Year |
Citation |
Score |
2017 |
Kandalkar SR, Ramaiah PA, Joshi M, Wavhal A, Waman Y, Raje AA, Tambe A, Ansari S, De S, Palle VP, Mookhtiar KA, Deshpande AM, Barawkar DA. Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2's-hydroxy-3's-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors. Bioorganic & Medicinal Chemistry. PMID 28951094 DOI: 10.1016/J.Bmc.2017.09.015 |
0.711 |
|
2017 |
Basu S, Barawkar DA, Ramdas V, Patel M, Waman Y, Panmand A, Kumar S, Thorat S, Naykodi M, Goswami A, Reddy BS, Prasad V, Chaturvedi S, Quraishi A, Menon S, et al. Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases. European Journal of Medicinal Chemistry. 134: 218-229. PMID 28415011 DOI: 10.1016/J.Ejmech.2017.04.014 |
0.352 |
|
2017 |
Koul S, Ramdas V, Barawkar DA, Waman YB, Prasad N, Madadi SK, Shejul YD, Bonagiri R, Basu S, Menon S, Reddy SB, Chaturvedi S, Chennamaneni SR, Bedse G, Thakare R, et al. Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation. Bioorganic & Medicinal Chemistry. PMID 28238512 DOI: 10.1016/J.Bmc.2017.02.029 |
0.336 |
|
2017 |
Basu S, Barawkar DA, Thorat S, Shejul YD, Patel M, Naykodi M, Jain V, Salve Y, Prasad V, Chaudhary S, Ghosh I, Bhat G, Quraishi A, Patil H, Ansari S, et al. Design, Synthesis of Novel, Potent, Selective, Orally Bio-available Adenosine A2A Receptor Antagonists and Their Biological Evaluation. Journal of Medicinal Chemistry. PMID 28055204 DOI: 10.1021/Acs.Jmedchem.6B01584 |
0.321 |
|
2016 |
Basu S, Barawkar DA, Ramdas V, Waman Y, Patel M, Panmand A, Kumar S, Thorat S, Bonagiri R, Jadhav D, Mukhopadhyay P, Prasad V, Reddy BS, Goswami A, Chaturvedi S, et al. A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives. European Journal of Medicinal Chemistry. PMID 27842891 DOI: 10.1016/J.Ejmech.2016.11.007 |
0.309 |
|
2014 |
Khose G, Shinde S, Panmand A, Kulkarni R, Munot Y, Bandyopadhyay A, Barawkar D, Patil SN. Synthesis of substituted esters of imidazoles, oxazoles, thiazoles, and diethyl pyrazine-2,5-dicarboxylate from a common acyclic precursor employing C-formylation strategy Tetrahedron Letters. 55: 2671-2674. DOI: 10.1016/J.Tetlet.2014.03.039 |
0.318 |
|
2013 |
Kandalkar SR, Kaduskar RD, Ramaiah PA, Barawkar DA, Bhuniya D, Deshpande AM. Highly efficient one-pot amination of carboxylate-substituted nitrogen-containing heteroaryl chlorides via Staudinger reaction Tetrahedron Letters. 54: 414-418. DOI: 10.1016/J.Tetlet.2012.11.027 |
0.709 |
|
2012 |
Barawkar DA, Bandyopadhyay A, Deshpande A, Koul S, Kandalkar S, Patil P, Khose G, Vyas S, Mone M, Bhosale S, Singh U, De S, Meru A, Gundu J, Chugh A, et al. Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain L-2-hydroxy acid oxidase. Bioorganic & Medicinal Chemistry Letters. 22: 4341-7. PMID 22658862 DOI: 10.1016/J.Bmcl.2012.05.020 |
0.723 |
|
2012 |
Basu S, Prasad UV, Barawkar DA, De S, Palle VP, Menon S, Patel M, Thorat S, Singh UP, Das Sarma K, Waman Y, Niranjan S, Pathade V, Gaur A, Reddy S, et al. Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors. Bioorganic & Medicinal Chemistry Letters. 22: 2843-9. PMID 22424978 DOI: 10.1016/J.Bmcl.2012.02.070 |
0.351 |
|
2011 |
Barawkar DA, Meru A, Bandyopadhyay A, Banerjee A, Deshpande AM, Athare C, Koduru C, Khose G, Gundu J, Mahajan K, Patil P, Kandalkar SR, Niranjan S, Bhosale S, De S, et al. Potent and Selective Inhibitors of Long Chain l-2-Hydroxy Acid Oxidase Reduced Blood Pressure in DOCA Salt-Treated Rats. Acs Medicinal Chemistry Letters. 2: 919-23. PMID 24900281 DOI: 10.1021/Ml2001938 |
0.715 |
|
2010 |
BARAWKAR DA, LINKLETTER B, BRUICE TC. ChemInform Abstract: Synthesis of Protected Guanidinium Linked Dinucleoside Incorporable into an Oligonucleotide Using Solid Phase DNA Methodology. Cheminform. 29: no-no. DOI: 10.1002/CHIN.199841236 |
0.458 |
|
2006 |
El Abdellaoui H, Varaprasad CVNS, Barawkar D, Chakravarty S, Maderna A, Tam R, Chen H, Allan M, Wu JZ, Appleby T, Yan S, Zhang W, Lang S, Yao N, Hamatake R, et al. Identification of isothiazole-4-carboxamidines derivatives as a novel class of allosteric MEK1 inhibitors Bioorganic and Medicinal Chemistry Letters. 16: 5561-5566. PMID 16934458 DOI: 10.1016/J.Bmcl.2006.08.048 |
0.306 |
|
2000 |
Barawkar DA, Kwok Y, Bruice TW, Bruice TC. Deoxynucleic guanidine/peptide nucleic acid chimeras: Synthesis, binding and invasion studies with DNA Journal of the American Chemical Society. 122: 5244-5250. DOI: 10.1021/Ja000022L |
0.573 |
|
1999 |
Jadhav VR, Barawkar DA, Ganesh KN. Polarity Sensing by Fluorescent Oligonucleotides: First Demonstration of Sequence-Dependent Microenvironmental Changes in the DNA Major Groove The Journal of Physical Chemistry B. 103: 7383-7385. DOI: 10.1021/Jp9914323 |
0.603 |
|
1999 |
Barawkar DA, Bruice TC. Deoxynucleic guanidines/PNA (DNG/PNA) chimeras: Oligonucleoside analogue containing cationic guanidinium and neutral amide linkages [2] Journal of the American Chemical Society. 121: 10418-10419. DOI: 10.1021/Ja9923540 |
0.493 |
|
1998 |
Barawkar DA, Linkletter B, Bruice TC. Synthesis of protected guanidinium linked dinucleoside incorporable into an oligonucleotide using solid phase DNA methodology. Bioorganic & Medicinal Chemistry Letters. 8: 1517-20. PMID 9873381 DOI: 10.1016/S0960-894X(98)00251-0 |
0.529 |
|
1998 |
Barawkar DA, Bruice TC. Synthesis, biophysical properties, and nuclease resistance properties of mixed backbone oligodeoxynucleotides containing cationic internucleoside guanidinium linkages: deoxynucleic guanidine/DNA chimeras. Proceedings of the National Academy of Sciences of the United States of America. 95: 11047-52. PMID 9736687 DOI: 10.1073/Pnas.95.19.11047 |
0.555 |
|
1998 |
Ganesh KN, Kumar V, Barawkar DA, Rajeev KG, Rana VS. Enhancing DNA triplex stability via nucleobase modification Pure and Applied Chemistry. 70: 289-292. DOI: 10.1351/Pac199870020289 |
0.737 |
|
1997 |
Ganesh KN, Rajeev KG, Pallan PS, Rana VS, Barawkar DA, Kumar VA. Modulation of DNA Triplex Stability Through Nucleobase Modifications Nucleosides and Nucleotides. 16: 1271-1278. DOI: 10.1080/07328319708006169 |
0.711 |
|
1997 |
Jadhav VR, Barawkar DA, Natu AA, Ganesh KN. 5-Amido-(carboxyfluorescein)-2′-dU-oligonucloetides: Novel Primers for Fluorescent Detection of PCR Amplified DNA Nucleosides and Nucleotides. 16: 107-114. DOI: 10.1080/07328319708002526 |
0.558 |
|
1996 |
Rana VS, Barawkar DA, Ganesh KN. Molecular Recognition of 5-Amino-dU in the Central Strand of a DNA Triplex: Formation of Triads AU(#):A in Parallel and GU(#):A in Antiparallel Motif(,). The Journal of Organic Chemistry. 61: 3578-3579. PMID 11667196 DOI: 10.1021/Jo9602074 |
0.747 |
|
1996 |
Barawkar DA, Rajeev KG, Kumar VA, Ganesh KN. Triplex formation at physiological pH by 5-Me-dC-N4-(spermine) [X] oligodeoxynucleotides: non protonation of N3 in X of X*G:C triad and effect of base mismatch/ionic strength on triplex stabilities. Nucleic Acids Research. 24: 1229-37. PMID 8614624 DOI: 10.1093/Nar/24.7.1229 |
0.704 |
|
1995 |
Barawkar DA, Ganesh KN. Fluorescent d(CGCGAATTCGCG): characterization of major groove polarity and study of minor groove interactions through a major groove semantophore conjugate. Nucleic Acids Research. 23: 159-64. PMID 7870581 DOI: 10.1093/Nar/23.1.159 |
0.589 |
|
1994 |
Barawkar DA, Ganesh KN. Exploring DNA minor groove interactions through a probe conjugate in major groove: fluorescence studies on netropsin complexation with dU-5-aminodansyl-DNA. Biochemical and Biophysical Research Communications. 203: 53-8. PMID 8074699 DOI: 10.1006/bbrc.1994.2147 |
0.516 |
|
1994 |
Barawkar DA, Kumar VA, Ganesh KN. Triplex formation at physiological pH by oligonucleotides incorporating 5-Me-dC-(N4-spermine). Biochemical and Biophysical Research Communications. 205: 1665-70. PMID 7811251 DOI: 10.1006/Bbrc.1994.2859 |
0.593 |
|
1994 |
Prakash T, Barawkar DA, Vaijayanti K, Ganesh K. Synthesis of site-specific oligonucleotide-polyamine conjugates Bioorganic & Medicinal Chemistry Letters. 4: 1733-1738. DOI: 10.1016/S0960-894X(00)80371-6 |
0.574 |
|
1993 |
Barawkar DA, Ganesh K. Solid phase synthesis of DNA containing 5-NH2-2′-deoxyuridine Bioorganic & Medicinal Chemistry Letters. 3: 347-352. DOI: 10.1016/S0960-894X(01)80908-2 |
0.591 |
|
Low-probability matches (unlikely to be authored by this person) |
2017 |
Basu S, Barawkar DA, Ramdas V, Naykodi M, Shejul YD, Patel M, Thorat S, Panmand A, Kashinath K, Bonagiri R, Prasad V, Bhat G, Quraishi A, Chaudhary S, Magdum A, et al. Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression. Acs Medicinal Chemistry Letters. 8: 835-840. PMID 28835798 DOI: 10.1021/Acsmedchemlett.7B00175 |
0.298 |
|
2003 |
Zhong W, An H, Barawkar D, Hong Z. Dinucleotide Analogues as Novel Inhibitors of RNA-Dependent RNA Polymerase of Hepatitis C Virus Antimicrobial Agents and Chemotherapy. 47: 2674-2681. PMID 12878540 DOI: 10.1128/Aac.47.8.2674-2681.2003 |
0.289 |
|
2006 |
Varaprasad CVNS, Barawkar D, Abdellaoui HE, Chakravarty S, Allan M, Chen H, Zhang W, Wu JZ, Tam R, Hamatake R, Lang S, Hong Z. Discovery of 3-hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles as potent MEK1 inhibitors. Bioorganic & Medicinal Chemistry Letters. 16: 3975-3980. PMID 16725322 DOI: 10.1016/J.Bmcl.2006.05.019 |
0.288 |
|
2014 |
Khose G, Shinde S, Panmand A, Kulkarni R, Munot Y, Bandyopadhyay A, Barawkar D, Patil SN. ChemInform Abstract: Synthesis of Substituted Esters of Imidazoles, Oxazoles, Thiazoles, and Diethylpyrazine-2,5-dicarboxylate from a Common Acyclic Precursor Employing C-Formylation Strategy. Cheminform. 45: no-no. DOI: 10.1002/CHIN.201440041 |
0.184 |
|
2013 |
Kandalkar SR, Kaduskar RD, Ramaiah PA, Barawkar DA, Bhuniya D, Deshpande AM. ChemInform Abstract: Highly Efficient One-Pot Amination of Carboxylate-Substituted Nitrogen-Containing Heteroaryl Chlorides via Staudinger Reaction. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201322153 |
0.165 |
|
Hide low-probability matches. |