363 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2023 Kushwaha M, Qayum A, Sharma N, Abrol V, Choudhary P, Murtaza M, Singh SK, Vishwakarma RA, Goutam U, Jain SK, Jaglan S. Correction to "LC-PDA-MS/MS-Based Dereplication Guided Isolation of a New Optical Isomer of 19,20-Epoxycytochalasin-N and Its Cytotoxic Activity". Acs Omega. 8: 7243. PMID 36844607 DOI: 10.1021/acsomega.3c00349  0.772
2022 Jain SK, Pathania AS, Parshad R, Raina C, Ali A, Gupta AP, Kushwaha M, Aravinda S, Bhushan S, Bharate SB, Vishwakarma RA. Correction: Chrysomycins A-C, antileukemic naphthocoumarins from . Rsc Advances. 12: 23680-23682. PMID 36125971 DOI: 10.1039/d2ra90078e  0.752
2022 Kushwaha M, Qayum A, Sharma N, Abrol V, Choudhary P, Murtaza M, Singh SK, Vishwakarma RA, Goutam U, Jain SK, Jaglan S. LC-PDA-MS/MS-Based Dereplication Guided Isolation of a New Optical Isomer of 19,20-Epoxycytochalasin-N and Its Cytotoxic Activity. Acs Omega. 7: 29135-29141. PMID 36033687 DOI: 10.1021/acsomega.2c03037  0.793
2022 Tripathi N, Goel B, Bhardwaj N, Vishwakarma RA, Jain SK. Exploring the Potential of Chemical Inhibitors for Targeting Post-translational Glycosylation of Coronavirus (SARS-CoV-2). Acs Omega. 7: 27038-27051. PMID 35937682 DOI: 10.1021/acsomega.2c02345  0.769
2022 Gupta R, Sharma S, Singh R, Vishwakarma RA, Mignani S, Singh PP. Functionalized Nitroimidazole Scaffold Construction and Their Pharmaceutical Applications: A 1950-2021 Comprehensive Overview. Pharmaceuticals (Basel, Switzerland). 15. PMID 35631389 DOI: 10.3390/ph15050561  0.287
2022 Kumar C, Akhter S, Satti NK, Gupta VK, Meena SR, Vishwakarma R, Hassan QP, Verma MK. Dereplication approach for the first time isolation of tatarinowin a and pentadecanoic acid from L. by using GC-MS. Natural Product Research. 1-6. PMID 35382654 DOI: 10.1080/14786419.2022.2061482  0.338
2022 Anand R, Cham PS, Gannedi V, Sharma S, Kumar M, Singh R, Vishwakarma RA, Singh PP. Stereoselective Synthesis of Nonpsychotic Natural Cannabidiol and Its Unnatural/Terpenyl/Tail-Modified Analogues. The Journal of Organic Chemistry. PMID 35289168 DOI: 10.1021/acs.joc.1c02571  0.785
2021 Shukla R, Rajpoot RK, Poddar A, Ahuja R, Beesetti H, Shanmugam RK, Chaturvedi S, Nayyar K, Singh D, Singamaneni V, Gupta P, Gupta AP, Gairola S, Kumar P, Bedi YS, ... ... Vishwakarma RA, et al. -Derived Phytopharmaceutical Drug Has Potent Anti-dengue Activity. Frontiers in Microbiology. 12: 746110. PMID 34912307 DOI: 10.3389/fmicb.2021.746110  0.296
2021 Joshi U, Naslund JA, Anand A, Tugnawat D, Vishwakarma R, Bhan A, Patel V, Lu C. Assessing costs of developing a digital program for training community health workers to deliver treatment for depression: A case study in rural India. Psychiatry Research. 307: 114299. PMID 34871874 DOI: 10.1016/j.psychres.2021.114299  0.189
2021 Girme A, Saste G, Pawar S, Ghule C, Mirgal A, Patel S, Tiwari A, Ghoshal S, Bharate SB, Bharate SS, Reddy DS, Vishwakarma RA, Hingorani L. Quantitative Determination and Characterization of a Kashmir Saffron ( L.)-Based Botanical Supplement Using Single-Laboratory Validation Study by HPLC-PDA with LC-MS/MS and HPTLC Investigations. Acs Omega. 6: 23460-23474. PMID 34549144 DOI: 10.1021/acsomega.1c03470  0.525
2021 Jamwal VL, Kumar N, Bhat R, Jamwal PS, Singh K, Dogra S, Kulkarni A, Bhadra B, Shukla MR, Saran S, Dasgupta S, Vishwakarma RA, Gandhi SG. Optimization and validation of RT-LAMP assay for diagnosis of SARS-CoV2 including the globally dominant Delta variant. Virology Journal. 18: 178. PMID 34461941 DOI: 10.1186/s12985-021-01642-9  0.23
2021 Prabhakara C, Godbole R, Sil P, Jahnavi S, Gulzar SE, van Zanten TS, Sheth D, Subhash N, Chandra A, Shivaraj A, Panikulam P, U I, Nuthakki VK, Puthiyapurayil TP, Ahmed R, ... ... Vishwakarma R, et al. Strategies to target SARS-CoV-2 entry and infection using dual mechanisms of inhibition by acidification inhibitors. Plos Pathogens. 17: e1009706. PMID 34252168 DOI: 10.1371/journal.ppat.1009706  0.642
2021 Gupta M, Wani A, Ahsan AU, Ali M, Chibber P, Singh S, Digra SK, Datt M, Bharate S, Vishwakarma RA, Singh G, Kumar A. Safranal inhibits NLRP3 inflammasome activation by preventing ASC oligomerization. Toxicology and Applied Pharmacology. 115582. PMID 34019860 DOI: 10.1016/j.taap.2021.115582  0.633
2021 Pathak S, Gokhroo A, Kumar Dubey A, Majumdar S, Gupta S, Almeida A, Mahajan GB, Kate A, Mishra P, Sharma R, Kumar S, Vishwakarma R, Balakrishnan A, Atreya H, Nandi D. 7-Hydroxy Frullanolide, a sesquiterpene lactone, increases intracellular calcium amounts, lowers CD4 T cell and macrophage responses, and ameliorates DSS-induced colitis. International Immunopharmacology. 97: 107655. PMID 33901737 DOI: 10.1016/j.intimp.2021.107655  0.267
2021 Raina D, Tiwari H, Sharma S, Deepika, Chinthakindi PK, Nargotra A, Sangwan PL, Eniyan K, Bajpai U, Vishwakarma RA, Khan FG, Saran S, Khan IA. Screening of compound library identifies novel inhibitors against the MurA enzyme of Escherichia coli. Applied Microbiology and Biotechnology. PMID 33860835 DOI: 10.1007/s00253-021-11272-4  0.358
2021 Singh VP, Pathania AS, Sharma S, Malik FA, Kumar A, Singh D, Vishwakarma RA. Total Synthesis and Conformational Analysis of Naturally Occurring Lipovelutibols along with Lead Optimization of Lipovelutibol D. Acs Omega. 6: 6070-6080. PMID 33718698 DOI: 10.1021/acsomega.0c04038  0.321
2021 Arora P, Kumar A, Vishwakarma RA, Riyaz-Ul-Hassan S. A natural association of a yeast with Aspergillus terreus and its impact on the host fungal biology. Fems Microbiology Letters. PMID 33713123 DOI: 10.1093/femsle/fnab032  0.26
2021 Manzoor MM, Goyal P, Pandotra P, Dar MS, Dar MJ, Misra P, Gupta AP, Vishwakarma RA, Ahuja A, Dhar MK, Gupta S. Transcriptome-wide identification of squalene epoxidase genes from Glycyrrhiza glabra L.: expression analysis and heterologous expression of GgSQE1 suggest important role in terpenoid biosynthesis. Protoplasma. PMID 33629144 DOI: 10.1007/s00709-021-01616-2  0.257
2021 Kushwaha M, Qayum A, Jain SK, Singh J, Srivastava AK, Srivastava S, Sharma N, Abrol V, Malik R, Singh SK, Vishwakarma RA, Jaglan S. Tandem MS-Based Metabolite Profiling of 19,20-Epoxycytochalasin C Reveals the Importance of a Hydroxy Group at the C7 Position for Biological Activity. Acs Omega. 6: 3717-3726. PMID 33585752 DOI: 10.1021/acsomega.0c05307  0.786
2021 Wani A, Al Rihani SB, Sharma A, Weadick B, Govindarajan R, Khan SU, Sharma PR, Dogra A, Nandi U, Reddy CN, Bharate SS, Singh G, Bharate SB, Vishwakarma RA, Kaddoumi A, et al. Crocetin promotes clearance of amyloid-β by inducing autophagy via the STK11/LKB1-mediated AMPK pathway. Autophagy. PMID 33404280 DOI: 10.1080/15548627.2021.1872187  0.502
2020 Sharma S, Anand R, Cham PS, Raina S, Vishwakarma RA, Singh PP. A concise and sequential synthesis of the nitroimidazooxazole based drug, Delamanid and related compounds. Rsc Advances. 10: 17085-17093. PMID 35521460 DOI: 10.1039/d0ra01662d  0.345
2020 Singh VP, Pathania AS, Kushwaha M, Singh S, Sharma V, Malik FA, Khan IA, Kumar A, Singh D, Vishwakarma RA. 14-Residue peptaibol velutibol A from : its structural and cytotoxic evaluation. Rsc Advances. 10: 31233-31242. PMID 35520634 DOI: 10.1039/d0ra05780k  0.329
2020 Bhardwaj M, Chib S, Kaur L, Kumar A, Chaudhuri B, Malik F, Vishwakarma RA, Saran S, Mukherjee D. Conversion of amino acids to aryl/heteroaryl ethanol metabolites using human CYP2D6-expressing live baker's yeast. Rsc Medicinal Chemistry. 11: 142-147. PMID 33479614 DOI: 10.1039/c9md00451c  0.325
2020 Girme A, Saste G, Pawar S, Balasubramaniam AK, Musande K, Darji B, Satti NK, Verma MK, Anand R, Singh R, Vishwakarma RA, Hingorani L. Investigating 11 Withanosides and Withanolides by UHPLC-PDA and Mass Fragmentation Studies from Ashwagandha (). Acs Omega. 5: 27933-27943. PMID 33163776 DOI: 10.1021/acsomega.0c03266  0.326
2020 Gani U, Vishwakarma RA, Misra P. Membrane transporters: the key drivers of transport of secondary metabolites in plants. Plant Cell Reports. PMID 32959124 DOI: 10.1007/S00299-020-02599-9  0.378
2020 Sharma S, Bhat R, Singh R, Sharma S, Wazir P, Singh PP, Vishwakarma RA, Khan IA. High-throughput screening of compounds library to identify novel inhibitors against latent Mycobacterium tuberculosis using streptomycin-dependent Mycobacterium tuberculosis 18b strain as a model. Tuberculosis (Edinburgh, Scotland). 124: 101958. PMID 32791471 DOI: 10.1016/J.Tube.2020.101958  0.414
2020 Visioni A, Rehman S, Viash SS, Singh SP, Vishwakarma R, Gyawali S, Al-Abdallat AM, Verma RPS. Genome Wide Association Mapping of Spot Blotch Resistance at Seedling and Adult Plant Stages in Barley. Frontiers in Plant Science. 11: 642. PMID 32670303 DOI: 10.3389/Fpls.2020.00642  0.232
2020 Gannedi V, Ali A, Singh PP, Vishwakarma RA. Total synthesis of phospholipomannan of the Candida albicans. The Journal of Organic Chemistry. PMID 32425042 DOI: 10.1021/Acs.Joc.0C00402  0.78
2020 Chibber P, Kumar C, Singh A, Assim Haq S, Ahmed I, Kumar A, Singh S, Vishwakarma R, Singh G. Anti-inflammatory and analgesic potential of OA-DHZ; a novel semisynthetic derivative of dehydrozingerone. International Immunopharmacology. 83: 106469. PMID 32251963 DOI: 10.1016/J.Intimp.2020.106469  0.411
2020 Kumar V, Bharate SS, Bhurta D, Gupta M, Gandhi SG, Singh D, Jaglan S, Kumar A, Vishwakarma RA, Bharate SB. Evaluation of rohitukine-enriched fraction of Dysoxylum binectariferum Hook.f. (leaves) as anti-arthritic phytopharmaceutical candidate: Chemical standardization, in-vivo validation, formulation development and oral pharmacokinetics. Journal of Ethnopharmacology. 112758. PMID 32165175 DOI: 10.1016/J.Jep.2020.112758  0.542
2020 Goyal P, Manzoor MM, Vishwakarma RA, Sharma D, Dhar MK, Gupta S. A Comprehensive Transcriptome-Wide Identification and Screening of WRKY Gene Family Engaged in Abiotic Stress in Glycyrrhiza glabra. Scientific Reports. 10: 373. PMID 31941983 DOI: 10.1038/S41598-019-57232-X  0.355
2020 Reddy CN, Bharate SB, Vishwakarma RA, Bharate SS. Chemical analysis of saffron by HPLC based crocetin estimation. Journal of Pharmaceutical and Biomedical Analysis. 181: 113094. PMID 31927167 DOI: 10.1016/J.Jpba.2020.113094  0.567
2020 Singh VP, Pathania AS, Kushwaha M, Singh S, Sharma V, Malik FA, Khan IA, Kumar A, Singh D, Vishwakarma RA. 14-Residue peptaibol velutibol A from Trichoderma velutinum: its structural and cytotoxic evaluation Rsc Advances. 10: 31233-31242. DOI: 10.1039/D0Ra05780K  0.424
2020 Sharma S, Anand R, Cham PS, Raina S, Vishwakarma RA, Singh PP. A concise and sequential synthesis of the nitroimidazooxazole based drug, Delamanid and related compounds Rsc Advances. 10: 17085-17093. DOI: 10.1039/D0Ra01662D  0.402
2020 Manzoor MM, Goyal P, Gupta AP, Khan S, Jaswal P, Misra P, Pandotra P, Ahuja A, Vishwakarma RA, Gupta S. Chemical and real-time based analysis revealed active gene machinery of glycyrrhizin biosynthesis and its accumulation in the aerial tissues of in-vitro regenerated Glycyrrhiza glabra L. Plant Growth Regulation. 1-9. DOI: 10.1007/S10725-020-00635-Y  0.368
2019 Ambala S, Singh R, Singh M, Cham PS, Gupta R, Munagala G, Yempalla KR, Vishwakarma RA, Singh PP. Metal-free, room temperature, acid-KSO mediated method for the nitration of olefins: an easy approach for the synthesis of nitroolefins. Rsc Advances. 9: 30428-30431. PMID 35530202 DOI: 10.1039/c9ra06414a  0.287
2019 Dar MI, Jan S, Reddy GL, Wani R, Syed M, Dar MJ, Sawant SD, Vishwakarma RA, Syed SH. Differentiation of human neuroblastoma cell line IMR-32 by sildenafil and its newly discovered analogue IS00384. Cellular Signalling. 65: 109425. PMID 31689507 DOI: 10.1016/J.Cellsig.2019.109425  0.416
2019 Reddy GL, Dar MI, Hudwekar AD, Mahajan P, Nargotra A, Baba AM, Nandi U, Wazir P, Singh G, Bharate SS, Vishwakarma RA, Syed SH, Sawant SD. Corrigendum to "Design, synthesis and biological evaluation of pyrazolopyrimidinone based potent and selective PDE5 inhibitors for treatment of erectile dysfunction" [Bioorg. Chem. 89 (2019) 103022]. Bioorganic Chemistry. 92: 103257. PMID 31525521 DOI: 10.1016/J.Bioorg.2019.103257  0.393
2019 Kumar V, Mintoo MJ, Mondhe DM, Bharate SB, Vishwakarma RA, Bharate SS. Binary and ternary solid dispersions of an anticancer preclinical lead, IIIM-290: In vitro and in vivo studies. International Journal of Pharmaceutics. 118683. PMID 31513869 DOI: 10.1016/J.Ijpharm.2019.118683  0.575
2019 Umar SA, Tanveer MA, Nazir LA, Divya G, Vishwakarma RA, Tasduq SA. Glycyrrhizic Acid Prevents Oxidative Stress Mediated DNA Damage Response through Modulation of Autophagy in Ultraviolet-B-Irradiated Human Primary Dermal Fibroblasts. Cellular Physiology and Biochemistry : International Journal of Experimental Cellular Physiology, Biochemistry, and Pharmacology. 53: 242-257. PMID 31313540 DOI: 10.33594/000000133  0.351
2019 Khan IA, Singh A, Mindala DP, Meena S, Vij B, Yadav AK, Roy S, Nandi U, Katare AK, Jaglan S, Singh D, Gupta AP, Gupta P, Singh S, Tikko MK, ... ... Vishwakarma RA, et al. Preclinical development of gastro-protective botanical candidate from Woodfordia fruticosa: Chemical standardization, efficacy, pharmacokinetics and safety pharmacology. Journal of Ethnopharmacology. 112023. PMID 31195031 DOI: 10.1016/J.Jep.2019.112023  0.379
2019 Reddy GL, Dar MI, Hudwekar AD, Mahajan P, Nargotra A, Baba AM, Nandi U, Wazir P, Singh G, Vishwakarma RA, Syed SH, Sawant SD. Design, synthesis and biological evaluation of pyrazolopyrimidinone based potent and selective PDE5 inhibitors for treatment of erectile dysfunction. Bioorganic Chemistry. 89: 103022. PMID 31181491 DOI: 10.1016/J.Bioorg.2019.103022  0.445
2019 Singh R, Mandrah K, Asati A, Patel DK, Goel B, Vishwakarma RA, Roy SK, Jain SK. Transformation of Santonin to a Naproxen Analogue with Anti-Inflammatory Activity. Journal of Natural Products. PMID 31125226 DOI: 10.1021/Acs.Jnatprod.8B00318  0.792
2019 Katoch M, Singh D, Kapoor KK, Vishwakarma RA. Trichoderma lixii (IIIM-B4), an endophyte of Bacopa monnieri L. producing peptaibols. Bmc Microbiology. 19: 98. PMID 31096902 DOI: 10.1186/S12866-019-1477-8  0.367
2019 Singh VP, Sharma R, Sharma V, Raina C, Kapoor KK, Kumar A, Chaubey A, Singh D, Vishwakarma RA. Isolation of depsipeptides and optimization for enhanced production of valinomycin from the North-Western Himalayan cold desert strain Streptomyces lavendulae. The Journal of Antibiotics. PMID 31073236 DOI: 10.1038/S41429-019-0183-Y  0.372
2019 Bharate SB, Kumar V, Bharate SS, Singh B, Singh G, Singh A, Gupta M, Singh D, Kumar A, Singh S, Vishwakarma RA. Discovery and preclinical development of IIIM-160, a Bergenia ciliata-based anti-inflammatory and anti-arthritic botanical drug candidate. Journal of Integrative Medicine. PMID 30898582 DOI: 10.1016/J.Joim.2019.03.001  0.565
2019 Abdullaha M, Mohammed S, Ali M, Kumar A, Vishwakarma RA, Bharate SB. Discovery of Quinazolin-4(3H)-ones as NLRP3 Inflammasome Inhibitors: Computational Design, Metal-free Synthesis and In-vitro Biological Evaluation. The Journal of Organic Chemistry. PMID 30896160 DOI: 10.1021/Acs.Joc.9B00138  0.689
2019 Wani A, Gupta M, Ahmad M, Shah AM, Ahsan AU, Hassan Qazi PH, Malik F, Singh G, Sharma PR, Kaddoumi A, Bharate SB, Vishwakarma RA, Kumar A. Alborixin clears amyloid-β by inducing autophagy through PTEN-mediated inhibition of the AKT pathway. Autophagy. PMID 30894052 DOI: 10.1080/15548627.2019.1596476  0.665
2019 Kumar A, Gannedi V, Rather SA, Vishwakarma RA, Ahmed QN. Introducing Oxo-Phenylacetyl (OPAc) as a Protecting Group for Carbohydrates. The Journal of Organic Chemistry. PMID 30888192 DOI: 10.1021/Acs.Joc.9B00126  0.778
2019 Nalli Y, Dar MS, Bano N, Rasool JU, Sarkar AR, Banday J, Bhat AQ, Rafia B, Vishwakarma RA, Dar MJ, Ali A. Analyzing the role of cannabinoids as modulators of Wnt/β-catenin signaling pathway for their use in the management of neuropathic pain. Bioorganic & Medicinal Chemistry Letters. PMID 30871771 DOI: 10.1016/J.Bmcl.2019.03.013  0.372
2019 Singh A, Chibber P, Kolimi P, Malik TA, Kapoor N, Kumar A, Kumar N, Gandhi SG, Singh S, Abdullah ST, Vishwakarma R, Singh G. Rohitukine inhibits NF-κB activation induced by LPS and other inflammatory agents. International Immunopharmacology. 69: 34-49. PMID 30665042 DOI: 10.1016/J.Intimp.2019.01.015  0.39
2019 Ambala S, Singh R, Singh M, Cham PS, Gupta R, Munagala G, Yempalla KR, Vishwakarma RA, Singh PP. Metal-free, room temperature, acid-K2S2O8 mediated method for the nitration of olefins: an easy approach for the synthesis of nitroolefins Rsc Advances. 9: 30428-30431. DOI: 10.1039/C9Ra06414A  0.388
2019 Kumar V, Vishwakarma RA, Bharate SS. Engineering solid dispersions of anticancer preclinical lead, IIIM-985: Physicochemical characterization and in vivo pharmacokinetics Journal of Drug Delivery Science and Technology. 49: 594-602. DOI: 10.1016/J.Jddst.2018.12.028  0.411
2019 Kumar M, Sharma S, Sil P, Kushwaha M, Mayor S, Vishwakarma RA, Singh PP. C-H Arylation of N -Heteroarenes under Metal-Free Conditions and its Application towards the Synthesis of Pentabromo- and Pentachloropseudilins European Journal of Organic Chemistry. 2019: 3591-3598. DOI: 10.1002/Ejoc.201900353  0.375
2019 Kumar Verma P, Vishwakarma RA, Sawant SD. Reaction Medium as the Installing Reservoir for Key Functionalities in the Molecules Asian Journal of Organic Chemistry. 8: 777-801. DOI: 10.1002/Ajoc.201900223  0.345
2018 Venkateswarlu V, Kour J, Kumar KAA, Verma PK, Reddy GL, Hussain Y, Tabassum A, Balgotra S, Gupta S, Hudwekar AD, Vishwakarma RA, Sawant SD. Direct N-heterocyclization of hydrazines to access styrylated pyrazoles: synthesis of 1,3,5-trisubstituted pyrazoles and dihydropyrazoles. Rsc Advances. 8: 26523-26527. PMID 35541044 DOI: 10.1039/c8ra04550j  0.33
2018 Bharate SS, Kumar V, Singh G, Singh A, Gupta M, Singh D, Kumar A, Vishwakarma RA, Bharate SB. Preclinical Development of -Based Botanical Lead IIIM-141 for Alzheimer's Disease: Chemical Standardization, Efficacy, Formulation Development, Pharmacokinetics, and Safety Pharmacology. Acs Omega. 3: 9572-9585. PMID 31459089 DOI: 10.1021/acsomega.8b00841  0.519
2018 Kumar V, Bhurta D, Sharma A, Kumar P, Bharate SB, Vishwakarma RA, Bharate SS. Impurity profiling of anticancer preclinical candidate, IIIM-290. Journal of Pharmaceutical and Biomedical Analysis. 166: 1-5. PMID 30590350 DOI: 10.1016/J.Jpba.2018.12.027  0.678
2018 Bharate SB, Mudududdla R, Mohanakrishnan D, Bharate SS, Vishwakarma RA, Sahal D. Orally Effective Aminoalkyl 10H-Indolo-[3,2-b]quinoline-11-carboxamide Kills the Malaria Parasite by Inhibiting Host Hemoglobin Uptake. Chemmedchem. PMID 30358112 DOI: 10.1002/Cmdc.201800579  0.688
2018 Thottacherry JJ, Kosmalska AJ, Kumar A, Vishen AS, Elosegui-Artola A, Pradhan S, Sharma S, Singh PP, Guadamillas MC, Chaudhary N, Vishwakarma R, Trepat X, Del Pozo MA, Parton RG, Rao M, et al. Mechanochemical feedback control of dynamin independent endocytosis modulates membrane tension in adherent cells. Nature Communications. 9: 4217. PMID 30310066 DOI: 10.1016/J.Bpj.2018.11.542  0.343
2018 Sharma S, Kumar M, Vishwakarma RA, Verma MK, Singh PP. Room Temperature, Metal-catalyzed Oxidative Acylation of Electron-deficient Heteroarenes with Alkynes, its Mechanism and Application Studies. The Journal of Organic Chemistry. PMID 30238752 DOI: 10.1021/Acs.Joc.8B01475  0.402
2018 Gupta M, Wani A, Ul Ahsan A, Chopra M, Vishwakarma RA, Singh G, Kumar A. Soluble Aβ suppresses TNF-α and activates NLRP3 inflammasome in THP-1 macrophages. Cytokine. 111: 84-87. PMID 30125779 DOI: 10.1016/J.Cyto.2018.07.026  0.375
2018 Kumar V, Bharate SB, Vishwakarma RA, Bharate SS. Selection of a Water-Soluble Salt Form of a Preclinical Candidate, IIIM-290: Multiwell-Plate Salt Screening and Characterization. Acs Omega. 3: 8365-8377. PMID 30087943 DOI: 10.1021/acsomega.8b00801  0.665
2018 Bharate SS, Mignani S, Vishwakarma RA. Why are the Majority of Active Compounds in the CNS Domain Natural Products? A Critical Analysis. Journal of Medicinal Chemistry. PMID 29989814 DOI: 10.1021/Acs.Jmedchem.7B01922  0.388
2018 Wani ZA, Ahmad T, Nalli Y, Ali A, Singh AP, Vishwakarma RA, Ashraf N, Riyaz-Ul-Hassan S. Porostereum sp., Associated with Saffron (Crocus sativus L.), is a Latent Pathogen Capable of Producing Phytotoxic Chlorinated Aromatic Compounds. Current Microbiology. PMID 29492649 DOI: 10.1007/S00284-018-1461-9  0.432
2018 Srinivas M, Singh Pathania A, Mahajan P, Verma PK, Chobe SS, Malik FA, Nargotra A, Vishwakarma RA, Sawant SD. Design and synthesis of 1,4-substituted 1H-1,2,3-triazolo-quinazolin-4(3H)-ones by Huisgen 1,3-dipolar cycloaddition with PI3Kγ isoform selective activity. Bioorganic & Medicinal Chemistry Letters. PMID 29486969 DOI: 10.1016/J.Bmcl.2018.02.032  0.461
2018 Singh VP, Yedukondalu N, Sharma V, Kushwaha M, Sharma R, Chaubey A, Kumar A, Singh D, Vishwakarma RA. Lipovelutibols A-D: Cytotoxic Lipopeptaibols from the Himalayan Cold Habitat Fungus Trichoderma velutinum. Journal of Natural Products. PMID 29373791 DOI: 10.1021/Acs.Jnatprod.6B00873  0.419
2018 Bharate SB, Kumar V, Jain SK, Mintoo MJ, Guru SK, Nuthakki VK, Sharma M, Bharate SS, Gandhi SG, Mondhe DM, Bhushan S, Vishwakarma RA. Discovery and Preclinical Development of IIIM-290, an Orally Active Potent Cyclin-dependent Kinase Inhibitor. Journal of Medicinal Chemistry. PMID 29370702 DOI: 10.1021/Acs.Jmedchem.7B01765  0.797
2018 Mignani S, Rodrigues J, Tomas H, Jalal R, Singh PP, Majoral JP, Vishwakarma RA. Present drug-likeness filters in medicinal chemistry during the hit and lead optimization process: how far can they be simplified? Drug Discovery Today. PMID 29330127 DOI: 10.1016/J.Drudis.2018.01.010  0.369
2018 Kushwaha M, Jain SK, Sharma N, Abrol V, Jaglan S, Vishwakarma RA. Establishment of LCMS Based Platform for Discovery of Quorum Sensing Inhibitors: Signal Detection in Pseudomonas aeruginosa PAO1. Acs Chemical Biology. PMID 29303546 DOI: 10.1021/Acschembio.7B00875  0.78
2018 Singh A, Thatikonda T, Kumar A, Wazir P, V V, Nandi U, Singh PP, Singh S, Gupta AP, Tikoo MK, Singh G, Vishwakarma R. Determination of ZSTK474, a novel Pan PI3K inhibitor in mouse plasma by LC-MS/MS and its application to Pharmacokinetics. Journal of Pharmaceutical and Biomedical Analysis. 149: 387-393. PMID 29175554 DOI: 10.1016/J.Jpba.2017.11.031  0.396
2018 Venkateswarlu V, Kour J, Kumar KAA, Verma PK, Reddy GL, Hussain Y, Tabassum A, Balgotra S, Gupta S, Hudwekar AD, Vishwakarma RA, Sawant SD. Direct N-heterocyclization of hydrazines to access styrylated pyrazoles: synthesis of 1,3,5-trisubstituted pyrazoles and dihydropyrazoles Rsc Advances. 8: 26523-26527. DOI: 10.1039/C8Ra04550J  0.397
2017 Awasthi P, Gupta AP, Bedi YS, Vishwakarma RA, Gandhi SG. Corrigendum: Mannitol Stress Directs Flavonoid Metabolism toward Synthesis of Flavones via Differential Regulation of Two Cytochrome P450 Monooxygenases in Coleus forskohlii. Frontiers in Plant Science. 8: 2222. PMID 29371862 DOI: 10.3389/fpls.2017.02222  0.239
2017 Magotra A, Sharma A, Singh S, Ojha PK, Kumar S, Bokolia N, Wazir P, Sharma S, Khan IA, Singh PP, Vishwakarma RA, Singh G, Nandi U. Physicochemical, pharmacokinetic, efficacy and toxicity profiling of a potential nitrofuranyl methyl piperazine derivative IIIM-MCD-211 for oral tuberculosis therapy via in-silico-in-vitro-in-vivo approach. Pulmonary Pharmacology & Therapeutics. PMID 29174840 DOI: 10.1016/J.Pupt.2017.11.006  0.425
2017 Sharma R, Gatchie L, Williams IS, Jain SK, Vishwakarma RA, Chaudhuri B, Bharate SB. Glycyrrhiza glabra extract and quercetin reverses cisplatin resistance in triple-negative MDA-MB-468 breast cancer cells via inhibition of cytochrome P450 1B1 enzyme. Bioorganic & Medicinal Chemistry Letters. PMID 29150398 DOI: 10.1016/J.Bmcl.2017.11.013  0.788
2017 Singh U, Chashoo G, Khan SU, Mahajan P, Nargotra A, Mahajan G, Singh A, Sharma A, Mintoo MJ, Guru SK, Aruri H, Thatikonda T, Sahu P, Chibber P, Kumar V, ... ... Vishwakarma RA, et al. Design of Novel 3-Pyrimidinylazaindole based CDK2/9 Inhibitors with Potent In-vitro and In-vivo Antitumor Efficacy in a Triple-Negative Breast Cancer Model. Journal of Medicinal Chemistry. PMID 29144137 DOI: 10.1021/Acs.Jmedchem.7B00663  0.434
2017 Sharma N, Kumar A, Sharma PR, Qayum A, Singh SK, Dutt P, Paul S, Gupta V, Verma MK, Satti NK, Vishwakarma R. A new clerodane furano diterpene glycoside from Tinospora cordifolia triggers autophagy and apoptosis in HCT-116 colon cancer cells. Journal of Ethnopharmacology. PMID 28962889 DOI: 10.1016/J.Jep.2017.09.034  0.378
2017 Singh R, Kumar V, Bharate SS, Vishwakarma RA. Synthesis, pH dependent, plasma and enzymatic stability of bergenin prodrugs for potential use against rheumatoid arthritis. Bioorganic & Medicinal Chemistry. PMID 28843845 DOI: 10.1016/J.Bmc.2017.08.011  0.396
2017 Williams IS, Chib S, Nuthakki V, Gatchie L, Joshi P, Narkhede N, Vishwakarma RA, Bharate SB, Saran S, Chaudhuri B. Biotransformation of chrysin to baicalein: Selective C6-hydroxylation of 5,7-dihydroxyflavone using whole yeast cells stably expressing human CYP1A1 enzyme. Journal of Agricultural and Food Chemistry. PMID 28782952 DOI: 10.1021/Acs.Jafc.7B02690  0.716
2017 Williams IS, Joshi P, Gatchie L, Sharma M, Satti NK, Vishwakarma RA, Chaudhuri B, Bharate SB. Synthesis and biological evaluation of pyrrole-based chalcones as CYP1 enzyme inhibitors, for possible prevention of cancer and overcoming cisplatin resistance. Bioorganic & Medicinal Chemistry Letters. PMID 28711350 DOI: 10.1016/J.Bmcl.2017.07.010  0.713
2017 Joshi P, Vishwakarma RA, Bharate SB. Natural alkaloids as P-gp inhibitors for multidrug resistance reversal in cancer. European Journal of Medicinal Chemistry. 138: 273-292. PMID 28675836 DOI: 10.1016/J.Ejmech.2017.06.047  0.678
2017 Nissar AU, Sharma L, Mudasir MA, Nazir LA, Umar SA, Sharma PR, Vishwakarma RA, Tasduq SA. Chemical chaperone 4-phenyl butyric acid (4PBA) reduces hepatocellular lipid accumulation and lipotoxicity through induction of autophagy. Journal of Lipid Research. PMID 28655725 DOI: 10.1194/Jlr.M077537  0.385
2017 Magotra A, Sharma A, Gupta AP, Wazir P, Sharma S, Singh PP, Tikoo MK, Vishwakarma RA, Singh G, Nandi U. Development and validation of a highly sensitive LC-ESI-MS/MS method for estimation of IIIM-MCD-211, a novel nitrofuranyl methyl piperazine derivative with potential activity against tuberculosis: Application to drug development. Journal of Chromatography. B, Analytical Technologies in the Biomedical and Life Sciences. 1060: 200-206. PMID 28623772 DOI: 10.1016/J.Jchromb.2017.06.015  0.389
2017 Sharma R, Jamwal V, Singh VP, Wazir P, Awasthi P, Singh D, Gandhi SG, Vishwakarma RA, Chaubey A. Revelation and cloning of valinomycin synthetase genes in Streptomyces lavendulae ACR-DA1 and their expression analysis under different fermentation and elicitation conditions. Journal of Biotechnology. PMID 28528783 DOI: 10.1016/J.Jbiotec.2017.05.008  0.407
2017 Joshi P, McCann GJP, Sonawane V, Vishwakarma RA, Chaudhuri B, Bharate SB. Identification of Potent and Selective CYP1A1 Inhibitors via Combined Ligand and Structure Based Virtual Screening and their In-vitro Validation in Sacchrosomes and Live human cells. Journal of Chemical Information and Modeling. PMID 28489395 DOI: 10.1021/Acs.Jcim.7B00095  0.699
2017 Batarseh YS, Bharate SS, Kumar V, Kumar A, Vishwakarma RA, Bharate SB, Kaddoumi A. Crocus sativus extract tighten the blood-brain barrier, reduces amyloid-β load and related toxicity in 5XFAD mice. Acs Chemical Neuroscience. PMID 28471166 DOI: 10.1021/Acschemneuro.7B00101  0.65
2017 Wadhwa B, Makhdoomi U, Vishwakarma R, Malik F. Protein kinase B: emerging mechanisms of isoform-specific regulation of cellular signaling in cancer. Anti-Cancer Drugs. PMID 28379898 DOI: 10.1097/Cad.0000000000000496  0.371
2017 Ahmad M, Aga MA, Bhat JA, Kumar B, Rouf A, Capalash N, Mintoo MJ, Kumar A, Mahajan P, Mondhe DM, Nargotra A, Sharma PR, Zargar MA, Vishwakarma RA, Shah BA, et al. Exploring derivatives of quinazoline alkaloid l-vasicine as cap groups in the design and biological mechanistic evaluation of novel antitumor histone deacetylase inhibitors. Journal of Medicinal Chemistry. PMID 28368585 DOI: 10.1021/Acs.Jmedchem.7B00322  0.422
2017 Vishwakarma R. Editorial: Medicinal Chemistry Research in India. Acs Medicinal Chemistry Letters. 8: 270-272. PMID 28337313 DOI: 10.1021/Acsmedchemlett.7B00064  0.313
2017 Baba SA, Vishwakarma RA, Ashraf N. Functional characterization of CsBGlu12, a β-glucosidase from Crocus sativus provides insights into its role in abiotic stress through accumulation of antioxidant flavonols. The Journal of Biological Chemistry. PMID 28154174 DOI: 10.1074/Jbc.M116.762161  0.389
2017 Singh A, Arvinda S, Singh S, Suri J, Koul S, Mondhe DM, Singh G, Vishwakarma R. IN0523 (Urs-12-ene-3α,24β-diol) a plant based derivative of boswellic acid protect Cisplatin induced urogenital toxicity. Toxicology and Applied Pharmacology. PMID 28122196 DOI: 10.1016/J.Taap.2017.01.011  0.392
2017 Kumar V, Gupta M, Gandhi SG, Bharate SS, Kumar A, Vishwakarma RA, Bharate SB. Anti-inflammatory chromone alkaloids and glycoside from Dysoxylum binectariferum Tetrahedron Letters. 58: 3974-3978. DOI: 10.1016/J.Tetlet.2017.09.005  0.617
2017 Razdan S, Bhat WW, Dhar N, Rana S, Pandith SA, Wani TA, Vishwakarma R, Lattoo SK. Molecular characterization of DWF1 from Withania somnifera (L.) Dunal: its implications in withanolide biosynthesis Journal of Plant Biochemistry and Biotechnology. 26: 52-63. DOI: 10.1007/S13562-016-0359-5  0.396
2016 Aruri H, Singh U, Kumar M, Sharma S, Aithagani SK, Gupta VK, Mignani S, Vishwakarma RA, Singh PP. Metal-free Cross-Dehydrogenative Coupling of HN-azoles with alpha-C(sp3)-H amides via C-H activation and its Mechanistic and Application studies. The Journal of Organic Chemistry. PMID 28013543 DOI: 10.1021/Acs.Joc.6B02448  0.405
2016 Saneja A, Nayak D, Srinivas M, Kumar A, Khare V, Katoch A, Goswami A, Vishwakarma RA, Sawant SD, Gupta PN. Development and mechanistic insight into enhanced cytotoxic potential of hyaluronic acid conjugated nanoparticles in CD44 overexpressing cancer cells. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 27989859 DOI: 10.1016/J.Ejps.2016.10.028  0.379
2016 Qadri M, Nalli Y, Jain SK, Chaubey A, Ali A, Strobel GA, Vishwakarma RA, Riyaz-Ul-Hassan S. An Insight into the Secondary Metabolism of Muscodor yucatanensis: Small-Molecule Epigenetic Modifiers Induce Expression of Secondary Metabolism-Related Genes and Production of New Metabolites in the Endophyte. Microbial Ecology. PMID 27924400 DOI: 10.1007/S00248-016-0901-Y  0.785
2016 Joshi P, Gupta M, Vishwakarma RA, Kumar A, Bharate SB. (Z)-2-(3-Chlorobenzylidene)-3,4-dihydro-N-(2-methoxyethyl)-3-oxo-2H-benzo[b][1,4]oxazine-6-carboxamide as GSK-3β inhibitor: Identification by virtual screening, and its validation in enzyme and cell-based assay. Chemical Biology & Drug Design. PMID 27896926 DOI: 10.1111/Cbdd.12913  0.683
2016 Pathania AS, Guru SK, Kumar S, Kumar A, Ahmad M, Bhushan S, Sharma PR, Mahajan P, Shah BA, Sharma S, Nargotra A, Vishwakarma R, Korkaya H, Malik F. Interplay between cell cycle and autophagy induced by boswellic acid analog. Scientific Reports. 6: 33146. PMID 27680387 DOI: 10.1038/Srep33146  0.409
2016 Yedukondalu N, Arora P, Wadhwa B, Malik FA, Vishwakarma RA, Gupta VK, Riyaz-Ul-Hassan S, Ali A. Diapolic acid A-B from an endophytic fungus, Diaporthe terebinthifolii depicting antimicrobial and cytotoxic activity. The Journal of Antibiotics. PMID 27599766 DOI: 10.1038/Ja.2016.109  0.392
2016 Padala AK, Wani A, Vishwakarma RA, Kumar A, Bharate SB. Functional induction of P-glycoprotein efflux pump by phenyl benzenesulfonamides: Synthesis and biological evaluation of T0901317 analogs. European Journal of Medicinal Chemistry. 122: 744-755. PMID 27497733 DOI: 10.1016/J.Ejmech.2016.07.005  0.69
2016 Yadav RR, Guru SK, Joshi P, Mahajan G, Mintoo MJ, Kumar V, Bharate SS, Mondhe DM, Vishwakarma RA, Bhushan S, Bharate SB. 6-Aryl substituted 4-(4-cyanomethyl) phenylamino quinazolines as a new class of isoform-selective PI3K-alpha inhibitors. European Journal of Medicinal Chemistry. 122: 731-743. PMID 27479483 DOI: 10.1016/J.Ejmech.2016.07.006  0.7
2016 Awasthi P, Gupta AP, Bedi YS, Vishwakarma RA, Gandhi SG. Mannitol Stress Directs Flavonoid Metabolism toward Synthesis of Flavones via Differential Regulation of Two Cytochrome P450 Monooxygenases in Coleus forskohlii. Frontiers in Plant Science. 7: 985. PMID 27458469 DOI: 10.3389/Fpls.2016.00985  0.409
2016 Kaur T, Bhat R, Khajuria M, Vyas R, Kumari A, Nadda G, Vishwakarma R, Vyas D. Dynamics of glucosinolate-myrosinase system during Plutella xylostella interaction to a novel host Lepidium latifolium L. Plant Science : An International Journal of Experimental Plant Biology. 250: 1-9. PMID 27457978 DOI: 10.1016/J.Plantsci.2016.05.012  0.364
2016 Gopalakrishna Pillai GK, Bharate SS, Awasthi A, Verma R, Mishra G, Singh AT, Jaggi M, Mithal A, Vishwakarma RA. Antidiabeticpotential of polyherbal formulation DB14201: Preclinical development, safety and efficacy studies. Journal of Ethnopharmacology. PMID 27457691 DOI: 10.1016/J.Jep.2016.07.062  0.349
2016 Kour G, Kumar A, Singh PP, Sharma S, Bhagat A, Vishwakarma RA, Ahmed Z. Preclinical comprehensive physicochemical and pharmacokinetic profiling of novel nitroimidazole derivative IIIM-019 - A potential oral treatment for tuberculosis. Pulmonary Pharmacology & Therapeutics. PMID 27457685 DOI: 10.1016/J.Pupt.2016.06.009  0.436
2016 Aruri H, Singh U, Kumar S, Kushwaha M, Gupta AP, Vishwakarma RA, Singh PP. I2/Aqueous TBHP-Catalyzed Coupling of Amides with Methylarenes/Aldehydes/Alcohols: Metal-Free Synthesis of Imides. Organic Letters. PMID 27434140 DOI: 10.1021/Acs.Orglett.6B01684  0.375
2016 Kumar V, Bharate SS, Vishwakarma RA. Modulating lipophilicity of rohitukine via prodrug approach: Preparation, characterization, and in vitro enzymatic hydrolysis in biorelevant media. European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 27422078 DOI: 10.1016/J.Ejps.2016.07.010  0.419
2016 Kumar V, Guru SK, Jain SK, Joshi P, Gandhi SG, Bharate SB, Bhushan S, Bharate SS, Vishwakarma RA. A chromatography-free isolation of rohitukine from leaves of Dysoxylum binectariferum: Evaluation for in vitro cytotoxicity, Cdk inhibition and physicochemical properties. Bioorganic & Medicinal Chemistry Letters. PMID 27363938 DOI: 10.1016/J.Bmcl.2016.06.046  0.801
2016 Aithagani SK, Kumar M, Yadav M, Vishwakarma RA, Singh PP. Metal-free, Phosphonium Salt-Mediated Sulfoximination of Azine N-oxides: Approach for the Synthesis of N-azine Sulfoximines. The Journal of Organic Chemistry. PMID 27304317 DOI: 10.1021/Acs.Joc.6B00593  0.386
2016 Gupta S, Kaul S, Singh B, Vishwakarma RA, Dhar MK. Production of Gentisyl Alcohol from Phoma herbarum Endophytic in Curcuma longa L. and Its Antagonistic Activity Towards Leaf Spot Pathogen Colletotrichum gloeosporioides. Applied Biochemistry and Biotechnology. PMID 27288000 DOI: 10.1007/S12010-016-2154-0  0.535
2016 Sharma R, Singh VP, Singh D, Yusuf F, Kumar A, Vishwakarma RA, Chaubey A. Optimization of nonribosomal peptides production by a psychrotrophic fungus: Trichoderma velutinum ACR-P1. Applied Microbiology and Biotechnology. PMID 27287849 DOI: 10.1007/S00253-016-7622-5  0.386
2016 Pandith SA, Dhar N, Rana S, Bhat WW, Kushwaha M, Gupta AP, Shah MA, Vishwakarma R, Lattoo SK. Characterization and functional promiscuity of two divergent paralogs of Type III plant polyketide synthases from Rheum emodi Wall ex. Meissn. Plant Physiology. PMID 27268960 DOI: 10.1104/pp.16.00003  0.297
2016 Bharate SB, Singh B, Kachler S, Oliveira A, Kumar V, Bharate SS, Vishwakarma RA, Klotz KN, Gutiérrez-de-Terán H. Discovery of 7-(prolinol-N-yl)-2-phenylamino-thiazolo[5,4-d]pyrimidines as novel non-nucleoside partial agonists for the A2A adenosine receptor: Prediction from molecular modeling. Journal of Medicinal Chemistry. PMID 27227326 DOI: 10.1021/Acs.Jmedchem.6B00552  0.715
2016 Bharate SS, Kumar V, Vishwakarma RA. Determining Partition Coefficient (Log P), Distribution Coefficient (Log D) and Ionization Constant (pKa) in Early Drug Discovery. Combinatorial Chemistry & High Throughput Screening. PMID 27137915 DOI: 10.2174/1386207319666160502123917  0.405
2016 Thatikonda T, Singh U, Ambala S, Vishwakarma RA, Singh PP. Metal free C-H functionalization of diazines and related heteroarenes with organoboron species and its application in the synthesis of a CDK inhibitor. Organic & Biomolecular Chemistry. PMID 27086946 DOI: 10.1039/C6Ob00526H  0.399
2016 Sharma N, Kumar C, Dutt P, Gupta S, Satti NK, Chandra S, Kitchlu S, Paul S, Vishwakarma RA, Verma MK. Isolation, Chemical Fingerprinting and Simultaneous Quantification of Four Compounds from Tanacetum gracile Using a Validated HPLC-ESI-QTOF-Mass Spectrometry Method. Journal of Chromatographic Science. PMID 26951542 DOI: 10.1093/Chromsci/Bmw013  0.409
2016 Kour G, Chandan BK, Khullar M, Munagala G, Singh PP, Bhagat A, Gupta AP, Vishwakarma RA, Ahmed Z. Development and validation of a highly sensitive LC-MS/MS-ESI method for quantification of IIIM-019-A novel nitroimidazole derivative with promising action against Tuberculosis: Application to drug development. Journal of Pharmaceutical and Biomedical Analysis. 124: 26-33. PMID 26922579 DOI: 10.1016/J.Jpba.2016.02.027  0.374
2016 Hussain A, Qazi AK, Mupparapu N, Guru SK, Kumar A, Sharma PR, Singh SK, Singh P, Dar MJ, Bharate SB, Zargar MA, Ahmed QN, Bhushan S, Vishwakarma RA, Hamid A. Modulation of glycolysis and lipogenesis by novel PI3K selective molecule represses tumor angiogenesis and decreases colorectal cancer growth. Cancer Letters. PMID 26921131 DOI: 10.1016/J.Canlet.2016.02.030  0.664
2016 Mehra R, Rani C, Mahajan P, Vishwakarma RA, Khan IA, Nargotra A. Computationally Guided Identification of Novel Mycobacterium tuberculosis GlmU Inhibitory Leads, Their Optimization, and in Vitro Validation. Acs Combinatorial Science. PMID 26812086 DOI: 10.1021/Acscombsci.5B00019  0.434
2016 Hussain A, Qazi AK, Mupparapu N, Kumar A, Mintoo MJ, Mahajan G, Sharma PR, Singh SK, Bharate SB, Zargar MA, Ahmed QN, Mondhe DM, Vishwakarma RA, Hamid A. A novel PI3K axis selective molecule exhibits potent tumor inhibition in colorectal carcinogenesis. Molecular Carcinogenesis. PMID 26764221 DOI: 10.1002/Mc.22457  0.687
2016 Manda S, Wani A, Bharate SS, Vishwakarma RA, Kumar A, Bharate SB. Design, synthesis and P-gp induction activity of aryl phosphonate esters: identification of tetraethyl-2-phenylethene-1,1-diyldiphosphonate as an orally bioavailable P-gp inducer Medchemcomm. 7: 1910-1915. DOI: 10.1039/C6Md00300A  0.592
2016 Meena S, Singh R, Vishwakarma RA, Aga MA, Jain SK. SeO2 mediated efficient synthesis of amides and α-ketoamides of secondary amines with wide substrate scope Tetrahedron Letters. 57: 3715-3717. DOI: 10.1016/J.Tetlet.2016.06.129  0.761
2016 Singh S, Munagala G, Reddy K, Bhola S, Chib R, Sharma R, Rani C, Singh P, Vishwakarma R, Khan I. Biological evaluation of a novel nitroimidazooxazole derivative, IIIM-MCD-019 against Mycobacterium tuberculosis and its in vivo efficacy International Journal of Infectious Diseases. 45: 414. DOI: 10.1016/J.Ijid.2016.02.883  0.356
2016 Magotra A, Nalli Y, Kushwaha M, Raina C, Gupta AP, Ali A, Vishwakarma RA, Chaubey A. An efficient liquid chromatography-tandem mass spectrometry method for the quantification of borrelidin from Streptomyces rochei (ATCC 10739) Journal of Chemical Technology and Biotechnology. 91: 198-203. DOI: 10.1002/Jctb.4562  0.374
2016 Sharma R, Vishwakarma RA, Bharate SB. Bimetallic Cu–Mn‐Catalyzed Synthesis of 2‐Arylquinazolin‐4(3H)‐ones: Aqueous Ammonia as Source of a Ring Nitrogen Atom European Journal of Organic Chemistry. 2016: 5227-5233. DOI: 10.1002/Ejoc.201601024  0.583
2016 Sharma R, Vishwakarma RA, Bharate SB. Ligand-Free Copper-Manganese Spinel Oxide-Catalyzed Tandem One-Pot C-H Amidation andN-Arylation of Benzylamines: A Facile Access to 2-Arylquinazolin-4(3H)-ones Advanced Synthesis & Catalysis. 358: 3027-3033. DOI: 10.1002/Adsc.201600549  0.576
2015 Khan S, Pandotra P, Manzoor MM, Kushwaha M, Sharma R, Jain S, Ahuja A, Amancha V, Bhushan S, Guru SK, Gupta AP, Vishwakarma R, Gupta S. Terpenoid and flavonoid spectrum of in vitro cultures of revealed high chemical heterogeneity: platform to understand biosynthesis. Plant Cell, Tissue and Organ Culture. 124: 507-516. PMID 32214564 DOI: 10.1007/s11240-015-0910-4  0.331
2015 Awasthi P, Mahajan V, Rather IA, Gupta AP, Rasool S, Bedi YS, Vishwakarma RA, Gandhi SG. Plant Omics: Isolation, Identification, and Expression Analysis of Cytochrome P450 Gene Sequences from Coleus forskohlii. Omics : a Journal of Integrative Biology. 19: 782-92. PMID 26669713 DOI: 10.1089/omi.2015.0148  0.289
2015 Dhar N, Razdan S, Rana S, Bhat WW, Vishwakarma R, Lattoo SK. A Decade of Molecular Understanding of Withanolide Biosynthesis and In vitro Studies in Withania somnifera (L.) Dunal: Prospects and Perspectives for Pathway Engineering. Frontiers in Plant Science. 6: 1031. PMID 26640469 DOI: 10.3389/Fpls.2015.01031  0.407
2015 Sharma R, Patel N, Vishwakarma RA, Bharatam PV, Bharate SB. Metal-free oxidative cyclization of acetophenones with diamines: a facile access to phenylpyridines. Chemical Communications (Cambridge, England). PMID 26593387 DOI: 10.1039/C5Cc08498A  0.666
2015 Saikam V, Dara S, Yadav M, Singh PP, Vishwakarma RA. Dimethyltin dichloride catalyzed regio-selective alkylation of cis-1,2-diols at room temperature. The Journal of Organic Chemistry. PMID 26569335 DOI: 10.1021/Acs.Joc.5B01898  0.361
2015 Aithagani SK, Dara S, Munagala G, Aruri H, Yadav M, Sharma S, Vishwakarma RA, Singh PP. Metal-Free Approach for the Synthesis of N-Aryl Sulfoximines via Aryne Intermediate. Organic Letters. PMID 26562479 DOI: 10.1021/Acs.Orglett.5B02804  0.367
2015 Manda S, Sharma S, Wani A, Joshi P, Kumar V, Guru SK, Bharate SS, Bhushan S, Vishwakarma RA, Kumar A, Bharate SB. Discovery of a marine-derived bis-indole alkaloid fascaplysin, as a new class of potent P-glycoprotein inducer and establishment of its structure-activity relationship. European Journal of Medicinal Chemistry. 107: 1-11. PMID 26560048 DOI: 10.1016/J.Ejmech.2015.10.049  0.695
2015 Yempalla KR, Munagala G, Singh S, Kour G, Sharma S, Chib R, Kumar S, Wazir P, Singh GD, Raina S, Bharate SS, Khan IA, Vishwakarma RA, Singh PP. Synthesis and Biological Evaluation of Polar Functionalities Containing Nitrodihydroimidazooxazoles as Anti-TB Agents. Acs Medicinal Chemistry Letters. 6: 1059-64. PMID 26487912 DOI: 10.1021/Acsmedchemlett.5B00202  0.439
2015 Yempalla KR, Munagala G, Singh S, Magotra A, Kumar S, Rajput VS, Bharate SS, Tikoo M, Singh GD, Khan IA, Vishwakarma RA, Singh PP. Nitrofuranyl Methyl Piperazines as New Anti-TB Agents: Identification, Validation, Medicinal Chemistry, and PK Studies. Acs Medicinal Chemistry Letters. 6: 1041-6. PMID 26487909 DOI: 10.1021/Acsmedchemlett.5B00141  0.445
2015 Sharma R, Vishwakarma RA, Bharate SB. An efficient transformation of furano-hydroxychalcones to furanoflavones via base mediated intramolecular tandem O-arylation and C-O bond cleavage: a new approach for the synthesis of furanoflavones. Organic & Biomolecular Chemistry. PMID 26426474 DOI: 10.1039/C5Ob01802A  0.663
2015 Ambala S, Thatikonda T, Sharma S, Munagala G, Yempalla KR, Vishwakarma RA, Singh PP. Cross-dehydrogenative coupling of α-C(sp(3))-H of ethers/alkanes with C(sp(2))-H of heteroarenes under metal-free conditions. Organic & Biomolecular Chemistry. PMID 26419479 DOI: 10.1039/C5Ob01268F  0.395
2015 Singh B, Jain SK, Bharate SB, Kushwaha M, Gupta AP, Vishwakarma RA. Simultaneous Quantification of Five Bioactive Flavonoids in High Altitude Plant Actinocarya tibetica by LC-ESI-MS/MS. Journal of Aoac International. 98: 907-12. PMID 26268971 DOI: 10.5740/Jaoacint.14-270  0.77
2015 Khazir J, Riley DL, Chashoo G, Mir BA, Liles D, Islam MA, Singh SK, Vishwakarma RA, Pilcher LA. Design, synthesis and anticancer activity of Michael-type thiol adducts of α-santonin analogue with exocyclic methylene. European Journal of Medicinal Chemistry. 101: 769-779. PMID 26222449 DOI: 10.1016/J.Ejmech.2015.07.022  0.47
2015 Qadri M, Deshidi R, Shah BA, Bindu K, Vishwakarma RA, Riyaz-Ul-Hassan S. An endophyte of Picrorhiza kurroa Royle ex. Benth, producing menthol, phenylethyl alcohol and 3-hydroxypropionic acid, and other volatile organic compounds. World Journal of Microbiology & Biotechnology. 31: 1647-54. PMID 26220851 DOI: 10.1007/S11274-015-1910-6  0.405
2015 Venkateswarlu V, Pathania AS, Aravinda Kumar KA, Mahajan P, Nargotra A, Vishwakarma RA, Malik FA, Sawant SD. 4-(N-Phenyl-N'-substituted benzenesulfonyl)-6-(4-hydroxyphenyl)quinolines as inhibitors of mammalian target of rapamycin. Bioorganic & Medicinal Chemistry. 23: 4237-47. PMID 26162498 DOI: 10.1016/J.Bmc.2015.06.046  0.468
2015 Sinha S, Amin H, Nayak D, Bhatnagar M, Kacker P, Chakraborty S, Kitchlu S, Vishwakarma R, Goswami A, Ghosal S. Assessment of microtubule depolymerization property of flavonoids isolated from Tanacetum gracile in breast cancer cells by biochemical and molecular docking approach. Chemico-Biological Interactions. 239: 1-11. PMID 26115782 DOI: 10.1016/J.Cbi.2015.06.034  0.45
2015 Venkateswarlu V, Aravinda Kumar KA, Gupta S, Singh D, Vishwakarma RA, Sawant SD. DMSO/I2 mediated C-C bond cleavage of α-ketoaldehydes followed by C-O bond formation: a metal-free approach for one-pot esterification. Organic & Biomolecular Chemistry. PMID 26110656 DOI: 10.1039/C5Ob01015B  0.395
2015 Bharate JB, Abbat S, Bharatam PV, Vishwakarma RA, Bharate SB. CuBr catalyzed aerobic oxidative coupling of 2-aminopyridines with cinnamaldehydes: direct access to 3-formyl-2-phenyl-imidazo[1,2-a]pyridines. Organic & Biomolecular Chemistry. 13: 7790-4. PMID 26103156 DOI: 10.1039/C5Ob00776C  0.675
2015 Mohammed S, Vishwakarma RA, Bharate SB. Iodine Catalyzed Oxidative Synthesis of Quinazolin-4(3H)-ones and Pyrazolo[4,3-d]pyrimidin-7(6H)-ones via Amination of sp3 C-H Bond Journal of Organic Chemistry. 80: 6915-6921. PMID 26067767 DOI: 10.1021/Acs.Joc.5B00989  0.677
2015 Yadav RR, Sharma S, Joshi P, Wani A, Vishwakarma RA, Kumar A, Bharate SB. Meridianin derivatives as potent Dyrk1A inhibitors and neuroprotective agents. Bioorganic & Medicinal Chemistry Letters. 25: 2948-52. PMID 26048785 DOI: 10.1016/J.Bmcl.2015.05.034  0.715
2015 Yadav RR, Khan SI, Singh S, Khan IA, Vishwakarma RA, Bharate SB. Synthesis, antimalarial and antitubercular activities of meridianin derivatives. European Journal of Medicinal Chemistry. 98: 160-9. PMID 26005918 DOI: 10.1016/J.Ejmech.2015.05.020  0.705
2015 Guru SK, Pathania AS, Kumar S, Ramesh D, Kumar M, Rana S, Kumar A, Malik F, Sharma PR, Chandan BK, Jaglan S, Sharma JP, Shah BA, Tasduq SA, Lattoo SK, ... ... Vishwakarma RA, et al. Secalonic Acid-D Represses HIF1α/VEGF-Mediated Angiogenesis by Regulating the Akt/mTOR/p70S6K Signaling Cascade. Cancer Research. 75: 2886-96. PMID 25977334 DOI: 10.1158/0008-5472.Can-14-2312  0.416
2015 Mahale S, Bharate SB, Manda S, Joshi P, Jenkins PR, Vishwakarma RA, Chaudhuri B. Antitumour potential of BPT: a dual inhibitor of cdk4 and tubulin polymerization. Cell Death & Disease. 6: e1743. PMID 25950473 DOI: 10.1038/Cddis.2015.96  0.612
2015 Raghupathy R, Anilkumar AA, Polley A, Singh PP, Yadav M, Johnson C, Suryawanshi S, Saikam V, Sawant SD, Panda A, Guo Z, Vishwakarma RA, Rao M, Mayor S. Transbilayer lipid interactions mediate nanoclustering of lipid-anchored proteins. Cell. 161: 581-94. PMID 25910209 DOI: 10.1016/J.Cell.2015.03.048  0.331
2015 Singh B, Kumar A, Joshi P, Guru SK, Kumar S, Wani ZA, Mahajan G, Hussain A, Qazi AK, Kumar A, Bharate SS, Gupta BD, Sharma PR, Hamid A, Saxena AK, ... ... Vishwakarma RA, et al. Colchicine derivatives with potent anticancer activity and reduced P-glycoprotein induction liability. Organic & Biomolecular Chemistry. 13: 5674-89. PMID 25895604 DOI: 10.1039/C5Ob00406C  0.736
2015 Bharate JB, Batarseh YS, Wani A, Sharma S, Vishwakarma RA, Kaddoumi A, Kumar A, Bharate SB. Synthesis and P-glycoprotein induction activity of colupulone analogs. Organic & Biomolecular Chemistry. 13: 5488-96. PMID 25875530 DOI: 10.1039/C5Ob00554J  0.681
2015 Bharate JB, Singh S, Wani A, Sharma S, Joshi P, Khan IA, Kumar A, Vishwakarma RA, Bharate SB. Discovery of 4-acetyl-3-(4-fluorophenyl)-1-(p-tolyl)-5-methylpyrrole as a dual inhibitor of human P-glycoprotein and Staphylococcus aureus Nor A efflux pump. Organic & Biomolecular Chemistry. 13: 5424-31. PMID 25865846 DOI: 10.1039/C5Ob00246J  0.693
2015 Bharate JB, Abbat S, Sharma R, Bharatam PV, Vishwakarma RA, Bharate SB. Cobalt(II) catalyzed C(sp)-H bond functionalization of alkynes with phenyl hydrazines: facile access to diaryl 1,2-diketones. Organic & Biomolecular Chemistry. 13: 5235-42. PMID 25856782 DOI: 10.1039/C5Ob00419E  0.679
2015 Kumar S, Guru SK, Venkateswarlu V, Malik F, Vishwakarma RA, Sawant SD, Bhushan S. A novel quinolinebased second-generation mTOR inhibitor that induces apoptosis and disruptsPI3K-Akt-mTOR signaling in human leukemia HL-60 cells. Anti-Cancer Agents in Medicinal Chemistry. PMID 25832358 DOI: 10.2174/1871520615666150402093558  0.419
2015 Sawant SD, Lakshma Reddy G, Dar MI, Srinivas M, Gupta G, Sahu PK, Mahajan P, Nargotra A, Singh S, Sharma SC, Tikoo M, Singh G, Vishwakarma RA, Syed SH. Discovery of novel pyrazolopyrimidinone analogs as potent inhibitors of phosphodiesterase type-5. Bioorganic & Medicinal Chemistry. 23: 2121-8. PMID 25801159 DOI: 10.1016/J.Bmc.2015.03.005  0.462
2015 Mudududdla R, Guru SK, Wani A, Sharma S, Joshi P, Vishwakarma RA, Kumar A, Bhushan S, Bharate SB. 3-(Benzo[d][1,3]dioxol-5-ylamino)-N-(4-fluorophenyl)thiophene-2-carboxamide overcomes cancer chemoresistance via inhibition of angiogenesis and P-glycoprotein efflux pump activity. Organic & Biomolecular Chemistry. 13: 4296-309. PMID 25758415 DOI: 10.1039/C5Ob00233H  0.719
2015 Bharate SS, Vishwakarma RA. Thermodynamic equilibrium solubility measurements in simulated fluids by 96-well plate method in early drug discovery. Bioorganic & Medicinal Chemistry Letters. 25: 1561-7. PMID 25740159 DOI: 10.1016/J.Bmcl.2015.02.013  0.406
2015 Munagala G, Yempalla KR, Singh S, Sharma S, Kalia NP, Rajput VS, Kumar S, Sawant SD, Khan IA, Vishwakarma RA, Singh PP. Synthesis of new generation triazolyl- and isoxazolyl-containing 6-nitro-2,3-dihydroimidazooxazoles as anti-TB agents: in vitro, structure-activity relationship, pharmacokinetics and in vivo evaluation. Organic & Biomolecular Chemistry. 13: 3610-24. PMID 25670502 DOI: 10.1039/C5Ob00054H  0.448
2015 Ashraf N, Jain D, Vishwakarma RA. Identification, cloning and characterization of an ultrapetala transcription factor CsULT1 from Crocus: a novel regulator of apocarotenoid biosynthesis. Bmc Plant Biology. 15: 25. PMID 25640597 DOI: 10.1186/S12870-015-0423-7  0.387
2015 Aruri H, Singh U, Sharma S, Gudup S, Bhogal M, Kumar S, Singh D, Gupta VK, Kant R, Vishwakarma RA, Singh PP. Cross-dehydrogenative coupling of azoles with α-C(sp3)-H of ethers and thioethers under metal-free conditions: functionalization of H-N azoles via C-H activation. The Journal of Organic Chemistry. 80: 1929-36. PMID 25588073 DOI: 10.1021/Jo502477R  0.38
2015 Kumar S, Guru SK, Pathania AS, Manda S, Kumar A, Bharate SB, Vishwakarma RA, Malik F, Bhushan S. Fascaplysin induces caspase mediated crosstalk between apoptosis and autophagy through the inhibition of PI3K/AKT/mTOR signaling cascade in human leukemia HL-60 cells. Journal of Cellular Biochemistry. 116: 985-97. PMID 25561006 DOI: 10.1002/Jcb.25053  0.669
2015 Rather IA, Awasthi P, Mahajan V, Bedi YS, Vishwakarma RA, Gandhi SG. Molecular cloning and functional characterization of an antifungal PR-5 protein from Ocimum basilicum. Gene. 558: 143-51. PMID 25550044 DOI: 10.1016/J.Gene.2014.12.055  0.361
2015 Mupparapu N, Battini N, Battula S, Khan S, Vishwakarma RA, Ahmed QN. Aminocatalytic cross-coupling approach via iminium ions to different C - C Bonds. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 2954-60. PMID 25524296 DOI: 10.1002/Chem.201405477  0.37
2015 Anil Kumar K, Kannaboina P, Dhaked DK, Vishwakarma RA, Bharatam PV, Das P. Cu-catalyzed arylation of the amino group in the indazole ring: regioselective synthesis of pyrazolo-carbazoles. Organic & Biomolecular Chemistry. 13: 1481-91. PMID 25474646 DOI: 10.1039/C4Ob02044H  0.407
2015 Mahajan V, Sharma N, Kumar S, Bhardwaj V, Ali A, Khajuria RK, Bedi YS, Vishwakarma RA, Gandhi SG. Production of rohitukine in leaves and seeds of Dysoxylum binectariferum: an alternate renewable resource. Pharmaceutical Biology. 53: 446-50. PMID 25472605 DOI: 10.3109/13880209.2014.923006  0.388
2015 Aravinda Kumar KA, Venkateswarlu V, Vishwakarma RA, Sawant SD. A Metal-Free Approach to Carboxylic Acids by Oxidation of Alkyl, Aryl, or Heteroaryl Alkyl Ketones or Arylalkynes Synthesis (Germany). 47: 3161-3168. DOI: 10.1055/S-0034-1381026  0.393
2015 Venkateswarlu V, Balgotra S, Aravinda Kumar KA, Vishwakarma RA, Sawant SD. Metal-free chemoselective ortho -C(sp<sup>2</sup>)-F bond hydroxylation and N-trifluoroacylation of fluoroarylamines for domino synthesis of 2-(N-trifluoroacyl)aminophenols Synlett. 26: 1258-1262. DOI: 10.1055/S-0034-1379905  0.39
2015 Bharate JB, Vishwakarma RA, Bharate SB. Metal-free domino one-pot protocols for quinoline synthesis Rsc Advances. 5: 42020-42053. DOI: 10.1039/C5Ra07798B  0.557
2015 Mohammed S, Vishwakarma RA, Bharate SB. Metal-free DBU promoted regioselective synthesis of isoxazoles and isoxazolines Rsc Advances. 5: 3470-3473. DOI: 10.1039/C4Ra14694H  0.586
2015 Sharma R, Guru SK, Jain SK, Pathania AS, Vishwakarma RA, Bhushan S, Bharate SB. 3-(2,6-Dichloro-benzyloxy)-11-oxo-olean-12-ene-29-oic acid, a semisynthetic derivative of glycyrrhetic acid: synthesis, antiproliferative, apoptotic and anti-angiogenesis activity Medchemcomm. 6: 564-575. DOI: 10.1039/C4Md00344F  0.805
2015 Srinivas M, Hudwekar AD, Venkateswarlu V, Reddy GL, Kumar KAA, Vishwakarma RA, Sawant SD. A metal-free approach for transamidation of amides with amines in aqueous media Tetrahedron Letters. 56: 4775-4779. DOI: 10.1016/J.Tetlet.2015.06.052  0.396
2015 Balgotra S, Venkateswarlu V, Vishwakarma RA, Sawant SD. Direct C-N bond cleavage of N-vinyl or N-allyl arylamines: A metal-free strategy for N-devinylation and N-deallylation Tetrahedron Letters. 56: 4289-4292. DOI: 10.1016/J.Tetlet.2015.05.042  0.366
2015 Sharma R, Abbat S, Mudududdla R, Vishwakarma RA, Bharatam PV, Bharate SB. ortho-Quinone methides: TFA-mediated generation in water and trapping with lactams and styrenes Tetrahedron Letters. 56: 4057-4059. DOI: 10.1016/J.Tetlet.2015.04.072  0.589
2015 Mupparapu N, Vishwakarma RA, Ahmed QN. Iodine-DMSO promoted C–H (SP3) functionalization approach to α-ketoamides Tetrahedron. 71: 3417-3421. DOI: 10.1016/J.Tet.2015.03.088  0.387
2015 Khan S, Pandotra P, Manzoor MM, Kushwaha M, Sharma R, Jain S, Ahuja A, Amancha V, Bhushan S, Guru SK, Gupta AP, Vishwakarma R, Gupta S. Terpenoid and flavonoid spectrum of in vitro cultures of Glycyrrhiza glabra revealed high chemical heterogeneity: platform to understand biosynthesis Plant Cell, Tissue and Organ Culture. 1-10. DOI: 10.1007/S11240-015-0910-4  0.765
2015 Yadav M, Dara S, Saikam V, Kumar M, Aithagani SK, Paul S, Vishwakarma RA, Singh PP. Regioselective Oxidative C-H Phosphonation of Imidazo[1,2-a]pyridines and Related Heteroarenes Mediated by Manganese(III) Acetate European Journal of Organic Chemistry. 2015: 6526-6533. DOI: 10.1002/Ejoc.201500984  0.41
2015 Padala AK, Mupparapu N, Singh D, Vishwakarma RA, Ahmed QN. α‐Carbonylimine to α‐Carbonylamide: An Efficient Oxidative Amidation Approach European Journal of Organic Chemistry. 2015: 3577-3586. DOI: 10.1002/Ejoc.201500251  0.43
2014 Kumar S, Guru SK, Pathania AS, Mupparapu N, Kumar A, Malik F, Bharate SB, Naveed Ahmed Q, Vishwakarma RA, Bhushan S. A novel quinazolinone derivative induces cytochrome c interdependent apoptosis and autophagy in human leukemia MOLT-4 cells. Toxicology Reports. 1: 1013-1025. PMID 28962314 DOI: 10.1016/J.Toxrep.2014.07.018  0.674
2014 Bharate JB, Vishwakarma RA, Bharate SB, Kushwaha M, Gupta AP. Quantification of the Polyisoprenylated Benzophenones Garcinol and Isogarcinol Using Multiple Reaction Monitoring LC/Electrospray Ionization-MS/MS Analysis of Ultrasound-Assisted Extracts of Garcinia indica Fruits. Journal of Aoac International. 97: 1317-22. PMID 25902981 DOI: 10.5740/Jaoacint.13-137  0.566
2014 Rana S, Bhat WW, Dhar N, Pandith SA, Razdan S, Vishwakarma R, Lattoo SK. Molecular characterization of two A-type P450s, WsCYP98A and WsCYP76A from Withania somnifera (L.) Dunal: expression analysis and withanolide accumulation in response to exogenous elicitations. Bmc Biotechnology. 14: 89. PMID 25416924 DOI: 10.1186/S12896-014-0089-5  0.37
2014 Pathania AS, Kumar S, Guru SK, Bhushan S, Sharma PR, Aithagani SK, Singh PP, Vishwakarma RA, Kumar A, Malik F. The synthetic tryptanthrin analogue suppresses STAT3 signaling and induces caspase dependent apoptosis via ERK up regulation in human leukemia HL-60 cells. Plos One. 9: e110411. PMID 25383546 DOI: 10.1371/Journal.Pone.0110411  0.409
2014 Mahale S, Bharate SB, Manda S, Joshi P, Bharate SS, Jenkins PR, Vishwakarma RA, Chaudhuri B. Biphenyl-4-carboxylic acid [2-(1H-indol-3-yl)-ethyl]-methylamide (CA224), a nonplanar analogue of fascaplysin, inhibits Cdk4 and tubulin polymerization: evaluation of in vitro and in vivo anticancer activity. Journal of Medicinal Chemistry. 57: 9658-72. PMID 25368960 DOI: 10.1021/Jm5014743  0.709
2014 Bharate JB, Bharate SB, Vishwakarma RA. Metal-free, ionic liquid-mediated synthesis of functionalized quinolines. Acs Combinatorial Science. 16: 624-30. PMID 25314670 DOI: 10.1021/Co500047W  0.588
2014 Singh B, Guru SK, Sharma R, Bharate SS, Khan IA, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis and anti-proliferative activities of new derivatives of embelin. Bioorganic & Medicinal Chemistry Letters. 24: 4865-70. PMID 25240254 DOI: 10.1016/J.Bmcl.2014.08.052  0.746
2014 Rao DN, Rasheed S, Vishwakarma RA, Das P. Copper-catalyzed sequential N-arylation of C-amino-NH-azoles. Chemical Communications (Cambridge, England). 50: 12911-4. PMID 25212901 DOI: 10.1039/C4Cc05628K  0.401
2014 Mudududdla R, Sharma R, Abbat S, Bharatam PV, Vishwakarma RA, Bharate SB. Synthesis of 2-phenylnaphthalenes from styryl-2-methoxybenzenes. Chemical Communications (Cambridge, England). 50: 12076-9. PMID 25163506 DOI: 10.1039/C4Cc05151C  0.684
2014 Jain SK, Singh S, Khajuria A, Guru SK, Joshi P, Meena S, Nadkarni JR, Singh A, Bharate SS, Bhushan S, Bharate SB, Vishwakarma RA. Pyrano-isochromanones as IL-6 inhibitors: synthesis, in vitro and in vivo antiarthritic activity. Journal of Medicinal Chemistry. 57: 7085-97. PMID 25111439 DOI: 10.1021/Jm500901E  0.797
2014 Jain SK, Aravinda Kumar KA, Bharate SB, Vishwakarma RA. Facile access to amides and hydroxamic acids directly from nitroarenes. Organic & Biomolecular Chemistry. 12: 6465-9. PMID 25019340 DOI: 10.1039/C4Ob01155D  0.774
2014 Bharate JB, Wani A, Sharma S, Reja SI, Kumar M, Vishwakarma RA, Kumar A, Bharate SB. Synthesis, and the antioxidant, neuroprotective and P-glycoprotein induction activity of 4-arylquinoline-2-carboxylates. Organic & Biomolecular Chemistry. 12: 6267-77. PMID 25007760 DOI: 10.1039/C4Ob00488D  0.711
2014 Manda S, Khan SI, Jain SK, Mohammed S, Tekwani BL, Khan IA, Vishwakarma RA, Bharate SB. Synthesis, antileishmanial and antitrypanosomal activities of N-substituted tetrahydro-β-carbolines. Bioorganic & Medicinal Chemistry Letters. 24: 3247-50. PMID 24980054 DOI: 10.1016/J.Bmcl.2014.06.030  0.7
2014 Bhat WW, Razdan S, Rana S, Dhar N, Wani TA, Qazi P, Vishwakarma R, Lattoo SK. A phenylalanine ammonia-lyase ortholog (PkPAL1) from Picrorhiza kurrooa Royle ex. Benth: molecular cloning, promoter analysis and response to biotic and abiotic elicitors. Gene. 547: 245-56. PMID 24979341 DOI: 10.1016/J.Gene.2014.06.046  0.389
2014 Jain SK, Meena S, Gupta AP, Kushwaha M, Uma Shaanker R, Jaglan S, Bharate SB, Vishwakarma RA. Dysoxylum binectariferum bark as a new source of anticancer drug camptothecin: bioactivity-guided isolation and LCMS-based quantification. Bioorganic & Medicinal Chemistry Letters. 24: 3146-9. PMID 24878199 DOI: 10.1016/J.Bmcl.2014.05.001  0.784
2014 Dara S, Saikam V, Yadav M, Singh PP, Vishwakarma RA. HClO4-silica-catalysed regioselective opening of benzylidene acetals and its application towards regioselective HO-4 glycosylation of benzylidene acetals in one-pot. Carbohydrate Research. 391: 93-6. PMID 24792317 DOI: 10.1016/J.Carres.2014.01.011  0.393
2014 Reddy GL, Guru SK, Srinivas M, Pathania AS, Mahajan P, Nargotra A, Bhushan S, Vishwakarma RA, Sawant SD. Synthesis of 5-substituted-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-one analogs and their biological evaluation as anticancer agents: mTOR inhibitors. European Journal of Medicinal Chemistry. 80: 201-8. PMID 24780597 DOI: 10.1016/J.Ejmech.2014.04.051  0.47
2014 Dhar N, Rana S, Razdan S, Bhat WW, Hussain A, Dhar RS, Vaishnavi S, Hamid A, Vishwakarma R, Lattoo SK. Cloning and functional characterization of three branch point oxidosqualene cyclases from Withania somnifera (L.) dunal. The Journal of Biological Chemistry. 289: 17249-67. PMID 24770414 DOI: 10.1074/Jbc.M114.571919  0.397
2014 Venkateswarlu V, Kumar KA, Balgotra S, Reddy GL, Srinivas M, Vishwakarma RA, Sawant SD. C-H oxygenation and N-trifluoroacylation of arylamines under metal-free conditions: a convenient approach to 2-aminophenols and N-trifluoroacyl-ortho-aminophenols. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 6641-5. PMID 24756872 DOI: 10.1002/Chem.201402411  0.397
2014 Zilla MK, Nayak D, Vishwakarma RA, Sharma PR, Goswami A, Ali A. A convergent synthesis of alkyne-azide cycloaddition derivatives of 4-α,β-2-propyne podophyllotoxin depicting potent cytotoxic activity. European Journal of Medicinal Chemistry. 77: 47-55. PMID 24607588 DOI: 10.1016/J.Ejmech.2014.02.030  0.46
2014 Qadri M, Rajput R, Abdin MZ, Vishwakarma RA, Riyaz-Ul-Hassan S. Diversity, molecular phylogeny, and bioactive potential of fungal endophytes associated with the Himalayan blue pine (Pinus wallichiana). Microbial Ecology. 67: 877-87. PMID 24563192 DOI: 10.1007/S00248-014-0379-4  0.389
2014 Bhat WW, Rana S, Dhar N, Razdan S, Pandith SA, Vishwakarma R, Lattoo SK. An inducible NADPH-cytochrome P450 reductase from Picrorhiza kurrooa - an imperative redox partner of cytochrome P450 enzymes. Functional & Integrative Genomics. 14: 381-99. PMID 24522789 DOI: 10.1007/S10142-014-0362-7  0.399
2014 Mupparapu N, Khan S, Battula S, Kushwaha M, Gupta AP, Ahmed QN, Vishwakarma RA. Metal-free oxidative amidation of 2-oxoaldehydes: a facile access to α-ketoamides. Organic Letters. 16: 1152-5. PMID 24490591 DOI: 10.1021/Ol5000204  0.397
2014 Yadav M, Raghupathy R, Saikam V, Dara S, Singh PP, Sawant SD, Mayor S, Vishwakarma RA. Synthesis of non-hydrolysable mimics of glycosylphosphatidylinositol (GPI) anchors. Organic & Biomolecular Chemistry. 12: 1163-72. PMID 24413835 DOI: 10.1039/C3Ob42116C  0.426
2014 Devari S, Jaglan S, Kumar M, Deshidi R, Guru S, Bhushan S, Kushwaha M, Gupta AP, Gandhi SG, Sharma JP, Taneja SC, Vishwakarma RA, Shah BA. Capsaicin production by Alternaria alternata, an endophytic fungus from Capsicum annum; LC-ESI-MS/MS analysis. Phytochemistry. 98: 183-9. PMID 24378219 DOI: 10.1016/J.Phytochem.2013.12.001  0.421
2014 Paul DJ, Laure NB, Guru SK, Khan IA, Ajit SK, Vishwakarma RA, Pierre T. Antiproliferative and antimicrobial activities of alkylbenzoquinone derivatives from Ardisia kivuensis. Pharmaceutical Biology. 52: 392-7. PMID 24192208 DOI: 10.3109/13880209.2013.837076  0.381
2014 Battula S, Vishwakarma RA, Ahmed QN. Cu–benzotriazole-catalyzed electrophilic cyclization of N-arylimines: a methodical tandem approach to O-protected-4hydroxyquinazolines- Rsc Advances. 4: 38375-38378. DOI: 10.1039/C4Ra07377K  0.377
2014 Aithagani SK, Yempalla KR, Munagala G, Vishwakarma RA, Singh PP. Metal-free, high yielding synthesis of unsymmetrical biaryl, bi(heteroaryl), aryl vinyl, aryl alkyl sulfones via coupling of aryne with sulfinic acid salts Rsc Advances. 4: 50208-50211. DOI: 10.1039/C4Ra07370C  0.4
2014 Rao DN, Rasheed S, Vishwakarma RA, Das P. Hypervalent iodine(III) catalyzed oxidative C–N bond formation in water: synthesis of benzimidazole-fused heterocycles Rsc Advances. 4: 25600-25604. DOI: 10.1039/C4Ra02279C  0.411
2014 Battini N, Padala AK, Mupparapu N, Vishwakarma RA, Ahmed QN. Unexplored reactivity of 2-oxoaldehydes towards Pictet–Spengler conditions: concise approach to β-carboline based marine natural products Rsc Advances. 4: 26258-26263. DOI: 10.1039/C4Ra01387E  0.411
2014 Joshi P, Singh S, Wani A, Sharma S, Jain SK, Singh B, Gupta BD, Satti NK, Koul S, Khan IA, Kumar A, Bharate SB, Vishwakarma RA. Osthol and curcumin as inhibitors of human Pgp and multidrug efflux pumps of Staphylococcus aureus: Reversing the resistance against frontline antibacterial drugs Medchemcomm. 5: 1540-1547. DOI: 10.1039/C4Md00196F  0.786
2014 Mudududdla R, Sharma R, Guru SK, Kushwaha M, Gupta AP, Bharate SS, Aravinda S, Kant R, Bhushan S, Vishwakarma RA, Bharate SB. Trifluoroacetic acid catalyzed thiophenylmethylation and thioalkylmethylation of lactams and phenols via domino three-component reaction in water Rsc Advances. 4: 14081-14088. DOI: 10.1039/C3Ra47874B  0.614
2014 Rasheed S, Rao DN, Reddy KR, Aravinda S, Vishwakarma RA, Das P. C-N bond formation via Cu-catalyzed cross-coupling with boronic acids leading to methyl carbazole-3-carboxylate: Synthesis of carbazole alkaloids Rsc Advances. 4: 4960-4969. DOI: 10.1039/C3Ra44903C  0.41
2014 Munagala G, Yempalla KR, Aithagani SK, Kalia NP, Ali F, Ali I, Rajput VS, Rani C, Chib R, Mehra R, Nargotra A, Khan IA, Vishwakarma RA, Singh PP. Synthesis and biological evaluation of substituted N-alkylphenyl-3,5-dinitrobenzamide analogs as anti-TB agents Medchemcomm. 5: 521-527. DOI: 10.1039/C3Md00366C  0.428
2014 Gannedi V, Ali A, Singh PP, Vishwakarma RA. Intramolecular aglycon delivery for (1 → 2)-β-mannosylation: towards the synthesis of phospholipomannan of Candida albicans Tetrahedron Letters. 55: 2945-2947. DOI: 10.1016/J.Tetlet.2014.03.099  0.378
2014 Dar BA, Dangroo NA, Gupta A, Wali A, Khuroo MA, Vishwakarma RA, Singh B. Iodine catalyzed solvent-free cross-dehydrogenative coupling of arylamines and H-phosphonates for the synthesis of N-arylphosphoramidates under atmospheric conditions Tetrahedron Letters. 55: 1544-1548. DOI: 10.1016/J.Tetlet.2014.01.064  0.383
2014 Sawant SD, Hudwekar AD, Aravinda Kumar KA, Venkateswarlu V, Singh PP, Vishwakarma RA. Ligand- and base-free synthesis of phenols by rapid oxidation of arylboronic acids using iron(III) oxide Tetrahedron Letters. 55: 811-814. DOI: 10.1016/J.Tetlet.2013.12.003  0.37
2014 Dar BA, Pandey N, Singh S, Bamezai RK, Sharma M, Vishwakarma RA, Singh B. Heterogeneous reusable catalyst, ultrasound energy, and no solvent: a quick and green recipe for one-pot synthesis of β-phosphonomalononitriles at room temperature Tetrahedron Letters. 55: 623-628. DOI: 10.1016/J.Tetlet.2013.11.095  0.378
2014 Dar BA, Singh S, Pandey N, Singh AP, Sharma P, Lazar A, Sharma M, Vishwakarma RA, Singh B. Clay encapsulated Cu(OH)x promoted homocoupling of arylboronic acids: An efficient and eco-friendly protocol Applied Catalysis a: General. 470: 232-238. DOI: 10.1016/J.Apcata.2013.10.048  0.365
2013 Gupta S, Pandotra P, Gupta AP, Verma MK, Ahuja A, Vishwakarma RA. Direct rhizogenesis, in vitro stolon proliferation and high-throughput regeneration of plantlets in . Acta Physiologiae Plantarum. 35: 2699-2705. PMID 32214545 DOI: 10.1007/s11738-013-1302-1  0.266
2013 Singh B, Guru SK, Kour S, Jain SK, Sharma R, Sharma PR, Singh SK, Bhushan S, Bharate SB, Vishwakarma RA. Synthesis, antiproliferative and apoptosis-inducing activity of thiazolo[5,4-d]pyrimidines. European Journal of Medicinal Chemistry. 70: 864-74. PMID 24262379 DOI: 10.1016/J.Ejmech.2013.10.039  0.79
2013 Dhar N, Rana S, Bhat WW, Razdan S, Pandith SA, Khan S, Dutt P, Dhar RS, Vaishnavi S, Vishwakarma R, Lattoo SK. Dynamics of withanolide biosynthesis in relation to temporal expression pattern of metabolic genes in Withania somnifera (L.) Dunal: a comparative study in two morpho-chemovariants. Molecular Biology Reports. 40: 7007-16. PMID 24190485 DOI: 10.1007/S11033-013-2820-Z  0.366
2013 Kannaboina P, Anilkumar K, Aravinda S, Vishwakarma RA, Das P. Direct C-2 arylation of 7-azaindoles: chemoselective access to multiarylated derivatives. Organic Letters. 15: 5718-21. PMID 24171392 DOI: 10.1021/Ol4027478  0.396
2013 Bhat WW, Dhar N, Razdan S, Rana S, Mehra R, Nargotra A, Dhar RS, Ashraf N, Vishwakarma R, Lattoo SK. Molecular characterization of UGT94F2 and UGT86C4, two glycosyltransferases from Picrorhiza kurrooa: comparative structural insight and evaluation of substrate recognition. Plos One. 8: e73804. PMID 24066073 DOI: 10.1371/Journal.Pone.0073804  0.401
2013 Jain SK, Pathania AS, Meena S, Sharma R, Sharma A, Singh B, Gupta BD, Bhushan S, Bharate SB, Vishwakarma RA. Semisynthesis of mallotus B from rottlerin: evaluation of cytotoxicity and apoptosis-inducing activity. Journal of Natural Products. 76: 1724-30. PMID 24041234 DOI: 10.1021/Np400433G  0.794
2013 Singh B, Vishwakarma RA, Bharate SB. QSAR and pharmacophore modeling of natural and synthetic antimalarial prodiginines. Current Computer-Aided Drug Design. 9: 350-9. PMID 24010933 DOI: 10.2174/15734099113099990020  0.721
2013 Agrawal M, Kharkar P, Moghe S, Mahajan T, Deka V, Thakkar C, Nair A, Mehta C, Bose J, Kulkarni-Almeida A, Bhedi D, Vishwakarma RA. Discovery of thiazolyl-phthalazinone acetamides as potent glucose uptake activators via high-throughput screening. Bioorganic & Medicinal Chemistry Letters. 23: 5740-3. PMID 23992862 DOI: 10.1016/J.Bmcl.2013.07.067  0.384
2013 Shakeel-U-Rehman, Sofi SN, Khuroo MA, Taneja SC, Bhat KA, Vishwakarma R. New natural compounds from Rhododendron lepidotum. Natural Product Research. 27: 2033-8. PMID 23941615 DOI: 10.1080/14786419.2013.824439  0.44
2013 Kaur T, Hussain K, Koul S, Vishwakarma R, Vyas D. Evaluation of nutritional and antioxidant status of Lepidium latifolium Linn.: a novel phytofood from Ladakh. Plos One. 8: e69112. PMID 23936316 DOI: 10.1371/Journal.Pone.0069112  0.39
2013 Zilla MK, Qadri M, Pathania AS, Strobel GA, Nalli Y, Kumar S, Guru SK, Bhushan S, Singh SK, Vishwakarma RA, Riyaz-Ul-Hassan S, Ali A. Bioactive metabolites from an endophytic Cryptosporiopsis sp. inhabiting Clidemia hirta. Phytochemistry. 95: 291-7. PMID 23870821 DOI: 10.1016/J.Phytochem.2013.06.021  0.461
2013 Kumar S, Pathania AS, Saxena AK, Vishwakarma RA, Ali A, Bhushan S. The anticancer potential of flavonoids isolated from the stem bark of Erythrina suberosa through induction of apoptosis and inhibition of STAT signaling pathway in human leukemia HL-60 cells. Chemico-Biological Interactions. 205: 128-37. PMID 23850732 DOI: 10.1016/J.Cbi.2013.06.020  0.419
2013 Singh B, Sidiq T, Joshi P, Jain SK, Lawaniya Y, Kichlu S, Khajuria A, Vishwakarma RA, Bharate SB. Anti-inflammatory and immunomodulatory flavones from Actinocarya tibetica Benth. Natural Product Research. 27: 2227-30. PMID 23768253 DOI: 10.1080/14786419.2013.805334  0.779
2013 Bharate SB, Sawant SD, Singh PP, Vishwakarma RA. Kinase inhibitors of marine origin. Chemical Reviews. 113: 6761-815. PMID 23679846 DOI: 10.1021/Cr300410V  0.647
2013 Dzoyem JP, Guru SK, Pieme CA, Kuete V, Sharma A, Khan IA, Saxena AK, Vishwakarma RA. Cytotoxic and antimicrobial activity of selected Cameroonian edible plants. Bmc Complementary and Alternative Medicine. 13: 78. PMID 23565827 DOI: 10.1186/1472-6882-13-78  0.372
2013 Bharate SS, Vishwakarma RA. Impact of preformulation on drug development. Expert Opinion On Drug Delivery. 10: 1239-57. PMID 23534681 DOI: 10.1517/17425247.2013.783563  0.38
2013 Bharate SB, Bharate JB, Khan SI, Tekwani BL, Jacob MR, Mudududdla R, Yadav RR, Singh B, Sharma PR, Maity S, Singh B, Khan IA, Vishwakarma RA. Discovery of 3,3'-diindolylmethanes as potent antileishmanial agents. European Journal of Medicinal Chemistry. 63: 435-43. PMID 23517732 DOI: 10.1016/J.Ejmech.2013.02.024  0.742
2013 Rana S, Lattoo SK, Dhar N, Razdan S, Bhat WW, Dhar RS, Vishwakarma R. NADPH-cytochrome P450 reductase: molecular cloning and functional characterization of two paralogs from Withania somnifera (L.) dunal. Plos One. 8: e57068. PMID 23437311 DOI: 10.1371/Journal.Pone.0057068  0.41
2013 Meena LS, Chopra P, Vishwakarma RA, Singh Y. Biochemical characterization of an S-adenosyll-methionine-dependent methyltransferase (Rv0469) of Mycobacterium tuberculosis Biological Chemistry. 394: 871-877. PMID 23435098 DOI: 10.1515/hsz-2013-0126  0.275
2013 Singh PP, Aithagani SK, Yadav M, Singh VP, Vishwakarma RA. Iron-catalyzed cross-coupling of electron-deficient heterocycles and quinone with organoboron species via innate C-H functionalization: application in total synthesis of pyrazine alkaloid botryllazine A. The Journal of Organic Chemistry. 78: 2639-48. PMID 23419207 DOI: 10.1021/Jo302797R  0.387
2013 Kumar M, Qadri M, Sharma PR, Kumar A, Andotra SS, Kaur T, Kapoor K, Gupta VK, Kant R, Hamid A, Johri S, Taneja SC, Vishwakarma RA, Riyaz-Ul-Hassan S, Shah BA. Tubulin inhibitors from an endophytic fungus isolated from Cedrus deodara. Journal of Natural Products. 76: 194-9. PMID 23387901 DOI: 10.1021/Np3006666  0.449
2013 Sinha S, Mishra P, Amin H, Rah B, Nayak D, Goswami A, Kumar N, Vishwakarma R, Ghosal S. A new cytotoxic quinolone alkaloid and a pentacyclic steroidal glycoside from the stem bark of Crataeva nurvala: study of anti-proliferative and apoptosis inducing property. European Journal of Medicinal Chemistry. 60: 490-6. PMID 23354071 DOI: 10.1016/J.Ejmech.2012.12.017  0.454
2013 Chinthakindi PK, Sangwan PL, Farooq S, Aleti RR, Kaul A, Saxena AK, Murthy YL, Vishwakarma RA, Koul S. Diminutive effect on T and B-cell proliferation of non-cytotoxic α-santonin derived 1,2,3-triazoles: a report. European Journal of Medicinal Chemistry. 60: 365-75. PMID 23314050 DOI: 10.1016/J.Ejmech.2012.12.018  0.455
2013 Razdan S, Bhat WW, Rana S, Dhar N, Lattoo SK, Dhar RS, Vishwakarma RA. Molecular characterization and promoter analysis of squalene epoxidase gene from Withania somnifera (L.) Dunal. Molecular Biology Reports. 40: 905-16. PMID 23065254 DOI: 10.1007/S11033-012-2131-9  0.377
2013 Ali A, Khajuria A, Sidiq T, Kumar A, Thakur NL, Naik D, Vishwakarma RA. Modulation of LPS induced inflammatory response by Lawsonyl monocyclic terpene from the marine derived Streptomyces sp. Immunology Letters. 150: 79-86. PMID 22975588 DOI: 10.1016/J.Imlet.2012.09.001  0.401
2013 Bharate JB, Vishwakarma RA, Bharate SB, Thite TB, Kushwaha M, Gupta AP. Quantification and Validation of Two Isomeric Anticancer Compounds, Garcinol and Isogarcinol, in Ultrasound- Assisted Extracts of Garcinia indica Fruits Using High- Performance Thin-Layer Chromatography Jpc-Journal of Planar Chromatography-Modern Tlc. 26: 480-485. DOI: 10.1556/Jpc.26.2013.6.4  0.581
2013 Bharate JB, Vishwakarma RA, Bharate SB, Kushwaha M, Gupta AP. Quantification Of Anticancer Polyisoprenylated Benzophenones Garcinol And Isogarcinol Using Multiple Reaction Monitoring Lc-Esi-Ms-Ms In Ultra-Sound Assisted Extracts Of Garcinia Indica Fruits Journal of Liquid Chromatography & Related Technologies. 150527103729000. DOI: 10.1080/10826076.2013.873872  0.565
2013 Tantry M, Khan I, Bedi Y, Vishwakarma R. Sulfated Triterpenes from Melissa officinalis L. Planta Medica. 79. DOI: 10.1055/S-0033-1348773  0.305
2013 Bharate JB, Sharma R, Aravinda S, Gupta VK, Singh B, Bharate SB, Vishwakarma RA. Montmorillonite clay catalyzed synthesis of functionalized pyrroles through domino four-component coupling of amines, aldehydes, 1,3-dicarbonyl compounds and nitroalkanes Rsc Advances. 3: 21736-21742. DOI: 10.1039/C3Ra43324B  0.588
2013 Jain SK, Pathania AS, Parshad R, Raina C, Ali A, Gupta AP, Kushwaha M, Aravinda S, Bhushan S, Bharate SB, Vishwakarma RA. Chrysomycins A-C, antileukemic naphthocoumarins from Streptomyces sporoverrucosus Rsc Advances. 3: 21046-21053. DOI: 10.1039/C3Ra42884B  0.802
2013 Bharate JB, Guru SK, Jain SK, Meena S, Singh PP, Bhushan S, Singh B, Bharate SB, Vishwakarma RA. Cu–Mn spinel oxide catalyzed synthesis of imidazo[1,2-a]pyridines through domino three-component coupling and 5-exo-dig cyclization in water Rsc Advances. 3: 20869-20876. DOI: 10.1039/C3Ra42046A  0.781
2013 Rao DN, Rasheed S, Aravinda S, Vishwakarma RA, Das P. Base and ligand free copper-catalyzed N-arylation of 2-amino-N-heterocycles with boronic acids in air Rsc Advances. 3: 11472-11475. DOI: 10.1039/C3Ra40735G  0.398
2013 Bharate SB, Yadav RR, Khan SI, Tekwani BL, Jacob MR, Khan IA, Vishwakarma RA. Meridianin G and its analogs as antimalarial agents Medchemcomm. 4: 1042-1048. DOI: 10.1039/C3Md00097D  0.607
2013 Jain SK, Meena S, Qazi AK, Hussain A, Bhola SK, Kshirsagar R, Pari K, Khajuria A, Hamid A, Shaanker RU, Bharate SB, Vishwakarma RA. Isolation and biological evaluation of chromone alkaloid dysoline, a new regioisomer of rohitukine from Dysoxylum binectariferum Tetrahedron Letters. 54: 7140-7143. DOI: 10.1016/J.Tetlet.2013.10.096  0.794
2013 Singh B, Parshad R, Khajuria R, Guru SK, Pathania AS, Sharma R, Chib R, Aravinda S, Gupta VK, Khan IA, Bhushan S, Bharate SB, Vishwakarma RA. Saccharonol B, a new cytotoxic methylated isocoumarin from Saccharomonospora azurea Tetrahedron Letters. 54: 6695-6699. DOI: 10.1016/J.Tetlet.2013.09.060  0.666
2013 Sawant SD, Srinivas M, Aravinda Kumar K, Lakshma Reddy G, Singh PP, Singh B, Sharma AK, Sharma P, Vishwakarma RA. Ligand-free C–N bond formation in aqueous medium using a reusable Cu–Mn bimetallic catalyst Tetrahedron Letters. 54: 5351-5354. DOI: 10.1016/J.Tetlet.2013.07.095  0.391
2013 Bharate SB, Padala AK, Dar BA, Yadav RR, Singh B, Vishwakarma RA. Montmorillonite clay Cu(II) catalyzed domino one-pot multicomponent synthesis of 3,5-disubstituted isoxazoles Tetrahedron Letters. 54: 3558-3561. DOI: 10.1016/J.Tetlet.2013.04.102  0.575
2013 Bharate SB, Mudududdla R, Sharma R, Vishwakarma RA. The first method for C-devinylation of aromatic systems Tetrahedron Letters. 54: 2913-2915. DOI: 10.1016/J.Tetlet.2013.03.064  0.579
2013 Gupta S, Pandotra P, Gupta AP, Verma MK, Ahuja A, Vishwakarma RA. Direct rhizogenesis, in vitro stolon proliferation and high-throughput regeneration of plantlets in Glycyrrhiza glabra Acta Physiologiae Plantarum. 35: 2699-2705. DOI: 10.1007/S11738-013-1302-1  0.373
2013 Sharma P, Kumar S, Ali F, Anthal S, Gupta VK, Khan IA, Singh S, Sangwan PL, Suri KA, Gupta BD, Gupta DK, Dutt P, Vishwakarma RA, Satti NK. Erratum to: Synthesis and biologic activities of some novel heterocyclic chalcone derivatives Medicinal Chemistry Research. 22: 4547-4547. DOI: 10.1007/S00044-012-0444-9  0.372
2013 Sharma P, Kumar S, Ali F, Anthal S, Gupta VK, Khan IA, Singh S, Sangwan PL, Suri KA, Gupta BD, Gupta DK, Dutt P, Vishwakarma RA, Satti NK. Synthesis and biologic activities of some novel heterocyclic chalcone derivatives Medicinal Chemistry Research. 22: 3969-3983. DOI: 10.1007/S00044-012-0401-7  0.466
2013 Mehra R, Nargotra A, Shah BA, Taneja SC, Vishwakarma RA, Koul S. Pro-apoptotic properties of parthenin analogs: A quantitative structure-activity relationship study Medicinal Chemistry Research. 22: 2303-2311. DOI: 10.1007/S00044-012-0225-5  0.416
2012 Mudududdla R, Jain SK, Bharate JB, Gupta AP, Singh B, Vishwakarma RA, Bharate SB. ortho-Amidoalkylation of phenols via tandem one-pot approach involving oxazine intermediate. The Journal of Organic Chemistry. 77: 8821-7. PMID 22970791 DOI: 10.1021/Jo3017132  0.782
2012 Bharate SB, Yadav RR, Vishwakarma RA. QSAR and Pharmacophore Study of Dyrk1A Inhibitory Meridianin Analogs as Potential Agents for Treatment of Neurodegenerative Diseases Medicinal Chemistry. 9: 152-161. PMID 22920091 DOI: 10.2174/157340613804488459  0.685
2012 Jadhav RD, Kadam KS, Kandre S, Guha T, Reddy MMK, Brahma MK, Deshmukh NJ, Dixit A, Doshi L, Potdar N, Enose AA, Vishwakarma RA, Sivaramakrishnan H, Srinivasan S, Nemmani KVS, et al. Synthesis and biological evaluation of isoxazole, oxazole, and oxadiazole containing heteroaryl analogs of biaryl ureas as DGAT1 inhibitors European Journal of Medicinal Chemistry. 54: 324-342. PMID 22683241 DOI: 10.1016/J.Ejmech.2012.05.016  0.462
2012 Singh PP, Thatikonda T, Kumar KA, Sawant SD, Singh B, Sharma AK, Sharma PR, Singh D, Vishwakarma RA. Cu-Mn spinel oxide catalyzed regioselective halogenation of phenols and N-heteroarenes. The Journal of Organic Chemistry. 77: 5823-8. PMID 22668006 DOI: 10.1021/Jo300731Z  0.393
2012 Bharate SB, Mudududdla R, Bharate JB, Battini N, Battula S, Yadav RR, Singh B, Vishwakarma RA. Tandem one-pot synthesis of flavans by recyclable silica-HClO4 catalyzed Knoevenagel condensation and [4 + 2]-Diels-Alder cycloaddition. Organic & Biomolecular Chemistry. 10: 5143-50. PMID 22648274 DOI: 10.1039/C2Ob25376C  0.601
2012 Ghosal S, Deb A, Mishra P, Vishwakarma R. Leishmanicidal compounds from the fruits of Piper longum. Planta Medica. 78: 906-8. PMID 22576441 DOI: 10.1055/S-0031-1298537  0.425
2012 Afnan Q, Adil MD, Nissar-Ul A, Rafiq AR, Amir HF, Kaiser P, Gupta VK, Vishwakarma R, Tasduq SA. Glycyrrhizic acid (GA), a triterpenoid saponin glycoside alleviates ultraviolet-B irradiation-induced photoaging in human dermal fibroblasts. Phytomedicine : International Journal of Phytotherapy and Phytopharmacology. 19: 658-64. PMID 22516896 DOI: 10.1016/J.Phymed.2012.03.007  0.391
2012 Jain SK, Bharate SB, Vishwakarma RA. Cyclin-dependent kinase inhibition by flavoalkaloids. Mini-Reviews in Medicinal Chemistry. 12: 632-649. PMID 22512551 DOI: 10.2174/138955712800626683  0.602
2012 Bharate SB, Yadav RR, Battula S, Vishwakarma RA. Meridianins: Marine-Derived Potent Kinase Inhibitors Mini-Reviews in Medicinal Chemistry. 12: 618-631. PMID 22512550 DOI: 10.2174/138955712800626728  0.625
2012 Bharate SB, Manda S, Mupparapu N, Battini N, Vishwakarma RA. Chemistry and biology of fascaplysin, a potent marine-derived CDK-4 inhibitor. Mini-Reviews in Medicinal Chemistry. 12: 650-664. PMID 22512549 DOI: 10.2174/138955712800626719  0.627
2012 Singh B, Nadkarni JR, Vishwakarma RA, Bharate SB, Nivsarkar M, Anandjiwala S. The hydroalcoholic extract of Cassia alata (Linn.) leaves and its major compound rhein exhibits antiallergic activity via mast cell stabilization and lipoxygenase inhibition. Journal of Ethnopharmacology. 141: 469-73. PMID 22449441 DOI: 10.1016/J.Jep.2012.03.012  0.65
2012 Bhat WW, Lattoo SK, Razdan S, Dhar N, Rana S, Dhar RS, Khan S, Vishwakarma RA. Molecular cloning, bacterial expression and promoter analysis of squalene synthase from Withania somnifera (L.) Dunal. Gene. 499: 25-36. PMID 22425978 DOI: 10.1016/J.Gene.2012.03.004  0.409
2012 Bharate SB, Singh B, Vishwakarma RA. Modulation of k-Ras signaling by natural products. Current Medicinal Chemistry. 19: 2273-2291. PMID 22414109 DOI: 10.2174/092986712800229050  0.628
2012 Singh PP, Gudup S, Aruri H, Singh U, Ambala S, Yadav M, Sawant SD, Vishwakarma RA. New method for C-H arylation/alkylation at α-position of cyclic aliphatic ethers by iron-oxide mediated reaction. Organic & Biomolecular Chemistry. 10: 1587-97. PMID 22222780 DOI: 10.1039/C1Ob06660A  0.407
2012 Bharate SB, Mupparapu N, Manda S, Bharate JB, Mudududdla R, Yadav RR, Vishwakarma RA. Efficient synthesis of 2,3-dihydroquinazolin-4(1H)-ones using heterogeneous solid acid catalysts: unexpected formation of 2,3-dihydro-2-(4-(tetrahydro-2H-pyran-2-yloxy)butyl)-quinazolin-4(1H)-one Arkivoc. 2012: 308-318. DOI: 10.3998/Ark.5550190.0013.826  0.589
2012 Jain SK, Meena S, Singh B, Bharate JB, Joshi P, Singh VP, Vishwakarma RA, Bharate SB. KF/alumina catalyzed regioselective benzylation and benzoylation using solvent-free grind-stone chemistry Rsc Advances. 2: 8929. DOI: 10.1039/C2Ra21154H  0.783
2012 Bharate SB, Manda S, Joshi P, Singh B, Vishwakarma RA. Total synthesis and anti-cholinesterase activity of marine-derived bis-indole alkaloid fascaplysin Medchemcomm. 3: 1098. DOI: 10.1039/C2Md20076G  0.674
2012 Sawant SD, Srinivas M, Lakshma Reddy G, Venkateswar Rao V, Singh PP, Vishwakarma RA. One-pot multicomponent synthesis of medicinally important purine quinazolinone derivatives Tetrahedron Letters. 53: 6195-6198. DOI: 10.1016/J.Tetlet.2012.08.137  0.471
2012 Yadav RR, Vishwakarma RA, Bharate SB. Catalyst-free ipso-nitration of aryl boronic acids using bismuth nitrate☆ Tetrahedron Letters. 53: 5958-5960. DOI: 10.1016/J.Tetlet.2012.08.121  0.575
2012 Yadav RR, Battini N, Mudududdla R, Bharate JB, Muparappu N, Bharate SB, Vishwakarma RA. Deformylation of indole and azaindole-3-carboxaldehydes using anthranilamide and solid acid heterogeneous catalyst via quinazolinone intermediate Tetrahedron Letters. 53: 2222-2225. DOI: 10.1016/J.Tetlet.2012.02.079  0.567
2012 Mohammed S, Padala AK, Dar BA, Singh B, Sreedhar B, Vishwakarma RA, Bharate SB. Recyclable clay supported Cu (II) catalyzed tandem one-pot synthesis of 1-aryl-1,2,3-triazoles ☆ Tetrahedron. 68: 8156-8162. DOI: 10.1016/J.Tet.2012.07.080  0.56
2012 Bhat WW, Lattoo SK, Rana S, Razdan S, Dhar N, Dhar RS, Vishwakarma RA. Efficient plant regeneration via direct organogenesis and Agrobacterium tumefaciens-mediated genetic transformation of Picrorhiza kurroa: An endangered medicinal herb of the alpine Himalayas In Vitro Cellular and Developmental Biology - Plant. 48: 295-303. DOI: 10.1007/S11627-012-9434-3  0.363
2012 Bharate SB, Singh B, Bharate JB, Jain SK, Meena S, Vishwakarma RA. QSAR and pharmacophore modeling of N-acetyl-2-aminobenzothiazole class of phosphoinositide-3-kinase-α inhibitors Medicinal Chemistry Research. 22: 890-899. DOI: 10.1007/S00044-012-0081-3  0.788
2011 Sen M, Shah B, Rakshit S, Singh V, Padmanabhan B, Ponnusamy M, Pari K, Vishwakarma R, Nandi D, Sadhale PP. UDP-glucose 4, 6-dehydratase activity plays an important role in maintaining cell wall integrity and virulence of Candida albicans. Plos Pathogens. 7: e1002384. PMID 22114559 DOI: 10.1371/Journal.Ppat.1002384  0.396
2011 Kulkarni-Almeida AA, Brahma MK, Padmanabhan P, Mishra PD, Parab RR, Gaikwad NV, Thakkar CS, Tokdar P, Ranadive PV, Nair AS, Damre AA, Bahirat UA, Deshmukh NJ, Doshi LS, Dixit AV, ... ... Vishwakarma RA, et al. Fermentation, Isolation, Structure, and antidiabetic activity of NFAT-133 produced by Streptomyces strain PM0324667. Amb Express. 1: 42. PMID 22104600 DOI: 10.1186/2191-0855-1-42  0.413
2011 Motiwala H, Kandre S, Birar V, Kadam KS, Rodge A, Jadhav RD, Mahesh Kumar Reddy M, Brahma MK, Deshmukh NJ, Dixit A, Doshi L, Gupte A, Gangopadhyay AK, Vishwakarma RA, Srinivasan S, et al. Exploration of pyridine containing heteroaryl analogs of biaryl ureas as DGAT1 inhibitors Bioorganic and Medicinal Chemistry Letters. 21: 5812-5817. PMID 21868220 DOI: 10.1016/J.Bmcl.2011.07.109  0.454
2011 Dhuru S, Bhedi D, Gophane D, Hirbhagat K, Nadar V, More D, Parikh S, Dalal R, Fonseca LC, Kharas F, Vadnal PY, Vishwakarma RA, Sivaramakrishnan H. Novel diarylheptanoids as inhibitors of TNF-α production. Bioorganic & Medicinal Chemistry Letters. 21: 3784-7. PMID 21600765 DOI: 10.1016/J.Bmcl.2011.04.040  0.438
2011 Singh PP, Gudup S, Ambala S, Singh U, Dadhwal S, Singh B, Sawant SD, Vishwakarma RA. Iron oxide mediated direct C-H arylation/alkylation at α-position of cyclic aliphatic ethers. Chemical Communications (Cambridge, England). 47: 5852-4. PMID 21503345 DOI: 10.1039/C1Cc11094B  0.392
2011 Mishra P, Sinha S, Guru SK, Bhushan S, Vishwakarma RA, Ghosal S. Two new amides with cytotoxic activity from the fruits of Piper longum. Journal of Asian Natural Products Research. 13: 143-8. PMID 21279878 DOI: 10.1080/10286020.2010.546789  0.468
2011 Balachandran S, Gadekar PK, Parkale S, Yadav VN, Kamath D, Ramaswamy S, Sharma S, Vishwakarma RA, Dagia NM. Synthesis and biological activity of novel MIF antagonists. Bioorganic & Medicinal Chemistry Letters. 21: 1508-11. PMID 21277206 DOI: 10.1016/J.Bmcl.2010.12.127  0.464
2011 Deore V, Lohar MK, Mundada R, Roychowdhury A, Vishwakarma R, Kumar S. Efficient synthesis of key intermediate toward liphagal synthesis Synthetic Communications. 41: 177-183. DOI: 10.1080/00397910903531920  0.406
2011 Saikam V, Raghupathy R, Yadav M, Gannedi V, Singh PP, Qazi NA, Sawant SD, Vishwakarma RA. Synthesis of new fluorescently labeled glycosylphosphatidylinositol (GPI) anchors Tetrahedron Letters. 52: 4277-4279. DOI: 10.1016/J.Tetlet.2011.06.005  0.389
2010 Adil MD, Kaiser P, Satti NK, Zargar AM, Vishwakarma RA, Tasduq SA. Effect of Emblica officinalis (fruit) against UVB-induced photo-aging in human skin fibroblasts. Journal of Ethnopharmacology. 132: 109-114. PMID 20688142 DOI: 10.1016/J.Jep.2010.07.047  0.385
2010 Chandra S, Ruhela D, Deb A, Vishwakarma RA. Glycobiology of the Leishmania parasite and emerging targets for antileishmanial drug discovery. Expert Opinion On Therapeutic Targets. 14: 739-57. PMID 20536412 DOI: 10.1517/14728222.2010.495125  0.342
2010 Ali A, Vishwakarma RA. Total synthesis of the fully lipidated glycosylphosphatidylinositol (GPI) anchor of malarial parasite Plasmodium falciparum Tetrahedron. 66: 4357-4369. DOI: 10.1016/J.Tet.2010.04.014  0.391
2009 Balachandran S, Rodge A, Gadekar PK, Yadav VN, Kamath D, Chetrapal-Kunwar A, Bhatt P, Srinivasan S, Sharma S, Vishwakarma RA, Dagia NM. Novel derivatives of ISO-1 as potent inhibitors of MIF biological function. Bioorganic & Medicinal Chemistry Letters. 19: 4773-6. PMID 19592246 DOI: 10.1016/J.Bmcl.2009.06.052  0.434
2009 Deshmukh SK, Mishra PD, Kulkarni-Almeida A, Verekar S, Sahoo MR, Periyasamy G, Goswami H, Khanna A, Balakrishnan A, Vishwakarma R. Anti-inflammatory and anticancer activity of ergoflavin isolated from an endophytic fungus Chemistry and Biodiversity. 6: 784-789. PMID 19479845 DOI: 10.1002/Cbdv.200800103  0.425
2009 Bharate SB, Nemmani KVS, Vishwakarma RA. Progress in the discovery and development of small-molecule modulators of G-protein-coupled receptor 40 (GPR40/FFA1/FFAR1): an emerging target for type 2 diabetes. Expert Opinion On Therapeutic Patents. 19: 237-264. PMID 19441920 DOI: 10.1517/13543770802665717  0.566
2009 Deore V, Yewalkar N, Bhatia D, Desai N, Gupte RD, Dadarkar SS, Jadhav MG, Tannu AA, Bhatt P, Nemmani KV, Vishwakarma RA, Sharma S, Roychowdhury A, Dagia NM, Bhonde MR, et al. Synthesis and therapeutic evaluation of pyridyl based novel mTOR inhibitors. Bioorganic & Medicinal Chemistry Letters. 19: 2949-52. PMID 19409777 DOI: 10.1016/J.Bmcl.2009.04.055  0.458
2009 Dagia NM, Kamath DV, Bhatt P, Gupte RD, Dadarkar SS, Fonseca L, Agarwal G, Chetrapal-Kunwar A, Balachandran S, Srinivasan S, Bose J, Pari K, B-Rao C, Parkale SS, Gadekar PK, ... ... Vishwakarma RA, et al. A fluorinated analog of ISO-1 blocks the recognition and biological function of MIF and is orally efficacious in a murine model of colitis. European Journal of Pharmacology. 607: 201-12. PMID 19239912 DOI: 10.1016/J.Ejphar.2009.02.031  0.412
2009 Vyas HK, Pal R, Vishwakarma R, Lohiya NK, Talwar GP. Selective killing of leukemia and lymphoma cells ectopically expressing hCGbeta by a conjugate of curcumin with an antibody against hCGbeta subunit. Oncology. 76: 101-11. PMID 19127081 DOI: 10.1159/000188665  0.231
2009 Singh A, Vishwakarma RA, Husain A. Evalutation of Artemisia annua strains for higher artemisinin production. Planta Medica. 54: 475-6. PMID 17265330 DOI: 10.1055/s-2006-962515  0.211
2009 Vishwakarma RA, Tyagi BR, Ahmed B, Husain A. Variation in forskolin content in the roots of Coleus forskohlii. Planta Medica. 54: 471-2. PMID 17265327 DOI: 10.1055/S-2006-962512  0.313
2009 Janardhanan KK, Meera CR, Nitha B, Vishwakarma RA. Anti-inflammatory and Free Radical Scavenging Activities of Polysaccharide−Protein Complex Isolated from Phellinus rimosus (Berk.) Pilát (Aphyllophoromycetideae) International Journal of Medicinal Mushrooms. 11: 365-373. DOI: 10.1615/Intjmedmushr.V11.I4.30  0.359
2009 Vishwakarma R, Ruhela D. Chapter 10 Chemical Synthesis of Glycosylphosphatidylinositol (GPI) Anchors The Enzymes. 26: 181-227. DOI: 10.1016/S1874-6047(09)26010-0  0.404
2008 Goswami D, Gowrishankar K, Bilgrami S, Ghosh S, Raghupathy R, Chadda R, Vishwakarma R, Rao M, Mayor S. Nanoclusters of GPI-anchored proteins are formed by cortical actin-driven activity. Cell. 135: 1085-97. PMID 19070578 DOI: 10.1016/J.Cell.2008.11.032  0.329
2008 Bharate SB, Rodge A, Joshi RK, Kaur J, Srinivasan S, Kumar SS, Kulkarni-Almeida A, Balachandran S, Balakrishnan A, Vishwakarma RA. Discovery of diacylphloroglucinols as a new class of GPR40 (FFAR1) agonists. Bioorganic & Medicinal Chemistry Letters. 18: 6357-61. PMID 18993064 DOI: 10.1016/J.Bmcl.2008.10.085  0.592
2008 Bhonde MR, Gupte RD, Dadarkar SD, Jadhav MG, Tannu AA, Bhatt P, Bhatia DR, Desai NK, Deore V, Yewalkar N, Vishwakarma RA, Sharma S, Kumar S, Dagia NM. A novel mTOR inhibitor is efficacious in a murine model of colitis. American Journal of Physiology. Gastrointestinal and Liver Physiology. 295: G1237-45. PMID 18927209 DOI: 10.14309/00000434-200809001-01044  0.451
2008 Subramaniam D, Giridharan P, Murmu N, Shankaranarayanan NP, May R, Houchen CW, Ramanujam RP, Balakrishnan A, Vishwakarma RA, Anant S. Activation of apoptosis by 1-hydroxy-5,7-dimethoxy-2-naphthalene-carboxaldehyde, a novel compound from Aegle marmelos. Cancer Research. 68: 8573-81. PMID 18922933 DOI: 10.1158/0008-5472.Can-08-2372  0.436
2008 Bharate SB, Mahajan TR, Gole YR, Nambiar M, Matan TT, Kulkarni-Almeida A, Balachandran S, Junjappa H, Balakrishnan A, Vishwakarma RA. Synthesis and evaluation of pyrazolo[3,4-b]pyridines and its structural analogues as TNF-alpha and IL-6 inhibitors. Bioorganic & Medicinal Chemistry. 16: 7167-76. PMID 18625560 DOI: 10.1016/J.Bmc.2008.06.042  0.677
2008 Kulkarni-Almeida A, Suthar A, Goswami H, Vishwakarma R, Chauhan VS, Balakrishnan A, Sharma S. Novel leads from Heliotropium ovalifolium, 4,7,8-trimethoxy-naphthalene-2-carboxylic acid and 6-hydroxy-5,7-dimethoxy-naphthalene-2-carbaldehyde show specific IL-6 inhibitory activity in THP-1 cells and primary human monocytes Phytomedicine. 15: 1079-1086. PMID 18583119 DOI: 10.1016/J.Phymed.2008.04.013  0.46
2008 Lohar MV, Mundada R, Bhonde M, Padgaonkar A, Deore V, Yewalkar N, Bhatia D, Rathos M, Joshi K, Vishwakarma RA, Kumar S. Design and synthesis of novel furoquinoline based inhibitors of multiple targets in the PI3K/Akt-mTOR pathway Bioorganic and Medicinal Chemistry Letters. 18: 3603-3606. PMID 18501601 DOI: 10.1016/J.Bmcl.2008.04.078  0.454
2007 Senthil V, Ramadevi S, Venkatakrishnan V, Giridharan P, Lakshmi BS, Vishwakarma RA, Balakrishnan A. Withanolide induces apoptosis in HL-60 leukemia cells via mitochondria mediated cytochrome c release and caspase activation Chemico-Biological Interactions. 167: 19-30. PMID 17328876 DOI: 10.1016/J.Cbi.2007.01.004  0.393
2006 Manjula N, Gayathri B, Vinaykumar KS, Shankernarayanan NP, Vishwakarma RA, Balakrishnan A. Inhibition of MAP kinases by crude extract and pure compound isolated from Commiphora mukul leads to down regulation of TNF-α, IL-1β and IL-2 International Immunopharmacology. 6: 122-132. PMID 16399617 DOI: 10.1016/J.Intimp.2005.07.001  0.447
2006 Vishwakarma RA, Anand MT, Arya R, Vats D, Bhattacharya A. Glycosylated inositol phospholipid from Entamoeba histolytica: Identification and structural characterization Molecular and Biochemical Parasitology. 145: 121-124. PMID 16242191 DOI: 10.1016/j.molbiopara.2005.09.009  0.235
2005 Vats D, Vishwakarma RA, Bhattacharya S, Bhattacharya A. Reduction of cell surface glycosylphosphatidylinositol conjugates in Entamoeba histolytica by antisense blocking of E. histolytica GlcNAc-phosphatidylinositol deacetylase expression: Effect on cell proliferation, endocytosis, and adhesion to target cells Infection and Immunity. 73: 8381-8392. PMID 16299336 DOI: 10.1128/IAI.73.12.8381-8392.2005  0.307
2005 Prasad T, Saini P, Gaur NA, Vishwakarma RA, Khan LA, Haq QM, Prasad R. Functional analysis of CaIPT1, a sphingolipid biosynthetic gene involved in multidrug resistance and morphogenesis of Candida albicans. Antimicrobial Agents and Chemotherapy. 49: 3442-52. PMID 16048959 DOI: 10.1128/AAC.49.8.3442-3452.2005  0.219
2005 Singh A, Gupta R, Vishwakarma RA, Narayanan PR, Paramasivan CN, Ramanathan VD, Tyagi AK. Requirement of the mymA Operon for Appropriate Cell Wall Ultrastructure and Persistence of Mycobacterium tuberculosis in the Spleens of Guinea Pigs Journal of Bacteriology. 187: 4173-4186. PMID 15937179 DOI: 10.1128/Jb.187.12.4173-4186.2005  0.37
2005 Vishwakarma RA, Vehring S, Mehta A, Sinha A, Pomorski T, Herrmann A, Menon AK. New fluorescent probes reveal that flippase-mediated flip-flop of phosphatidylinositol across the endoplasmic reticulum membrane does not depend on the stereochemistry of the lipid. Organic & Biomolecular Chemistry. 3: 1275-83. PMID 15785818 DOI: 10.1039/B500300H  0.346
2005 Ruhela D, Chatterjee P, Vishwakarma RA. 1-Oxabicyclic beta-lactams as new inhibitors of elongating MPT--a key enzyme responsible for assembly of cell-surface phosphoglycans of Leishmania parasite. Organic & Biomolecular Chemistry. 3: 1043-8. PMID 15750647 DOI: 10.1039/B418247B  0.382
2005 Anandharajan R, Pathmanathan K, Shankernarayanan NP, Vishwakarma RA, Balakrishnan A. Upregulation of Glut-4 and PPARγ by an isoflavone from Pterocarpus marsupium on L6 myotubes: a possible mechanism of action Journal of Ethnopharmacology. 97: 253-260. PMID 15707762 DOI: 10.1016/J.Jep.2004.11.023  0.37
2005 Ali A, Gowda DC, Vishwakarma RA. A new approach to construct full-length glycosylphosphatidylinositols of parasitic protozoa and [4-deoxy-Man-III]-GPI analogues. Chemical Communications (Cambridge, England). 519-21. PMID 15654389 DOI: 10.1039/B414119A  0.401
2005 Vishwakarma RA, Menon AK. Flip-flop of glycosylphosphatidylinositols (GPI's) across the ER. Chemical Communications (Cambridge, England). 453-5. PMID 15654367 DOI: 10.1039/B413196G  0.342
2004 Ruhela D, Vishwakarma RA. A facile and novel route to the antigenic branched phosphoglycan of the protozoan Leishmania major parasite Tetrahedron Letters. 45: 2589-2592. DOI: 10.1016/J.Tetlet.2004.01.155  0.376
2003 Ruhela D, Vishwakarma RA. Iterative synthesis of Leishmania phosphoglycans by solution, solid-phase, and polycondensation approaches without involving any glycosylation. Journal of Organic Chemistry. 68: 4446-4456. PMID 12762750 DOI: 10.1021/Jo0341867  0.395
2003 Chawla M, Vishwakarma RA. Alkylacylglycerolipid domain of GPI molecules of Leishmania is responsible for inhibition of PKC-mediated c-fos expression. Journal of Lipid Research. 44: 594-600. PMID 12562866 DOI: 10.1194/Jlr.M200296-Jlr200  0.392
2003 Arya R, Mehra A, Bhattacharya S, Vishwakarma RA, Bhattacharya A. Biosynthesis of Entamoeba histolytica proteophosphoglycan in vitro. Molecular and Biochemical Parasitology. 126: 1-8. PMID 12554078 DOI: 10.1016/S0166-6851(02)00252-9  0.35
2002 Giridharan P, Somasundaram ST, Perumal K, Vishwakarma RA, Karthikeyan NP, Velmurugan R, Balakrishnan A. Novel substituted methylenedioxy lignan suppresses proliferation of cancer cells by inhibiting telomerase and activation of c-myc and caspases leading to apoptosis. British Journal of Cancer. 87: 98-105. PMID 12085264 DOI: 10.1038/Sj.Bjc.6600422  0.476
2001 Ruhela D, Vishwakarma RA. Efficient synthesis of the antigenic phosphoglycans of the Leishmania parasite. Chemical Communications. 2024-5. PMID 12240271 DOI: 10.1039/B106634J  0.373
2000 Nakra P, Manivel V, Vishwakarma RA, Rao KVS. B Cell Responses to a Peptide Epitope. X. Epitope Selection in a Primary Response Is Thermodynamically Regulated Journal of Immunology. 164: 5615-5625. PMID 10820236 DOI: 10.4049/Jimmunol.164.11.5615  0.358
2000 Sahai P, Chawla M, Vishwakarma RA. 13C Labelling and electrospray mass spectrometry reveal a de novo route for inositol biosynthesis in Leishmania donovani parasite Journal of the Chemical Society-Perkin Transactions 1. 1283-1290. DOI: 10.1039/B000262N  0.385
2000 Upreti M, Ruhela D, Vishwakarma RA. Synthesis of the Tetrasaccharide Cap Domain of the Antigenic Lipophosphoglycan of Leishmania donovani Parasite Tetrahedron. 56: 6577-6584. DOI: 10.1016/S0040-4020(00)00609-8  0.398
1999 Upreti M, Vishwakarma RA. Synthesis of the phosphodisaccharide repeat of antigenic lipophosphoglycan of Leishmania donovani parasite Tetrahedron Letters. 40: 2619-2622. DOI: 10.1016/S0040-4039(99)00231-2  0.403
1998 Bharel S, Gulati A, Abdin MZ, Srivastava PS, Vishwakarma RA, Jain SK. Enzymatic Synthesis of Artemisinin from Natural and Synthetic Precursors Journal of Natural Products. 61: 633-636. PMID 9599263 DOI: 10.1021/Np970024S  0.404
1998 Bharel S, Vishwakarma RA, Jain SK. Artemisinin mediated alteration of haemin to a δ-meso oxidation product: relevance to mechanism of action Journal of the Chemical Society-Perkin Transactions 1. 2163-2166. DOI: 10.1039/A802423E  0.389
1998 and PS, Vishwakarma RA, Bharel S, Gulati A, Abdin MZ, Srivastava aPS, Jain SK. HPLC−Electrospray Ionization Mass Spectrometric Analysis of Antimalarial Drug Artemisinin Analytical Chemistry. 70: 3084-3087. DOI: 10.1021/Ac970944F  0.382
1998 Tyagi AK, Vishwakarma RA. Recombinant Bacillus subtilis whole cell system as a catalyst for enzymatic synthesis of cyclic inositol phosphate Tetrahedron Letters. 39: 6069-6072. DOI: 10.1016/S0040-4039(98)01250-7  0.416
1997 Tripathi R, Vishwakarma RA, Dutta GP. Plasmodium fragile: efficacy of arteether (alpha/beta) against cerebral malaria model. Experimental Parasitology. 87: 290-2. PMID 9371096 DOI: 10.1006/Expr.1997.4239  0.302
1997 Sahai P, Vishwakarma RA. Phospholipase-A2-mediated stereoselective synthesis of(R)-1-O-alkylglycero-3-phosphate and alkyl-acylanalogues: application for synthesis of radiolabelled biosyntheticprecursors of cell surface glycoconjugates of Leishmaniadonovani Journal of the Chemical Society-Perkin Transactions 1. 1845-1850. DOI: 10.1039/A700353F  0.403
1997 Ghosal S, Vishwakarma RA. Tinocordiside, a new rearranged cadinane sesquiterpene glycoside from Tinospora cordifolia Journal of Natural Products. 60: 839-841. DOI: 10.1021/Np970169Z  0.405
1997 Zamir LO, Balachandran S, Zheng YF, Nedea ME, Caron G, Nikolakakis A, Vishwakarma RA, Sauriol F, Mamer O. Acid catalyzed rearrangement and acyl migration studies on 9-dihydro-13-acetylbaccatin-III, a major taxane from Taxus canadensis Tetrahedron. 53: 15991-16008. DOI: 10.1016/S0040-4020(97)10069-2  0.387
1996 Tripathi R, Dutta GP, Vishwakarma RA. Gametocytocidal activity of alpha/beta arteether by the oral route of administration. The American Journal of Tropical Medicine and Hygiene. 54: 652-4. PMID 8686787 DOI: 10.4269/Ajtmh.1996.54.652  0.341
1995 Pandey M, Vishwakarma RA, Khatri AK, Roy SK, Shukla VK. Bile, bacteria, and gallbladder carcinogenesis. Journal of Surgical Oncology. 58: 282-3. PMID 7723375 DOI: 10.1002/JSO.2930580417  0.196
1995 Gupta S, Ghosh PK, Dutta GP, Vishwakarma RA. In vivo Study of Artemisinin and Its Derivatives against Primary Amebic Meningoencephalitis Caused by Naegleria fowleri The Journal of Parasitology. 81: 1012. DOI: 10.2307/3284060  0.261
1995 Vishwakarma R, Gupta S, Shukla V, Khan M. 572 Bile, bacteria and carcinona of gall bladder European Journal of Cancer. 31: S122. DOI: 10.1016/0959-8049(95)95826-R  0.188
1994 Balachandran S, Vishwakarma RA, Monaghan SM, Prelle A, Stamford NPJ, Leeper FJ, Battersby AR. Biosynthesis of porphyrins and related macrocycles. Part 42. Pulse labelling experiments concerning the timing of cobalt insertion during vitamin B12 biosynthesis Journal of the Chemical Society, Perkin Transactions 1. 487-491. DOI: 10.1039/P19940000487  0.628
1994 Li Y, Alanine AID, Vishwakarma RA, Balachandran S, Leeper FJ, Battersby AR. Biosynthesis of vitamin B12: Mechanistic studies on the transfer of a methyl group from C-11 to C-12 and incorporation of 18O Journal of the Chemical Society - Series Chemical Communications. 2507-2508. DOI: 10.1039/C39940002507  0.638
1993 Vishwakarma RA, Balachandran S, Alanine AID, Stamford NPJ, Kiuchi F, Leeper FJ, Battersby AR. Biosynthesis of porphyrins and related macrocycles. Part 41. Fate of oxygen atoms as precorrin-2 carrying eight labelled carboxyl groups ( 13C18O2H) is enzymatically converted into cobyrinic acid Journal of the Chemical Society, Perkin Transactions 1. 2893-2899. DOI: 10.1039/P19930002893  0.638
1992 Vishwakarma RA, Mehrotra R, Tripathi R, Dutta GP. Stereoselective Synthesis and Antimalarial Activity of α-Artelinic Acid from Artemisinin Journal of Natural Products. 55: 1142-1144. PMID 1431937 DOI: 10.1021/Np50086A018  0.394
1992 Tandon JS, Roy R, Balachandran S, Vishwakarma RA. Epi-deoxycoleonol, a new antihypertensive labdane diterpenoid from Coleus forskohlii Bioorganic and Medicinal Chemistry Letters. 2: 249-254. DOI: 10.1016/S0960-894X(01)81074-X  0.367
1991 Tripathi R, Dutta GP, Vishwakarma RA. Gametocytocidal activity of the antimalarial alpha/beta arteether against Plasmodium cynomolgi B. The American Journal of Tropical Medicine and Hygiene. 43: 571-5. PMID 2267960 DOI: 10.4269/AJTMH.1990.43.571  0.253
1991 Tripathi R, Dutta GP, Vishwakarma RA. Comparison of antimalarial efficacy of alpha, beta, and alpha/beta arteether against Plasmodium cynomolgi B infection in monkeys. The American Journal of Tropical Medicine and Hygiene. 44: 560-3. PMID 2063959 DOI: 10.4269/AJTMH.1991.44.560  0.2
1991 Agrawal PK, Vishwakarma RA, Jain DC, Roy R. High field NMR spectroscopic studies of arteannuin B and a reappraisal of the structure of arteannuin C Phytochemistry. 30: 3469-3471. DOI: 10.1016/0031-9422(91)83234-C  0.368
1990 Roy R, Vishwakarma RA, Varma N, Tandon JS. Coleonolic acid, a rearranged ursane triterpenoid from coleus forskohlII Tetrahedron Letters. 31: 3467-3470. DOI: 10.1016/S0040-4039(00)97424-0  0.383
1990 Vishwakarma RA, Tandon JS. Stereoisomers of coleonol (forskolin) and related diterpenoids Tetrahedron Letters. 31: 7493-7494. DOI: 10.1016/S0040-4039(00)88525-1  0.364
1989 Dutta GP, Bajpai R, Vishwakarma RA. Antimalarial efficacy of arteether against multiple drug resistant strain of plasmodium yoelii nigeriensis Pharmacological Research. 21: 415-419. PMID 2771860 DOI: 10.1016/1043-6618(89)90159-X  0.344
1989 Dutta GP, Bajpai R, Vishwakarma RA. Artemisinin (Qinghaosu)-a new gametocytocidal drug for malaria Chemotherapy. 35: 200-207. PMID 2766860 DOI: 10.1159/000238671  0.343
1989 Bajpai R, Dutta GP, Vishwakarma RA. Blood schizontocidal activity of a new antimalarial drug, arteether (α/β), against plasmodium knowlesi in rhesus monkeys Transactions of the Royal Society of Tropical Medicine and Hygiene. 83: 484-484. PMID 2617597 DOI: 10.1016/0035-9203(89)90257-5  0.364
1989 Kar K, Nath A, Bajpai R, Dutta GP, Vishwakarma RA. Pharmacology of alpha/beta arteether--a potential antimalarial drug. Journal of Ethnopharmacology. 27: 297-305. PMID 2615435 DOI: 10.1016/0378-8741(89)90004-4  0.384
1989 Dutta GP, Bajpai R, Vishwakarma RA. Comparison of antimalarial efficacy of artemisinin (Qinghaosu) and arteether against plasmodium cynomolgi b infection in monkeys Transactions of the Royal Society of Tropical Medicine and Hygiene. 83: 56-57. PMID 2603208 DOI: 10.1016/0035-9203(89)90704-9  0.357
1989 Mehrotra R, Ahmed B, Vishwakarma RA, Thakur RS. Verbacoside: A New Luteolin Glycoside from Verbascum thapsus Journal of Natural Products. 52: 640-643. DOI: 10.1021/Np50063A028  0.352
1989 Vishwakarma RA. Spiroforskolin: acid-catalysed rearrangement product of forskolin Tetrahedron Letters. 30: 131-132. DOI: 10.1016/S0040-4039(01)80343-9  0.369
1989 Mehrotra R, Vishwakarma R, Thakur R. Abietane diterpenoids from Coleus zeylanicus Phytochemistry. 28: 3135-3137. DOI: 10.1016/0031-9422(89)80293-6  0.352
1988 Ahmed B, Vishwakarma RA. Coleoside, a monoterpene glycoside from Coleus forskohlii Phytochemistry. 27: 3309-3310. DOI: 10.1016/0031-9422(88)80050-5  0.371
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