Truong Thanh Tung, Ph.D - Related publications

2014-2018 Drug Design and Pharmacology University of Copenhagen, København, Denmark 
 2018- Chemistry University of Pittsburgh, Pittsburgh, PA, United States 
Medicinal chemistry
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50 most relevant papers in past 60 days:
Year Citation  Score
2021 Zhou TS, He LL, He J, Yang ZK, Zhou ZY, Du AQ, Yu JB, Li YS, Wang SJ, Wei B, Cui ZN, Wang H. Discovery of a series of 5-phenyl-2-furan derivatives containing 1,3-thiazole moiety as potent Escherichia coli β-glucuronidase inhibitors. Bioorganic Chemistry. 116: 105306. PMID 34521047 DOI: 10.1016/j.bioorg.2021.105306   
2021 Hamdy R, Fayed B, Mostafa A, Shama NMA, Mahmoud SH, Mehta CH, Nayak Y, M Soliman SS. Iterated Virtual Screening-Assisted Antiviral and Enzyme Inhibition Assays Reveal the Discovery of Novel Promising Anti-SARS-CoV-2 with Dual Activity. International Journal of Molecular Sciences. 22. PMID 34445763 DOI: 10.3390/ijms22169057   
2021 Hernández-Ochoa B, Navarrete-Vázquez G, Aguayo-Ortiz R, Ortiz-Ramírez P, Morales-Luna L, Martínez-Rosas V, González-Valdez A, Gómez-Chávez F, Enríquez-Flores S, Wong-Baeza C, Baeza-Ramírez I, Pérez de la Cruz V, Gómez-Manzo S. Identification and In Silico Characterization of Novel Glucose-6-Phosphate Dehydrogenase Inhibitors. Molecules (Basel, Switzerland). 26. PMID 34443540 DOI: 10.3390/molecules26164955   
2021 Li J, Li Z, Chen T, Ye G, Qiu L, Long Y. New azaphilones from mangrove endophytic fungus SCNU-F0040. Natural Product Research. 1-9. PMID 34498957 DOI: 10.1080/14786419.2021.1959580   
2021 Wichur T, Pasieka A, Godyń J, Panek D, Góral I, Latacz G, Honkisz-Orzechowska E, Bucki A, Siwek A, Głuch-Lutwin M, Knez D, Brazzolotto X, Gobec S, Kołaczkowski M, Sabate R, et al. Discovery of 1-(phenylsulfonyl)-1H-indole-based multifunctional ligands targeting cholinesterases and 5-HT receptor with anti-aggregation properties against amyloid-beta and tau. European Journal of Medicinal Chemistry. 225: 113783. PMID 34461507 DOI: 10.1016/j.ejmech.2021.113783   
2021 Afzal O, Altamimi ASA, Shahroz MM, Sharma HK, Riadi Y, Hassan MQ. Analgesic and Anticancer Activity of Benzoxazole Clubbed 2-Pyrrolidinones as Novel Inhibitors of Monoacylglycerol Lipase. Molecules (Basel, Switzerland). 26. PMID 33924091 DOI: 10.3390/molecules26082389   
2021 Zhang L, Feng XZ, Xiao ZQ, Fan GR, Chen SX, Liao SL, Luo H, Wang ZD. Design, Synthesis, Antibacterial, Antifungal and Anticancer Evaluations of Novel -Pinene Quaternary Ammonium Salts. International Journal of Molecular Sciences. 22. PMID 34681957 DOI: 10.3390/ijms222011299   
2021 Ma S, Jiang W, Li Q, Li T, Wu W, Bai H, Shi B. Design, Synthesis, and Study of the Insecticidal Activity of Novel Steroidal 1,3,4-Oxadiazoles. Journal of Agricultural and Food Chemistry. PMID 34554742 DOI: 10.1021/acs.jafc.1c00088   
2021 Legru A, Verdirosa F, Hernandez JF, Tassone G, Sannio F, Benvenuti M, Conde PA, Bossis G, Thomas CA, Crowder MW, Dillenberger M, Becker K, Pozzi C, Mangani S, Docquier JD, et al. 1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-β-lactamase inhibitors with re-sensitization activity. European Journal of Medicinal Chemistry. 226: 113873. PMID 34626878 DOI: 10.1016/j.ejmech.2021.113873   
2021 Qi X, Chen WH, Lin XP, Liao SR, Yang B, Zhou XF, Liu YH, Wang JF, Li Y. A glyoxylate-containing benzene derivative and butenolides from a marine algicolous fungus sp. SCSIO 41304. Natural Product Research. 1-8. PMID 34542359 DOI: 10.1080/14786419.2021.1978994   
2021 Zhang JH, Xie HX, Li Y, Wang KM, Song Z, Zhu KK, Fang L, Zhang J, Jiang CS. Design, synthesis and biological evaluation of novel (E)-2-benzylidene-N-(3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophen-2-yl)hydrazine-1-carboxamide derivatives as α-glucosidase inhibitors. Bioorganic & Medicinal Chemistry Letters. 128413. PMID 34634473 DOI: 10.1016/j.bmcl.2021.128413   
2021 Mancuso F, De Luca L, Bucolo F, Vrabel M, Angeli A, Capasso C, Supuran CT, Gitto R. 4-Sulfamoylphenylalkylamides as Inhibitors of Carbonic Anhydrases Expressed in Vibrio cholerae. Chemmedchem. PMID 34592052 DOI: 10.1002/cmdc.202100510   
2021 Song L, Merceron R, Hulpia F, Lucía A, Gracia B, Jian Y, Risseeuw MDP, Verstraelen T, Cos P, Aínsa JA, Boshoff HI, Munier-Lehmann H, Savvides SN, Van Calenbergh S. Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors. European Journal of Medicinal Chemistry. 225: 113784. PMID 34450493 DOI: 10.1016/j.ejmech.2021.113784   
2021 Ghosh AK, Shahabi D, Yadav M, Kovela S, Anson BJ, Lendy EK, Bonham C, Sirohi D, Brito-Sierra CA, Hattori SI, Kuhn R, Mitsuya H, Mesecar AD. Chloropyridinyl Esters of Nonsteroidal Anti-Inflammatory Agents and Related Derivatives as Potent SARS-CoV-2 3CL Protease Inhibitors. Molecules (Basel, Switzerland). 26. PMID 34641337 DOI: 10.3390/molecules26195782   
2021 de Magalhães LS, Cotta Cardoso Reis A, Nakao IA, Péret VAC, Reis RCFM, Silva NC, Dias ALT, Carvalho DT, Dias DF, Brandão GC, Braga SFP, de Souza TB. Glucosyl-1,2,3-triazoles derived from eugenol and analogues: synthesis, anti-Candida activity and molecular modeling studies in CYP-51. Chemical Biology & Drug Design. PMID 34480517 DOI: 10.1111/cbdd.13948   
2021 Pokhrel S, Bouback TA, Samad A, Nur SM, Alam R, Abdullah-Al-Mamun M, Nain Z, Imon RR, Talukder MEK, Tareq MMI, Hossen MS, Karpiński TM, Ahammad F, Qadri I, Rahman MS. Spike protein recognizer receptor ACE2 targeted identification of potential natural antiviral drug candidates against SARS-CoV-2. International Journal of Biological Macromolecules. PMID 34592225 DOI: 10.1016/j.ijbiomac.2021.09.146   
2021 Mou H, Shi J, Chen J, Hu D. Synthesis, antibacterial activity and mechanism of new butenolides derivatives containing an amide moiety. Pesticide Biochemistry and Physiology. 178: 104913. PMID 34446189 DOI: 10.1016/j.pestbp.2021.104913   
2021 Chen YJ, Ma KY, Du SS, Zhang ZJ, Wu TL, Sun Y, Liu YQ, Yin XD, Zhou R, Yan YF, Wang RX, He YH, Chu QR, Tang C. Antifungal Exploration of Quinoline Derivatives against Phytopathogenic Fungi Inspired by Quinine Alkaloids. Journal of Agricultural and Food Chemistry. PMID 34623798 DOI: 10.1021/acs.jafc.1c05677   
2021 Li H, He YH, Hu YM, Chu QR, Chen YJ, Wu ZR, Zhang ZJ, Liu YQ, Yang CJ, Liang HJ, Yan YF. Design, Synthesis, and Structure-Activity Relationship Studies of Magnolol Derivatives as Antifungal Agents. Journal of Agricultural and Food Chemistry. PMID 34582205 DOI: 10.1021/acs.jafc.1c01838   
2021 Khan IA, Ahmad M, Ashfaq UA, Sultan S, Zaki MEA. Discovery of Amide-Functionalized Benzimidazolium Salts as Potent α-Glucosidase Inhibitors. Molecules (Basel, Switzerland). 26. PMID 34443347 DOI: 10.3390/molecules26164760   
2021 Hu YW, Chen WH, Song MM, Pang XY, Tian XP, Wang FZ, Liu YH, Wang JF. Indole diketopiperazine alkaloids and aromatic polyketides from the Antarctic fungus sp. SCSIO 05705. Natural Product Research. 1-9. PMID 34498972 DOI: 10.1080/14786419.2021.1973460   
2021 Barbosa da Silva E, Rocha DA, Fortes IS, Yang W, Monti L, Siqueira-Neto JL, Caffrey CR, McKerrow J, Andrade SF, Ferreira RS. Structure-Based Optimization of Quinazolines as Cruzain and CATL Inhibitors. Journal of Medicinal Chemistry. PMID 34461718 DOI: 10.1021/acs.jmedchem.1c01151   
2021 Zheng PF, Xiong Z, Liao CY, Zhang X, Feng M, Wu XZ, Lin J, Lei LS, Zhang YC, Wang SH, Xu XT. and studies of bis (indol-3-yl) methane derivatives as potential α-glucosidase and α-amylase inhibitors. Journal of Enzyme Inhibition and Medicinal Chemistry. 36: 1938-1951. PMID 34459690 DOI: 10.1080/14756366.2021.1971976   
2021 Wang Y, Wang J, Wang S, Cao Z, Gu D, Wang Y, Tian J, Yang Y. An efficient method based on an inhibitor-enzyme complex to screen an active compound against lipase from . Food & Function. PMID 34617090 DOI: 10.1039/d1fo01542g   
2021 Malani A, Makwana A, Monapara J, Ahmad I, Patel H, Desai N. Synthesis, molecular docking, DFT study, and in vitro antimicrobial activity of some 4-(biphenyl-4-yl)-1,4-dihydropyridine and 4-(biphenyl-4-yl)pyridine derivatives. Journal of Biochemical and Molecular Toxicology. e22903. PMID 34459052 DOI: 10.1002/jbt.22903   
2021 Wang Z, Zang R, Niu Z, Wang W, Wang X, Tang Y. Synthesis and antiviral effect of phosphamide modified vidarabine for treating HSV 1 infections. Bioorganic & Medicinal Chemistry Letters. 128405. PMID 34624489 DOI: 10.1016/j.bmcl.2021.128405   
2021 Suwanhom P, Saetang J, Khongkow P, Nualnoi T, Tipmanee V, Lomlim L. Synthesis, Biological Evaluation, and In Silico Studies of New Acetylcholinesterase Inhibitors Based on Quinoxaline Scaffold. Molecules (Basel, Switzerland). 26. PMID 34443482 DOI: 10.3390/molecules26164895   
2021 Zhang XW, Bian GL, Kang PY, Cheng XJ, Yan K, Liu YL, Gao YX, Li DQ. Recent advance in the discovery of tyrosinase inhibitors from natural sources via separation methods. Journal of Enzyme Inhibition and Medicinal Chemistry. 36: 2104-2117. PMID 34579614 DOI: 10.1080/14756366.2021.1983559   
2021 Chen T, Li WQ, Liu Z, Jiang W, Liu T, Yang Q, Zhu XL, Yang GF. Discovery of Biphenyl-Sulfonamides as Novel β--Acetyl-d-Hexosaminidase Inhibitors via Structure-Based Virtual Screening. Journal of Agricultural and Food Chemistry. PMID 34587743 DOI: 10.1021/acs.jafc.1c01642   
2021 Ghosh AK, Raghavaiah J, Shahabi D, Yadav M, Anson BJ, Lendy EK, Hattori SI, Higashi-Kuwata N, Mitsuya H, Mesecar AD. Indole Chloropyridinyl Ester-Derived SARS-CoV-2 3CLpro Inhibitors: Enzyme Inhibition, Antiviral Efficacy, Structure-Activity Relationship, and X-ray Structural Studies. Journal of Medicinal Chemistry. PMID 34528437 DOI: 10.1021/acs.jmedchem.1c01214   
2021 Taha M, Alrashedy AS, Almandil NB, Iqbal N, Anouar EH, Nawaz M, Uddin N, Chigurupati S, Wadood A, Rahim F, Das S, Venugopal V, Nawaz F, Khan KM. Synthesis of indole derivatives as diabetics II inhibitors and enzymatic kinetics study of α-glucosidase and α-amylase along with their in-silico study. International Journal of Biological Macromolecules. 190: 301-318. PMID 34481854 DOI: 10.1016/j.ijbiomac.2021.08.207   
2021 Sadiq Butt AR, Abbasi MA, Rehman AU, Siddiqui SZ, Raza H, Hassan M, Shah SAA, Seo SY. Synthesis, Kinetics, Binding Conformations and Structure-activity Relationship of Potent Tyrosinase Inhibitors: Aralkylated 2-aminothiazole-ethyltriazole Hybrids. Iranian Journal of Pharmaceutical Research : Ijpr. 20: 206-228. PMID 34567157 DOI: 10.22037/ijpr.2020.15521.13145   
2021 Hua X, Liu W, Chen Y, Ru J, Guo S, Yu X, Cui Y, Liu X, Gu Y, Xue C, Liu Y, Sui J, Wang G. Synthesis, Fungicidal Activity, and Mechanism of Action of Pyrazole Amide and Ester Derivatives Based on Natural Products l-Serine and Waltherione Alkaloids. Journal of Agricultural and Food Chemistry. PMID 34543010 DOI: 10.1021/acs.jafc.1c01346   
2021 Wu C, Cui X, Sun L, Lu J, Li F, Song M, Zhang Y, Hao X, Tian C, Song M, Liu X. Aspulvinones Suppress Postprandial Hyperglycemia as Potent α-Glucosidase Inhibitors From ASM-1. Frontiers in Chemistry. 9: 736070. PMID 34485249 DOI: 10.3389/fchem.2021.736070   
2021 Cui J, Jia J. Discovery of juglone and its derivatives as potent SARS-CoV-2 main proteinase inhibitors. European Journal of Medicinal Chemistry. 225: 113789. PMID 34438124 DOI: 10.1016/j.ejmech.2021.113789   
2021 Česnek M, Šafránek M, Dračínský M, Tloušťová E, Mertlíková-Kaiserová H, Hayes MP, Watts VJ, Janeba Z. Halogen Dance-Based Synthesis of Phosphonomethoxyethyl (PME) Substituted 2-Aminothiazoles as Potent Inhibitors of Bacterial Adenylate Cyclases. Chemmedchem. PMID 34636150 DOI: 10.1002/cmdc.202100568   
2021 Kanada R, Suzuki T, Murata T, Miyazaki M, Shimada T, Kuroha M, Minami M, Higuchi S, Tominaga Y, Naito H. 4-Pyridone-3-carboxylic acid as a benzoic acid bioisostere: Design, synthesis, and evaluation of EP300/CBP histone acetyltransferase inhibitors. Bioorganic & Medicinal Chemistry Letters. 128358. PMID 34534674 DOI: 10.1016/j.bmcl.2021.128358   
2021 Dissanayake AA, Mills GL, Bonito G, Rennick B, Nair MG. Chemical Composition and Anti-Inflammatory and Antioxidant Activities of Extracts from Cultivated Morel Mushrooms, Species of Genus Morchella (Ascomycota). International Journal of Medicinal Mushrooms. 23: 73-83. PMID 34591400 DOI: 10.1615/IntJMedMushrooms.2021039297   
2021 Kim JH, Vinh LB, Hur M, Koo SC, Park WT, Moon YH, Lee YJ, Kim YH, Huh YC, Yang SY. Inhibitory activity of 4-O-benzoyl-3'-O-(-methylsinapoyl)sucrose from on β-glucuronidase. Journal of Microbiology and Biotechnology. 31. PMID 34528918 DOI: 10.4014/jmb.2108.08004   
2021 Friday SN, Cheng DW, Zagler SG, Zanella BS, Dietz JD, Calbat CN, Roach LT, Bagnal C, Faile IS, Halkides CJ, Viola RE. Design and testing of selective inactivators against an antifungal enzyme target. Drug Development Research. PMID 34469014 DOI: 10.1002/ddr.21875   
2021 Zhang B, Duan Y, Yang Y, Mao Q, Lin F, Gao J, Dai X, Zhang P, Li Q, Li J, Dai R, Wang S. Design, synthesis, and biological evaluation of N-(3-cyano-1H-indol-5/6-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides and 5-(6-oxo-1,6-dihydropyrimidin-2-yl)-1H-indole-3-carbonitriles as novel xanthine oxidase inhibitors. European Journal of Medicinal Chemistry. 227: 113928. PMID 34688012 DOI: 10.1016/j.ejmech.2021.113928   
2021 Nadeem MS, Khan JA, Rashid U. Fluoxetine and sertraline based multitarget inhibitors of cholinesterases and monoamine oxidase-A/B for the treatment of Alzheimer's disease: Synthesis, pharmacology and molecular modeling studies. International Journal of Biological Macromolecules. PMID 34687762 DOI: 10.1016/j.ijbiomac.2021.10.102   
2021 Ali JS, Riaz N, Mannan A, Latif M, Zia M. Antioxidant, antimicrobial, enzyme inhibition, and cytotoxicity guided investigation of (A.DC.) T.D. Penn. leaves extracts. Natural Product Research. 1-4. PMID 34498973 DOI: 10.1080/14786419.2021.1973461   
2021 Zhu X, Chen S, Zheng Y, Zhang Y, Hsiang T, Huang R, Qi J, Gan T, Chang Y, Li J. Antifungal and insecticidal activities of rhein derivatives: synthesis, characterization and preliminary structure-activity relationship studies. Natural Product Research. 1-7. PMID 34533080 DOI: 10.1080/14786419.2021.1977804   
2021 Rocha K, Magallon J, Reeves C, Phan K, Vu P, Oakley-Havens CL, Kwan S, Ramirez MS, LaVoi T, Donow H, Chapagain P, Santos R, Pinilla C, Giulianotti MA, Tolmasky ME. Inhibition of Aminoglycoside 6'--acetyltransferase Type Ib (AAC(6')-Ib): Structure-Activity Relationship of Substituted Pyrrolidine Pentamine Derivatives as Inhibitors. Biomedicines. 9. PMID 34572404 DOI: 10.3390/biomedicines9091218   
2021 Ryan MD, Parkes AL, Corbett D, Dickie AP, Southey M, Andersen OA, Stein DB, Barbeau OR, Sanzone A, Thommes P, Barker J, Cain R, Compper C, Dejob M, Dorali A, et al. Discovery of Novel UDP--Acetylglucosamine Acyltransferase (LpxA) Inhibitors with Activity against . Journal of Medicinal Chemistry. PMID 34569791 DOI: 10.1021/acs.jmedchem.1c00888   
2021 Gao Z, Huang XY, Geng CA, Li TZ, Chen JJ. Artemicapillasins A-N, cytotoxic coumaric acid analogues against hepatic stellate cell LX2 from Artemisia capillaris (Yin-Chen). Bioorganic Chemistry. 117: 105441. PMID 34695731 DOI: 10.1016/j.bioorg.2021.105441   
2021 Hamad A, Khan MA, Ahmad I, Khalil R, Khalid M, Abbas U, Azhar R, Uddin J, Batiha GE, Khan A, Shafiq Z, Al-Harrasi A. Bio-oriented synthesis of new sulphadiazine derivatives for urease inhibition and their pharmacokinetic analysis. Scientific Reports. 11: 18973. PMID 34556784 DOI: 10.1038/s41598-021-98413-x   
2021 Nhoek P, Ahn S, Park IG, Pel P, Huh J, Kim HW, Ahn J, Khiev P, Choi YH, Lee K, Noh M, Chin YW. Salicinoyl Quinic Acids and Their Prostaglandin E Production Inhibitory Activities from the Fruits of . Journal of Natural Products. PMID 34463498 DOI: 10.1021/acs.jnatprod.1c00343   
2021 Wang S, Chen J, Shi J, Wang Z, Hu D, Song B. Novel Cinnamic Acid Derivatives Containing the 1,3,4-Oxadiazole Moiety: Design, Synthesis, Antibacterial Activities, and Mechanisms. Journal of Agricultural and Food Chemistry. PMID 34597041 DOI: 10.1021/acs.jafc.1c03087