| Year |
Citation |
Score |
| 2021 |
Bahuguna A, Rawat S, Rawat DS. QcrB in Mycobacterium tuberculosis: The new drug target of antitubercular agents. Medicinal Research Reviews. PMID 33400275 DOI: 10.1002/med.21779 |
1 |
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| 2020 |
Bahuguna A, Bharatam PV, Rawat DS. 3D QSAR studies on amphiphilic indoles for antimycobacterial activity. Journal of Biochemical and Molecular Toxicology. e22675. PMID 33347664 DOI: 10.1002/jbt.22675 |
1 |
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| 2020 |
Gagandeep, Kumar P, Kandi SK, Mukhopadhyay K, Rawat DS. Synthesis of novel monocarbonyl curcuminoids, evaluation of their efficacy against MRSA, including ex vivo infection model and their mechanistic studies. European Journal of Medicinal Chemistry. 195: 112276. PMID 32279050 DOI: 10.1016/j.ejmech.2020.112276 |
1 |
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| 2019 |
Arora G, Gagandeep, Behura A, Gosain TP, Shaliwal RP, Kidwai S, Singh P, Kandi SK, Dhiman R, Rawat DS, Singh R. NSC 18725, a Pyrazole Derivative Inhibits Growth of Intracellular by Induction of Autophagy. Frontiers in Microbiology. 10: 3051. PMID 32063889 DOI: 10.3389/fmicb.2019.03051 |
1 |
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| 2019 |
Bahuguna A, Rawat DS. An overview of new antitubercular drugs, drug candidates, and their targets. Medicinal Research Reviews. PMID 31254295 DOI: 10.1002/med.21602 |
1 |
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| 2019 |
Tripathi M, Taylor D, Khan SI, Tekwani BL, Ponnan P, Das US, Velpandian T, Rawat DS. Hybridization of Fluoro-amodiaquine (FAQ) with Pyrimidines: Synthesis and Antimalarial Efficacy of FAQ-Pyrimidines. Acs Medicinal Chemistry Letters. 10: 714-719. PMID 31097988 DOI: 10.1021/acsmedchemlett.8b00496 |
1 |
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| 2018 |
Maurya SS, Bahuguna A, Khan SI, Kumar D, Kholiya R, Rawat DS. N-Substituted aminoquinoline-pyrimidine hybrids: Synthesis, in vitro antimalarial activity evaluation and docking studies. European Journal of Medicinal Chemistry. 162: 277-289. PMID 30448417 DOI: 10.1016/j.ejmech.2018.11.021 |
1 |
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| 2018 |
Negi B, Poonan P, Ansari MF, Kumar D, Aggarwal S, Singh R, Azam A, Rawat DS. Synthesis, antiamoebic activity and docking studies of metronidazole-triazole-styryl hybrids. European Journal of Medicinal Chemistry. 150: 633-641. PMID 29558734 DOI: 10.1016/j.ejmech.2018.03.033 |
1 |
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| 2017 |
Rawat DS, Ponnan P. Editorial: Peptide Science at the Chemistry and Biology Interface. Current Protein & Peptide Science. 18: 884. PMID 28758599 DOI: 10.2174/138920371809170706181108 |
1 |
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| 2017 |
Joshi R, Rohil V, Arora S, Manral S, Kumar A, Goel S, Priya N, Singh P, Ponnan P, Chatterji S, Dwarakanath BS, Saluja D, Rawat DS, Prasad AK, Saso L, et al. Corrigendum to The Competence of 7,8-Diacetoxy-4-Methylcoumarin and Other Polyphenolic Acetates in Mitigating the Oxidative Stress and their Role in Angiogenesis. Current Topics in Medicinal Chemistry. 17: 1115. PMID 28406076 DOI: 10.2174/156802661709170213214101 |
1 |
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| 2017 |
Reddy PL, Tripathi M, Arundhathi R, Rawat DS. Chemoselective Hydrazine-mediated Transfer Hydrogenation of Nitroarenes by Co3 O4 Nanoparticles Immobilized on an Al/Si-mixed Oxide Support. Chemistry, An Asian Journal. PMID 28328163 DOI: 10.1002/asia.201700025 |
1 |
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| 2017 |
Kholiya R, Khan SI, Bahuguna A, Tripathi M, Rawat DS. N-Piperonyl substitution on aminoquinoline-pyrimidine hybrids: Effect on the antiplasmodial potency. European Journal of Medicinal Chemistry. 131: 126-140. PMID 28315598 DOI: 10.1016/j.ejmech.2017.03.007 |
1 |
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| 2017 |
Maurya SS, Khan SI, Bahuguna A, Kumar D, Rawat DS. Synthesis, antimalarial activity, heme binding and docking studies of N-substituted 4-aminoquinoline-pyrimidine molecular hybrids. European Journal of Medicinal Chemistry. 129: 175-185. PMID 28222317 DOI: 10.1016/j.ejmech.2017.02.024 |
1 |
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| 2016 |
Reddy PL, Khan SI, Ponnan P, Tripathi M, Rawat DS. Design, synthesis and evaluation of 4-aminoquinoline-purine hybrids as potential antiplasmodial agents. European Journal of Medicinal Chemistry. 126: 675-686. PMID 27936446 DOI: 10.1016/j.ejmech.2016.11.057 |
1 |
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| 2016 |
Negi B, Kumar D, Rawat DS. Marine Peptides As Anticancer Agents: A Remedy To Mankind By Nature. Current Protein & Peptide Science. PMID 27455970 |
1 |
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| 2016 |
Negi B, Kumar D, Kumbukgolla W, Jayaweera S, Ponnan P, Singh R, Agarwal S, Rawat DS. Anti-methicillin resistant Staphylococcus aureus activity, synergism with oxacillin and molecular docking studies of metronidazole-triazole hybrids. European Journal of Medicinal Chemistry. 115: 426-437. PMID 27046397 DOI: 10.1016/j.ejmech.2016.03.041 |
1 |
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| 2016 |
Anthwal A, Singh K, Rawat MS, Tyagi AK, Haque A, Ali I, Rawat DS. Synthesis of 4-piperidone Based Curcuminoids with Anti-inflammatory and Anti-Proliferation Potential in Human Cancer Cell Lines. Anti-Cancer Agents in Medicinal Chemistry. 16: 841-51. PMID 26567619 |
1 |
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| 2015 |
Kumar D, Negi B, Rawat DS. The anti-tuberculosis agents under development and the challenges ahead. Future Medicinal Chemistry. PMID 26505682 DOI: 10.4155/fmc.15.128 |
1 |
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| 2015 |
Joshi R, Arora S, Kumar A, Manral S, Rohil V, Goel S, Priya N, Singh P, Ponnan P, Chatterji S, Dwarakanath BS, Saluja D, Rawat DS, Prasad AK, Saso L, et al. The Competence of 7,8-Diacetoxy-4-Methylcoumarin and Other Polyphenolic Acetates in Mitigating the Oxidative Stress and their Role in Angiogenesis. Current Topics in Medicinal Chemistry. 15: 179-86. PMID 25547104 |
1 |
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| 2015 |
Kumar D, Khan SI, Tekwani BL, Ponnan P, Rawat DS. 4-Aminoquinoline-pyrimidine hybrids: synthesis, antimalarial activity, heme binding and docking studies. European Journal of Medicinal Chemistry. 89: 490-502. PMID 25462261 DOI: 10.1016/j.ejmech.2014.10.061 |
1 |
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| 2015 |
Joshi S, Dewangan RP, Yar MS, Rawat DS, Pasha S. N-terminal aromatic tag induced self assembly of tryptophan-arginine rich ultra short sequences and their potent antibacterial activity Rsc Advances. 5: 68610-68620. DOI: 10.1039/c5ra12095k |
1 |
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| 2015 |
Kandi SK, Manohar S, Vélez Gerena CE, Zayas B, Malhotra SV, Rawat DS. C5-curcuminoid-4-aminoquinoline based molecular hybrids: Design, synthesis and mechanistic investigation of anticancer activity New Journal of Chemistry. 39: 224-234. DOI: 10.1039/c4nj00936c |
1 |
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| 2015 |
Kumar D, Khare G, Beena, Kidwai S, Tyagi AK, Singh R, Rawat DS. Novel isoniazid-amidoether derivatives: Synthesis, characterization and antimycobacterial activity evaluation Medchemcomm. 6: 131-137. DOI: 10.1039/c4md00288a |
1 |
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| 2014 |
Joshi R, Arora S, Kumar A, Manral S, Rohil V, Goel S, Priya N, Singh P, Ponnan P, Chatterji S, Dwarakanath BS, Saluja D, Rawat DS, Prasad AK, Saso L, et al. The Competence Of 7,8-Diacetoxy-4-Methylcoumarinand Other Polyphenolic Acetates In Mitigating The Oxidative Stress And Their Role In Angiogenesis. Current Topics in Medicinal Chemistry. PMID 25496273 |
1 |
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| 2014 |
Anthwal A, Thakur BK, Rawat MS, Rawat DS, Tyagi AK, Aggarwal BB. Synthesis, characterization and in vitro anticancer activity of C-5 curcumin analogues with potential to inhibit TNF-α-induced NF-κB activation. Biomed Research International. 2014: 524161. PMID 25157362 DOI: 10.1155/2014/524161 |
1 |
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| 2014 |
Negi B, Raj KK, Siddiqui SM, Ramachandran D, Azam A, Rawat DS. In vitro antiamoebic activity evaluation and docking studies of metronidazole-triazole hybrids. Chemmedchem. 9: 2439-44. PMID 25146853 DOI: 10.1002/cmdc.201402240 |
1 |
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| 2014 |
Manohar S, Tripathi M, Rawat DS. 4-aminoquinoline based molecular hybrids as antimalarials: an overview. Current Topics in Medicinal Chemistry. 14: 1706-33. PMID 25116580 |
1 |
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| 2014 |
Kumar D, Beena, Khare G, Kidwai S, Tyagi AK, Singh R, Rawat DS. Synthesis of novel 1,2,3-triazole derivatives of isoniazid and their in vitro and in vivo antimycobacterial activity evaluation. European Journal of Medicinal Chemistry. 81: 301-13. PMID 24852277 DOI: 10.1016/j.ejmech.2014.05.005 |
1 |
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| 2014 |
Anthwal A, Rajesh UC, Rawat MS, Kushwaha B, Maikhuri JP, Sharma VL, Gupta G, Rawat DS. Novel metronidazole-chalcone conjugates with potential to counter drug resistance in Trichomonas vaginalis. European Journal of Medicinal Chemistry. 79: 89-94. PMID 24727243 DOI: 10.1016/j.ejmech.2014.03.076 |
1 |
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| 2014 |
Kumar D, Khan SI, Tekwani BL, Ponnan P, Rawat DS. Synthesis, antimalarial activity, heme binding and docking studies of 4-aminoquinoline-pyrimidine based molecular hybrids Rsc Advances. 4: 63655-63669. DOI: 10.1039/c4ra09768h |
1 |
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| 2014 |
Manohar S, Pepe A, Vélez Gerena CE, Zayas B, Malhotra SV, Rawat DS. Anticancer activity of 4-aminoquinoline-triazine based molecular hybrids Rsc Advances. 4: 7062-7067. DOI: 10.1039/c3ra45333b |
1 |
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| 2014 |
Thakur A, Manohar S, Vélez Gerena CE, Zayas B, Kumar V, Malhotra SV, Rawat DS. Novel 3,5-bis(arylidiene)-4-piperidone based monocarbonyl analogs of curcumin: Anticancer activity evaluation and mode of action study Medchemcomm. 5: 576-586. DOI: 10.1039/c3md00399j |
1 |
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| 2013 |
Rawat DS, Singh R. Plant derived secondary metabolites as anti-cancer agents. Anti-Cancer Agents in Medicinal Chemistry. 13: 1551. PMID 24341389 DOI: 10.2174/187152061310131206154445 |
1 |
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| 2013 |
Joshi R, Kumar A, Manral S, Sinha R, Arora S, Sharma A, Goel S, Kalra N, Chatterji S, Dwarakanath BS, Rawat DS, Depass AL, Rohil V, Saluja D, Parmar VS, et al. Calreticulin transacetylase mediated upregulation of thioredoxin by 7,8-diacetoxy-4-methylcoumarin enhances the antioxidant potential and the expression of vascular endothelial growth factor in peripheral blood mononuclear cells. Chemico-Biological Interactions. 206: 327-36. PMID 24103856 DOI: 10.1016/j.cbi.2013.09.017 |
1 |
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| 2013 |
Rawat DS, Singh R. Plant-Derived Secondary Metabolites as Anticancer Agents. Anti-Cancer Agents in Medicinal Chemistry. PMID 23438829 |
1 |
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| 2013 |
Kumar D, Raj KK, Bailey M, Alling T, Parish T, Rawat DS. Antimycobacterial activity evaluation, time-kill kinetic and 3D-QSAR study of C-(3-aminomethyl-cyclohexyl)-methylamine derivatives. Bioorganic & Medicinal Chemistry Letters. 23: 1365-9. PMID 23357633 DOI: 10.1016/j.bmcl.2012.12.083 |
1 |
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| 2013 |
Manohar S, Khan SI, Rawat DS. 4-aminoquinoline-triazine-based hybrids with improved in vitro antimalarial activity against CQ-sensitive and CQ-resistant strains of Plasmodium falciparum. Chemical Biology & Drug Design. 81: 625-30. PMID 23331618 DOI: 10.1111/cbdd.12108 |
1 |
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| 2013 |
Beena, Kumar D, Rawat DS. Synthesis and antioxidant activity of thymol and carvacrol based Schiff bases. Bioorganic & Medicinal Chemistry Letters. 23: 641-5. PMID 23273412 DOI: 10.1016/j.bmcl.2012.12.001 |
1 |
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| 2013 |
Manohar S, Khan SI, Kandi SK, Raj K, Sun G, Yang X, Calderon Molina AD, Ni N, Wang B, Rawat DS. Synthesis, antimalarial activity and cytotoxic potential of new monocarbonyl analogues of curcumin. Bioorganic & Medicinal Chemistry Letters. 23: 112-6. PMID 23218718 DOI: 10.1016/j.bmcl.2012.11.004 |
1 |
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| 2013 |
Beena, Rawat DS. Antituberculosis drug research: a critical overview. Medicinal Research Reviews. 33: 693-764. PMID 22622957 DOI: 10.1002/med.21262 |
1 |
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| 2013 |
Rajesh UC, Manohar S, Rawat DS. Hydromagnesite as an efficient recyclable heterogeneous solid base catalyst for the synthesis of flavanones, flavonols and 1,4-dihydropyridines in water Advanced Synthesis and Catalysis. 355: 3170-3178. DOI: 10.1002/adsc.201300555 |
1 |
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| 2012 |
Manohar S, Rajesh UC, Khan SI, Tekwani BL, Rawat DS. Novel 4-aminoquinoline-pyrimidine based hybrids with improved in vitro and in vivo antimalarial activity. Acs Medicinal Chemistry Letters. 3: 555-9. PMID 24900509 DOI: 10.1021/ml3000808 |
1 |
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| 2012 |
Joshi S, Dewangan RP, Yadav S, Rawat DS, Pasha S. Synthesis, antibacterial activity and mode of action of novel linoleic acid-dipeptide-spermidine conjugates. Organic & Biomolecular Chemistry. 10: 8326-35. PMID 22986997 DOI: 10.1039/c2ob26393a |
1 |
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| 2012 |
Beena, Joshi S, Kumar N, Kidwai S, Singh R, Rawat DS. Synthesis and antitubercular activity evaluation of novel unsymmetrical cyclohexane-1,2-diamine derivatives. Archiv Der Pharmazie. 345: 896-901. PMID 22945019 DOI: 10.1002/ardp.201200219 |
1 |
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| 2012 |
Joshi S, Bisht GS, Rawat DS, Maiti S, Pasha S. Comparative mode of action of novel hybrid peptide CS-1a and its rearranged amphipathic analogue CS-2a. The Febs Journal. 279: 3776-90. PMID 22883393 DOI: 10.1111/j.1742-4658.2012.08738.x |
1 |
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| 2012 |
Kumar N, Singh R, Rawat DS. Tetraoxanes: synthetic and medicinal chemistry perspective. Medicinal Research Reviews. 32: 581-610. PMID 22675731 |
1 |
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| 2012 |
Joshi MC, Rawat DS. Recent developments in enediyne chemistry. Chemistry & Biodiversity. 9: 459-98. PMID 22422520 DOI: 10.1002/cbdv.201100047 |
1 |
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| 2011 |
Sharma M, Joshi MC, Kumar V, Malhotra SV, Rawat DS. Synthesis and anticancer activity of 13-membered cyclic enediynes. Archiv Der Pharmazie. 344: 564-71. PMID 21887797 DOI: 10.1002/ardp.201000309 |
1 |
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| 2011 |
Kumar N, Sharma M, Rawat DS. Medicinal chemistry perspectives of trioxanes and tetraoxanes. Current Medicinal Chemistry. 18: 3889-928. PMID 21824099 DOI: 10.2174/092986711803414340 |
1 |
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| 2011 |
Kumar N, Khan SI, Atheaya H, Mamgain R, Rawat DS. Synthesis and in vitro antimalarial activity of tetraoxane-amine/amide conjugates. European Journal of Medicinal Chemistry. 46: 2816-27. PMID 21530018 DOI: 10.1016/j.ejmech.2011.04.002 |
1 |
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| 2011 |
Manohar S, Khan SI, Rawat DS. Synthesis of 4-aminoquinoline-1,2,3-triazole and 4-aminoquinoline-1,2,3-triazole-1,3,5-triazine hybrids as potential antimalarial agents. Chemical Biology & Drug Design. 78: 124-36. PMID 21457474 DOI: 10.1111/j.1747-0285.2011.01115.x |
1 |
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| 2011 |
Sharma M, Joshi P, Kumar N, Joshi S, Rohilla RK, Roy N, Rawat DS. Synthesis, antimicrobial activity and structure-activity relationship study of N,N-dibenzyl-cyclohexane-1,2-diamine derivatives. European Journal of Medicinal Chemistry. 46: 480-7. PMID 21163555 DOI: 10.1016/j.ejmech.2010.11.027 |
1 |
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| 2010 |
Kumar N, Singh R, Rawat DS. Tetraoxanes: synthetic and medicinal chemistry perspective. Medicinal Research Reviews. PMID 21064188 DOI: 10.1002/med.20223 |
1 |
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| 2010 |
Joshi S, Bisht GS, Rawat DS, Kumar A, Kumar R, Maiti S, Pasha S. Interaction studies of novel cell selective antimicrobial peptides with model membranes and E. coli ATCC 11775. Biochimica Et Biophysica Acta. 1798: 1864-75. PMID 20599694 DOI: 10.1016/j.bbamem.2010.06.016 |
1 |
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| 2010 |
Kumar D, Joshi S, Rohilla RK, Roy N, Rawat DS. Synthesis and antibacterial activity of benzyl-[3-(benzylamino-methyl)-cyclohexylmethyl]-amine derivatives. Bioorganic & Medicinal Chemistry Letters. 20: 893-5. PMID 20047831 DOI: 10.1016/j.bmcl.2009.12.074 |
1 |
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| 2010 |
Manohar S, Khan SI, Rawat DS. Synthesis, antimalarial activity and cytotoxicity of 4-aminoquinoline-triazine conjugates. Bioorganic & Medicinal Chemistry Letters. 20: 322-5. PMID 19910192 DOI: 10.1016/j.bmcl.2009.10.106 |
1 |
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| 2009 |
Aggarwal N, Kumar R, Dureja P, Rawat DS. Schiff bases as potential fungicides and nitrification inhibitors. Journal of Agricultural and Food Chemistry. 57: 8520-5. PMID 19702271 DOI: 10.1021/jf902035w |
1 |
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| 2009 |
Kumar N, Khan SI, Beena, Rajalakshmi G, Kumaradhas P, Rawat DS. Synthesis, antimalarial activity and cytotoxicity of substituted 3,6-diphenyl-[1,2,4,5]tetraoxanes. Bioorganic & Medicinal Chemistry. 17: 5632-8. PMID 19574054 DOI: 10.1016/j.bmc.2009.06.020 |
1 |
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| 2009 |
Kumar N, Khan SI, Sharma M, Atheaya H, Rawat DS. Iodine-catalyzed one-pot synthesis and antimalarial activity evaluation of symmetrically and asymmetrically substituted 3,6-diphenyl[1,2,4,5]tetraoxanes. Bioorganic & Medicinal Chemistry Letters. 19: 1675-7. PMID 19231182 DOI: 10.1016/j.bmcl.2009.01.103 |
1 |
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| 2009 |
Beena, Kumar N, Rohilla RK, Roy N, Rawat DS. Synthesis and antibacterial activity evaluation of metronidazole-triazole conjugates. Bioorganic & Medicinal Chemistry Letters. 19: 1396-8. PMID 19195884 DOI: 10.1016/j.bmcl.2009.01.037 |
1 |
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| 2008 |
Singh R, Sharma M, Joshi P, Rawat DS. Clinical status of anti-cancer agents derived from marine sources. Anti-Cancer Agents in Medicinal Chemistry. 8: 603-17. PMID 18690825 |
1 |
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| 2008 |
Atheaya H, Khan SI, Mamgain R, Rawat DS. Synthesis, thermal stability, antimalarial activity of symmetrically and asymmetrically substituted tetraoxanes. Bioorganic & Medicinal Chemistry Letters. 18: 1446-9. PMID 18248990 DOI: 10.1016/j.bmcl.2007.12.069 |
1 |
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| 2008 |
Rawat DS, Krzysiak AJ, Gibbs RA. Synthesis and biochemical evaluation of 3,7-disubstituted farnesyl diphosphate analogues. The Journal of Organic Chemistry. 73: 1881-7. PMID 18225915 DOI: 10.1021/jo701725b |
1 |
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| 2007 |
Bisht GS, Rawat DS, Kumar A, Kumar R, Pasha S. Antimicrobial activity of rationally designed amino terminal modified peptides. Bioorganic & Medicinal Chemistry Letters. 17: 4343-6. PMID 17553680 DOI: 10.1016/j.bmcl.2007.05.015 |
1 |
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| 2007 |
Krzysiak AJ, Rawat DS, Scott SA, Pais JE, Handley M, Harrison ML, Fierke CA, Gibbs RA. Combinatorial modulation of protein prenylation. Acs Chemical Biology. 2: 385-9. PMID 17530735 DOI: 10.1021/cb700062b |
1 |
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| 2007 |
Joshi MC, Bisht GS, Rawat DS. Syntheses and antibacterial activity of phendioxy substituted cyclic enediynes. Bioorganic & Medicinal Chemistry Letters. 17: 3226-30. PMID 17433674 DOI: 10.1016/j.bmcl.2007.03.007 |
1 |
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| 2006 |
Singh R, Sharma R, Tewari N, Rawat DS. Nitrilase and its application as a 'green' catalyst. Chemistry & Biodiversity. 3: 1279-87. PMID 17193242 DOI: 10.1002/cbdv.200690131 |
1 |
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| 2006 |
Rawat DS, Joshi MC, Joshi P, Atheaya H. Marine peptides and related compounds in clinical trial. Anti-Cancer Agents in Medicinal Chemistry. 6: 33-40. PMID 16475925 |
1 |
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| 2004 |
McFarland MJ, Porter AC, Rakhshan FR, Rawat DS, Gibbs RA, Barker EL. A role for caveolae/lipid rafts in the uptake and recycling of the endogenous cannabinoid anandamide. The Journal of Biological Chemistry. 279: 41991-7. PMID 15292270 DOI: 10.1074/jbc.M407250200 |
1 |
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| 2003 |
Benites PJ, Holmberg RC, Rawat DS, Kraft BJ, Klein LJ, Peters DG, Thorp HH, Zaleski JM. Metal-ligand charge-transfer-promoted photoelectronic Bergman cyclization of copper metalloenediynes: photochemical DNA cleavage via C-4' H-atom abstraction. Journal of the American Chemical Society. 125: 6434-46. PMID 12785783 DOI: 10.1021/ja020939f |
1 |
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| 2002 |
Rawat DS, Gibbs RA. Synthesis of 7-substituted farnesyl diphosphate analogues. Organic Letters. 4: 3027-30. PMID 12201708 DOI: 10.1021/ol026176i |
1 |
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