, Part 4, A Convergent Synthesis of Ethynediyl-Linked Adenosine Tetramers Helvetica Chimica Acta. 83: 3229-3245. DOI: 10.1002/1522-2675(20001220)83:12<3229::Aid-Hlca3229>3.0.Co;2-S |
0.386 |
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| 2000 |
Gunji H, Vasella A. Oligonucleosides with a Nucleobase-Including Backbone, Part 3, Synthesis of Acetyleno-Linked Adenosine Dimers Helvetica Chimica Acta. 83: 2975-2992. DOI: 10.1002/1522-2675(20001108)83:11<2975::Aid-Hlca2975>3.0.Co;2-2 |
0.435 |
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| 2000 |
Venkata Ramana C, Vasella A. Sugar-Derived Di- and Tetrahydropyridazinones: Synthesis of New Glycosidase Inhibitors Helvetica Chimica Acta. 83: 1599-1610. DOI: 10.1002/1522-2675(20000705)83:7<1599::Aid-Hlca1599>3.0.Co;2-0 |
0.402 |
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| 2000 |
Gunji H, Vasella A. Oligonucleosides with a Nucleobase-Including Backbone, Part 2, Synthesis and Structure Determination of Adenosine-Derived Monomers Helvetica Chimica Acta. 83: 1331-1345. DOI: 10.1002/1522-2675(20000705)83:7<1331::Aid-Hlca1331>3.0.Co;2-Z |
0.427 |
|
| 2000 |
Eppacher S, Solladié N, Bernet B, Vasella A. Oligonucleosides with a Nucleobase-Including Backbone, Part 1, Concept, Force-Field Calculations, and Synthesis of Uridine-Derived Monomers and Dimers Helvetica Chimica Acta. 83: 1311-1330. DOI: 10.1002/1522-2675(20000705)83:7<1311::Aid-Hlca1311>3.0.Co;2-2 |
0.388 |
|
| 2000 |
Bernet B, Vasella A. 1H-NMR Analysis of Intra- and Intermolecular H-Bonds of Alcohols in DMSO: Chemical Shift of Hydroxy Groups and Aspects of Conformational Analysis of Selected Monosaccharides, Inositols, and Ginkgolides Helvetica Chimica Acta. 83: 995-1021. DOI: 10.1002/(Sici)1522-2675(20000510)83:5<995::Aid-Hlca995>3.0.Co;2-Q |
0.314 |
|
| 2000 |
Panday N, Canac Y, Vasella A. Very Strong Inhibition of Glucosidases byC(2)-Substituted Tetrahydroimidazopyridines Helvetica Chimica Acta. 83: 58-79. DOI: 10.1002/(Sici)1522-2675(20000119)83:1<58::Aid-Hlca58>3.0.Co;2-K |
0.362 |
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| 2000 |
Mohan H, Vasella A. An Improved Synthesis of 2-Acetamido-2-deoxy-D-gluconohydroximolactone (PUGNAc), A Strong Inhibitor ofβ-N-Acetylglucosaminidases Helvetica Chimica Acta. 83: 114-118. DOI: 10.1002/(Sici)1522-2675(20000119)83:1<114::Aid-Hlca114>3.0.Co;2-9 |
0.389 |
|
| 1999 |
Vonhoff S, Vasella A. An Advantageous Synthesis of 5,6,7,8-Tetra-Hydrotetrazolo[1,5-a]Pyridines Synthetic Communications. 29: 551-560. DOI: 10.1080/00397919908085802 |
0.408 |
|
| 1999 |
Vasella A, Wenger W, Rajamannar T. Synthesis of glycosyl boranes and glycosyl borinates Chemical Communications. 2215-2216. DOI: 10.1039/A906400A |
0.357 |
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| 1999 |
Scheffler G, Justus M, Vasella A, Wessel HP. A multicomponent one-pot reaction integrating a bis-functional carbohydrate derivative Tetrahedron Letters. 40: 5845-5848. DOI: 10.1016/S0040-4039(99)01146-6 |
0.331 |
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| 1999 |
Storz T, Bernet B, Vasella A. β-Lactams fromD-Erythrose-Derived Imines: A Convenient Synthesis of 2,3-Diamino-2,3-dideoxy-D-mannonic-Acid Derivatives Helvetica Chimica Acta. 82: 2380-2412. DOI: 10.1002/(Sici)1522-2675(19991215)82:12<2380::Aid-Hlca2380>3.0.Co;2-P |
0.427 |
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| 1999 |
Xu J, Vasella A. Oligosaccharide Analogues of Polysaccharides, Part 19, Synthesis of 2-(Naphthalen-1-yl)ethyl Cellooligoglycosides and [(Naphthalene-1,8-diyl)di(ethane-2,1-diyl)] Bis[cellooligoglycosides] Helvetica Chimica Acta. 82: 1728-1752. DOI: 10.1002/(Sici)1522-2675(19991006)82:10<1728::Aid-Hlca1728>3.0.Co;2-A |
0.459 |
|
| 1999 |
Billault I, Vasella A. Synthesis ofgluco-Configured Tetrahydroimidazopyridine-2phosphonate-Derived Lipids, Potential Glucosyl Transferase Inhibitors Helvetica Chimica Acta. 82: 1137-1149. DOI: 10.1002/(Sici)1522-2675(19990804)82:8<1137::Aid-Hlca1137>3.0.Co;2-N |
0.444 |
|
| 1999 |
Vonhoff S, Piens K, Pipelier M, Braet C, Claeyssens M, Vasella A. Inhibition of Cellobiohydrolases fromTrichoderma reesei. Synthesis and Evaluation of Some Glucose-, Cellobiose-, and Cellotriose-Derived Hydroximolactams andImidazoles Helvetica Chimica Acta. 82: 963-980. DOI: 10.1002/(Sici)1522-2675(19990707)82:7<963::Aid-Hlca963>3.0.Co;2-V |
0.347 |
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| 1999 |
Peer A, Vasella A. Synthesis of anL-Fucose-Derived Cyclic Nitrone and its Conversion toα-L-Fucosidase Inhibitors Helvetica Chimica Acta. 82: 1044-1065. DOI: 10.1002/(Sici)1522-2675(19990707)82:7<1044::Aid-Hlca1044>3.0.Co;2-3 |
0.413 |
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| 1999 |
Kapferer P, Sarabia F, Vasella A. Carbasaccharidesvia Ring-Closing Alkene Metathesis. A Synthesis of (+)-Valienamine fromD-Glucose Helvetica Chimica Acta. 82: 645-656. DOI: 10.1002/(Sici)1522-2675(19990505)82:5<645::Aid-Hlca645>3.0.Co;2-K |
0.443 |
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| 1999 |
Bürli R, Vasella A. Oligosaccharide Analogues of Polysaccharides, Part 18 , Synthesis of Cyclic Hybrids of 2,2′-Bipyridine and Acetylenosaccharides Helvetica Chimica Acta. 82: 485-493. DOI: 10.1002/(Sici)1522-2675(19990407)82:4<485::Aid-Hlca485>3.0.Co;2-A |
0.394 |
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| 1999 |
Bohner T, Becker O, Vasella A. Oligosaccharide Analogues of Polysaccharides, Part 17, Synthesis and Characterization of a Hexadecamer: Evidence for the Essential Structural Role of the Intramolecular, Interresidue C(3)−OH⋅⋅⋅O−C(5) Hydrogen Bond in Celluloses Helvetica Chimica Acta. 82: 198-228. DOI: 10.1002/(Sici)1522-2675(19990210)82:2<198::Aid-Hlca198>3.0.Co;2-Y |
0.412 |
|
| 1998 |
Vorwerk S, Vasella A. Carbocyclic Analogues of N-Acetyl-2,3-didehydro-2-deoxy-D-neuraminic Acid (Neu5Ac2en, DANA): Synthesis and Inhibition of Viral and Bacterial Neuraminidases. Angewandte Chemie (International Ed. in English). 37: 1732-1734. PMID 29711519 DOI: 10.1002/(Sici)1521-3773(19980703)37:12<1732::Aid-Anie1732>3.0.Co;2-I |
0.427 |
|
| 1998 |
Widauer C, Bernet B, Vasella A. Synthesis of Enantiomerically Pure Carbohydrate–Derived Annulated Cyclopentadienes and of a Ferrocene Synthetic Communications. 28: 593-602. DOI: 10.1080/00397919808005930 |
0.418 |
|
| 1998 |
Carcano M, Vasella A. Aldehyde-Promoted Addition of 2-(Trimethylsilyl)thiazole to ?,??-Dialkoxy Ketones: A new way to branched-chain monosaccharides Helvetica Chimica Acta. 81: 889-901. DOI: 10.1002/Hlca.19980810510 |
0.405 |
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| 1998 |
Granier T, Vasella A. Synthesis and Some Transformations of 2-Acetamido-5-amino-3,4,6-tri-O-benzyl-2,5-dideoxy-D-glucono-1,5-lactam Helvetica Chimica Acta. 81: 865-880. DOI: 10.1002/Hlca.19980810508 |
0.457 |
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| 1998 |
Heightman TD, Vasella A, Tsitsanou KE, Zographos SE, Skamnaki VT, Oikonomakos NG. Cooperative Interactions of the Catalytic Nucleophile and the Catalytic Acid in the Inhibition of ?-Glycosidases. Calculations and their validation by comparative kinetic and structural studies of the inhibition of glycogen phosphorylaseb Helvetica Chimica Acta. 81: 853-864. DOI: 10.1002/Hlca.19980810507 |
0.329 |
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| 1998 |
Biamonte MA, Vasella A. Glycosylidene Carbenes part 26. The intramolecular F…︁HO hydrogen bond of 1,3‐diaxial 3‐fluorocyclohexanols Helvetica Chimica Acta. 81: 695-717. DOI: 10.1002/Hlca.19980810320 |
0.354 |
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| 1998 |
Biamonte MA, Vasella A. An Advantageous Synthesis Of 1D- And 1L-1,2,3,5/4-Cyclohexanepentol Helvetica Chimica Acta. 81: 688-694. DOI: 10.1002/Hlca.19980810319 |
0.37 |
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| 1998 |
Panday N, Granier T, Vasella A. Synthesis and Evaluation of Indolizine‐Type Inhibitors of N‐acetyl‐β‐D‐glucosaminidases Helvetica Chimica Acta. 81: 475-490. DOI: 10.1002/Hlca.19980810303 |
0.442 |
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| 1998 |
Storz T, Vasella A. N-Monoalkylation of Tetra-O-benzyl-D-arabinonamide: Synthesis of Some Open-Chain Analogues ofN-Acetylneuraminic Acid and Their Evaluation as Sialidase Inhibitors Helvetica Chimica Acta. 81: 1896-1907. DOI: 10.1002/(Sici)1522-2675(19981007)81:10<1896::Aid-Hlca1896>3.0.Co;2-5 |
0.41 |
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| 1998 |
Vonhoff S, Heightman T, Vasella A. Inhibition of Glycosidases by Lactam Oximes: Influence of the Aglycon in Disaccharide Analogues Helvetica Chimica Acta. 81: 1710-1725. DOI: 10.1002/(Sici)1522-2675(19980909)81:9<1710::Aid-Hlca1710>3.0.Co;2-I |
0.37 |
|
| 1998 |
Vorwerk S, Vasella A. Carbocyclische Analoga vonN-Acetyl-2,3- didehydro-2-desoxy-D-neuraminsäure (Neu5Ac2en, DANA): Synthese und Hemmwirkung auf virale und bakterielle Neuraminidasen Angewandte Chemie. 110: 1765-1767. DOI: 10.1002/(Sici)1521-3757(19980619)110:12<1765::Aid-Ange1765>3.0.Co;2-Y |
0.314 |
|
| 1997 |
Hoos R, Vasella A, Rupitz K, Withers SG. d-Glyconhydroximolactams strongly inhibit α-glycosidases Carbohydrate Research. 298: 291-298. DOI: 10.1016/S0008-6215(96)00320-5 |
0.37 |
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| 1997 |
Bürli R, Vasella A. Oligosaccharide analogues of polysaccharides. Part 14:. Carbocyclic cyclodextrin analogues. Synthesis of all trimeric and tetrameric isomers by homo- and heterocoupling of 1,4-cis-diethynylated 1,5-anhydroglucitols Helvetica Chimica Acta. 80: 2215-2237. DOI: 10.1002/Hlca.19970800720 |
0.407 |
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| 1997 |
Waldraff C, Bernet B, Vasella A. Glycosylidene Carbenes. Part 24 Reactivity modulation by protecting groups of the addition of glycosylidene carbenes to electron-rich alkenes Helvetica Chimica Acta. 80: 1882-1900. DOI: 10.1002/Hlca.19970800612 |
0.364 |
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| 1997 |
Granier T, Gaiser F, Hintermann L, Vasella A. Synthesis via a Carbohydrate‐Derived Münchnone of Pyrrolopyridines (Indolizines) and imidazopyridines, and their evaluation as inhibitors of β‐D‐glucosidases Helvetica Chimica Acta. 80: 1443-1456. DOI: 10.1002/Hlca.19970800509 |
0.409 |
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| 1997 |
Bernet B, Mäder T, Vasella A. Glyconothio-O-lactones. Part III. Thermolysis of a 4,5-Dihydro-1,2,3- and a 2,5-Dihydro-1,3,4-thiadiazole Helvetica Chimica Acta. 80: 1260-1279. DOI: 10.1002/Hlca.19970800422 |
0.389 |
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| 1997 |
Bürli R, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 12. Synthesis of ‘acetyleno-saccharide’-derived cyclodextrin analogues Helvetica Chimica Acta. 80: 1027-1052. DOI: 10.1002/Hlca.19970800403 |
0.381 |
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| 1997 |
Granier T, Panday N, Vasella A. Structure-Activity Relations for Imidazo-pyridine-Type Inhibitors of ?-D-Glucosidases Helvetica Chimica Acta. 80: 979-987. DOI: 10.1002/Hlca.19970800329 |
0.429 |
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| 1997 |
Bürli R, Vasella A. Cyclic“Acetylenosaccharides”—Novel Cyclodextrin Analogues Angewandte Chemie International Edition in English. 36: 1852-1853. DOI: 10.1002/Anie.199718521 |
0.388 |
|
| 1996 |
Crennell SJ, Garman EF, Philippon C, Vasella A, Laver WG, Vimr ER, Taylor GL. The structures of Salmonella typhimurium LT2 neuraminidase and its complexes with three inhibitors at high resolution Journal of Molecular Biology. 259: 264-280. PMID 8656428 DOI: 10.1006/Jmbi.1996.0318 |
0.349 |
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| 1996 |
Ernst A, Gobbi L, Vasella A. Orthogonally protected dialkynes Tetrahedron Letters. 37: 7959-7962. DOI: 10.1016/0040-4039(96)01838-2 |
0.339 |
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| 1996 |
Li Z, Vasella A. Synthesis of Enantiomerically Pure Carbohydrate‐Derived Annulated Cyclopentadienes and Ferrocenes Helvetica Chimica Acta. 79: 2201-2218. DOI: 10.1002/Hlca.19960790815 |
0.408 |
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| 1996 |
Heightman TD, Locatelli M, Vasella A. Synthesis of Fused Triazoles as Probes for the Active Site of Retaining ?-Glycosidases: From Which Direction Is the Glycoside Protonated? Helvetica Chimica Acta. 79: 2190-2200. DOI: 10.1002/Hlca.19960790814 |
0.35 |
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| 1996 |
Xu J, Egger A, Bernet B, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 9. Synthesis and Thermolysis of Acetylenosaccharide‐Derived 1,2‐Dialkynylbenzenes Helvetica Chimica Acta. 79: 2004-2022. DOI: 10.1002/Hlca.19960790722 |
0.447 |
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| 1996 |
Hoos R, Huixin J, Vasella A, Weiss P. Synthesis and Enzymatic Evaluation of Substrates and Inhibitors of ?-Glucuronidases Helvetica Chimica Acta. 79: 1757-1784. DOI: 10.1002/Hlca.19960790703 |
0.336 |
|
| 1996 |
Ernst A, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 8. Orthogonally Protected Cellobiose-Derived Dialkynes. A Convenient Method for the Regioselective Bromo- and Protodegermylation of Trimethylgermyl- and Trimethylsilyl-protected Dialkynes Helvetica Chimica Acta. 79: 1279-1294. DOI: 10.1002/Hlca.19960790505 |
0.746 |
|
| 1996 |
Zapata A, Bernet B, Vasella A. Glycosylidene Carbenes. Part 23. Regioselective glycosidation of deoxy- and fluorodeoxy-myo-inositol derivatives Helvetica Chimica Acta. 79: 1169-1191. DOI: 10.1002/Hlca.19960790424 |
0.384 |
|
| 1996 |
Bürli R, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 7. Synthesis of a monosaccharide‐derived monomer for amylose and cyclodextrin analogues Helvetica Chimica Acta. 79: 1159-1168. DOI: 10.1002/Hlca.19960790423 |
0.471 |
|
| 1996 |
Fowler P, Bernet B, Vasella A. A1H-NMR Spectroscopic Investigation of the Conformation of the Acetamido Group in Some Derivatives ofN-Acetyl-D-allosamine and -D-glucosamine Helvetica Chimica Acta. 79: 269-287. DOI: 10.1002/Hlca.19960790127 |
0.373 |
|
| 1996 |
Cai C, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 6. Orthogonal protecting/activating groups in an improved binomial synthesis of ?acetyleno-oligosaccharides? Helvetica Chimica Acta. 79: 255-268. DOI: 10.1002/Hlca.19960790126 |
0.676 |
|
| 1995 |
Cai C, Vasella A. Oligosaccharide analogues of polysaccharides. Part 5. Studies on the cross-coupling of alkynes and haloalkynes Helvetica Chimica Acta. 78: 2053-2064. DOI: 10.1002/Hlca.19950780814 |
0.611 |
|
| 1995 |
Vasella A, Witzig C. Glycosylidene Carbenes. Part 22. ?-D-Selectivity in the Glycosidation by Carbenes Derived from 2-Acetamido-hexoses Helvetica Chimica Acta. 78: 1971-1982. DOI: 10.1002/Hlca.19950780806 |
0.427 |
|
| 1995 |
Granier T, Vasella A. Synthesis and Evaluation as Glycosidase Inhibitors of 1H-Imidazol-2-ylC-Glycopyranosides Helvetica Chimica Acta. 78: 1738-1746. DOI: 10.1002/Hlca.19950780707 |
0.384 |
|
| 1995 |
Alzeer J, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 4. Synthesis of a monosaccharide-derived octamer Helvetica Chimica Acta. 78: 1219-1237. DOI: 10.1002/Hlca.19950780515 |
0.762 |
|
| 1995 |
Mangholz SE, Vasella A. Glycosylidene Carbenes. Part 21. Synthesis of N-tosylglycono-1,4-lactone hydrazones as precursors of glycofuranosylidene carbenes Helvetica Chimica Acta. 78: 1020-1035. DOI: 10.1002/Hlca.19950780424 |
0.429 |
|
| 1995 |
Palme M, Vasella A. O-(1-Phenyl-1H-tetrazol-5-yl) Glycosides: Alternative synthesis and transformation into glycosyl fluorides Helvetica Chimica Acta. 78: 959-969. DOI: 10.1002/Hlca.19950780418 |
0.382 |
|
| 1995 |
Cai C, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 3. A new protecting group for alkynes: Orthogonally protected dialkynes Helvetica Chimica Acta. 78: 732-757. DOI: 10.1002/Hlca.19950780319 |
0.659 |
|
| 1995 |
Heightman TD, Ermert P, Klein D, Vasella A. Synthesis of Galactose‐ and N‐Acetylglucosamine‐Derived Tetrazoles and their evaluation as β‐glycosidase inhibitors Helvetica Chimica Acta. 78: 514-532. DOI: 10.1002/Hlca.19950780221 |
0.346 |
|
| 1995 |
Alzeer J, Cai C, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 1. Concept and synthesis of monosaccharide-derived monomers Helvetica Chimica Acta. 78: 242-264. DOI: 10.1002/Hlca.19950780122 |
0.797 |
|
| 1995 |
Alzeer J, Vasella A. Oligosaccharide Analogues of Polysaccharides. Part 2. Regioselective deprotection of monosaccharide-derived monomers and dimers Helvetica Chimica Acta. 78: 177-193. DOI: 10.1002/Hlca.19950780117 |
0.752 |
|
| 1995 |
Jonas U, Cardullo F, Belik P, Diederich F, Gügel A, Harth E, Herrmann A, Isaacs L, Müllen K, Ringsdorf H, Thilgen C, Uhlmann P, Vasella A, Waldraff CAA, Walter M. Synthesis of a Fullerene[60] Cryptate and Systematic Langmuir-Blodgett and Thin-Film Investigations of Amphiphilic Fullerene Derivatives Chemistry - a European Journal. 1: 243-251. DOI: 10.1002/Chem.19950010408 |
0.646 |
|
| 1994 |
Langston S, Bernet B, Vasella A. Temporary Protection and Activation in the Regioselective Synthesis of Saccharide Sulfates Helvetica Chimica Acta. 77: 2341-2353. DOI: 10.1002/Hlca.19940770821 |
0.305 |
|
| 1994 |
Uhlmann P, Harth E, Naughton AB, Vasella A. Glycosylidene Carbenes. Part 20. Synthesis of deprotected, spiro‐linked C‐glycosides of C60 Helvetica Chimica Acta. 77: 2335-2340. DOI: 10.1002/Hlca.19940770820 |
0.686 |
|
| 1994 |
Frey O, Hoffmann M, Wittmann V, Kessler H, Uhlmann P, Vasella A. Preparation and Transmetallation of a Triphenylstannyl ?-D-Glucopyranoside: A highly stereoselective route to ?-D-C-glycosidesvia glycosyl dianions Helvetica Chimica Acta. 77: 2060-2069. DOI: 10.1002/Hlca.19940770730 |
0.443 |
|
| 1994 |
Briner K, Bernet B, Maloisel J, Vasella A. Glycosylidene Carbenes. Part 19. Regioselective glycosidation of allyl 2-deoxy-2-phthalimido-D-allopyranosides Helvetica Chimica Acta. 77: 1969-1984. DOI: 10.1002/Hlca.19940770724 |
0.355 |
|
| 1994 |
Vedø P, Chauvin R, Li Z, Bernet B, Vasella A. Synthesis of Enantiomerically Pure Ferrocenes from Glycofuranosyl-cyclopentadienes, synthetic equivalents of (alkoxyalkyl)fulvenes Helvetica Chimica Acta. 77: 1631-1659. DOI: 10.1002/Hlca.19940770620 |
0.627 |
|
| 1994 |
Uhlmann P, Nanz D, Bozó E, Vasella A. Glycosylidene Carbenes. Part 18. Insertion of glycosylidene carbenes into the SnH bond of tributyl- and triphenylstannane: A synthesis of stannoglycosides Helvetica Chimica Acta. 77: 1430-1440. DOI: 10.1002/Hlca.19940770521 |
0.419 |
|
| 1994 |
Uhlmann P, Vasella A. Glycosylidene Carbenes. Part 17. Glycosidation of benzyl ?-D- and ?-L-ribopyranosides. Further evidence for the effect of stereoelectronic control on the regioselectivity of glycosidation Helvetica Chimica Acta. 77: 1175-1192. DOI: 10.1002/Hlca.19940770426 |
0.381 |
|
| 1994 |
Engstler M, Ferrero-Garcia MA, Parodi AJ, Schauer R, Storz-Eckerlin T, Vasella A, Witzig C, Zhu X. N-(4-Nitrophenyl)oxamic acid and related N-acylanilines are non-competitive inhibitors of Vibrio cholerae sialidase but do not inhibit Trypanosoma cruzi or Trypanosoma brucei trans-sialidases Helvetica Chimica Acta. 77: 1166-1174. DOI: 10.1002/Hlca.19940770425 |
0.318 |
|
| 1994 |
Schnabelrauch M, Vasella A, Withers SG. Synthesis and Evaluation as Irreversible Glycosidase Inhibitors of Mono- and Oligo(glycosylthio)benzoquinones Helvetica Chimica Acta. 77: 778-799. DOI: 10.1002/Hlca.19940770319 |
0.37 |
|
| 1994 |
Bozó E, Vasella A. Glycosylidene Carbenes. Part 16. Glycosidation of methyl 6-O-trityl-α-D-altropyranoside Helvetica Chimica Acta. 77: 745-753. DOI: 10.1002/Hlca.19940770316 |
0.411 |
|
| 1994 |
Muddasani PR, Bernet B, Vasella A. Glycosylidene Carbenes. Part 15. Synthesis of disaccharides from allopyranose-derived vicinal 1,2-diols. Evidence for the protonation by a H-bonded hydroxy group in the ?-plane of the intermediate carbene, followed by attack on the oxycarbenium ion in the ?-plane Helvetica Chimica Acta. 77: 334-350. DOI: 10.1002/Hlca.19940770133 |
0.409 |
|
| 1994 |
Muddasani PR, Bozó E, Bernet B, Vasella A. Glycosylidene Carbenes. Part 14. Glycosidation of partially protected galactopyranose-, glucopyranose-, and mannopyranose-derived vicinal diols Helvetica Chimica Acta. 77: 257-290. DOI: 10.1002/Hlca.19940770128 |
0.384 |
|
| 1993 |
Ermert P, Vasella A, Weber M, Rupitz K, Withers SG. Configurationally selective transition state analogue inhibitors of glycosidases. A study with nojiritetrazoles, a new class of glycosidase inhibitors Carbohydrate Research. 250: 113-128. DOI: 10.1016/0008-6215(93)84160-8 |
0.359 |
|
| 1993 |
Braun H, Felber H, Kresze G, Schmidtchen FP, Prewo R, Vasella A. Diastereoselektive Diels-Alder-Reaktionen mit α-Chlornitrososacchariden Liebigs Annalen Der Chemie. 1993: 261-268. DOI: 10.1002/Jlac.199319930146 |
0.364 |
|
| 1993 |
Vasella A, Witzig C, Waldraff C, Uhlmann P, Briner K, Bernet B, Panza L, Husi R. Glycosylidene Carbenes. Part 13. Synthesis and thermolysis of representative 1-azi-glycoses Helvetica Chimica Acta. 76: 2847-2875. DOI: 10.1002/Hlca.19930760811 |
0.409 |
|
| 1993 |
Ermert P, Vasella A. A New Approach to 5-Thiosugars: 5-Thio-D-Gluconhydroximo-1,5-lactone, Synthesis and Evaluation as ?-Glucosidase Inhibitor Helvetica Chimica Acta. 76: 2687-2699. DOI: 10.1002/Hlca.19930760724 |
0.466 |
|
| 1993 |
Hoos R, Naughton AB, Thiel W, Vasella A, Weber W, Rupitz K, Withers SG. D-Gluconhydroximo-1,5-lactam and RelatedN-Arylcarbamates Theoretical Calculations, Structure, Synthesis, and Inhibitory Effect on ?-Glucosidases Helvetica Chimica Acta. 76: 2666-2686. DOI: 10.1002/Hlca.19930760723 |
0.353 |
|
| 1993 |
Hoos R, Naughton AB, Vasella A. A Convenient Procedure for he Synthesis o 2,3,4,6-Tetra-O-benzyl-D-gluconolactam and D-Nojirilactam Helvetica Chimica Acta. 76: 1802-1807. DOI: 10.1002/Hlca.19930760435 |
0.396 |
|
| 1993 |
Vasella A, Dhar P, Witzig C. Glycosylidene Carbenes Part 12. A new synthesis and some reactions of spirooxiranes Helvetica Chimica Acta. 76: 1767-1778. DOI: 10.1002/Hlca.19930760433 |
0.445 |
|
| 1993 |
Czollner L, Baudin G, Bernet B, Vasella A. Synthese eines 1,2-trans-konfigurierten, äquatorialen Glycosyl-phosphonat-Analogen vonD-myo-Inositol-1,4,5-trisphosphat Helvetica Chimica Acta. 76: 1013-1025. DOI: 10.1002/Hlca.19930760224 |
0.435 |
|
| 1993 |
Hürzeler M, Bernet B, Vasella A. Glyconothio-O-lactones. Part I. Preparation and reactions with nucleophiles Helvetica Chimica Acta. 76: 995-1012. DOI: 10.1002/Hlca.19930760223 |
0.392 |
|
| 1993 |
Li C, Vasella A. A New Synthesis of Benzylidene Acetals Helvetica Chimica Acta. 76: 211-221. DOI: 10.1002/Hlca.19930760115 |
0.365 |
|
| 1993 |
Li C, Vasella A. Intramolecular Addition of Nucleophilic Carbenes to Acceptor-Substituted Alkenyl Groups: Synthesis and transformation of homobenzofurans and synthesis of a homoindole Helvetica Chimica Acta. 76: 197-210. DOI: 10.1002/Hlca.19930760114 |
0.392 |
|
| 1993 |
?opusi?ski A, Bernet B, Linden A, Vasella A. Synthesis of Glycosylphosphine Oxides and Related Compounds Helvetica Chimica Acta. 76: 94-112. DOI: 10.1002/Hlca.19930760104 |
0.364 |
|
| 1992 |
Maloisel J, Vasella A, Trost BM, Van Vranken DL. Synthesis of Allosamidin Helvetica Chimica Acta. 75: 1515-1526. DOI: 10.1039/C39910001099 |
0.412 |
|
| 1992 |
Li C, Bernet B, Vasella A, Broger EA, Meili A. Synthesis and evaluation in asymmetric hydrogenation of carbohydrate-derived 1,3-bisphosphines Carbohydrate Research. 216: 149-169. DOI: 10.1016/0008-6215(92)84158-O |
0.37 |
|
| 1992 |
Bozó E, Vasella A. Glycosylidene Carbenes. Part 10. Regioselective Glycosidation of 4,6-O-Benzylidene-D-altropyranosides Helvetica Chimica Acta. 75: 2613-2633. DOI: 10.1002/Hlca.19920750816 |
0.406 |
|
| 1992 |
Uhlmann P, Vasella A. Glycosylidene Carbenes. Part 9. Regioselective glycosidation of diols and triols: Intra- and intermolecular hydrogen bonds Helvetica Chimica Acta. 75: 1979-1994. DOI: 10.1002/Hlca.19920750623 |
0.358 |
|
| 1992 |
Linden A, Vasella A, Witzig C. Glycosylidene Carbenes. Part 8. Crystal Structure of a Cyclic, N‐Acetylallosamine‐Derived Alkoxy‐alkyl‐diazirine Helvetica Chimica Acta. 75: 1572-1577. DOI: 10.1002/Hlca.19920750511 |
0.328 |
|
| 1992 |
Takahashi Y, Vasella A. Glycosylidene Carbenes. Part 7. Neighbouring‐group participation by the 2‐benzyloxy group in the glycosidation of strongly acidic hydroxy compounds Helvetica Chimica Acta. 75: 1563-1571. DOI: 10.1002/Hlca.19920750510 |
0.35 |
|
| 1992 |
Maloisel J, Vasella A. Synthesis ofN-Acetylallosamine-Derived Disaccharides Helvetica Chimica Acta. 75: 1491-1514. DOI: 10.1002/Hlca.19920750505 |
0.439 |
|
| 1992 |
Briner K, Vasella A. Glycosylidene Carbenes. Part 6. Synthesis of alkyl and fluoroalkyl glycosides Helvetica Chimica Acta. 75: 621-637. DOI: 10.1002/Hlca.19920750218 |
0.39 |
|
| 1992 |
Wolk DR, Vasella A, Schweikart F, Peter MG. Synthesis and Enzyme-Inhibition Studies of Phenylsemicarbazones derived from D-glucono-1,5-lactone and 2-acetamido-2-deoxy-D-glucono-1,5-lactone Helvetica Chimica Acta. 75: 323-334. DOI: 10.1002/Hlca.19920750129 |
0.387 |
|
| 1992 |
Vasella A, Uhlmann P, Waldraff CAA, Diederich F, Thilgen C. Fullerene Sugars: Preparation of Enantiomerically Pure, Spiro-LinkedC-Glycosides of C60 Angewandte Chemie International Edition in English. 31: 1388-1390. DOI: 10.1002/Anie.199213881 |
0.342 |
|
| 1991 |
Horsch M, Hoesch L, Vasella A, Rast DM. N-acetylglucosaminono-1,5-lactone oxime and the corresponding (phenylcarbamoyl)oxime. Novel and potent inhibitors of beta-N-acetylglucosaminidase. European Journal of Biochemistry / Febs. 197: 815-8. PMID 2029909 DOI: 10.1111/J.1432-1033.1991.Tb15976.X |
0.317 |
|
| 1991 |
Papageorgiou AC, Oikonomakos NG, Leonidas DD, Bernet B, Beer D, Vasella A. The binding of D-gluconohydroximo-1,5-lactone to glycogen phosphorylase. Kinetic, ultracentrifugation and crystallographic studies. Biochemical Journal. 274: 329-338. PMID 1900987 DOI: 10.1042/Bj2740329 |
0.335 |
|
| 1991 |
Vasella A, Witzig C, Chiara J, Martin-Lomas M. Convenient Synthesis of 2-Azido-2-deoxy-aldoses by Diazo Transfer Helvetica Chimica Acta. 74: 2073-2077. DOI: 10.1002/Hlca.19910740842 |
0.389 |
|
| 1991 |
Ermert P, Vasella A. Synthesis of a Glucose-Derived Tetrazole as a New ?-Glucosidase Inhibitor. A New Synthesis of 1-Deoxynojirimycin Helvetica Chimica Acta. 74: 2043-2053. DOI: 10.1002/Hlca.19910740839 |
0.385 |
|
| 1991 |
Fritschi S, Vasella A. Synthesis of N,N‐Disubstituted Lactone Hydrazones via (Sulfonylimino)‐ethers Helvetica Chimica Acta. 74: 2024-2034. DOI: 10.1002/Hlca.19910740837 |
0.391 |
|
| 1991 |
Mahmood K, Vasella A, Bernet B. Deoxy-nitrosugars. 17th communication. Synthesis of ketose-derived nucleosides from 1-deoxy-1-nitroribose Helvetica Chimica Acta. 74: 1555-1584. DOI: 10.1002/Hlca.19910740719 |
0.319 |
|
| 1991 |
Wallimann K, Vasella A. C-Glykoside derN-Acetylneuraminsäure. Synthese und Untersuchung ihrer Wirkung auf dieVibrio choleraeSialidase Helvetica Chimica Acta. 74: 1520-1532. DOI: 10.1002/Hlca.19910740716 |
0.403 |
|
| 1991 |
Vasella A, Witzig C, Husi R. Glycosylidene Carbenes. Part 4. Synthesis of Spirocyclopropanes from Acetamidoglycosylidene-Derived Diazirines Helvetica Chimica Acta. 74: 1362-1372. DOI: 10.1002/Hlca.19910740625 |
0.427 |
|
| 1991 |
Vasella A, Waldraff CAA. Glycosylidene Carbenes. Part 3. Synthesis of Spirocyclopropanes Helvetica Chimica Acta. 74: 585-593. DOI: 10.1002/Hlca.19910740316 |
0.451 |
|
| 1991 |
Vasella A, Wyler R. Synthesis of a Phosphonic Acid Analogue ofN-Acetyl-2,3-didehydro-2-deoxyneuraminic Acid, an Inhibitor ofVibrio cholerae Sialidase Helvetica Chimica Acta. 74: 451-463. DOI: 10.1002/Hlca.19910740223 |
0.422 |
|
| 1991 |
Glänzer BI, Györgydeák Z, Bernet B, Vasella A. Analogues of Sialic Acids as Potential Sialidase Inhibitors. Synthesis of C6and C7Analogues ofN-Acetyl-6-amino-2,6-dideoxyneuraminic Acid Helvetica Chimica Acta. 74: 343-369. DOI: 10.1002/Hlca.19910740214 |
0.385 |
|
| 1991 |
Vasella A, Baudin G, Panza L. Synthesis of glycosyl phosphonates and related compounds Heteroatom Chemistry. 2: 151-161. DOI: 10.1002/Hc.520020117 |
0.438 |
|
| 1990 |
Huber R, Vasella A. The kinetic anomeric effect. Additions of nucleophiles and of dipolarophiles to N-glycosylnitrones and to N-pseudoglycosylnitrones Tetrahedron. 46: 33-58. DOI: 10.1016/S0040-4020(01)97582-9 |
0.35 |
|
| 1990 |
Brade W, Vasella A. Synthese von Pyrano[3,2-b][1]benzopyranen aus 1-Nitroglycalen Helvetica Chimica Acta. 73: 1923-1930. DOI: 10.1002/Hlca.19900730715 |
0.4 |
|
| 1990 |
Beer D, Maloisel J, Rast DM, Vasella A. Synthesis of 2-Acetamido-2-deoxy-D-gluconhydroximolactone- and Chitobionhydroximolactone-DerivedN-Phenylcarbamates, Potential Inhibitors of ?-N-Acetylglucosaminidase Helvetica Chimica Acta. 73: 1918-1922. DOI: 10.1002/Hlca.19900730714 |
0.415 |
|
| 1990 |
Briner K, Vasella A. Glycosylidene Carbenes. Part 2. Synthesis ofO-Aryl Glycosides Helvetica Chimica Acta. 73: 1764-1778. DOI: 10.1002/Hlca.19900730621 |
0.379 |
|
| 1990 |
Vasella A, Wyler R. Synthesis of the 6-C-Methyl and 6-C-(Hydroxymethyl) Analogues ofN-Acetylneuraminic Acid and ofN-Acetyl-2,3-didehydro-2-deoxyneuraminic Acid Helvetica Chimica Acta. 73: 1742-1763. DOI: 10.1002/Hlca.19900730620 |
0.355 |
|
| 1990 |
Wallimann K, Vasella A. Phosphonic-Acid Analogues of the N-Acetyl-2-deoxyneiiraniinic Acids: Synthesis and Inhibition ofVibrio cholerae Sialidase Helvetica Chimica Acta. 73: 1359-1372. DOI: 10.1002/Hlca.19900730523 |
0.422 |
|
| 1990 |
Czollner L, Kuszmann J, Vasella A. Synthesis of Pyrrolidine Analogues ofN-Acetylneuraminic Acid as Potential Sialidase Inhibitors Helvetica Chimica Acta. 73: 1338-1358. DOI: 10.1002/Hlca.19900730522 |
0.432 |
|
| 1990 |
Huber R, Molleyres L, Vasella A. Synthesis of Potential Glucosidase-Inhibitors:D-Xylopyranoside-5-spiro-l?-cyclopropanes Helvetica Chimica Acta. 73: 1329-1337. DOI: 10.1002/Hlca.19900730521 |
0.407 |
|
| 1990 |
Bernet B, Murty ARCB, Vasella A. Analogues of Sialic Acids as Potential Sialidase Inhibitors Synthesis of 2-C-Hydroxymethyl Derivatives ofN-Acetyl-6-amino-2,6-dideoxy-neuraminic Acid Helvetica Chimica Acta. 73: 940-958. DOI: 10.1002/Hlca.19900730422 |
0.408 |
|
| 1989 |
Brade W, Vasella A. Synthesis of Naphtho[2,3-b]pyrandiones: (?)-Cryptosporin Helvetica Chimica Acta. 72: 1649-1657. DOI: 10.1002/Hlca.19890720802 |
0.378 |
|
| 1989 |
Briner K, Vasella A. Glycosylidene Carbenes a new approach to glycoside synthesis. Part 1. Preparation of glycosylidene-derived diaziridines and diazirines Helvetica Chimica Acta. 72: 1371-1382. DOI: 10.1002/Hlca.19890720626 |
0.481 |
|
| 1988 |
Dessinges A, Vasella A. Synthesis of a non-isosteric, isopolar monophosphonate analogue of β-d-fructose 2,6-bisphosphate Carbohydrate Research. 174: 47-59. DOI: 10.1016/0008-6215(88)85080-8 |
0.403 |
|
| 1988 |
Baudin G, Glänzer BI, Swaminathan KS, Vasella A. A Synthesis of 1D- and 1L-myo-Inositol 1,3,4,5,-Tetraphosphate Helvetica Chimica Acta. 71: 1367-1378. DOI: 10.1002/Hlca.19880710548 |
0.303 |
|
| 1988 |
Csuk R, Hugener M, Vasella A. A new synthesis ofN-acetylneuraminic acid Helvetica Chimica Acta. 71: 609-618. DOI: 10.1002/Hlca.19880710314 |
0.42 |
|
| 1988 |
Baumberger F, Vasella A, Schauer R. Synthesis of New Sialidase Inhibitors, 6-Amino-6-Deoxysialic Acids Helvetica Chimica Acta. 71: 429-445. DOI: 10.1002/Hlca.19880710216 |
0.437 |
|
| 1987 |
Julina R, Müller I, Vasella A, Wyler R. A synthesis of N-acetylneuraminic acid and [6-2H]-N-acetylneuraminic acid from N-acetyl-D-glucosamine. Carbohydrate Research. 164: 415-32. PMID 3621240 DOI: 10.1016/0008-6215(87)80145-3 |
0.423 |
|
| 1987 |
Clinch K, Vasella A, Schauer R. Synthesis of (2R,4S,5S)-5-acetamido-4-hydroxy-pipecolinic acid as a potential inhibitor of sialidases Tetrahedron Letters. 28: 6425-6428. DOI: 10.1016/S0040-4039(00)96878-3 |
0.338 |
|
| 1987 |
Schauer R, Stoll S, Zbiral E, Schreiner E, Brandstetter HH, Vasella A, Baumberger F. Interaction of N-acetyl-4-, 7-, 8- or 9-deoxyneuraminic acids and N-acetyl-4-, 7- or 8-mono-epi- and-7,8-di-epineuraminic acids with N-acetylneuraminate lyase Glycoconjugate Journal. 4: 361-369. DOI: 10.1007/Bf01048369 |
0.323 |
|
| 1987 |
Huber R, Vasella A. Nucleophilic additions toN-glycosylnitrones part IV Asymmetric synthesis ofN-hydroxy-?-aminophosphonic and ?-aminophosphonic acids Helvetica Chimica Acta. 70: 1461-1476. DOI: 10.1002/Hlca.19870700603 |
0.331 |
|
| 1987 |
Briner K, Vasella A. Glycosylphosphonates of 2-Amino-2-deoxy-aldoses. Synthesis of a Phosphonate Analogue of Lipid X Helvetica Chimica Acta. 70: 1341-1356. DOI: 10.1002/Hlca.19870700516 |
0.445 |
|
| 1986 |
Baumberger F, Vasella A, Schauer R. 4-Methylumbelliferyl 5-Acetamido-3,4,5-trideoxy-?-D-manno-2-nonulopyranosidonic Acid: Synthesis and Resistance to Bacterial Sialidases Helvetica Chimica Acta. 69: 1927-1935. DOI: 10.1002/Hlca.19860690820 |
0.42 |
|
| 1986 |
Baumberger F, Vasella A. Deoxy-nitrosugars. 16th Communication. Synthesis ofN-acetyl-4-deoxyneuraminic acid Helvetica Chimica Acta. 69: 1535-1541. DOI: 10.1002/Hlca.19860690702 |
0.43 |
|
| 1986 |
Baumberger F, Vasella A. Deoxy-nitrosugars 15th communication Synthesis ofN-acetylneuraminic acid andN-acetyl-4-epineuraminic Acid Helvetica Chimica Acta. 69: 1205-1215. DOI: 10.1002/Hlca.19860690528 |
0.452 |
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| 1986 |
Baumberger F, Beer D, Christen M, Prewo R, Vasella A. Desoxy-nitrozucker 14. Mitteilung 1-C-Nitroglycale. Herstellung und Umsetzung mit einigen Stickstoff-Nucleophilen Helvetica Chimica Acta. 69: 1191-1204. DOI: 10.1002/Hlca.19860690527 |
0.409 |
|
| 1986 |
Beer D, Bieri JH, Macher I, Prewo R, Vasella A. Desoxy-nitrozucker. 13. Mitteilung. Herstellung ungeschützter und partiell geschützter 1-Desoxy-1-nitro-D-aldosen sowie Röntgenstrukturanalysen einiger ihrer Vertreter Helvetica Chimica Acta. 69: 1172-1190. DOI: 10.1002/Hlca.19860690526 |
0.407 |
|
| 1986 |
Meuwly R, Vasella A. Deoxy-nitrosugars 12th communication Synthesis of isosteric mono-phosphonate analogues of ?-and ?-D-fructose 2,6-bisphosphate Helvetica Chimica Acta. 69: 751-760. DOI: 10.1002/Hlca.19860690402 |
0.45 |
|
| 1986 |
Julina R, Herzig T, Bernet B, Vasella A. Enantioselective Synthesis ofD-erythro-Sphingosine and of Ceramide Helvetica Chimica Acta. 69: 368-373. DOI: 10.1002/Hlca.19860690216 |
0.394 |
|
| 1986 |
BAUMBERGER F, BEER D, CHRISTEN M, PREWO R, VASELLA A. ChemInform Abstract: Deoxynitro Sugars. Part 14. 1-C-Nitroglycals. Preparation and Reaction with Some Nitrogen Nucleophiles. Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198646326 |
0.344 |
|
| 1986 |
BEER D, BIERI JH, MACHER I, PREWO R, VASELLA A. ChemInform Abstract: Deoxynitro Sugars. Part 13. Preparation of Unprotected and Partially Protected 1-Deoxy-1-nitro-D-aldoses and Some Representative X-Ray Structure Analyses. Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198646325 |
0.315 |
|
| 1986 |
MEUWLY R, VASELLA A. ChemInform Abstract: Deoxy-Nitrosugars. Part 12. Synthesis of Isosteric Mono-Phosphonate Analogues of β- and α-D-Fructose 2,6-Bisphosphate, Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198639330 |
0.394 |
|
| 1986 |
HUBER R, KNIERZINGER A, KRAWCZYK E, OBRECHT JP, VASELLA A. ChemInform Abstract: Kinetic Anomeric Effect in Asymmetric Synthesis: A New Approach to Aminophosphonic Acids Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198634377 |
0.351 |
|
| 1986 |
Julina R, Herzig T, Bernet B, Vasella A. Enantioselective Synthesis of D‐erythro‐Sphingosine and of Ceramide. Cheminform. 17. DOI: 10.1002/Chin.198624333 |
0.407 |
|
| 1986 |
Meuwly R, Vasella A. Synthesis of 1,2-cis-Configurated Glycosylphosphonates Helvetica Chimica Acta. 69: 25-34. DOI: 10.1002/Chin.198618352 |
0.312 |
|
| 1985 |
Julina R, Vasella A. Deoxy-nitrosugars. 10th Communication. Synthesis of Isosteric Phosphonate Analogues of Ulose-1-Phosphates Helvetica Chimica Acta. 68: 819-830. DOI: 10.1002/Hlca.19850680402 |
0.395 |
|
| 1985 |
Bernet B, Krawczyk E, Vasella A. Diastereoselectivity in the Reaction ofN-Glycosyl-nitrones: 1,3-Dipolar Cycloaddition and Addition of Phosphite Anion Helvetica Chimica Acta. 68: 2299-2311. DOI: 10.1002/Chin.198611349 |
0.314 |
|
| 1985 |
Beer D, Vasella A. Aldonhydroximo-lactones. Preparation and Determination of Configuration Helvetica Chimica Acta. 68: 2254-2274. DOI: 10.1002/Chin.198611348 |
0.339 |
|
| 1985 |
Huber R, Knierzinger A, Obrecht J, Vasella A. Nucleophilic Additions toN-Glycosylnitrones. Asymmetric Synthesis of ?-Aminophosphonic Acids Helvetica Chimica Acta. 68: 1730-1747. DOI: 10.1002/Chin.198551236 |
0.387 |
|
| 1985 |
Mirza S, Molleyres L, Vasella A. Synthesis of a Glyoxalase I Inhibitor fromStreptomyces griseosporeus NIIDAet OGASAWARA Helvetica Chimica Acta. 68: 988-996. DOI: 10.1002/Chin.198539361 |
0.363 |
|
| 1984 |
Knierzinger A, Vasella A. Synthesis of 6-epithienamycin Journal of the Chemical Society, Chemical Communications. 9-11. DOI: 10.1039/C39840000009 |
0.397 |
|
| 1984 |
Felber H, Kresze G, Braun H, Vasella A. Asymmetric diels - alder reacrions with α-chloronitroso compounds- II. The use of a carbohydrate derived α-chloro-α-nitroso ether Tetrahedron Letters. 25: 5381-5382. DOI: 10.1016/S0040-4039(01)91289-4 |
0.347 |
|
| 1984 |
Mirza S, Vasella A. Deoxy-nitrosugars, 7th communication Synthesis of methyl shikimate and of diethyl phosphashikimate from D-ribose Helvetica Chimica Acta. 67: 1562-1567. DOI: 10.1002/Hlca.19840670621 |
0.411 |
|
| 1984 |
Bernet B, Vasella A. Fragmentation of 6-Deoxy-6-halo-hexono-1,5-ortholactones: A Concerted, Nonstereospecific Process Helvetica Chimica Acta. 67: 1328-1347. DOI: 10.1002/Hlca.19840670519 |
0.385 |
|
| 1984 |
Meuwly R, Vasella A. Deoxy-nitrosugars 8th communication Convenient preparation of 1-C-nitroglycosyl chlorides. Halonitro ethers from hydroxy oximes Helvetica Chimica Acta. 67: 1568-1571. DOI: 10.1002/Chin.198452348 |
0.303 |
|
| 1984 |
Knierzinger A, Vasella A. Synthesis Of 6-Epithienamycin Cheminform. 15. DOI: 10.1002/Chin.198419343 |
0.397 |
|
| 1984 |
VASELLA A, VOEFFRAY R, PLESS J, HUGUENIN R. ChemInform Abstract: SYNTHESIS OF D- AND L-5-OXAPROLINE AND A NEW CAPTOPRIL ANALOG Chemischer Informationsdienst. 15. DOI: 10.1002/Chin.198401200 |
0.359 |
|
| 1983 |
Bernet B, Vasella A. Enantioselective synthesis of D-erythro-sphingosine Tetrahedron Letters. 24: 5491-5494. DOI: 10.1016/S0040-4039(00)94120-0 |
0.421 |
|
| 1983 |
Baumberger F, Vasella A. Deoxy-nitrosugars. 6th communication. Stereoelectronic control in the reductive denitration of tertiary nitro ethers. A synthesis of ?C-glycosides? Helvetica Chimica Acta. 66: 2210-2222. DOI: 10.1002/Hlca.19830660733 |
0.452 |
|
| 1983 |
Vasella A, Voeffray R, Pless J, Huguenin R. Synthesis ofD- andL-5-Oxaproline and of a New Captopril Analogue Helvetica Chimica Acta. 66: 1241-1252. DOI: 10.1002/Hlca.19830660424 |
0.437 |
|
| 1983 |
Aebischer B, Vasella A. Deoxy-nitrosugars. 4th communication. Convenient synthesis of 1-deoxy-1-nitroaldoses Helvetica Chimica Acta. 66: 789-794. DOI: 10.1002/Hlca.19830660310 |
0.372 |
|
| 1983 |
AEBISCHER B, BIERI JH, PREWO R, VASELLA A. ChemInform Abstract: DEOXYNITROSUGARS. PART 3. SYNTHESIS OF KETOSES BY CHAIN ELONGATION OF 1-DEOXY-1-NITROALDOSES. NUCLEOPHILIC ADDITIONS AND SOLVOLYSIS OF NITRO ETHERS Chemischer Informationsdienst. 14. DOI: 10.1002/Chin.198313341 |
0.403 |
|
| 1982 |
Aebischer B, Bieri JH, Prewo R, Vasella A. Desoxy-nitrozucker. 3. Mitteilung. Synthese von Ketosen durch Kettenverlängerung von 1-Desoxy-1-nitro-aldosen. Nucleophile Additionen und Solvolyse von Nitroaethern Helvetica Chimica Acta. 65: 2251-2272. DOI: 10.1002/Hlca.19820650730 |
0.439 |
|
| 1982 |
Vasella A, Voeffray R. Totalsynthese von Nojirimycin Helvetica Chimica Acta. 65: 1134-1144. DOI: 10.1002/Hlca.19820650403 |
0.397 |
|
| 1982 |
Aebischer B, Vasella A, Weber H. Desoxy-nitrozucker. 2. Mitteilung Herstellung geschützter 1-Desoxy-1-nitroaldosen Helvetica Chimica Acta. 65: 621-634. DOI: 10.1002/Hlca.19820650302 |
0.37 |
|
| 1982 |
Beer D, Meuwly R, Vasella A. L-Erythruronic Acid Derivatives as Building Blocks for Nucleoside Analogs. Synthesis of 4?-C-Aryl-D-ribonucleosides Helvetica Chimica Acta. 65: 2570-2582. DOI: 10.1002/Chin.198315350 |
0.415 |
|
| 1982 |
AEBISCHER B, VASELLA A, WEBER HP. ChemInform Abstract: DEOXYNITROSUGARS. PART 2. SYNTHESIS OF PROTECTED 1-DEOXY-1-NITROALDOSES Chemischer Informationsdienst. 13. DOI: 10.1002/Chin.198236312 |
0.408 |
|
| 1981 |
Vasella A, Voeffray R. Asymmetric synthesis of a new proline analogue Journal of the Chemical Society, Chemical Communications. 97-98. DOI: 10.1039/C39810000097 |
0.425 |
|
| 1979 |
Bernet B, Vasella A. Carbocyclen aus Monosacchariden. III. Zur Diastereoselektivität der Bildung von Cyclopentanderivaten. Umsetzungen in der Galactosereihe Helvetica Chimica Acta. 62: 2411-2431. DOI: 10.1002/Hlca.19790620737 |
0.405 |
|
| 1979 |
Bernet B, Vasella A. Carbocyclische Verbindungen aus Monosacchariden. I. Umsetzungen in der glucosereihe Helvetica Chimica Acta. 62: 1990-2016. DOI: 10.1002/Hlca.19790620629 |
0.382 |
|
| 1979 |
Steinlin H, Camarda L, Vasella A. Über die Herstellung des Methyl-α-D-fructopyranosides und die Struktur der dabei gebildeten Orthoester† Helvetica Chimica Acta. 62: 378-390. DOI: 10.1002/Hlca.19790620204 |
0.388 |
|
| 1979 |
STEINLIN H, CAMARDA L, VASELLA A. ChemInform Abstract: PREPARATION OF METHYL α-D-FRUCTOPYRANOSIDES AND THE STRUCTURE OF THE ORTHOESTER BY-PRODUCTS Chemischer Informationsdienst. 10. DOI: 10.1002/Chin.197922307 |
0.361 |
|
| 1977 |
Vasella A. Stereoselektivität und Reaktivität bei der 1,3‐dipolaren Cycloaddition chiraler N‐(Alkoxyalkyl)nitrone Helvetica Chimica Acta. 60: 1273-1295. DOI: 10.1002/Hlca.19770600417 |
0.399 |
|
| 1977 |
Vasella A. Synthese und Umwandlungen von Isoxazolidin-Nucleosiden Helvetica Chimica Acta. 60: 426-446. DOI: 10.1002/Hlca.19770600214 |
0.404 |
|
| 1971 |
Spichtig AM, Vasella A. [Synthesis of alpha-methylsordarose]. Helvetica Chimica Acta. 54: 1191-1194. PMID 5095218 DOI: 10.1002/Hlca.19710540428 |
0.378 |
|
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