Dinesh A Barawkar - Publications

Affiliations: 
CSIR-National Chemical Laboratory, Pune, India 
Area:
Bio-organic chemistry

27/32 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2017 Kandalkar SR, Ramaiah PA, Joshi M, Wavhal A, Waman Y, Raje AA, Tambe A, Ansari S, De S, Palle VP, Mookhtiar KA, Deshpande AM, Barawkar DA. Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2's-hydroxy-3's-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors. Bioorganic & Medicinal Chemistry. PMID 28951094 DOI: 10.1016/J.Bmc.2017.09.015  0.711
2017 Basu S, Barawkar DA, Ramdas V, Patel M, Waman Y, Panmand A, Kumar S, Thorat S, Naykodi M, Goswami A, Reddy BS, Prasad V, Chaturvedi S, Quraishi A, Menon S, et al. Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases. European Journal of Medicinal Chemistry. 134: 218-229. PMID 28415011 DOI: 10.1016/J.Ejmech.2017.04.014  0.352
2017 Koul S, Ramdas V, Barawkar DA, Waman YB, Prasad N, Madadi SK, Shejul YD, Bonagiri R, Basu S, Menon S, Reddy SB, Chaturvedi S, Chennamaneni SR, Bedse G, Thakare R, et al. Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A1 receptor antagonists and their biological evaluation. Bioorganic & Medicinal Chemistry. PMID 28238512 DOI: 10.1016/J.Bmc.2017.02.029  0.336
2017 Basu S, Barawkar DA, Thorat S, Shejul YD, Patel M, Naykodi M, Jain V, Salve Y, Prasad V, Chaudhary S, Ghosh I, Bhat G, Quraishi A, Patil H, Ansari S, et al. Design, Synthesis of Novel, Potent, Selective, Orally Bio-available Adenosine A2A Receptor Antagonists and Their Biological Evaluation. Journal of Medicinal Chemistry. PMID 28055204 DOI: 10.1021/Acs.Jmedchem.6B01584  0.321
2016 Basu S, Barawkar DA, Ramdas V, Waman Y, Patel M, Panmand A, Kumar S, Thorat S, Bonagiri R, Jadhav D, Mukhopadhyay P, Prasad V, Reddy BS, Goswami A, Chaturvedi S, et al. A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives. European Journal of Medicinal Chemistry. PMID 27842891 DOI: 10.1016/J.Ejmech.2016.11.007  0.309
2014 Khose G, Shinde S, Panmand A, Kulkarni R, Munot Y, Bandyopadhyay A, Barawkar D, Patil SN. Synthesis of substituted esters of imidazoles, oxazoles, thiazoles, and diethyl pyrazine-2,5-dicarboxylate from a common acyclic precursor employing C-formylation strategy Tetrahedron Letters. 55: 2671-2674. DOI: 10.1016/J.Tetlet.2014.03.039  0.318
2013 Kandalkar SR, Kaduskar RD, Ramaiah PA, Barawkar DA, Bhuniya D, Deshpande AM. Highly efficient one-pot amination of carboxylate-substituted nitrogen-containing heteroaryl chlorides via Staudinger reaction Tetrahedron Letters. 54: 414-418. DOI: 10.1016/J.Tetlet.2012.11.027  0.709
2012 Barawkar DA, Bandyopadhyay A, Deshpande A, Koul S, Kandalkar S, Patil P, Khose G, Vyas S, Mone M, Bhosale S, Singh U, De S, Meru A, Gundu J, Chugh A, et al. Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain L-2-hydroxy acid oxidase. Bioorganic & Medicinal Chemistry Letters. 22: 4341-7. PMID 22658862 DOI: 10.1016/J.Bmcl.2012.05.020  0.723
2012 Basu S, Prasad UV, Barawkar DA, De S, Palle VP, Menon S, Patel M, Thorat S, Singh UP, Das Sarma K, Waman Y, Niranjan S, Pathade V, Gaur A, Reddy S, et al. Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors. Bioorganic & Medicinal Chemistry Letters. 22: 2843-9. PMID 22424978 DOI: 10.1016/J.Bmcl.2012.02.070  0.351
2011 Barawkar DA, Meru A, Bandyopadhyay A, Banerjee A, Deshpande AM, Athare C, Koduru C, Khose G, Gundu J, Mahajan K, Patil P, Kandalkar SR, Niranjan S, Bhosale S, De S, et al. Potent and Selective Inhibitors of Long Chain l-2-Hydroxy Acid Oxidase Reduced Blood Pressure in DOCA Salt-Treated Rats. Acs Medicinal Chemistry Letters. 2: 919-23. PMID 24900281 DOI: 10.1021/Ml2001938  0.715
2010 BARAWKAR DA, LINKLETTER B, BRUICE TC. ChemInform Abstract: Synthesis of Protected Guanidinium Linked Dinucleoside Incorporable into an Oligonucleotide Using Solid Phase DNA Methodology. Cheminform. 29: no-no. DOI: 10.1002/CHIN.199841236  0.458
2006 El Abdellaoui H, Varaprasad CVNS, Barawkar D, Chakravarty S, Maderna A, Tam R, Chen H, Allan M, Wu JZ, Appleby T, Yan S, Zhang W, Lang S, Yao N, Hamatake R, et al. Identification of isothiazole-4-carboxamidines derivatives as a novel class of allosteric MEK1 inhibitors Bioorganic and Medicinal Chemistry Letters. 16: 5561-5566. PMID 16934458 DOI: 10.1016/J.Bmcl.2006.08.048  0.306
2000 Barawkar DA, Kwok Y, Bruice TW, Bruice TC. Deoxynucleic guanidine/peptide nucleic acid chimeras: Synthesis, binding and invasion studies with DNA Journal of the American Chemical Society. 122: 5244-5250. DOI: 10.1021/Ja000022L  0.573
1999 Jadhav VR, Barawkar DA, Ganesh KN. Polarity Sensing by Fluorescent Oligonucleotides:  First Demonstration of Sequence-Dependent Microenvironmental Changes in the DNA Major Groove The Journal of Physical Chemistry B. 103: 7383-7385. DOI: 10.1021/Jp9914323  0.603
1999 Barawkar DA, Bruice TC. Deoxynucleic guanidines/PNA (DNG/PNA) chimeras: Oligonucleoside analogue containing cationic guanidinium and neutral amide linkages [2] Journal of the American Chemical Society. 121: 10418-10419. DOI: 10.1021/Ja9923540  0.493
1998 Barawkar DA, Linkletter B, Bruice TC. Synthesis of protected guanidinium linked dinucleoside incorporable into an oligonucleotide using solid phase DNA methodology. Bioorganic & Medicinal Chemistry Letters. 8: 1517-20. PMID 9873381 DOI: 10.1016/S0960-894X(98)00251-0  0.529
1998 Barawkar DA, Bruice TC. Synthesis, biophysical properties, and nuclease resistance properties of mixed backbone oligodeoxynucleotides containing cationic internucleoside guanidinium linkages: deoxynucleic guanidine/DNA chimeras. Proceedings of the National Academy of Sciences of the United States of America. 95: 11047-52. PMID 9736687 DOI: 10.1073/Pnas.95.19.11047  0.555
1998 Ganesh KN, Kumar V, Barawkar DA, Rajeev KG, Rana VS. Enhancing DNA triplex stability via nucleobase modification Pure and Applied Chemistry. 70: 289-292. DOI: 10.1351/Pac199870020289  0.737
1997 Ganesh KN, Rajeev KG, Pallan PS, Rana VS, Barawkar DA, Kumar VA. Modulation of DNA Triplex Stability Through Nucleobase Modifications Nucleosides and Nucleotides. 16: 1271-1278. DOI: 10.1080/07328319708006169  0.711
1997 Jadhav VR, Barawkar DA, Natu AA, Ganesh KN. 5-Amido-(carboxyfluorescein)-2′-dU-oligonucloetides: Novel Primers for Fluorescent Detection of PCR Amplified DNA Nucleosides and Nucleotides. 16: 107-114. DOI: 10.1080/07328319708002526  0.558
1996 Rana VS, Barawkar DA, Ganesh KN. Molecular Recognition of 5-Amino-dU in the Central Strand of a DNA Triplex: Formation of Triads AU(#):A in Parallel and GU(#):A in Antiparallel Motif(,). The Journal of Organic Chemistry. 61: 3578-3579. PMID 11667196 DOI: 10.1021/Jo9602074  0.747
1996 Barawkar DA, Rajeev KG, Kumar VA, Ganesh KN. Triplex formation at physiological pH by 5-Me-dC-N4-(spermine) [X] oligodeoxynucleotides: non protonation of N3 in X of X*G:C triad and effect of base mismatch/ionic strength on triplex stabilities. Nucleic Acids Research. 24: 1229-37. PMID 8614624 DOI: 10.1093/Nar/24.7.1229  0.704
1995 Barawkar DA, Ganesh KN. Fluorescent d(CGCGAATTCGCG): characterization of major groove polarity and study of minor groove interactions through a major groove semantophore conjugate. Nucleic Acids Research. 23: 159-64. PMID 7870581 DOI: 10.1093/Nar/23.1.159  0.589
1994 Barawkar DA, Ganesh KN. Exploring DNA minor groove interactions through a probe conjugate in major groove: fluorescence studies on netropsin complexation with dU-5-aminodansyl-DNA. Biochemical and Biophysical Research Communications. 203: 53-8. PMID 8074699 DOI: 10.1006/bbrc.1994.2147  0.516
1994 Barawkar DA, Kumar VA, Ganesh KN. Triplex formation at physiological pH by oligonucleotides incorporating 5-Me-dC-(N4-spermine). Biochemical and Biophysical Research Communications. 205: 1665-70. PMID 7811251 DOI: 10.1006/Bbrc.1994.2859  0.593
1994 Prakash T, Barawkar DA, Vaijayanti K, Ganesh K. Synthesis of site-specific oligonucleotide-polyamine conjugates Bioorganic & Medicinal Chemistry Letters. 4: 1733-1738. DOI: 10.1016/S0960-894X(00)80371-6  0.574
1993 Barawkar DA, Ganesh K. Solid phase synthesis of DNA containing 5-NH2-2′-deoxyuridine Bioorganic & Medicinal Chemistry Letters. 3: 347-352. DOI: 10.1016/S0960-894X(01)80908-2  0.591
Low-probability matches (unlikely to be authored by this person)
2017 Basu S, Barawkar DA, Ramdas V, Naykodi M, Shejul YD, Patel M, Thorat S, Panmand A, Kashinath K, Bonagiri R, Prasad V, Bhat G, Quraishi A, Chaudhary S, Magdum A, et al. Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression. Acs Medicinal Chemistry Letters. 8: 835-840. PMID 28835798 DOI: 10.1021/Acsmedchemlett.7B00175  0.298
2003 Zhong W, An H, Barawkar D, Hong Z. Dinucleotide Analogues as Novel Inhibitors of RNA-Dependent RNA Polymerase of Hepatitis C Virus Antimicrobial Agents and Chemotherapy. 47: 2674-2681. PMID 12878540 DOI: 10.1128/Aac.47.8.2674-2681.2003  0.289
2006 Varaprasad CVNS, Barawkar D, Abdellaoui HE, Chakravarty S, Allan M, Chen H, Zhang W, Wu JZ, Tam R, Hamatake R, Lang S, Hong Z. Discovery of 3-hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles as potent MEK1 inhibitors. Bioorganic & Medicinal Chemistry Letters. 16: 3975-3980. PMID 16725322 DOI: 10.1016/J.Bmcl.2006.05.019  0.288
2014 Khose G, Shinde S, Panmand A, Kulkarni R, Munot Y, Bandyopadhyay A, Barawkar D, Patil SN. ChemInform Abstract: Synthesis of Substituted Esters of Imidazoles, Oxazoles, Thiazoles, and Diethylpyrazine-2,5-dicarboxylate from a Common Acyclic Precursor Employing C-Formylation Strategy. Cheminform. 45: no-no. DOI: 10.1002/CHIN.201440041  0.184
2013 Kandalkar SR, Kaduskar RD, Ramaiah PA, Barawkar DA, Bhuniya D, Deshpande AM. ChemInform Abstract: Highly Efficient One-Pot Amination of Carboxylate-Substituted Nitrogen-Containing Heteroaryl Chlorides via Staudinger Reaction. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201322153  0.165
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