Year |
Citation |
Score |
2023 |
Lazo JS, Isbell KN, Vasa SA, Llaneza DC, Rastelli EJ, Wipf P, Sharlow ER. Disruption of ovarian cancer STAT3 and p38 signaling with a small molecule inhibitor of PTP4A3 phosphatase. The Journal of Pharmacology and Experimental Therapeutics. PMID 36627205 DOI: 10.1124/jpet.122.001401 |
0.335 |
|
2021 |
Lazo JS, Sharlow ER, Cornelison R, Hart DJ, Llaneza DC, Mendelson AJ, Rastelli EJ, Tasker NR, Landen CN, Wipf P. Credentialing and Pharmacologically Targeting PTP4A3 Phosphatase as a Molecular Target for Ovarian Cancer. Biomolecules. 11. PMID 34209460 DOI: 10.3390/biom11070969 |
0.354 |
|
2021 |
Rastelli EJ, Sannino S, Hart DJ, Sharlow ER, Lazo JS, Brodsky JL, Wipf P. Synthesis and evaluation of bifunctional PTP4A3 phosphatase inhibitors activating the ER stress pathway. Bioorganic & Medicinal Chemistry Letters. 46: 128167. PMID 34089839 DOI: 10.1016/j.bmcl.2021.128167 |
0.36 |
|
2020 |
Czub MP, Boulton AM, Rastelli EJ, Tasker NR, Maskrey TS, Blanco IK, McQueeney KE, Bushweller JH, Minor W, Wipf P, Sharlow ER, Lazo JS. Structure of the complex of an iminopyridinedione PTP4A3 phosphatase inhibitor with human serum albumin. Molecular Pharmacology. PMID 32978326 DOI: 10.1124/molpharm.120.000131 |
0.336 |
|
2019 |
Coltart DM, Uddin N, Knight J, Rastelli E, Soubra-Ghaoui C, Albright T, Wu CH, Wu J. On the Mechanism of the Asymmetric Aldol Addition of Chiral N-Amino Cyclic Carbamate Hydrazones: Evidence of Non-Curtin-Hammett Behavior. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 31650641 DOI: 10.1002/Chem.201902388 |
0.67 |
|
2019 |
Lazo JS, Blanco IK, Tasker NR, Rastelli EJ, Burnett JC, Garrott SR, Hart DJ, McCloud RL, Hsu KL, Wipf P, Sharlow ER. Next-Generation Cell-active Inhibitors of the Undrugged Oncogenic PTP4A3 Phosphatase. The Journal of Pharmacology and Experimental Therapeutics. PMID 31601683 DOI: 10.1124/Jpet.119.262188 |
0.43 |
|
2019 |
Tasker NR, Rastelli EJ, Burnett JC, Sharlow ER, Lazo JS, Wipf P. Tapping the therapeutic potential of protein tyrosine phosphatase 4A with small molecule inhibitors. Bioorganic & Medicinal Chemistry Letters. PMID 31307888 DOI: 10.1016/J.Bmcl.2019.06.048 |
0.418 |
|
2019 |
Ferguson MW, Gerak CAN, Chow CCT, Rastelli EJ, Elmore KE, Stahl F, Hosseini-Farahabadi S, Baradaran-Heravi A, Coltart DM, Roberge M. The antimalarial drug mefloquine enhances TP53 premature termination codon readthrough by aminoglycoside G418. Plos One. 14: e0216423. PMID 31120902 DOI: 10.1371/Journal.Pone.0216423 |
0.58 |
|
2019 |
Tasker NR, Rastelli EJ, Blanco IK, Burnett JC, Sharlow ER, Lazo JS, Wipf P. In-flow photooxygenation of aminothienopyridinones generates iminopyridinedione PTP4A3 phosphatase inhibitors. Organic & Biomolecular Chemistry. PMID 30746541 DOI: 10.1039/C9Ob00025A |
0.438 |
|
2018 |
Rastelli EJ, Coltart, DM. Synthesis and biological activity of apratoxin derivatives Tetrahedron. 74: 2269-2290. DOI: 10.1016/J.Tet.2017.11.004 |
0.483 |
|
2018 |
Rastelli EJ, Bolinger AA, Coltart DM. Stereodivergent Synthesis of β,γ-Fused Bicyclic γ-Lactones via a Multicomponent Ring-Expansion Cascade Chem. 4: 2228-2238. DOI: 10.1016/J.Chempr.2018.08.007 |
0.656 |
|
2016 |
Rastelli EJ, Truong NT, Coltart DM. Asymmetric Induction in Hydroacylation by Cooperative Iminium Ion-Transition-Metal Catalysis. Organic Letters. PMID 27767317 DOI: 10.1021/Acs.Orglett.6B02825 |
0.617 |
|
2016 |
Rastelli EJ, Coltart DM. Asymmetric Synthesis of (+)-anti- and (-)-syn-Mefloquine Hydrochloride. The Journal of Organic Chemistry. PMID 27657347 DOI: 10.1021/Acs.Joc.6B01476 |
0.68 |
|
2015 |
Rastelli EJ, Coltart DM. A Concise and Highly Enantioselective Total Synthesis of (+)-anti- and (-)-syn-Mefloquine Hydrochloride: Definitive Absolute Stereochemical Assignment of the Mefloquines. Angewandte Chemie (International Ed. in English). PMID 26422780 DOI: 10.1002/Anie.201507304 |
0.687 |
|
2015 |
Tarsis EM, Rastelli EJ, Wengryniuk SE, Coltart DM. The apratoxin marine natural products: isolation, structure determination, and asymmetric total synthesis Tetrahedron. 71: 5029-5044. DOI: 10.1016/j.tet.2015.05.047 |
0.497 |
|
2015 |
Tarsis EM, Rastelli EJ, Wengryniuk SE, Coltart DM. The apratoxin marine natural products: Isolation, structure determination, and asymmetric total synthesis Tetrahedron. 71: 5029-5044. DOI: 10.1016/J.Tet.2015.05.047 |
0.515 |
|
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