Diwan S Rawat, PhD - Publications

Affiliations: 
1994-1997 Chemistry University of Delhi 

71 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 Bahuguna A, Rawat S, Rawat DS. QcrB in Mycobacterium tuberculosis: The new drug target of antitubercular agents. Medicinal Research Reviews. PMID 33400275 DOI: 10.1002/med.21779  1
2020 Bahuguna A, Bharatam PV, Rawat DS. 3D QSAR studies on amphiphilic indoles for antimycobacterial activity. Journal of Biochemical and Molecular Toxicology. e22675. PMID 33347664 DOI: 10.1002/jbt.22675  1
2020 Gagandeep, Kumar P, Kandi SK, Mukhopadhyay K, Rawat DS. Synthesis of novel monocarbonyl curcuminoids, evaluation of their efficacy against MRSA, including ex vivo infection model and their mechanistic studies. European Journal of Medicinal Chemistry. 195: 112276. PMID 32279050 DOI: 10.1016/j.ejmech.2020.112276  1
2019 Arora G, Gagandeep, Behura A, Gosain TP, Shaliwal RP, Kidwai S, Singh P, Kandi SK, Dhiman R, Rawat DS, Singh R. NSC 18725, a Pyrazole Derivative Inhibits Growth of Intracellular by Induction of Autophagy. Frontiers in Microbiology. 10: 3051. PMID 32063889 DOI: 10.3389/fmicb.2019.03051  1
2019 Bahuguna A, Rawat DS. An overview of new antitubercular drugs, drug candidates, and their targets. Medicinal Research Reviews. PMID 31254295 DOI: 10.1002/med.21602  1
2019 Tripathi M, Taylor D, Khan SI, Tekwani BL, Ponnan P, Das US, Velpandian T, Rawat DS. Hybridization of Fluoro-amodiaquine (FAQ) with Pyrimidines: Synthesis and Antimalarial Efficacy of FAQ-Pyrimidines. Acs Medicinal Chemistry Letters. 10: 714-719. PMID 31097988 DOI: 10.1021/acsmedchemlett.8b00496  1
2018 Maurya SS, Bahuguna A, Khan SI, Kumar D, Kholiya R, Rawat DS. N-Substituted aminoquinoline-pyrimidine hybrids: Synthesis, in vitro antimalarial activity evaluation and docking studies. European Journal of Medicinal Chemistry. 162: 277-289. PMID 30448417 DOI: 10.1016/j.ejmech.2018.11.021  1
2018 Negi B, Poonan P, Ansari MF, Kumar D, Aggarwal S, Singh R, Azam A, Rawat DS. Synthesis, antiamoebic activity and docking studies of metronidazole-triazole-styryl hybrids. European Journal of Medicinal Chemistry. 150: 633-641. PMID 29558734 DOI: 10.1016/j.ejmech.2018.03.033  1
2017 Rawat DS, Ponnan P. Editorial: Peptide Science at the Chemistry and Biology Interface. Current Protein & Peptide Science. 18: 884. PMID 28758599 DOI: 10.2174/138920371809170706181108  1
2017 Joshi R, Rohil V, Arora S, Manral S, Kumar A, Goel S, Priya N, Singh P, Ponnan P, Chatterji S, Dwarakanath BS, Saluja D, Rawat DS, Prasad AK, Saso L, et al. Corrigendum to The Competence of 7,8-Diacetoxy-4-Methylcoumarin and Other Polyphenolic Acetates in Mitigating the Oxidative Stress and their Role in Angiogenesis. Current Topics in Medicinal Chemistry. 17: 1115. PMID 28406076 DOI: 10.2174/156802661709170213214101  1
2017 Reddy PL, Tripathi M, Arundhathi R, Rawat DS. Chemoselective Hydrazine-mediated Transfer Hydrogenation of Nitroarenes by Co3 O4 Nanoparticles Immobilized on an Al/Si-mixed Oxide Support. Chemistry, An Asian Journal. PMID 28328163 DOI: 10.1002/asia.201700025  1
2017 Kholiya R, Khan SI, Bahuguna A, Tripathi M, Rawat DS. N-Piperonyl substitution on aminoquinoline-pyrimidine hybrids: Effect on the antiplasmodial potency. European Journal of Medicinal Chemistry. 131: 126-140. PMID 28315598 DOI: 10.1016/j.ejmech.2017.03.007  1
2017 Maurya SS, Khan SI, Bahuguna A, Kumar D, Rawat DS. Synthesis, antimalarial activity, heme binding and docking studies of N-substituted 4-aminoquinoline-pyrimidine molecular hybrids. European Journal of Medicinal Chemistry. 129: 175-185. PMID 28222317 DOI: 10.1016/j.ejmech.2017.02.024  1
2016 Reddy PL, Khan SI, Ponnan P, Tripathi M, Rawat DS. Design, synthesis and evaluation of 4-aminoquinoline-purine hybrids as potential antiplasmodial agents. European Journal of Medicinal Chemistry. 126: 675-686. PMID 27936446 DOI: 10.1016/j.ejmech.2016.11.057  1
2016 Negi B, Kumar D, Rawat DS. Marine Peptides As Anticancer Agents: A Remedy To Mankind By Nature. Current Protein & Peptide Science. PMID 27455970  1
2016 Negi B, Kumar D, Kumbukgolla W, Jayaweera S, Ponnan P, Singh R, Agarwal S, Rawat DS. Anti-methicillin resistant Staphylococcus aureus activity, synergism with oxacillin and molecular docking studies of metronidazole-triazole hybrids. European Journal of Medicinal Chemistry. 115: 426-437. PMID 27046397 DOI: 10.1016/j.ejmech.2016.03.041  1
2016 Anthwal A, Singh K, Rawat MS, Tyagi AK, Haque A, Ali I, Rawat DS. Synthesis of 4-piperidone Based Curcuminoids with Anti-inflammatory and Anti-Proliferation Potential in Human Cancer Cell Lines. Anti-Cancer Agents in Medicinal Chemistry. 16: 841-51. PMID 26567619  1
2015 Kumar D, Negi B, Rawat DS. The anti-tuberculosis agents under development and the challenges ahead. Future Medicinal Chemistry. PMID 26505682 DOI: 10.4155/fmc.15.128  1
2015 Joshi R, Arora S, Kumar A, Manral S, Rohil V, Goel S, Priya N, Singh P, Ponnan P, Chatterji S, Dwarakanath BS, Saluja D, Rawat DS, Prasad AK, Saso L, et al. The Competence of 7,8-Diacetoxy-4-Methylcoumarin and Other Polyphenolic Acetates in Mitigating the Oxidative Stress and their Role in Angiogenesis. Current Topics in Medicinal Chemistry. 15: 179-86. PMID 25547104  1
2015 Kumar D, Khan SI, Tekwani BL, Ponnan P, Rawat DS. 4-Aminoquinoline-pyrimidine hybrids: synthesis, antimalarial activity, heme binding and docking studies. European Journal of Medicinal Chemistry. 89: 490-502. PMID 25462261 DOI: 10.1016/j.ejmech.2014.10.061  1
2015 Joshi S, Dewangan RP, Yar MS, Rawat DS, Pasha S. N-terminal aromatic tag induced self assembly of tryptophan-arginine rich ultra short sequences and their potent antibacterial activity Rsc Advances. 5: 68610-68620. DOI: 10.1039/c5ra12095k  1
2015 Kandi SK, Manohar S, Vélez Gerena CE, Zayas B, Malhotra SV, Rawat DS. C5-curcuminoid-4-aminoquinoline based molecular hybrids: Design, synthesis and mechanistic investigation of anticancer activity New Journal of Chemistry. 39: 224-234. DOI: 10.1039/c4nj00936c  1
2015 Kumar D, Khare G, Beena, Kidwai S, Tyagi AK, Singh R, Rawat DS. Novel isoniazid-amidoether derivatives: Synthesis, characterization and antimycobacterial activity evaluation Medchemcomm. 6: 131-137. DOI: 10.1039/c4md00288a  1
2014 Joshi R, Arora S, Kumar A, Manral S, Rohil V, Goel S, Priya N, Singh P, Ponnan P, Chatterji S, Dwarakanath BS, Saluja D, Rawat DS, Prasad AK, Saso L, et al. The Competence Of 7,8-Diacetoxy-4-Methylcoumarinand Other Polyphenolic Acetates In Mitigating The Oxidative Stress And Their Role In Angiogenesis. Current Topics in Medicinal Chemistry. PMID 25496273  1
2014 Anthwal A, Thakur BK, Rawat MS, Rawat DS, Tyagi AK, Aggarwal BB. Synthesis, characterization and in vitro anticancer activity of C-5 curcumin analogues with potential to inhibit TNF-α-induced NF-κB activation. Biomed Research International. 2014: 524161. PMID 25157362 DOI: 10.1155/2014/524161  1
2014 Negi B, Raj KK, Siddiqui SM, Ramachandran D, Azam A, Rawat DS. In vitro antiamoebic activity evaluation and docking studies of metronidazole-triazole hybrids. Chemmedchem. 9: 2439-44. PMID 25146853 DOI: 10.1002/cmdc.201402240  1
2014 Manohar S, Tripathi M, Rawat DS. 4-aminoquinoline based molecular hybrids as antimalarials: an overview. Current Topics in Medicinal Chemistry. 14: 1706-33. PMID 25116580  1
2014 Kumar D, Beena, Khare G, Kidwai S, Tyagi AK, Singh R, Rawat DS. Synthesis of novel 1,2,3-triazole derivatives of isoniazid and their in vitro and in vivo antimycobacterial activity evaluation. European Journal of Medicinal Chemistry. 81: 301-13. PMID 24852277 DOI: 10.1016/j.ejmech.2014.05.005  1
2014 Anthwal A, Rajesh UC, Rawat MS, Kushwaha B, Maikhuri JP, Sharma VL, Gupta G, Rawat DS. Novel metronidazole-chalcone conjugates with potential to counter drug resistance in Trichomonas vaginalis. European Journal of Medicinal Chemistry. 79: 89-94. PMID 24727243 DOI: 10.1016/j.ejmech.2014.03.076  1
2014 Kumar D, Khan SI, Tekwani BL, Ponnan P, Rawat DS. Synthesis, antimalarial activity, heme binding and docking studies of 4-aminoquinoline-pyrimidine based molecular hybrids Rsc Advances. 4: 63655-63669. DOI: 10.1039/c4ra09768h  1
2014 Manohar S, Pepe A, Vélez Gerena CE, Zayas B, Malhotra SV, Rawat DS. Anticancer activity of 4-aminoquinoline-triazine based molecular hybrids Rsc Advances. 4: 7062-7067. DOI: 10.1039/c3ra45333b  1
2014 Thakur A, Manohar S, Vélez Gerena CE, Zayas B, Kumar V, Malhotra SV, Rawat DS. Novel 3,5-bis(arylidiene)-4-piperidone based monocarbonyl analogs of curcumin: Anticancer activity evaluation and mode of action study Medchemcomm. 5: 576-586. DOI: 10.1039/c3md00399j  1
2013 Rawat DS, Singh R. Plant derived secondary metabolites as anti-cancer agents. Anti-Cancer Agents in Medicinal Chemistry. 13: 1551. PMID 24341389 DOI: 10.2174/187152061310131206154445  1
2013 Joshi R, Kumar A, Manral S, Sinha R, Arora S, Sharma A, Goel S, Kalra N, Chatterji S, Dwarakanath BS, Rawat DS, Depass AL, Rohil V, Saluja D, Parmar VS, et al. Calreticulin transacetylase mediated upregulation of thioredoxin by 7,8-diacetoxy-4-methylcoumarin enhances the antioxidant potential and the expression of vascular endothelial growth factor in peripheral blood mononuclear cells. Chemico-Biological Interactions. 206: 327-36. PMID 24103856 DOI: 10.1016/j.cbi.2013.09.017  1
2013 Rawat DS, Singh R. Plant-Derived Secondary Metabolites as Anticancer Agents. Anti-Cancer Agents in Medicinal Chemistry. PMID 23438829  1
2013 Kumar D, Raj KK, Bailey M, Alling T, Parish T, Rawat DS. Antimycobacterial activity evaluation, time-kill kinetic and 3D-QSAR study of C-(3-aminomethyl-cyclohexyl)-methylamine derivatives. Bioorganic & Medicinal Chemistry Letters. 23: 1365-9. PMID 23357633 DOI: 10.1016/j.bmcl.2012.12.083  1
2013 Manohar S, Khan SI, Rawat DS. 4-aminoquinoline-triazine-based hybrids with improved in vitro antimalarial activity against CQ-sensitive and CQ-resistant strains of Plasmodium falciparum. Chemical Biology & Drug Design. 81: 625-30. PMID 23331618 DOI: 10.1111/cbdd.12108  1
2013 Beena, Kumar D, Rawat DS. Synthesis and antioxidant activity of thymol and carvacrol based Schiff bases. Bioorganic & Medicinal Chemistry Letters. 23: 641-5. PMID 23273412 DOI: 10.1016/j.bmcl.2012.12.001  1
2013 Manohar S, Khan SI, Kandi SK, Raj K, Sun G, Yang X, Calderon Molina AD, Ni N, Wang B, Rawat DS. Synthesis, antimalarial activity and cytotoxic potential of new monocarbonyl analogues of curcumin. Bioorganic & Medicinal Chemistry Letters. 23: 112-6. PMID 23218718 DOI: 10.1016/j.bmcl.2012.11.004  1
2013 Beena, Rawat DS. Antituberculosis drug research: a critical overview. Medicinal Research Reviews. 33: 693-764. PMID 22622957 DOI: 10.1002/med.21262  1
2013 Rajesh UC, Manohar S, Rawat DS. Hydromagnesite as an efficient recyclable heterogeneous solid base catalyst for the synthesis of flavanones, flavonols and 1,4-dihydropyridines in water Advanced Synthesis and Catalysis. 355: 3170-3178. DOI: 10.1002/adsc.201300555  1
2012 Manohar S, Rajesh UC, Khan SI, Tekwani BL, Rawat DS. Novel 4-aminoquinoline-pyrimidine based hybrids with improved in vitro and in vivo antimalarial activity. Acs Medicinal Chemistry Letters. 3: 555-9. PMID 24900509 DOI: 10.1021/ml3000808  1
2012 Joshi S, Dewangan RP, Yadav S, Rawat DS, Pasha S. Synthesis, antibacterial activity and mode of action of novel linoleic acid-dipeptide-spermidine conjugates. Organic & Biomolecular Chemistry. 10: 8326-35. PMID 22986997 DOI: 10.1039/c2ob26393a  1
2012 Beena, Joshi S, Kumar N, Kidwai S, Singh R, Rawat DS. Synthesis and antitubercular activity evaluation of novel unsymmetrical cyclohexane-1,2-diamine derivatives. Archiv Der Pharmazie. 345: 896-901. PMID 22945019 DOI: 10.1002/ardp.201200219  1
2012 Joshi S, Bisht GS, Rawat DS, Maiti S, Pasha S. Comparative mode of action of novel hybrid peptide CS-1a and its rearranged amphipathic analogue CS-2a. The Febs Journal. 279: 3776-90. PMID 22883393 DOI: 10.1111/j.1742-4658.2012.08738.x  1
2012 Kumar N, Singh R, Rawat DS. Tetraoxanes: synthetic and medicinal chemistry perspective. Medicinal Research Reviews. 32: 581-610. PMID 22675731  1
2012 Joshi MC, Rawat DS. Recent developments in enediyne chemistry. Chemistry & Biodiversity. 9: 459-98. PMID 22422520 DOI: 10.1002/cbdv.201100047  1
2011 Sharma M, Joshi MC, Kumar V, Malhotra SV, Rawat DS. Synthesis and anticancer activity of 13-membered cyclic enediynes. Archiv Der Pharmazie. 344: 564-71. PMID 21887797 DOI: 10.1002/ardp.201000309  1
2011 Kumar N, Sharma M, Rawat DS. Medicinal chemistry perspectives of trioxanes and tetraoxanes. Current Medicinal Chemistry. 18: 3889-928. PMID 21824099 DOI: 10.2174/092986711803414340  1
2011 Kumar N, Khan SI, Atheaya H, Mamgain R, Rawat DS. Synthesis and in vitro antimalarial activity of tetraoxane-amine/amide conjugates. European Journal of Medicinal Chemistry. 46: 2816-27. PMID 21530018 DOI: 10.1016/j.ejmech.2011.04.002  1
2011 Manohar S, Khan SI, Rawat DS. Synthesis of 4-aminoquinoline-1,2,3-triazole and 4-aminoquinoline-1,2,3-triazole-1,3,5-triazine hybrids as potential antimalarial agents. Chemical Biology & Drug Design. 78: 124-36. PMID 21457474 DOI: 10.1111/j.1747-0285.2011.01115.x  1
2011 Sharma M, Joshi P, Kumar N, Joshi S, Rohilla RK, Roy N, Rawat DS. Synthesis, antimicrobial activity and structure-activity relationship study of N,N-dibenzyl-cyclohexane-1,2-diamine derivatives. European Journal of Medicinal Chemistry. 46: 480-7. PMID 21163555 DOI: 10.1016/j.ejmech.2010.11.027  1
2010 Kumar N, Singh R, Rawat DS. Tetraoxanes: synthetic and medicinal chemistry perspective. Medicinal Research Reviews. PMID 21064188 DOI: 10.1002/med.20223  1
2010 Joshi S, Bisht GS, Rawat DS, Kumar A, Kumar R, Maiti S, Pasha S. Interaction studies of novel cell selective antimicrobial peptides with model membranes and E. coli ATCC 11775. Biochimica Et Biophysica Acta. 1798: 1864-75. PMID 20599694 DOI: 10.1016/j.bbamem.2010.06.016  1
2010 Kumar D, Joshi S, Rohilla RK, Roy N, Rawat DS. Synthesis and antibacterial activity of benzyl-[3-(benzylamino-methyl)-cyclohexylmethyl]-amine derivatives. Bioorganic & Medicinal Chemistry Letters. 20: 893-5. PMID 20047831 DOI: 10.1016/j.bmcl.2009.12.074  1
2010 Manohar S, Khan SI, Rawat DS. Synthesis, antimalarial activity and cytotoxicity of 4-aminoquinoline-triazine conjugates. Bioorganic & Medicinal Chemistry Letters. 20: 322-5. PMID 19910192 DOI: 10.1016/j.bmcl.2009.10.106  1
2009 Aggarwal N, Kumar R, Dureja P, Rawat DS. Schiff bases as potential fungicides and nitrification inhibitors. Journal of Agricultural and Food Chemistry. 57: 8520-5. PMID 19702271 DOI: 10.1021/jf902035w  1
2009 Kumar N, Khan SI, Beena, Rajalakshmi G, Kumaradhas P, Rawat DS. Synthesis, antimalarial activity and cytotoxicity of substituted 3,6-diphenyl-[1,2,4,5]tetraoxanes. Bioorganic & Medicinal Chemistry. 17: 5632-8. PMID 19574054 DOI: 10.1016/j.bmc.2009.06.020  1
2009 Kumar N, Khan SI, Sharma M, Atheaya H, Rawat DS. Iodine-catalyzed one-pot synthesis and antimalarial activity evaluation of symmetrically and asymmetrically substituted 3,6-diphenyl[1,2,4,5]tetraoxanes. Bioorganic & Medicinal Chemistry Letters. 19: 1675-7. PMID 19231182 DOI: 10.1016/j.bmcl.2009.01.103  1
2009 Beena, Kumar N, Rohilla RK, Roy N, Rawat DS. Synthesis and antibacterial activity evaluation of metronidazole-triazole conjugates. Bioorganic & Medicinal Chemistry Letters. 19: 1396-8. PMID 19195884 DOI: 10.1016/j.bmcl.2009.01.037  1
2008 Singh R, Sharma M, Joshi P, Rawat DS. Clinical status of anti-cancer agents derived from marine sources. Anti-Cancer Agents in Medicinal Chemistry. 8: 603-17. PMID 18690825  1
2008 Atheaya H, Khan SI, Mamgain R, Rawat DS. Synthesis, thermal stability, antimalarial activity of symmetrically and asymmetrically substituted tetraoxanes. Bioorganic & Medicinal Chemistry Letters. 18: 1446-9. PMID 18248990 DOI: 10.1016/j.bmcl.2007.12.069  1
2008 Rawat DS, Krzysiak AJ, Gibbs RA. Synthesis and biochemical evaluation of 3,7-disubstituted farnesyl diphosphate analogues. The Journal of Organic Chemistry. 73: 1881-7. PMID 18225915 DOI: 10.1021/jo701725b  1
2007 Bisht GS, Rawat DS, Kumar A, Kumar R, Pasha S. Antimicrobial activity of rationally designed amino terminal modified peptides. Bioorganic & Medicinal Chemistry Letters. 17: 4343-6. PMID 17553680 DOI: 10.1016/j.bmcl.2007.05.015  1
2007 Krzysiak AJ, Rawat DS, Scott SA, Pais JE, Handley M, Harrison ML, Fierke CA, Gibbs RA. Combinatorial modulation of protein prenylation. Acs Chemical Biology. 2: 385-9. PMID 17530735 DOI: 10.1021/cb700062b  1
2007 Joshi MC, Bisht GS, Rawat DS. Syntheses and antibacterial activity of phendioxy substituted cyclic enediynes. Bioorganic & Medicinal Chemistry Letters. 17: 3226-30. PMID 17433674 DOI: 10.1016/j.bmcl.2007.03.007  1
2006 Singh R, Sharma R, Tewari N, Rawat DS. Nitrilase and its application as a 'green' catalyst. Chemistry & Biodiversity. 3: 1279-87. PMID 17193242 DOI: 10.1002/cbdv.200690131  1
2006 Rawat DS, Joshi MC, Joshi P, Atheaya H. Marine peptides and related compounds in clinical trial. Anti-Cancer Agents in Medicinal Chemistry. 6: 33-40. PMID 16475925  1
2004 McFarland MJ, Porter AC, Rakhshan FR, Rawat DS, Gibbs RA, Barker EL. A role for caveolae/lipid rafts in the uptake and recycling of the endogenous cannabinoid anandamide. The Journal of Biological Chemistry. 279: 41991-7. PMID 15292270 DOI: 10.1074/jbc.M407250200  1
2003 Benites PJ, Holmberg RC, Rawat DS, Kraft BJ, Klein LJ, Peters DG, Thorp HH, Zaleski JM. Metal-ligand charge-transfer-promoted photoelectronic Bergman cyclization of copper metalloenediynes: photochemical DNA cleavage via C-4' H-atom abstraction. Journal of the American Chemical Society. 125: 6434-46. PMID 12785783 DOI: 10.1021/ja020939f  1
2002 Rawat DS, Gibbs RA. Synthesis of 7-substituted farnesyl diphosphate analogues. Organic Letters. 4: 3027-30. PMID 12201708 DOI: 10.1021/ol026176i  1
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