| Year |
Citation |
Score |
| 2023 |
Inokuma T, Yamada KI. Remote Electronic Tuning of Chiral N-Heterocyclic Carbenes. Chemical Record (New York, N.Y.). e202300103. PMID 37255345 DOI: 10.1002/tcr.202300103 |
0.318 |
|
| 2021 |
Inokuma T. Synthesis of Non-canonical Amino Acids and Peptide Containing Them for Establishment of the Template for Drug Discovery. Chemical & Pharmaceutical Bulletin. 69: 303-313. PMID 33790076 DOI: 10.1248/cpb.c21-00031 |
0.371 |
|
| 2019 |
Inokuma T, Sakakibara T, Someno T, Masui K, Shigenaga A, Otaka A, Yamada KI. Asymmetric Synthesis of α-Amino Phosphonic Acids Using Stable Imino Phosphonate as a Universal Precursor. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 31449339 DOI: 10.1002/Chem.201903572 |
0.395 |
|
| 2019 |
Komiya C, Shigenaga A, Tsukimoto J, Ueda M, Morisaki T, Inokuma T, Itoh K, Otaka A. Traceless synthesis of protein thioesters using enzyme-mediated hydrazinolysis and subsequent self-editing of the cysteinyl prolyl sequence. Chemical Communications (Cambridge, England). 55: 7029-7032. PMID 31140482 DOI: 10.1039/C9Cc03583D |
0.389 |
|
| 2019 |
Kiyama H, Inokuma T, Kuroda Y, Yamaoka Y, Takasu K, Yamada K. Optical resolution via catalytic generation of chiral auxiliary Tetrahedron Letters. 60: 175-177. DOI: 10.1016/J.Tetlet.2018.12.006 |
0.304 |
|
| 2018 |
Inokuma T. [Asymmetric Synthesis of Unnatural Amino Acid-containing Peptides via Direct Asymmetric Reaction of Peptidyl Compounds]. Yakugaku Zasshi : Journal of the Pharmaceutical Society of Japan. 138: 1371-1379. PMID 30381645 DOI: 10.1248/Yakushi.18-00143 |
0.456 |
|
| 2018 |
Naruse N, Ohkawachi K, Inokuma T, Shigenaga A, Otaka A. Resin-Bound Crypto-Thioester for Native Chemical Ligation. Organic Letters. PMID 29629775 DOI: 10.1021/Acs.Orglett.8B00795 |
0.389 |
|
| 2018 |
Inokuma T, Sato S. [Chemical Biology for Pharmaceutical Sciences (Development of Practical Chemical Biotechnology)]. Yakugaku Zasshi : Journal of the Pharmaceutical Society of Japan. 138: 37-38. PMID 29311463 DOI: 10.1248/Yakushi.17-00186-F |
0.392 |
|
| 2018 |
Otaka A, Yamada K, Inokuma T, Nishida K. Direct Enantioselective Indolylation of Peptidyl Imine for the Synthesis of Indolyl Glycine-Containing Peptides Heterocycles. 97: 1269. DOI: 10.3987/Com-18-S(T)86 |
0.415 |
|
| 2018 |
Jichu T, Inokuma T, Aihara K, Kohiki T, Nishida K, Shigenaga A, Yamada K, Otaka A. A Recyclable Hydrophobic Anchor‐Tagged Asymmetric Amino Thiourea Catalyst Chemcatchem. 10: 3402-3405. DOI: 10.1002/Cctc.201800714 |
0.321 |
|
| 2017 |
Kohiki T, Nishikawa Y, Inokuma T, Shigenaga A, Otaka A. Chemical Synthetic Platform for Chlorpromazine Oligomers That Were Reported as Photo-degradation Products of Chlorpromazine. Chemical & Pharmaceutical Bulletin. 65: 1161-1166. PMID 29199220 DOI: 10.1248/Cpb.C17-00692 |
0.346 |
|
| 2017 |
Inokuma T, Jichu T, Nishida K, Shigenaga A, Otaka A. A Convenient Method for Preparation of α-Imino Carboxylic Acid Derivatives and Application to the Asymmetric Synthesis of Unnatural α-Amino Acid Derivative. Chemical & Pharmaceutical Bulletin. 65: 573-581. PMID 28566650 DOI: 10.1248/Cpb.C17-00158 |
0.377 |
|
| 2017 |
Shigenaga A, Yamamoto J, Kohiki T, Inokuma T, Otaka A. Invention of stimulus-responsive peptide-bond-cleaving residue (Spr) and its application to chemical biology tools. Journal of Peptide Science : An Official Publication of the European Peptide Society. PMID 28105728 DOI: 10.1002/Psc.2961 |
0.392 |
|
| 2017 |
Aihara K, Inokuma T, Jichu T, Lin Z, Fu F, Yamaoka K, Shigenaga A, Hutchins DA, Schmidt EW, Otaka A. Cysteine-Free Intramolecular Ligation of N-Sulfanylethylanilide Peptide Using 4-Mercaptobenzylphosphonic Acid: Synthesis of Cyclic Peptide Trichamide Synlett. 28: 1944-1949. DOI: 10.1055/S-0036-1589055 |
0.434 |
|
| 2016 |
Eto M, Naruse N, Morimoto K, Yamaoka K, Sato K, Tsuji K, Inokuma T, Shigenaga A, Otaka A. Development of an Anilide-Type Scaffold for the Thioester Precursor N-Sulfanylethylcoumarinyl Amide. Organic Letters. PMID 27529363 DOI: 10.1021/Acs.Orglett.6B02207 |
0.409 |
|
| 2016 |
Nakamura T, Sato K, Naruse N, Kitakaze K, Inokuma T, Hirokawa T, Shigenaga A, Itoh K, Otaka A. Tailored Synthesis of 162-Residue S-Monoglycosylated GM2-Activator Protein (GM2AP) Analogues that Allows Facile Access to Protein Library. Chembiochem : a European Journal of Chemical Biology. PMID 27428709 DOI: 10.1002/Cbic.201600400 |
0.462 |
|
| 2016 |
Denda M, Morisaki T, Kohiki T, Yamamoto J, Sato K, Sagawa I, Inokuma T, Sato Y, Yamauchi A, Shigenaga A, Otaka A. Labelling of endogenous target protein via N-S acyl transfer-mediated activation of N-sulfanylethylanilide. Organic & Biomolecular Chemistry. PMID 27264675 DOI: 10.1039/C6Ob01014H |
0.379 |
|
| 2016 |
Morisaki T, Denda M, Yamamoto J, Tsuji D, Inokuma T, Itoh K, Shigenaga A, Otaka A. An N-sulfanylethylanilide-based traceable linker for enrichment and selective labelling of target proteins. Chemical Communications (Cambridge, England). PMID 27146590 DOI: 10.1039/C6Cc01229A |
0.33 |
|
| 2016 |
Aihara K, Yamaoka K, Naruse N, Inokuma T, Shigenaga A, Otaka A. One-Pot/Sequential Native Chemical Ligation Using Photocaged Crypto-thioester. Organic Letters. PMID 26753720 DOI: 10.1021/Acs.Orglett.5B03661 |
0.401 |
|
| 2016 |
Nakamura T, Sato K, Naruse N, Kitakaze K, Inokuma T, Hirokawa T, Shigenaga A, Itoh K, Otaka A. Back Cover: Tailored Synthesis of 162‐Residue S‐Monoglycosylated GM2‐Activator Protein (GM2AP) Analogues that Allows Facile Access to a Protein Library (ChemBioChem 20/2016) Chembiochem. 17: 1994-1994. DOI: 10.1002/Cbic.201600521 |
0.325 |
|
| 2015 |
Itoh Y, Aihara K, Mellini P, Tojo T, Ota Y, Tsumoto H, Solomon VR, Zhan P, Suzuki M, Ogasawara D, Shigenaga A, Inokuma T, Nakagawa H, Miyata N, Mizukami T, et al. Identification of SNAIL1 Peptide-Based Irreversible Lysine Specific Demethylase 1-Selective Inactivators. Journal of Medicinal Chemistry. PMID 26700437 DOI: 10.1021/Acs.Jmedchem.5B01323 |
0.368 |
|
| 2015 |
Komiya C, Aihara K, Morishita K, Ding H, Inokuma T, Shigenaga A, Otaka A. Development of an intein-inspired amide cleavage chemical device. The Journal of Organic Chemistry. PMID 26646813 DOI: 10.1021/Acs.Joc.5B02399 |
0.336 |
|
| 2015 |
Miyajima R, Tsuda Y, Inokuma T, Shigenaga A, Imanishi M, Futaki S, Otaka A. Preparation of peptide thioesters from naturally occurring sequences using reaction sequence consisting of regioselective S-cyanylation and hydrazinolysis†. Biopolymers. PMID 26501985 DOI: 10.1002/Bip.22757 |
0.442 |
|
| 2015 |
Tsuda Y, Shigenaga A, Tsuji K, Denda M, Sato K, Kitakaze K, Nakamura T, Inokuma T, Itoh K, Otaka A. Development of a Chemical Methodology for the Preparation of Peptide Thioesters Applicable to Naturally Occurring Peptides Using a Sequential Quadruple Acyl Transfer System. Chemistryopen. 4: 448-52. PMID 26478838 DOI: 10.1002/Open.201500086 |
0.42 |
|
| 2015 |
Tsuji K, Tanegashima K, Sato K, Sakamoto K, Shigenaga A, Inokuma T, Hara T, Otaka A. Efficient one-pot synthesis of CXCL14 and its derivative using an N-sulfanylethylanilide peptide as a peptide thioester equivalent and their biological evaluation. Bioorganic & Medicinal Chemistry. 23: 5909-14. PMID 26187016 DOI: 10.1016/J.Bmc.2015.06.064 |
0.378 |
|
| 2015 |
Sato K, Kitakaze K, Nakamura T, Naruse N, Aihara K, Shigenaga A, Inokuma T, Tsuji D, Itoh K, Otaka A. The total chemical synthesis of the monoglycosylated GM2 ganglioside activator using a novel cysteine surrogate. Chemical Communications (Cambridge, England). 51: 9946-8. PMID 26006093 DOI: 10.1039/C5Cc02967H |
0.435 |
|
| 2015 |
Inokuma T, Fuller RP, Barbas CF. N-Sulfonyl-β-lactam hapten as an effective labeling reagent for aldolase mAb. Bioorganic & Medicinal Chemistry Letters. 25: 1684-7. PMID 25791455 DOI: 10.1016/J.Bmcl.2015.03.011 |
0.328 |
|
| 2015 |
Aihara K, Komiya C, Shigenaga A, Inokuma T, Takahashi D, Otaka A. Liquid-phase synthesis of bridged peptides using olefin metathesis of a protected peptide with a long aliphatic chain anchor. Organic Letters. 17: 696-9. PMID 25629979 DOI: 10.1021/Ol503718J |
0.371 |
|
| 2015 |
Kita M, Yamamoto J, Morisaki T, Komiya C, Inokuma T, Miyamoto L, Tsuchiya K, Shigenaga A, Otaka A. Design and synthesis of a hydrogen peroxide-responsive amino acid that induces peptide bond cleavage after exposure to hydrogen peroxide Tetrahedron Letters. 56: 4228-4231. DOI: 10.1016/J.Tetlet.2015.05.060 |
0.386 |
|
| 2015 |
Aihara K, Inokuma T, Komiya C, Shigenaga A, Otaka A. Synthesis of lactam-bridged cyclic peptides using sequential olefin metathesis and diimide reduction reactions Tetrahedron. 71: 4183-4191. DOI: 10.1016/J.Tet.2015.04.093 |
0.444 |
|
| 2014 |
Tsuji N, Stadler M, Kazumi N, Inokuma T, Kobayashi Y, Takemoto Y. Catalytic asymmetric synthesis of the pentacyclic core of (-)-nakadomarin A via oxazolidine as an iminium cation equivalent. Organic & Biomolecular Chemistry. 12: 7919-22. PMID 25216237 DOI: 10.1039/C4Ob01678E |
0.355 |
|
| 2014 |
Azuma T, Murata A, Kobayashi Y, Inokuma T, Takemoto Y. A dual arylboronic acid--aminothiourea catalytic system for the asymmetric intramolecular hetero-Michael reaction of α,β-unsaturated carboxylic acids. Organic Letters. 16: 4256-9. PMID 25075571 DOI: 10.1021/Ol501954R |
0.42 |
|
| 2014 |
Ebisuno K, Denda M, Ogura K, Inokuma T, Shigenaga A, Otaka A. Development of caged non-hydrolyzable phosphoamino acids and application to photo-control of binding affinity of phosphopeptide mimetic to phosphopeptide-recognizing protein. Bioorganic & Medicinal Chemistry. 22: 2984-91. PMID 24768166 DOI: 10.1016/J.Bmc.2014.04.002 |
0.408 |
|
| 2013 |
Kobayashi Y, Taniguchi Y, Hayama N, Inokuma T, Takemoto Y. A powerful hydrogen-bond-donating organocatalyst for the enantioselective intramolecular oxa-Michael reaction of α,β-unsaturated amides and esters. Angewandte Chemie (International Ed. in English). 52: 11114-8. PMID 24039087 DOI: 10.1002/Anie.201305492 |
0.376 |
|
| 2013 |
Sato S, Inokuma T, Otsubo N, Burton DR, Barbas CF. Chemically Programmed Antibodies AS HIV-1 Attachment Inhibitors. Acs Medicinal Chemistry Letters. 4: 460-465. PMID 23750312 DOI: 10.1021/Ml400097Z |
0.423 |
|
| 2013 |
Ban H, Nagano M, Gavrilyuk J, Hakamata W, Inokuma T, Barbas CF. Facile and stabile linkages through tyrosine: bioconjugation strategies with the tyrosine-click reaction. Bioconjugate Chemistry. 24: 520-32. PMID 23534985 DOI: 10.1021/Bc300665T |
0.668 |
|
| 2013 |
Kobayashi Y, Inokuma T, Takemoto Y. Development of innovative hydrogen-bond-donor catalysts based on heterocyclic scaffolds and their applications to asymmetric reactions Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry. 71: 491-502. DOI: 10.5059/Yukigoseikyokaishi.71.491 |
0.322 |
|
| 2012 |
Uno T, Inokuma T, Takemoto Y. NHC-catalyzed thioesterification of aldehydes by external redox activation. Chemical Communications (Cambridge, England). 48: 1901-3. PMID 22228405 DOI: 10.1039/C2Cc17183J |
0.318 |
|
| 2011 |
Sakamoto S, Inokuma T, Takemoto Y. Organocatalytic asymmetric Neber reaction for the synthesis of 2H-azirine carboxylic esters. Organic Letters. 13: 6374-7. PMID 22107059 DOI: 10.1021/Ol2026747 |
0.418 |
|
| 2011 |
Inokuma T, Suzuki Y, Sakaeda T, Takemoto Y. Synthesis of optically active N-aryl amino acid derivatives through the asymmetric petasis reaction catalyzed by a novel hydroxy-thiourea catalyst. Chemistry, An Asian Journal. 6: 2902-6. PMID 21815270 DOI: 10.1002/Asia.201100453 |
0.411 |
|
| 2011 |
Inokuma T, Furukawa M, Uno T, Suzuki Y, Yoshida K, Yano Y, Matsuzaki K, Takemoto Y. Bifunctional hydrogen-bond donors that bear a quinazoline or benzothiadiazine skeleton for asymmetric organocatalysis. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 10470-7. PMID 21812044 DOI: 10.1002/Chem.201101338 |
0.301 |
|
| 2010 |
Yoshida K, Inokuma T, Takasu K, Takemoto Y. Catalytic asymmetric synthesis of both enantiomers of 4‑substituted 1,4-dihydropyridines with the use of bifunctional thiourea-ammonium salts bearing different counterions. Molecules (Basel, Switzerland). 15: 8305-26. PMID 21079568 DOI: 10.3390/Molecules15118305 |
0.368 |
|
| 2010 |
Yoshida K, Inokuma T, Takasu K, Takemoto Y. Brønsted acid-thiourea co-catalysis: Asymmetric synthesis of functionalized 1,4-dihydropyridines from β-enamino esters and α,β-unsaturated aldehydes Synlett. 1865-1869. DOI: 10.1055/S-0030-1258090 |
0.326 |
|
| 2009 |
Inokuma T, Takasu K, Sakaeda T, Takemoto Y. Hydroxyl group-directed organocatalytic asymmetric Michael addition of alpha,beta-unsaturated ketones with alkenylboronic acids. Organic Letters. 11: 2425-8. PMID 19402642 DOI: 10.1021/Ol9006053 |
0.315 |
|
| 2009 |
Inokuma T, Nagamoto Y, Sakamoto S, Miyabe H, Takasu K, Takemoto Y. Asymmetric synthesis of 4-substituted 2,6-dioxopiperidine-3-carbonitrile by using thioureacatalyzed asymmetric michael addition Heterocycles. 79: 573-582. DOI: 10.3987/Com-08-S(D)18 |
0.358 |
|
| 2009 |
Inokuma T, Sakamoto S, Takemoto Y. Enantioselective nitrocyclopropanation of α,β-unsaturated α-cyanoimides catalyzed by bifunctional thiourea Synlett. 1627-1630. DOI: 10.1055/S-0029-1217331 |
0.373 |
|
| 2006 |
Inokuma T, Hoashi Y, Takemoto Y. Thiourea-catalyzed asymmetric michael addition of activated methylene compounds to alpha,beta-unsaturated imides: dual activation of imide by intra- and intermolecular hydrogen bonding. Journal of the American Chemical Society. 128: 9413-9. PMID 16848477 DOI: 10.1021/Ja061364F |
0.391 |
|
| 2005 |
Yanada R, Obika S, Inokuma T, Yanada K, Yamashita M, Ohta S, Takemoto Y. Stereoselective synthesis of 3-alkylideneoxindoles via palladium-catalyzed domino reactions. The Journal of Organic Chemistry. 70: 6972-5. PMID 16095329 DOI: 10.1021/Jo0508604 |
0.4 |
|
| 2005 |
Yanada R, Obika S, Kobayashi Y, Inokuma T, Oyama M, Yanada K, Takemoto Y. Stereoselective synthesis of 3-alkylideneoxindoles using tandem indium-mediated carbometallation and palladium-catalyzed cross-coupling reactions Advanced Synthesis and Catalysis. 347: 1632-1642. DOI: 10.1002/Adsc.200505147 |
0.352 |
|
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