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L.-C. Campeau - Publications

Affiliations: 
2007- Process Chemistry Merck & Co., Inc. 
Area:
Drug Discovery & Development
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40/75 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Davison EK, Petrone DA, Meanwell M, Nodwell MB, Silverman SM, Campeau LC, Britton R. Practical and concise synthesis of nucleoside analogs. Nature Protocols. PMID 35788720 DOI: 10.1038/s41596-022-00705-7  0.337
2022 Gabbey AL, Michel NWM, Hughes JME, Campeau LC, Rousseaux SAL. Synthesis of α-Aryl Secondary Amides via Nickel-Catalyzed Reductive Coupling of Redox-Active Esters. Organic Letters. PMID 35471845 DOI: 10.1021/acs.orglett.2c00918  0.607
2021 Meanwell M, Fehr G, Ren W, Adluri B, Rose V, Lehmann J, Silverman SM, Rowshanpour R, Adamson C, Bergeron-Brlek M, Foy H, Challa VR, Campeau LC, Dudding T, Britton R. Diversity-oriented synthesis of glycomimetics. Communications Chemistry. 4: 96. PMID 36697548 DOI: 10.1038/s42004-021-00520-3  0.317
2021 Piou T, Campeau LC. Bringing amines back into aziridination. Nature Chemistry. 13: 1027-1028. PMID 34697398 DOI: 10.1038/s41557-021-00819-7  0.416
2021 Klapars A, Chung JYL, Limanto J, Calabria R, Campeau LC, Campos KR, Chen W, Dalby SM, Davis TA, DiRocco DA, Hyde AM, Kassim AM, Larsen MU, Liu G, Maligres PE, et al. Efficient synthesis of antiviral agent uprifosbuvir enabled by new synthetic methods. Chemical Science. 12: 9031-9036. PMID 34276931 DOI: 10.1039/d1sc01978c  0.367
2020 Meanwell M, Silverman SM, Lehmann J, Adluri B, Wang Y, Cohen R, Campeau LC, Britton R. A short de novo synthesis of nucleoside analogs. Science (New York, N.Y.). 369: 725-730. PMID 32764073 DOI: 10.1126/Science.Abb3231  0.412
2019 Campeau LC, Hazari N. Cross-Coupling and Related Reactions: Connecting Past Success to the Development of New Reactions for the Future. Organometallics. 38: 3-35. PMID 31741548 DOI: 10.1021/acs.organomet.8b00720  0.461
2017 Ji Y, Li H, Hyde AM, Chen Q, Belyk KM, Lexa KW, Yin J, Sherer EC, Williamson RT, Brunskill A, Ren S, Campeau LC, Davies IW, Ruck RT. A rational pre-catalyst design for bis-phosphine mono-oxide palladium catalyzed reactions. Chemical Science. 8: 2841-2851. PMID 28553522 DOI: 10.1039/C6Sc05472B  0.409
2017 DiRocco DA, Ji Y, Sherer EC, Klapars A, Reibarkh M, Dropinski J, Mathew R, Maligres P, Hyde AM, Limanto J, Brunskill A, Ruck RT, Campeau LC, Davies IW. A multifunctional catalyst that stereoselectively assembles prodrugs. Science (New York, N.Y.). 356: 426-430. PMID 28450641 DOI: 10.1126/Science.Aam7936  0.319
2016 Yayla HG, Peng F, Mangion IK, McLaughlin M, Campeau LC, Davies IW, DiRocco DA, Knowles RR. Discovery and mechanistic study of a photocatalytic indoline dehydrogenation for the synthesis of elbasvir. Chemical Science. 7: 2066-2073. PMID 29899932 DOI: 10.1039/C5Sc03350K  0.309
2016 Kutchukian PS, Dropinski JF, Dykstra KD, Li B, DiRocco DA, Streckfuss EC, Campeau LC, Cernak T, Vachal P, Davies IW, Krska SW, Dreher SD. Chemistry informer libraries: a chemoinformatics enabled approach to evaluate and advance synthetic methods. Chemical Science. 7: 2604-2613. PMID 28660032 DOI: 10.1039/C5Sc04751J  0.304
2016 Joshi-Pangu A, Lévesque F, Roth HG, Oliver SF, Campeau LC, Nicewicz D, DiRocco DA. Acridinium-Based Photocatalysts: A Sustainable Option in Photoredox Catalysis. The Journal of Organic Chemistry. PMID 27454776 DOI: 10.1021/Acs.Joc.6B01240  0.332
2016 Williams MJ, Kong J, Chung CK, Brunskill A, Campeau LC, McLaughlin M. The Discovery of Quinoxaline-Based Metathesis Catalysts from Synthesis of Grazoprevir (MK-5172). Organic Letters. PMID 27123552 DOI: 10.1021/Acs.Orglett.6B00070  0.337
2016 Shevlin M, Friedfeld MR, Sheng H, Pierson NA, Hoyt JM, Campeau LC, Chirik PJ. Nickel-Catalyzed Asymmetric Alkene Hydrogenation of α,β-Unsaturated Esters: High-Throughput Experimentation-Enabled Reaction Discovery, Optimization, and Mechanistic Elucidation. Journal of the American Chemical Society. PMID 26890979 DOI: 10.1021/Jacs.6B00519  0.381
2016 Friedfeld MR, Shevlin M, Margulieux GW, Campeau LC, Chirik PJ. Cobalt-Catalyzed Enantioselective Hydrogenation of Minimally Functionalized Alkenes: Isotopic Labeling Provides Insight into the Origin of Stereoselectivity and Alkene Insertion Preferences. Journal of the American Chemical Society. PMID 26854359 DOI: 10.1021/Jacs.5B10148  0.361
2016 Kutchukian PS, Dropinski JF, Dykstra KD, Li B, Dirocco DA, Streckfuss EC, Campeau LC, Cernak T, Vachal P, Davies IW, Krska SW, Dreher SD. Chemistry informer libraries: A chemoinformatics enabled approach to evaluate and advance synthetic methods Chemical Science. 7: 2604-2613. DOI: 10.1039/c5sc04751j  0.305
2016 Yayla HG, Peng F, Mangion IK, McLaughlin M, Campeau LC, Davies IW, Dirocco DA, Knowles RR. Discovery and mechanistic study of a photocatalytic indoline dehydrogenation for the synthesis of elbasvir Chemical Science. 7: 2066-2073. DOI: 10.1039/c5sc03350k  0.324
2015 Halperin SD, Kwon D, Holmes M, Regalado EL, Campeau LC, DiRocco DA, Britton R. Development of a Direct Photocatalytic C-H Fluorination for the Preparative Synthesis of Odanacatib. Organic Letters. 17: 5200-3. PMID 26484983 DOI: 10.1021/Acs.Orglett.5B02532  0.376
2015 Li H, Belyk KM, Yin J, Chen Q, Hyde A, Ji Y, Oliver S, Tudge MT, Campeau LC, Campos KR. Enantioselective Synthesis of Hemiaminals via Pd-Catalyzed C-N Coupling with Chiral Bisphosphine Mono-Oxides. Journal of the American Chemical Society. PMID 26414910 DOI: 10.1021/jacs.5b05934  0.422
2015 Buitrago Santanilla A, Christensen M, Campeau LC, Davies IW, Dreher SD. P2Et Phosphazene: A Mild, Functional Group Tolerant Base for Soluble, Room Temperature Pd-Catalyzed C-N, C-O, and C-C Cross-Coupling Reactions. Organic Letters. PMID 26099020 DOI: 10.1021/acs.orglett.5b01648  0.345
2015 Buitrago Santanilla A, Regalado EL, Pereira T, Shevlin M, Bateman K, Campeau LC, Schneeweis J, Berritt S, Shi ZC, Nantermet P, Liu Y, Helmy R, Welch CJ, Vachal P, Davies IW, et al. Organic chemistry. Nanomole-scale high-throughput chemistry for the synthesis of complex molecules. Science (New York, N.Y.). 347: 49-53. PMID 25554781 DOI: 10.1126/Science.1259203  0.415
2014 McCabe Dunn JM, Kuethe JT, Orr RK, Tudge M, Campeau LC. Development of a palladium-catalyzed α-arylation of cyclopropyl nitriles. Organic Letters. 16: 6314-7. PMID 25474721 DOI: 10.1021/ol5030426  0.438
2010 Sun HY, Gorelsky SI, Stuart DR, Campeau LC, Fagnou K. Mechanistic analysis of azine N-oxide direct arylation: evidence for a critical role of acetate in the Pd(OAc)2 precatalyst. The Journal of Organic Chemistry. 75: 8180-9. PMID 21053903 DOI: 10.1021/Jo101821R  0.695
2010 Sun HY, Gorelsky SI, Stuart DR, Campeau LC, Fagnou K. Mechanistic analysis of azine N-oxide direct arylation: Evidence for a critical role of acetate in the Pd(OAc)2 precatalyst Journal of Organic Chemistry. 75: 8180-8189. DOI: 10.1021/jo101821r  0.603
2009 Campeau LC, Stuart DR, Leclerc JP, Bertrand-Laperle M, Villemure E, Sun HY, Lasserre S, Guimond N, Lecavallier M, Fagnou K. Palladium-catalyzed direct arylation of azine and azole N-oxides: Reaction development, scope and applications in synthesis Journal of the American Chemical Society. 131: 3291-3306. PMID 19215128 DOI: 10.1021/Ja808332K  0.723
2009 Schipper DJ, Campeau LC, Fagnou K. Catalyst and base controlled site-selective sp2 and sp3 direct arylation of azine N-oxides Tetrahedron. 65: 3155-3164. DOI: 10.1016/J.Tet.2008.12.004  0.755
2009 Schipper DJ, Campeau L, Fagnou K. ChemInform Abstract: Catalyst and Base Controlled Site-Selective sp2and sp3Direct Arylation of Azine N-Oxides. Cheminform. 40. DOI: 10.1002/CHIN.200932097  0.645
2008 Caron L, Campeau LC, Fagnou K. Palladium-catalyzed direct arylation of nitro-substituted aromatics with aryl halides. Organic Letters. 10: 4533-6. PMID 18811176 DOI: 10.1021/Ol801839W  0.741
2008 Campeau LC, Bertrand-Laperle M, Leclerc JP, Villemure E, Gorelsky S, Fagnou K. C2, C5, and C4 azole N-oxide direct arylation including room-temperature reactions Journal of the American Chemical Society. 130: 3276-3277. PMID 18302383 DOI: 10.1021/Ja7107068  0.606
2008 Campeau LC, Schipper DJ, Fagnou K. Site-selective sp2 and benzylic sp3 palladium-catalyzed direct arylation. Journal of the American Chemical Society. 130: 3266-7. PMID 18293986 DOI: 10.1021/Ja710451S  0.739
2008 Caron L, Campeau LC, Fagnou K. Palladium-catalyzed direct arylation of nitro-substituted aromatics with aryl halides Organic Letters. 10: 4533-4536. DOI: 10.1021/ol801839w  0.726
2007 Campeau LC, Fagnou K. Applications of and alternatives to π-electron-deficient azine organometallics in metal catalyzed cross-coupling reactions Chemical Society Reviews. 36: 1058-1068. PMID 17576474 DOI: 10.1039/B616082D  0.642
2006 Campeau LC, Fagnou K. Palladium-catalyzed direct arylation of simple arenes in synthesis of biaryl molecules Chemical Communications. 1253-1264. PMID 16538241 DOI: 10.1039/B515481M  0.728
2006 Campeau LC, Parisien M, Jean A, Fagnou K. Catalytic direct arylation with aryl chlorides, bromides, and iodides: intramolecular studies leading to new intermolecular reactions. Journal of the American Chemical Society. 128: 581-90. PMID 16402846 DOI: 10.1021/Ja055819X  0.757
2006 Campeau LC, Parisien M, Jean A, Fagnou K. Catalytic direct arylation with aryl chlorides, bromides, and iodides: Intramolecular studies leading to new intermolecular reactions Journal of the American Chemical Society. 128: 581-590. DOI: 10.1021/ja055819x  0.738
2005 Campeau LC, Rousseaux S, Fagnou K. A solution to the 2-pyridyl organometallic cross-coupling problem: regioselective catalytic direct arylation of pyridine N-oxides. Journal of the American Chemical Society. 127: 18020-1. PMID 16366550 DOI: 10.1021/Ja056800X  0.752
2005 Campeau LC, Thansandote P, Fagnou K. High-yielding intramolecular direct arylation reactions with aryl chlorides. Organic Letters. 7: 1857-60. PMID 15844924 DOI: 10.1021/Ol050501V  0.752
2005 Campeau LC, Thansandote P, Fagnou K. High-yielding intramolecular direct arylation reactions with aryl chlorides Organic Letters. 7: 1857-1860. DOI: 10.1021/ol050501v  0.725
2004 Campeau LC, Parisien M, Leblanc M, Fagnou K. Biaryl synthesis via direct arylation: establishment of an efficient catalyst for intramolecular processes. Journal of the American Chemical Society. 126: 9186-7. PMID 15281800 DOI: 10.1021/Ja049017Y  0.659
2004 Campeau LC, Parisien M, Leblanc M, Fagnou K. Biaryl synthesis via direct arylation: Establishment of an efficient catalyst for intramolecular processes Journal of the American Chemical Society. 126: 9186-9187. DOI: 10.1021/ja049017y  0.65
Low-probability matches (unlikely to be authored by this person)
2011 Campeau LC, Dolman SJ, Gauvreau D, Corley E, Liu J, Guidry EN, Ouellet SG, Steinhuebel D, Weisel M, O'Shea PD. Convergent kilo-scale synthesis of a potent renin inhibitor for the treatment of hypertension Organic Process Research and Development. 15: 1138-1148. DOI: 10.1021/Op2001063  0.284
2022 Nesic M, Ryffel DB, Maturano J, Shevlin M, Pollack SR, Gauthier DR, Trigo-Mouriño P, Zhang LK, Schultz DM, McCabe Dunn JM, Campeau LC, Patel NR, Petrone DA, Sarlah D. Total Synthesis of Darobactin A. Journal of the American Chemical Society. PMID 35900216 DOI: 10.1021/jacs.2c05891  0.239
2013 Girardin M, Ouellet SG, Gauvreau D, Moore JC, Hughes G, Devine PN, O'Shea PD, Campeau LC. Convergent kilogram-scale synthesis of dual orexin receptor antagonist Organic Process Research and Development. 17: 61-68. DOI: 10.1021/Op3002678  0.236
2016 Orr R, Campeau L, Chobanian H, McCabe Dunn J, Pio B, Plummer C, Nolting A, Ruck R. A Modular Synthesis of 2-Alkyl- and 2-Arylchromans via a Three-Step Sequence Synthesis. 49: 657-666. DOI: 10.1055/s-0036-1588075  0.231
2022 McIntosh JA, Liu Z, Andresen BM, Marzijarani NS, Moore JC, Marshall NM, Borra-Garske M, Obligacion JV, Fier PS, Peng F, Forstater JH, Winston MS, An C, Chang W, Lim J, ... ... Campeau LC, et al. A kinase-cGAS cascade to synthesize a therapeutic STING activator. Nature. 603: 439-444. PMID 35296845 DOI: 10.1038/s41586-022-04422-9  0.223
2011 Koay N, Campeau L. ChemInform Abstract: Efficient Preparation of 3-Substituted Quinazolinediones Directly from Anthranilic Acids and Isocyanates. Cheminform. 42: no-no. DOI: 10.1002/CHIN.201133162  0.215
2010 Koay N, Campeau L. Efficient preparation of 3-substituted quinazolinediones directly from anthranilic acids and isocyanates Journal of Heterocyclic Chemistry. 48: 473-478. DOI: 10.1002/JHET.551  0.201
2016 Campeau LC, Chen Q, Gauvreau D, Girardin M, Belyk K, Maligres P, Zhou G, Gu C, Zhang W, Tan L, O'Shea PD. A Robust Kilo-Scale Synthesis of Doravirine Organic Process Research and Development. 20: 1476-1481. DOI: 10.1021/acs.oprd.6b00163  0.188
2016 Christensen M, Nolting A, Shevlin M, Weisel M, Maligres PE, Lee J, Orr RK, Plummer CW, Tudge MT, Campeau LC, Ruck RT. Enantioselective Synthesis of α-Methyl-β-Cyclopropyldihydrocinnamates. The Journal of Organic Chemistry. PMID 26743694 DOI: 10.1021/acs.joc.5b02296  0.184
2020 Nilova A, Campeau LC, Sherer EC, Stuart DR. Analysis of Benzenoid Substitution Patterns in Small Molecule Active Pharmaceutical Ingredients. Journal of Medicinal Chemistry. PMID 32786676 DOI: 10.1021/Acs.Jmedchem.0C00915  0.179
2015 Liu P, Hu Z, DuBois BG, Moyes CR, Hunter DN, Zhu C, Kar NF, Zhu Y, Garfunkle J, Kang L, Chicchi G, Ehrhardt A, Woods A, Seo T, Woods M, ... ... Campeau LC, et al. Design of Potent and Orally Active GPR119 Agonists for the Treatment of Type II Diabetes. Acs Medicinal Chemistry Letters. 6: 936-41. PMID 26288697 DOI: 10.1021/acsmedchemlett.5b00207  0.154
2012 Ouellet SG, Gauvreau D, Cameron M, Dolman S, Campeau LC, Hughes G, O'Shea PD, Davies IW. Convergent, fit-for-purpose, kilogram-scale synthesis of a 5-lipoxygenase inhibitor Organic Process Research and Development. 16: 214-219. DOI: 10.1021/op200299p  0.13
2024 Michel NWM, Gabbey AL, Edjoc RK, Fagbola E, Hughes JME, Campeau LC, Rousseaux SAL. Nickel-Catalyzed Reductive Arylation of Redox Active Esters for the Synthesis of α-Aryl Nitriles: Investigation of a Chlorosilane Additive. The Journal of Organic Chemistry. PMID 38197128 DOI: 10.1021/acs.joc.3c02354  0.12
2024 Campeau LC, Horwitz MA, Schultz DM. Should You Start a Chemistry Podcast? Organic Letters. PMID 38169530 DOI: 10.1021/acs.orglett.3c04181  0.12
2011 Chen A, Campeau LC, Cauchon E, Chefson A, Ducharme Y, Dubé D, Falgueyret JP, Fournier PA, Gagné S, Grimm E, Han Y, Houle R, Huang JQ, Lacombe P, Laliberté S, et al. Renin inhibitors for the treatment of hypertension: design and optimization of a novel series of pyridone-substituted piperidines. Bioorganic & Medicinal Chemistry Letters. 21: 3970-5. PMID 21621998 DOI: 10.1016/j.bmcl.2011.05.013  0.117
2015 Meng D, Andre P, Bateman TJ, Berger R, Chen YH, Desai K, Dewnani S, Ellsworth K, Feng D, Geissler WM, Guo L, Hruza A, Jian T, Li H, Metzger J, ... ... Campeau LC, et al. Development of a novel tricyclic class of potent and selective FIXa inhibitors. Bioorganic & Medicinal Chemistry Letters. PMID 26318999 DOI: 10.1016/J.Bmcl.2015.07.078  0.109
2015 Zhang T, Andre P, Bateman TJ, Chen YH, Desai K, Ellsworth K, Geissler WM, Guo L, Hruza A, Jian T, Meng D, Parker DL, Qian X, Reichert P, Sherer EC, ... ... Campeau LC, et al. Development of a novel class of potent and selective FIXa inhibitors. Bioorganic & Medicinal Chemistry Letters. PMID 25978966 DOI: 10.1016/J.Bmcl.2015.04.057  0.107
2017 Zhu C, Wang L, Zhu Y, Guo ZZ, Liu P, Hu Z, Szewczyk JW, Kang L, Chicchi G, Ehrhardt A, Woods A, Seo T, Woods M, van Heek M, Dingley KH, ... ... Campeau LC, et al. Discovery of phenyl acetamides as potent and selective GPR119 agonists. Bioorganic & Medicinal Chemistry Letters. PMID 28185720 DOI: 10.1016/j.bmcl.2017.01.091  0.1
2012 Campeau L, Dolman SJ, Gauvreau D, Corley E, Liu J, Guidry EN, Ouellet SG, Steinhuebel D, Weisel M, O’Shea PD. Correction to Convergent Kilo-Scale Synthesis of a Potent Renin Inhibitor for the Treatment of Hypertension Organic Process Research & Development. 16: 1241-1241. DOI: 10.1021/op300123u  0.096
2017 Plummer CW, Clements MJ, Chen H, Rajagopalan M, Josien H, Hagmann WK, Miller M, Trujillo ME, Kirkland M, Kosinski D, Mane J, Pachanski M, Cheewatrakoolpong B, Nolting AF, Orr R, ... ... Campeau LC, et al. Design and Synthesis of Novel, Selective GPR40 AgoPAMs. Acs Medicinal Chemistry Letters. 8: 221-226. PMID 28197316 DOI: 10.1021/acsmedchemlett.6b00443  0.095
2019 Campeau L, Fogg DE. The Roles of Organometallic Chemistry in Pharmaceutical Research and Development Organometallics. 38: 1-2. DOI: 10.1021/Acs.Organomet.8B00918  0.095
2017 Boga SB, Christensen M, Perrotto N, Krska SW, Dreher S, Tudge MT, Ashley ER, Poirier M, Reibarkh M, Liu Y, Streckfuss E, Campeau L, Ruck RT, Davies IW, Vachal P. Selective functionalization of complex heterocycles via an automated strong base screening platform Reaction Chemistry & Engineering. 2: 446-450. DOI: 10.1039/C7Re00057J  0.095
2017 Schreier JD, Embrey MW, Raheem IT, Barbe G, Campeau LC, Dubost D, McCabe Dunn J, Grobler J, Hartingh TJ, Hazuda DJ, Klein D, Miller MD, Moore KP, Nguyen N, Pajkovic N, et al. Discovery and optimization of 2-pyridinone aminal integrase strand transfer inhibitors for the treatment of HIV. Bioorganic & Medicinal Chemistry Letters. PMID 28285916 DOI: 10.1016/j.bmcl.2017.02.039  0.087
2011 Levesque E, Campeau L, Gauvreau D. ChemInform Abstract: Convergent Approach to Nonsymmetrical 2,5-Diester Pyrroles. Cheminform. 42: no-no. DOI: 10.1002/CHIN.201117114  0.087
2011 Chen A, Aspiotis R, Campeau LC, Cauchon E, Chefson A, Ducharme Y, Falgueyret JP, Gagné S, Han Y, Houle R, Laliberté S, Larouche G, Lévesque JF, McKay D, Percival D. Renin inhibitors for the treatment of hypertension: design and optimization of a novel series of spirocyclic piperidines. Bioorganic & Medicinal Chemistry Letters. 21: 7399-404. PMID 22071301 DOI: 10.1016/j.bmcl.2011.10.013  0.083
2010 Campeau L, O'Shea P. Chemoselective Staudinger Strategy in the Practical, Fit for Purpose, Gram-Scale Synthesis of an HCV RNA Polymerase Inhibitor Synlett. 2011: 57-60. DOI: 10.1055/S-0030-1259085  0.076
2021 Vachal P, Duffy JL, Campeau LC, Amin RP, Mitra K, Murphy BA, Shao PP, Sinclair PJ, Ye F, Katipally R, Lu Z, Ondeyka D, Chen YH, Zhao K, Sun W, et al. Invention of MK-8262, a Cholesteryl Ester Transfer Protein (CETP) Inhibitor Backup to Anacetrapib with Best-in-Class Properties. Journal of Medicinal Chemistry. PMID 34375108 DOI: 10.1021/acs.jmedchem.1c00959  0.065
2010 Gauvreau D, Lévesque É, Campeau L. Convergent Approach to Nonsymmetrical 2,5-Diester Pyrroles Synlett. 2010: 3086-3088. DOI: 10.1055/S-0030-1259074  0.051
2014 Sheridan RP, Zorn N, Sherer EC, Campeau LC, Chang CZ, Cumming J, Maddess ML, Nantermet PG, Sinz CJ, O'Shea PD. Modeling a crowdsourced definition of molecular complexity. Journal of Chemical Information and Modeling. 54: 1604-16. PMID 24802889 DOI: 10.1021/Ci5001778  0.045
2014 Lai MT, Feng M, Falgueyret JP, Tawa P, Witmer M, DiStefano D, Li Y, Burch J, Sachs N, Lu M, Cauchon E, Campeau LC, Grobler J, Yan Y, Ducharme Y, et al. In vitro characterization of MK-1439, a novel HIV-1 nonnucleoside reverse transcriptase inhibitor Antimicrobial Agents and Chemotherapy. 58: 1652-1663. PMID 24379202 DOI: 10.1128/AAC.02403-13  0.04
2014 Côté B, Burch JD, Asante-Appiah E, Bayly C, Bédard L, Blouin M, Campeau LC, Cauchon E, Chan M, Chefson A, Coulombe N, Cromlish W, Debnath S, Deschênes D, Dupont-Gaudet K, et al. Discovery of MK-1439, an orally bioavailable non-nucleoside reverse transcriptase inhibitor potent against a wide range of resistant mutant HIV viruses. Bioorganic & Medicinal Chemistry Letters. 24: 917-22. PMID 24412110 DOI: 10.1016/J.Bmcl.2013.12.070  0.038
2020 Ren H, Maloney KM, Basu K, Di Maso MJ, Humphrey G, Peng F, Desmond R, Otte DAL, Alwdi E, Liu W, Zhang SW, Song S, Arvary RA, Zompa MA, Lehnherr D, ... ... Campeau LC, et al. Development of a Green & Sustainable Manufacturing Process for Gefapixant Citrate (MK-7264) Part 1: Introduction and Process Overview Org. Process Res. Dev.. DOI: 10.1021/acs.oprd.0c00248  0.037
2023 Johns DG, Campeau LC, Banka P, Bautmans A, Bueters T, Bianchi E, Branca D, Bulger PG, Crevecoeur I, Ding FX, Garbaccio RM, Guetschow ED, Guo Y, Ha SN, Johnston JM, et al. Orally Bioavailable Macrocyclic Peptide That Inhibits Binding of PCSK9 to the Low Density Lipoprotein Receptor. Circulation. PMID 37125593 DOI: 10.1161/CIRCULATIONAHA.122.063372  0.027
2015 Liu P, Hu Z, Dubois BG, Moyes CR, Hunter DN, Zhu C, Kar NF, Zhu Y, Garfunkle J, Kang L, Chicchi G, Ehrhardt A, Woods A, Seo T, Woods M, ... ... Campeau LC, et al. Design of Potent and Orally Active GPR119 Agonists for the Treatment of Type II Diabetes Acs Medicinal Chemistry Letters. 6: 936-941. DOI: 10.1021/acsmedchemlett.5b00207  0.02
2020 Schultz D, Campeau LC. Harder, better, faster. Nature Chemistry. PMID 32651465 DOI: 10.1038/S41557-020-0510-8  0.01
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