Jean Martinez - Publications

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500 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2021 Zajdel P, Grychowska K, Mogilski S, Kurczab R, Satała G, Bugno R, Kos T, Gołębiowska J, Malikowska-Racia N, Nikiforuk A, Chaumont-Dubel S, Bantreil X, Pawłowski M, Martinez J, Subra G, et al. Structure-Based Design and Optimization of FPPQ, a Dual-Acting 5-HT and 5-HT Receptor Antagonist with Antipsychotic and Procognitive Properties. Journal of Medicinal Chemistry. PMID 34467765 DOI: 10.1021/acs.jmedchem.1c00224  0.771
2021 Laconde G, Amblard M, Martinez J. Synthesis of α-Amino Acid -Carboxyanhydrides. Organic Letters. PMID 34369154 DOI: 10.1021/acs.orglett.1c02224  0.339
2021 Drop M, Jacquot F, Canale V, Chaumont-Dubel S, Walczak M, Satała G, Nosalska K, Mahoro GU, Słoczyńska K, Piska K, Lamoine S, Pękala E, Masurier N, Bojarski AJ, Pawłowski M, ... Martinez J, et al. Neuropathic pain-alleviating activity of novel 5-HT receptor inverse agonists derived from 2-aryl-1H-pyrrole-3-carboxamide. Bioorganic Chemistry. 115: 105218. PMID 34365058 DOI: 10.1016/j.bioorg.2021.105218  0.758
2021 Bourbiaux K, Legrand B, Verdié P, Mallart S, Manette G, Minoletti C, Stepp JD, Prigent P, Le Bail JC, Gauzy-Lazo L, Duclos O, Martinez J, Amblard M. Potent Lys Patch-Containing Stapled Peptides Targeting PCSK9. Journal of Medicinal Chemistry. PMID 34266235 DOI: 10.1021/acs.jmedchem.0c02051  0.349
2021 Valot L, Maumus M, Brunel L, Martinez J, Amblard M, Noël D, Mehdi A, Subra G. A Collagen-Mimetic Organic-Inorganic Hydrogel for Cartilage Engineering. Gels (Basel, Switzerland). 7. PMID 34203914 DOI: 10.3390/gels7020073  0.42
2021 Drop M, Canale V, Chaumont-Dubel S, Kurczab R, Satała G, Bantreil X, Walczak M, Koczurkiewicz-Adamczyk P, Latacz G, Gwizdak A, Krawczyk M, Gołębiowska J, Grychowska K, Bojarski AJ, Nikiforuk A, ... ... Martinez J, et al. 2-Phenyl-1-pyrrole-3-carboxamide as a New Scaffold for Developing 5-HT Receptor Inverse Agonists with Cognition-Enhancing Activity. Acs Chemical Neuroscience. PMID 33705101 DOI: 10.1021/acschemneuro.1c00061  0.798
2021 Malki Y, Martinez J, Masurier N. 1,3-Diazepine: A privileged scaffold in medicinal chemistry. Medicinal Research Reviews. PMID 33645848 DOI: 10.1002/med.21795  0.492
2021 Milbeo P, Martinez J, Amblard M, Calmès M, Legrand B. 1-Aminobicyclo[2.2.2]octane-2-carboxylic Acid and Derivatives As Chiral Constrained Bridged Scaffolds for Foldamers and Chiral Catalysts. Accounts of Chemical Research. PMID 33464823 DOI: 10.1021/acs.accounts.0c00680  0.811
2021 Maurel M, Montheil T, Martin J, Chaar L, Guzman-Gonzalez V, Couvet M, Jacquet T, Jia T, Eymin B, Parra K, Dumy P, Martinez J, Ruggiero F, Vaganay E, Mehdi A, et al. Design of PEGylated Three Ligands Silica Nanoparticles for Multi-Receptor Targeting. Nanomaterials (Basel, Switzerland). 11. PMID 33445812 DOI: 10.3390/nano11010177  0.699
2021 Yeboue Y, Jean M, Subra G, Martinez J, Lamaty F, Métro TX. Epimerization-Free C-Term Activation of Peptide Fragments by Ball Milling. Organic Letters. PMID 33393789 DOI: 10.1021/acs.orglett.0c03209  0.608
2020 Besserer-Offroy É, Tétreault P, Brouillette RL, René A, Murza A, Fanelli R, Kirby K, Parent A, Dubuc I, Beaudet N, Côté J, Longpré JM, Martinez J, Cavelier F, Sarret P. Data set describing the biological activity of JMV2009, a novel silylated neurotensin(8-13) analog. Data in Brief. 31: 105884. PMID 32637491 DOI: 10.1016/J.Dib.2020.105884  0.804
2020 Tétreault P, Besserer-Offroy É, Brouillette RL, René A, Murza A, Fanelli R, Kirby K, Parent AJ, Dubuc I, Beaudet N, Côté J, Longpré JM, Martinez J, Cavelier F, Sarret P. Pain relief devoid of opioid side effects following central action of a silylated neurotensin analog. European Journal of Pharmacology. 173174. PMID 32534076 DOI: 10.1016/J.Ejphar.2020.173174  0.787
2020 Milbeo P, Simon M, Didierjean C, Wenger E, Aubert E, Martinez J, Amblard M, Calmès M, Legrand B. A bicyclic unit reversal to stabilize the 12/14-helix in mixed homochiral oligoureas. Chemical Communications (Cambridge, England). PMID 32529998 DOI: 10.1039/D0Cc02902E  0.783
2020 Mehdi A, Julie M, Wehbi M, Echalier C, Hunger S, Bethry A, Garric X, Pinese C, Martinez J, Vezenkov L, Subra G. Direct synthesis of peptide-containing silicone. A new way for bioactive materials. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32516440 DOI: 10.1002/Chem.202001571  0.317
2020 Montheil T, Maumus M, Valot L, Lebrun A, Martinez J, Amblard M, Noël D, Mehdi A, Subra G. Inorganic Sol-Gel Polymerization for Hydrogel Bioprinting. Acs Omega. 5: 2640-2647. PMID 32095687 DOI: 10.1021/acsomega.9b03100  0.27
2020 Touati-Jallabe Y, Tintillier T, Mauchauffée E, Boucher JL, Leroy J, Ramassamy B, Hamzé A, Mezghenna K, Bouzekrini A, Verna C, Martinez J, Lajoix AD, Hernandez JF. Solid Phase Synthesis and Evaluation of Substrate-based Dipeptides and Heterocyclic Pseudo-dipeptides as Potential NO Synthases Inhibitors. Chemmedchem. PMID 32027778 DOI: 10.1002/Cmdc.201900659  0.505
2020 Moulat L, Martinez J, Salom-Roig XJ. Efficient monoacylation of symmetrical secondary alkanediamines and synthesis of unsymmetrical diacylated alkanediamines. A new L-proline-based organocatalyst Arkivoc. 2019: 336-349. DOI: 10.24820/Ark.5550190.P011.054  0.266
2020 Martinez J, Fehrentz J. From JMV-1843 to Macrilen Australian Journal of Chemistry. 73: 334-337. DOI: 10.1071/Ch19530  0.602
2020 Jebors S, Pinese C, Montheil T, Bethry A, Verquin S, Plais L, Moulin M, Dupont C, Garric X, Mehdi A, Martinez J, Subra G. Turning peptides into bioactive nylons European Polymer Journal. 135: 109886. DOI: 10.1016/J.Eurpolymj.2020.109886  0.338
2019 Valot L, Maumus M, Montheil T, Martinez J, Noël D, Mehdi A, Subra G. Biocompatible Glycine-Assisted Catalysis of the Sol-Gel Process: Development of Cell-Embedded Hydrogels. Chempluschem. 84: 1720-1729. PMID 31943873 DOI: 10.1002/Cplu.201900509  0.431
2019 Tourné-Péteilh C, Robin B, Lions M, Martinez J, Mehdi A, Subra G, Devoisselle JM. Combining sol-gel and microfluidics processes for the synthesis of protein-containing hybrid microgels. Chemical Communications (Cambridge, England). PMID 31612874 DOI: 10.1039/C9Cc04963K  0.425
2019 Martin J, Martinez J, Mehdi A, Subra G. Silicone grafted bioactive peptides and their applications. Current Opinion in Chemical Biology. 52: 125-135. PMID 31386969 DOI: 10.1016/J.Cbpa.2019.06.012  0.514
2019 Jia T, Ciccione J, Jacquet T, Maurel M, Montheil T, Mehdi A, Martinez J, Eymin B, Subra G, Coll JL. The presence of PEG on nanoparticles presenting the c[RGDfK]- and/or ATWLPPR peptides deeply affects the RTKs-AKT-GSK3β-eNOS signaling pathway and endothelial cells survival. International Journal of Pharmaceutics. 118507. PMID 31299336 DOI: 10.1016/J.Ijpharm.2019.118507  0.601
2019 Valot L, Martinez J, Mehdi A, Subra G. Chemical insights into bioinks for 3D printing. Chemical Society Reviews. PMID 31271159 DOI: 10.1039/C7Cs00718C  0.429
2019 Beillard A, Bantreil X, Métro TX, Martinez J, Lamaty F. Alternative Technologies That Facilitate Access to Discrete Metal Complexes. Chemical Reviews. PMID 31059243 DOI: 10.1021/Acs.Chemrev.8B00479  0.648
2019 Jebors S, Valot L, Echalier C, Legrand B, Mikhaleff R, Lee AVD, Arenal R, Dumy P, Amblard M, Martinez J, Mehdi A, Subra G. Self-mineralization and assembly of a bis-silylated Phe–Phe pseudodipeptide to a structured bioorganic–inorganic material Materials Horizons. 6: 2040-2046. DOI: 10.1039/C9Mh00580C  0.273
2019 Laconde G, Amblard M, Martinez J. A simple and versatile method to synthesize N-acyl-benzotriazoles Tetrahedron Letters. 60: 341-343. DOI: 10.1016/J.Tetlet.2018.12.046  0.345
2019 Echalier C, Valot L, Martinez J, Mehdi A, Subra G. Chemical cross-linking methods for cell encapsulation in hydrogels Materials Today Communications. 20: 100536. DOI: 10.1016/J.Mtcomm.2019.05.012  0.227
2019 Laconde G, Amblard M, Martinez J. Unexpected Reactivity of N‐Acyl‐Benzotriazoles with Aromatic Amines in Acidic Medium (ABAA Reaction) European Journal of Organic Chemistry. 2019: 85-90. DOI: 10.1002/Ejoc.201801567  0.266
2018 Montheil T, Echalier C, Martinez J, Subra G, Mehdi A. Inorganic polymerization: an attractive route to biocompatible hybrid hydrogels. Journal of Materials Chemistry. B. 6: 3434-3448. PMID 32254441 DOI: 10.1039/C8Tb00456K  0.237
2018 Masurier N, Tissot JB, Boukhriss D, Jebors S, Pinese C, Verdié P, Amblard M, Mehdi A, Martinez J, Humblot V, Subra G. Site-specific grafting on titanium surfaces with hybrid temporin antibacterial peptides. Journal of Materials Chemistry. B. 6: 1782-1790. PMID 32254250 DOI: 10.1039/C8Tb00051D  0.307
2018 Turolla EA, Valtorta S, Bresciani E, Fehrentz JA, Giuliano L, Stucchi S, Belloli S, Rainone P, Sudati F, Rizzi L, Molteni L, Verdiè P, Martinez J, Torsello A, Moresco RM, et al. Study of the Tissue Distribution of TLQP-21 in Mice Using [F]JMV5763, a Radiolabeled Analog Prepared via [F]Aluminum Fluoride Chelation Chemistry. Frontiers in Pharmacology. 9: 1274. PMID 30542281 DOI: 10.3389/Fphar.2018.01274  0.576
2018 Cheignon C, Cordeau E, Prache N, Cantel S, Martinez J, Subra G, Arnaudguilhem C, Bouyssiere B, Enjalbal C. Receptor-Ligand Interaction Measured by Inductively Coupled Plasma Mass Spectrometry and Selenium Labeling. Journal of Medicinal Chemistry. PMID 30395477 DOI: 10.1021/Acs.Jmedchem.8B01320  0.471
2018 Calmes M, Legrand B, Simon M, Aubert E, Milbeo P, Lui H, André C, Wenger E, Amblard M, Martinez J. 12/10-helix in mixed b-peptides alternating bicyclic and acyclic b-amino acids: probing the relationship between bicyclic side chain and helix stability. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30277633 DOI: 10.1002/Chem.201804404  0.792
2018 Ben Haj Salah K, Das S, Ruiz N, Andreu V, Martinez J, Wenger E, Amblard M, Didierjean C, Legrand B, Inguimbert N. How are 1,2,3-triazoles accommodated in helical secondary structures? Organic & Biomolecular Chemistry. PMID 29693098 DOI: 10.1039/C8Ob00686E  0.795
2018 Damian M, Pons V, Renault P, M'Kadmi C, Delort B, Hartmann L, Kaya AI, Louet M, Gagne D, Ben Haj Salah K, Denoyelle S, Ferry G, Boutin JA, Wagner R, Fehrentz JA, ... Martinez J, et al. GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation. Proceedings of the National Academy of Sciences of the United States of America. PMID 29632174 DOI: 10.1073/Pnas.1712725115  0.779
2018 Van der Poorten O, Legrand B, Vezenkov L, Garcia-Pindado J, Bettache N, Knuhtsen A, Sejer Pedersen D, Sanchez-Navarro M, Martinez J, Teixido M, Garcia M, Tourwe D, Amblard M, Ballet S. Indoloazepinone-Constrained Oligomers as Cell-Penetrating and Blood-Brain Barrier Permeable Compounds. Chembiochem : a European Journal of Chemical Biology. PMID 29377388 DOI: 10.1002/Cbic.201700678  0.453
2018 Chaubet G, Berthet M, Pasco M, Cazals G, Lebrun A, Martinez J, Parrot I. Fused Bis-lactams to Spirolactams: A New Member of the Family of Ring- Contraction Reaction Letters in Organic Chemistry. 15: 1046-1055. DOI: 10.2174/1570178615666180326160131  0.266
2018 Beillard A, Bantreil X, Métro T, Martinez J, Lamaty F. A more sustainable and efficient access to IMes·HCl and IPr·HCl by ball-milling Green Chemistry. 20: 964-968. DOI: 10.1039/C7Gc03539J  0.582
2018 Yeboue Y, Gallard B, Moigne NL, Jean M, Lamaty F, Martinez J, Métro T. Peptide Couplings by Reactive Extrusion: Solid-Tolerant and Free from Carcinogenic, Mutagenic and Reprotoxic Chemicals Acs Sustainable Chemistry & Engineering. 6: 16001-16004. DOI: 10.1021/Acssuschemeng.8B04509  0.59
2018 Milbeo P, Moulat L, Didierjean C, Aubert E, Martinez J, Calmès M. C1‐Symmetric 1,2‐Diaminobicyclo[2.2.2]octane Ligands in Copper‐Catalyzed Asymmetric Henry Reaction: Catalyst Development and DFT Studies European Journal of Organic Chemistry. 2018: 178-187. DOI: 10.1002/Ejoc.201701452  0.788
2017 Maurin O, Verdié P, Subra G, Lamaty F, Martinez J, Métro TX. Peptide synthesis: ball-milling, in solution, or on solid support, what is the best strategy? Beilstein Journal of Organic Chemistry. 13: 2087-2093. PMID 33613776 DOI: 10.3762/Bjoc.13.206  0.601
2017 Kulakova AN, Bilyachenko AN, Levitsky MM, Khrustalev VN, Korlyukov AA, Zubavichus YV, Dorovatovskii PV, Lamaty F, Bantreil X, Villemejeanne B, Martinez J, Shul'pina LS, Shubina ES, Gutsul EI, Mikhailov IA, et al. Si10Cu6N4 Cage Hexacoppersilsesquioxanes Containing N Ligands: Synthesis, Structure, and High Catalytic Activity in Peroxide Oxidations. Inorganic Chemistry. 56: 15026-15040. PMID 29185729 DOI: 10.1021/Acs.Inorgchem.7B02320  0.665
2017 Jia T, Choi J, Ciccione J, Henry M, Mehdi A, Martinez J, Eymin B, Subra G, Coll JL. Heteromultivalent targeting of integrin αvβ3 and neuropilin 1 promotes cell survival via the activation of the IGF-1/insulin receptors. Biomaterials. 155: 64-79. PMID 29169039 DOI: 10.1016/J.Biomaterials.2017.10.042  0.778
2017 Pétry N, Benakki H, Clot E, Retailleau P, Guenoun F, Asserar F, Sekkat C, Métro TX, Martinez J, Lamaty F. A mechanochemical approach to access the proline-proline diketopiperazine framework. Beilstein Journal of Organic Chemistry. 13: 2169-2178. PMID 29114324 DOI: 10.3762/Bjoc.13.217  0.754
2017 Rodriguez JA, Fehrentz JA, Martinez J, Salah KBH, Wellman PJ. The GHR-R antagonist JMV 2959 neither induces malaise nor alters the malaise property of LiCl in the adult male rat. Physiology & Behavior. PMID 29056353 DOI: 10.1016/J.Physbeh.2017.10.017  0.769
2017 Sirago G, Conte E, Fracasso F, Cormio A, Fehrentz JA, Martinez J, Musicco C, Camerino GM, Fonzino A, Rizzi L, Torsello A, Lezza AMS, Liantonio A, Cantatore P, Pesce V. Growth hormone secretagogues hexarelin and JMV2894 protect skeletal muscle from mitochondrial damages in a rat model of cisplatin-induced cachexia. Scientific Reports. 7: 13017. PMID 29026190 DOI: 10.1038/S41598-017-13504-Y  0.622
2017 Lucchi C, Costa AM, Giordano C, Curia G, Piat M, Leo G, Vinet J, Brunel L, Fehrentz JA, Martinez J, Torsello A, Biagini G. Involvement of PPARγ in the Anticonvulsant Activity of EP-80317, a Ghrelin Receptor Antagonist. Frontiers in Pharmacology. 8: 676. PMID 29018345 DOI: 10.3389/Fphar.2017.00676  0.746
2017 Bonnel C, Legrand B, Simon M, Martinez J, Bantignies JL, Kang YK, Wenger E, Hoh F, Masurier N, Maillard LT. C9/12-ribbon-like structure in hybrid peptides alternating α- and thiazole-based γ-amino acids. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28990697 DOI: 10.1002/Chem.201704001  0.725
2017 Das S, Ben Haj Salah K, Wenger E, Martinez J, Kotarba J, Andreu V, Ruiz N, Savini F, Stella L, Didierjean C, Legrand B, Inguimbert N. Enhancing the antimicrobial activity of alamethicin F50/5 by incorporating N-terminal hydrophobic triazole substituents. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28922505 DOI: 10.1002/Chem.201703569  0.803
2017 Amblard MC, Vezenkov LL, Martin V, Bettache N, Simon M, Messerschmitt A, Legrand B, Bantignies JL, Subra G, Maynadier M, Bellet V, Garcia M, Martinez J. Ribbon-like foldamers for cellular uptake and drug delivery. Chembiochem : a European Journal of Chemical Biology. PMID 28863239 DOI: 10.1002/Cbic.201700455  0.802
2017 Zayed M, Tourne-Peteilh C, Ramonda M, Rethore G, Weiss P, Martinez J, Subra G, Mehdi A, Devoisselle JM, Legrand P. Microgels of silylated HPMC as a multimodal system for drug co-encapsulation. International Journal of Pharmaceutics. PMID 28755992 DOI: 10.1016/J.Ijpharm.2017.07.074  0.719
2017 Konnert L, Lamaty F, Martinez J, Colacino E. Recent Advances in the Synthesis of Hydantoins: The State of the Art of a Valuable Scaffold. Chemical Reviews. 117: 13757-13809. PMID 28644621 DOI: 10.1021/Acs.Chemrev.7B00067  0.567
2017 Martinez J. Unexpected functions of angiotensin converting enzyme, beyond its enzymatic activity. Journal of Peptide Science : An Official Publication of the European Peptide Society. PMID 28626916 DOI: 10.1002/Psc.3022  0.483
2017 Fanelli R, Berthomieu D, Didierjean C, Doudouh A, Lebrun A, Martinez J, Cavelier F. Hydrophobic α,α-Disubstituted Disilylated TESDpg Induces Incipient 310-Helix in Short Tripeptide Sequence. Organic Letters. PMID 28514165 DOI: 10.1021/Acs.Orglett.7B01172  0.66
2017 Sevaille L, Gavara L, Bebrone C, De Luca F, Nauton L, Achard M, Mercuri P, Tanfoni S, Borgianni L, Guyon C, Lonjon P, Turan-Zitouni G, Dzieciolowski J, Becker K, Bénard L, ... ... Martinez J, et al. 1,2,4-Triazole-3-thione compounds as inhibitors of di-zinc metallo-β-lactamases. Chemmedchem. PMID 28505394 DOI: 10.1002/Cmdc.201700186  0.482
2017 Beillard A, Métro TX, Bantreil X, Martinez J, Lamaty F. Cu(0), O2 and mechanical forces: a saving combination for efficient production of Cu-NHC complexes. Chemical Science. 8: 1086-1089. PMID 28451247 DOI: 10.1039/C6Sc03182J  0.612
2017 Molteni L, Rizzi L, Bresciani E, Possenti R, Petrocchi Passeri P, Ghè C, Muccioli G, Fehrentz JA, Verdié P, Martinez J, Omeljaniuk RJ, Biagini G, Binda A, Rivolta I, Locatelli V, et al. Pharmacological and Biochemical Characterization of TLQP-21 Activation of a Binding Site on CHO Cells. Frontiers in Pharmacology. 8: 167. PMID 28424618 DOI: 10.3389/Fphar.2017.00167  0.772
2017 Denis RG, Joly-Amado A, Webber E, Langlet F, Schaeffer M, Padilla SL, Cansell C, Dehouck B, Castel J, Delbès AS, Martinez S, Lacombe A, Rouch C, Kassis N, Fehrentz JA, ... Martinez J, et al. Palatability Can Drive Feeding Independent of AgRP Neurons. Cell Metabolism. 25: 975. PMID 28380385 DOI: 10.1016/J.Cmet.2017.03.001  0.773
2017 Fanelli R, Floquet N, Besserer-Offroy É, Delort B, Vivancos M, Longpré JM, Renault P, Martinez J, Sarret P, Cavelier F. Use of Molecular Modeling to Design Selective-NTS2 Neurotensin Analogues. Journal of Medicinal Chemistry. PMID 28368584 DOI: 10.1021/Acs.Jmedchem.6B01848  0.801
2017 Conte E, Camerino GM, Mele A, De Bellis M, Pierno S, Rana F, Fonzino A, Caloiero R, Rizzi L, Bresciani E, Ben Haj Salah K, Fehrentz JA, Martinez J, Giustino A, Mariggiò MA, et al. Growth hormone secretagogues prevent dysregulation of skeletal muscle calcium homeostasis in a rat model of cisplatin-induced cachexia. Journal of Cachexia, Sarcopenia and Muscle. PMID 28294567 DOI: 10.1002/Jcsm.12185  0.625
2017 Rivolta I, Binda A, Molteni L, Rizzi L, Bresciani E, Possenti R, Fehrentz JA, Verdié P, Martinez J, Omeljaniuk RJ, Locatelli V, Torsello A. JMV5656, A Novel Derivative of TLQP-21, Triggers the Activation of a Calcium-Dependent Potassium Outward Current in Microglial Cells. Frontiers in Cellular Neuroscience. 11: 41. PMID 28280458 DOI: 10.3389/Fncel.2017.00041  0.647
2017 Delort B, Renault P, Charlier L, Raussin F, Martinez J, Floquet N. Coarse-Grained Prediction of Peptide Binding to G-Protein Coupled Receptors. Journal of Chemical Information and Modeling. PMID 28230370 DOI: 10.1021/Acs.Jcim.6B00503  0.492
2017 Milbeo P, Moulat L, Didierjean C, Aubert E, Martinez J, Calmès M. Synthesis of enantiopure DABO derivatives, C1-symmetric chiral 1,2-diamines with a rigid bicyclic backbone. The Journal of Organic Chemistry. PMID 28198182 DOI: 10.1021/Acs.Joc.7B00122  0.809
2017 Mascitti A, Lupacchini M, Guerra R, Taydakov I, Tonucci L, d'Alessandro N, Lamaty F, Martinez J, Colacino E. Poly(ethylene glycol)s as grinding additives in the mechanochemical preparation of highly functionalized 3,5-disubstituted hydantoins. Beilstein Journal of Organic Chemistry. 13: 19-25. PMID 28179944 DOI: 10.3762/Bjoc.13.3  0.637
2017 Karageorgis A, Claron M, Jugé R, Aspord C, Thoreau F, Leloup C, Kucharczak J, Plumas J, Henry M, Hurbin A, Verdié P, Martinez J, Subra G, Dumy P, Boturyn D, et al. Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model. Molecular Therapy : the Journal of the American Society of Gene Therapy. 25: 534-546. PMID 28153100 DOI: 10.1016/J.Ymthe.2016.11.002  0.479
2017 Berthet M, Legrand B, Martinez J, Parrot I. A General Approach to the Aza-Diketomorpholine Scaffold. Organic Letters. PMID 28093918 DOI: 10.1021/Acs.Orglett.6B03656  0.51
2017 Yalymov A, Bilyachenko A, Levitsky M, Korlyukov A, Khrustalev V, Shul’pina L, Dorovatovskii P, Es’kova M, Lamaty F, Bantreil X, Villemejeanne B, Martinez J, Shubina E, Kozlov Y, Shul’pin G. High Catalytic Activity of Heterometallic (Fe6Na7 and Fe6Na6) Cage Silsesquioxanes in Oxidations with Peroxides Catalysts. 7: 101. DOI: 10.3390/Catal7040101  0.671
2017 Drop M, Bantreil X, Grychowska K, Mahoro GU, Colacino E, Pawłowski M, Martinez J, Subra G, Zajdel P, Lamaty F. Continuous flow ring-closing metathesis, an environmentally-friendly route to 2,5-dihydro-1H-pyrrole-3-carboxylates Green Chemistry. 19: 1647-1652. DOI: 10.1039/C7Gc00235A  0.586
2017 Echalier C, Levato R, Mateos-Timoneda MA, Castano O, Dejean S, Garric X, Pinese C, Noel D, Engel E, Martinez J, Mehdi A, Subra G. Modular bioink for 3D printing of biocompatible hydrogels: sol–gel polymerization of hybrid peptides and polymers Rsc Advances. 7: 12231-12235. DOI: 10.1039/C6Ra28540F  0.266
2017 Beillard A, Bantreil X, Métro T, Martinez J, Lamaty F. Mechanochemistry for facilitated access to N,N-diaryl NHC metal complexes New Journal of Chemistry. 41: 1057-1063. DOI: 10.1039/C6Nj02895K  0.556
2017 Métro T, Martinez J, Lamaty F. 1,1′-Carbonyldiimidazole and Mechanochemistry: A Shining Green Combination Acs Sustainable Chemistry & Engineering. 5: 9599-9602. DOI: 10.1021/Acssuschemeng.7B03260  0.591
2017 Gonnet L, Tintillier T, Venturini N, Konnert L, Hernandez J, Lamaty F, Laconde G, Martinez J, Colacino E. N-Acyl Benzotriazole Derivatives for the Synthesis of Dipeptides and Tripeptides and Peptide Biotinylation by Mechanochemistry Acs Sustainable Chemistry & Engineering. 5: 2936-2941. DOI: 10.1021/Acssuschemeng.6B02439  0.616
2017 Lupacchini M, Mascitti A, Giachi G, Tonucci L, d'Alessandro N, Martinez J, Colacino E. Sonochemistry in non-conventional, green solvents or solvent-free reactions Tetrahedron. 73: 609-653. DOI: 10.1016/J.Tet.2016.12.014  0.269
2017 Pinese C, Jebors S, Stoebner PE, Humblot V, Verdié P, Causse L, Garric X, Taillades H, Martinez J, Mehdi A, Subra G. Bioactive peptides grafted silicone dressings: A simple and specific method Materials Today Chemistry. 4: 73-83. DOI: 10.1016/J.Mtchem.2017.02.007  0.312
2017 Echalier C, Jebors S, Laconde G, Brunel L, Verdié P, Causse L, Bethry A, Legrand B, Berghe HVD, Garric X, Noël D, Martinez J, Mehdi A, Subra G. Sol–gel synthesis of collagen-inspired peptide hydrogel Materials Today. 20: 59-66. DOI: 10.1016/J.Mattod.2017.02.001  0.269
2017 Ali-Moussa H, Amador RN, Martinez J, Lamaty F, Carboni M, Bantreil X. Synthesis and post-synthetic modification of UiO-67 type metal-organic frameworks by mechanochemistry Materials Letters. 197: 171-174. DOI: 10.1016/J.Matlet.2017.03.140  0.566
2017 Beillard A, Métro T, Bantreil X, Martinez J, Lamaty F. A3-Coupling Reaction and [Ag(IPr)2]PF6: A Successful Couple European Journal of Organic Chemistry. 2017: 4642-4647. DOI: 10.1002/Ejoc.201700985  0.565
2017 Bilyachenko AN, Kulakova AN, Levitsky MM, Korlyukov AA, Khrustalev VN, Vologzhanina AV, Titov AA, Dorovatovskii PV, Shul'pina LS, Lamaty F, Bantreil X, Villemejeanne B, Ruiz C, Martinez J, Shubina ES, et al. Ionic Complexes of Tetra- and Nonanuclear Cage Copper(II) Phenylsilsesquioxanes: Synthesis and High Activity in Oxidative Catalysis Chemcatchem. 9: 4437-4447. DOI: 10.1002/Cctc.201701063  0.679
2016 Giordano C, Costa AM, Lucchi C, Leo G, Brunel L, Fehrentz JA, Martinez J, Torsello A, Biagini G. Progressive Seizure Aggravation in the Repeated 6-Hz Corneal Stimulation Model Is Accompanied by Marked Increase in Hippocampal p-ERK1/2 Immunoreactivity in Neurons. Frontiers in Cellular Neuroscience. 10: 281. PMID 28018175 DOI: 10.3389/Fncel.2016.00281  0.731
2016 Berthet M, Cheviet T, Dujardin G, Parrot I, Martinez J. Isoxazolidine: A Privileged Scaffold for Organic and Medicinal Chemistry. Chemical Reviews. PMID 27981833 DOI: 10.1021/Acs.Chemrev.6B00543  0.509
2016 Konnert L, Gonnet L, Halasz I, Suppo JS, de Figueiredo RM, Campagne JM, Lamaty F, Martinez J, Colacino E. Correction to Mechanochemical Preparation of 3,5-Disubstituted Hydantoins from Dipeptides and Unsymmetrical Ureas of Amino Acid Derivatives. The Journal of Organic Chemistry. 81: 12071. PMID 27934473 DOI: 10.1021/Acs.Joc.6B02671  0.726
2016 Rossato M, Miralles G, M'Kadmi C, Maingot M, Amblard M, Mouillac B, Gagne D, Martinez J, Subra G, Enjalbal C, Cantel S. Quantitative MALDI-MS Binding Assays: An Alternative to Radiolabeling. Chemmedchem. 11: 2582-2587. PMID 27922213 DOI: 10.1002/Cmdc.201600447  0.663
2016 Bresciani E, Rizzi L, Molteni L, Ravelli M, Liantonio A, Ben Haj Salah K, Fehrentz JA, Martinez J, Omeljaniuk RJ, Biagini G, Locatelli V, Torsello A. JMV2894, a novel growth hormone secretagogue, accelerates body mass recovery in an experimental model of cachexia. Endocrine. PMID 27896546 DOI: 10.1007/S12020-016-1184-2  0.736
2016 Bellet V, Lichon L, Arama DP, Gallud A, Lisowski V, Maillard LT, Garcia M, Martinez J, Masurier N. Imidazopyridine-fused [1,3]-diazepinones part 2: Structure-activity relationships and antiproliferative activity against melanoma cells. European Journal of Medicinal Chemistry. 125: 1225-1234. PMID 27871038 DOI: 10.1016/J.Ejmech.2016.11.023  0.79
2016 Pinese C, Jebors S, Echalier C, Licznar-Fajardo P, Garric X, Humblot V, Calers C, Martinez J, Mehdi A, Subra G. Simple and Specific Grafting of Antibacterial Peptides on Silicone Catheters. Advanced Healthcare Materials. PMID 27792296 DOI: 10.1002/Adhm.201600757  0.445
2016 Beillard A, Bantreil X, Métro TX, Martinez J, Lamaty F. Unraveling the synthesis of homoleptic [Ag(N,N-diaryl-NHC)2]Y (Y = BF4, PF6) complexes by ball-milling. Dalton Transactions (Cambridge, England : 2003). PMID 27774541 DOI: 10.1039/C6Dt03564G  0.63
2016 Bonnel C, Legrand B, Bantignies JL, Petitjean H, Martinez J, Masurier N, Maillard LT. FT-IR and NMR structural markers for thiazole-based γ-peptide foldamers. Organic & Biomolecular Chemistry. 14: 8664-8669. PMID 27714174 DOI: 10.1039/C6Ob01594H  0.478
2016 Konnert L, Gonnet L, Halasz I, Suppo JS, de Figueiredo RM, Campagne JM, Lamaty F, Martinez J, Colacino E. Mechanochemical preparation of 3,5-disubstituted Hydantoins from Dipeptides and Unsymmetrical Ureas of Amino Acid Derivatives. The Journal of Organic Chemistry. PMID 27679874 DOI: 10.1021/Acs.Joc.6B01832  0.764
2016 Salom-Roig XJ, Grenet E, Martinez J. Lewis Acid Induced-Switch of Torquoselectivity in the Nazarov Cyclization of Activated Dienones Bearing a Chiral Sulfoxide. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27618730 DOI: 10.1002/Chem.201603920  0.789
2016 Rémond E, Martin C, Martinez J, Cavelier F. Silicon-Containing Amino Acids: Synthetic Aspects, Conformational Studies, and Applications to Bioactive Peptides. Chemical Reviews. PMID 27529497 DOI: 10.1021/Acs.Chemrev.6B00122  0.506
2016 Knuhtsen A, Legrand B, Van der Poorten O, Amblard M, Martinez J, Ballet S, Kristensen JL, Pedersen DS. Conformationally Constrained Peptidomimetics as Inhibitors of the Protein Arginine Methyl Transferases. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27515561 DOI: 10.1002/Chem.201602518  0.513
2016 Cordeau E, Cantel S, Gagne D, Lebrun A, Martinez J, Subra G, Enjalbal C. Selenazolidine: a selenium containing proline surrogate in peptide science. Organic & Biomolecular Chemistry. PMID 27506250 DOI: 10.1039/C6Ob01450J  0.532
2016 Berthet M, Martinez J, Parrot I. MgI2 -Chemoselective Cleavage for removal of amino acid protecting groups: A Fresh Vision for Peptide Synthesis. Biopolymers. PMID 27390871 DOI: 10.1002/Bip.22908  0.486
2016 Coppens J, Aourz N, Walrave L, Fehrentz JA, Martinez J, De Bundel D, Portelli J, Smolders I. Anticonvulsant effect of a ghrelin receptor agonist in 6Hz corneally kindled mice. Epilepsia. PMID 27378373 DOI: 10.1111/Epi.13463  0.635
2016 Cordeau E, Arnaudguilhem C, Bouyssiere B, Hagège A, Martinez J, Subra G, Cantel S, Enjalbal C. Investigation of Elemental Mass Spectrometry in Pharmacology for Peptide Quantitation at Femtomolar Levels. Plos One. 11: e0157943. PMID 27336163 DOI: 10.1371/Journal.Pone.0157943  0.464
2016 Amblard MC, Legrand B, André C, Moulat L, Didierjean C, Hermet P, Bantignies JL, Martinez J, Calmès M. 12/14/14-Helix Formation in 2:1 α/β-hybrid peptides containing bicyclo[2.2.2]octane ring constraints. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27311099 DOI: 10.1002/Chem.201602746  0.798
2016 Grychowska K, Satała G, Kos T, Partyka A, Colacino E, Chaumont-Dubel S, Bantreil X, Wesołowska A, Pawlowski MH, Martinez J, Marin P, Subra G, Bojarski AJ, Lamaty F, Popik P, et al. Novel 1H-pyrrolo[3,2-c]quinoline based 5-HT6 receptor antagonists with potential application for the treatment of cognitive disorders associated with Alzheimer's disease. Acs Chemical Neuroscience. PMID 27100049 DOI: 10.1021/Acschemneuro.6B00090  0.795
2016 Maingot M, Blayo AL, Denoyelle S, M'Kadmi C, Damian M, Mary S, Gagne D, Sanchez P, Aicher B, Schmidt P, Müller G, Teifel M, Günther E, Marie J, Banères JL, ... Martinez J, et al. New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center. Bioorganic & Medicinal Chemistry Letters. PMID 27072910 DOI: 10.1016/J.Bmcl.2016.04.003  0.78
2016 Neasta J, Valmalle C, Coyne AC, Carnazzi E, Subra G, Galleyrand JC, Gagne D, M'Kadmi C, Bernad N, Bergé G, Cantel S, Marin P, Marie J, Banères JL, Kemel ML, ... ... Martinez J, et al. The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release. British Journal of Pharmacology. 173: 1314-28. PMID 27027724 DOI: 10.1111/Bph.13424  0.719
2016 Kalistratova A, Legrand B, Verdié P, Naydenova E, Amblard M, Martinez J, Subra G. A switchable stapled peptide. Journal of Peptide Science : An Official Publication of the European Peptide Society. 22: 143-8. PMID 26785930 DOI: 10.1002/Psc.2851  0.362
2016 Chatalic KL, Konijnenberg M, Nonnekens J, de Blois E, Hoeben S, de Ridder C, Brunel L, Fehrentz JA, Martinez J, van Gent DC, Nock BA, Maina T, van Weerden WM, de Jong M. In Vivo Stabilization of a Gastrin-Releasing Peptide Receptor Antagonist Enhances PET Imaging and Radionuclide Therapy of Prostate Cancer in Preclinical Studies. Theranostics. 6: 104-17. PMID 26722377 DOI: 10.7150/Thno.13580  0.588
2016 Haeck JC, Bol K, de Ridder CMA, Brunel L, Fehrentz JA, Martinez J, van Weerden WM, Bernsen MR, de Jong M, Veenland JF. Imaging heterogeneity of peptide delivery and binding in solid tumors using SPECT imaging and MRI Ejnmmi Research. 6: 1-9. DOI: 10.1186/S13550-016-0160-4  0.454
2016 Neasta J, Valmalle C, Coyne AC, Carnazzi E, Subra G, Galleyrand JC, Gagne D, M'Kadmi C, Bernad N, Bergé G, Cantel S, Marin P, Marie J, Banères JL, Kemel ML, ... ... Martinez J, et al. The novel nonapeptide acein targets angiotensin converting enzyme in the brain and induces dopamine release British Journal of Pharmacology. DOI: 10.1111/bph.13424  0.76
2016 Fanelli R, Martinez J, Cavelier F. Expedient Synthesis of Fmoc-(S)-γ-Fluoroleucine and Late-Stage Fluorination of Peptides Synlett. DOI: 10.1055/S-0035-1561568  0.744
2016 Bilyachenko AN, Levitsky MM, Yalymov AI, Korlyukov AA, Vologzhanina AV, Kozlov YN, Shul'pina LS, Nesterov DS, Pombeiro AJL, Lamaty F, Bantreil X, Fetre A, Liu D, Martinez J, Long J, et al. A heterometallic (Fe6Na8) cage-like silsesquioxane: synthesis, structure, spin glass behavior and high catalytic activity Rsc Advances. 6: 48165-48180. DOI: 10.1039/C6Ra07081G  0.775
2016 Echalier C, Kalistratova A, Ciccione J, Lebrun A, Legrand B, Naydenova E, Gagne D, Fehrentz J, Marie J, Amblard M, Mehdi A, Martinez J, Subra G. Selective homodimerization of unprotected peptides using hybrid hydroxydimethylsilane derivatives Rsc Advances. 6: 32905-32914. DOI: 10.1039/C6Ra06075G  0.598
2016 Konnert L, Dimassi M, Gonnet L, Lamaty F, Martinez J, Colacino E. Poly(ethylene) glycols and mechanochemistry for the preparation of bioactive 3,5-disubstituted hydantoins Rsc Advances. 6: 36978-36986. DOI: 10.1039/C6Ra03222B  0.596
2016 Echalier C, Pinese C, Garric X, Van Den Berghe H, Jumas Bilak E, Martinez J, Mehdi A, Subra G. Easy Synthesis of Tunable Hybrid Bioactive Hydrogels Chemistry of Materials. 28: 1261-1265. DOI: 10.1021/Acs.Chemmater.5B04881  0.447
2016 Ciccione J, Jia T, Coll JL, Parra K, Amblard M, Jebors S, Martinez J, Mehdi A, Subra G. Unambiguous and Controlled One-Pot Synthesis of Multifunctional Silica Nanoparticles Chemistry of Materials. 28: 885-889. DOI: 10.1021/Acs.Chemmater.5B04398  0.645
2016 Géant P, Grenet E, Martínez J, Salom-Roig XJ. Stereoselective divergent synthesis of 1,2-aminoalcohol-containing heterocycles from a common chiral nonracemic building block Tetrahedron-Asymmetry. 27: 22-30. DOI: 10.1016/J.Tetasy.2015.11.008  0.783
2016 Grychowska K, Kubica B, Drop M, Colacino E, Bantreil X, Pawłowski M, Martinez J, Subra G, Zajdel P, Lamaty F. Application of the ring-closing metathesis to the formation of 2-aryl-1H-pyrrole-3-carboxylates as building blocks for biologically active compounds Tetrahedron. 72: 7462-7469. DOI: 10.1016/J.Tet.2016.09.059  0.599
2016 Milbeo P, Maurent K, Moulat L, Lebrun A, Didierjean C, Aubert E, Martinez J, Calmès M. N-Pyrrolidine-based α/β-peptides incorporating ABOC, a constrained bicyclic β-amino acid, for asymmetric aldol reaction catalysis Tetrahedron. 72: 1706-1715. DOI: 10.1016/J.Tet.2016.02.027  0.805
2016 Porte V, Thioloy M, Pigoux T, Métro T, Martinez J, Lamaty F. Peptide Mechanosynthesis by Direct Coupling of N‐Protected α‐Amino Acids with Amino Esters European Journal of Organic Chemistry. 2016: 3505-3508. DOI: 10.1002/Ejoc.201600617  0.619
2016 Hapəu D, Rémond E, Fanelli R, Vivancos M, René A, Côté J, Besserer-Offroy É, Longpré JM, Martinez J, Zaharia V, Sarret P, Cavelier F. Stereoselective Synthesis of β-(5-Arylthiazolyl) α-Amino Acids and Use in Neurotensin Analogues European Journal of Organic Chemistry. 2016: 1017-1024. DOI: 10.1002/Ejoc.201501495  0.818
2016 Grenet E, Martinez J, Salom-Roig XJ. Torquoselective Nazarov Cyclization Mediated by a Chiral Sulfoxide: First Enantioselective Synthesis of two Known Anticancer Agents Asian Journal of Organic Chemistry. 6: 189-198. DOI: 10.1002/Ajoc.201600471  0.766
2015 Pozzi F, Rizzi L, Zambelli V, Molteni L, Cavagna M, Verdie P, Fehrentz JA, Martinez J, Torsello A, Bellani G, Pesenti A. TLQP-21 modulate inflammation and fibrosis in a model of ards. Intensive Care Medicine Experimental. 3: A562. PMID 27290127 DOI: 10.1186/2197-425X-3-S1-A562  0.396
2015 Logez C, Damian M, Legros C, Dupré C, Guéry M, Mary S, Wagner R, M'Kadmi C, Nosjean O, Fould B, Marie J, Fehrentz JA, Martinez J, Ferry G, Boutin JA, et al. Detergent-free Isolation of Functional G Protein-Coupled Receptors into Nanometric Lipid Particles. Biochemistry. PMID 26701065 DOI: 10.1021/Acs.Biochem.5B01040  0.783
2015 Vezenkov LL, Sanchez CA, Bellet V, Martin V, Maynadier M, Bettache N, Lisowski V, Martinez J, Garcia M, Amblard M, Hernandez JF. Structure-Activity Relationships of JMV4463, a Vectorized Cathepsin D Inhibitor with Antiproliferative Properties: The Unique Role of the AMPA-Based Vector. Chemmedchem. PMID 26639308 DOI: 10.1002/Cmdc.201500457  0.787
2015 Beillard A, Golliard E, Gillet V, Bantreil X, Métro TX, Martinez J, Lamaty F. Expedient Mechanosynthesis of N,N-Dialkyl Imidazoliums and Silver(I)-Carbene Complexes in a Ball-Mill. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26489706 DOI: 10.1002/Chem.201503472  0.649
2015 Ramakrishnan SK, Jebors S, Martin M, Cloitre T, Agarwal V, Mehdi A, Martinez J, Subra G, Gergely C. Engineered adhesion peptides for improved silicon adsorption. Langmuir : the Acs Journal of Surfaces and Colloids. PMID 26440047 DOI: 10.1021/Acs.Langmuir.5B02857  0.789
2015 Martin V, Legrand B, Vezenkov LL, Berthet M, Subra G, Calmès M, Bantignies JL, Martinez J, Amblard M. Turning Peptide Sequences into Ribbon Foldamers by a Straightforward Multicyclization Reaction. Angewandte Chemie (International Ed. in English). PMID 26398631 DOI: 10.1002/Anie.201506955  0.796
2015 M'Kadmi C, Leyris JP, Onfroy L, Galés C, Saulière A, Gagne D, Damian M, Mary S, Maingot M, Denoyelle S, Verdié P, Fehrentz JA, Martinez J, Banères JL, Marie J. Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling. The Journal of Biological Chemistry. 290: 27021-39. PMID 26363071 DOI: 10.1074/Jbc.M115.659250  0.787
2015 Fanelli R, Besserer-Offroy É, René A, Côté J, Tétreault P, Collerette-Tremblay J, Longpré JM, Leduc R, Martinez J, Sarret P, Cavelier F. Synthesis and Characterization in Vitro and in Vivo of (l)-(Trimethylsilyl)alanine Containing Neurotensin Analogues. Journal of Medicinal Chemistry. 58: 7785-95. PMID 26348111 DOI: 10.1021/Acs.Jmedchem.5B00841  0.802
2015 Fanelli R, Salah KB, Inguimbert N, Didierjean C, Martinez J, Cavelier F. Access to α,α-Disubstituted Disilylated Amino Acids and Their Use in Solid-Phase Peptide Synthesis. Organic Letters. 17: 4498-501. PMID 26347940 DOI: 10.1021/Acs.Orglett.5B02175  0.813
2015 Denis RG, Joly-Amado A, Webber E, Langlet F, Schaeffer M, Padilla SL, Cansell C, Dehouck B, Castel J, Delbès AS, Martinez S, Lacombe A, Rouch C, Kassis N, Fehrentz JA, ... Martinez J, et al. Palatability Can Drive Feeding Independent of AgRP Neurons. Cell Metabolism. PMID 26278050 DOI: 10.1016/J.Cmet.2015.07.011  0.764
2015 Floquet N, Costa MG, Batista PR, Renault P, Bisch PM, Raussin F, Martinez J, Morris MC, Perahia D. Conformational Equilibrium of CDK/Cyclin Complexes by Molecular Dynamics with Excited Normal Modes. Biophysical Journal. 109: 1179-89. PMID 26255588 DOI: 10.1016/J.Bpj.2015.07.003  0.773
2015 Métro TX, Bonnamour J, Reidon T, Duprez A, Sarpoulet J, Martinez J, Lamaty F. Comprehensive study of the organic-solvent-free CDI-mediated acylation of various nucleophiles by mechanochemistry. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 12787-96. PMID 26177831 DOI: 10.1002/Chem.201501325  0.586
2015 Cavalier M, Crouzin N, Ben Sedrine A, de Jesus Ferreira MC, Guiramand J, Cohen-Solal C, Fehrentz JA, Martinez J, Barbanel G, Vignes M. Involvement of PKA and ERK pathways in ghrelin-induced long-lasting potentiation of excitatory synaptic transmission in the CA1 area of rat hippocampus. The European Journal of Neuroscience. 42: 2568-76. PMID 26153524 DOI: 10.1111/Ejn.13013  0.581
2015 Berthet M, Davanier F, Dujardin G, Martinez J, Parrot I. MgI2 -mediated chemoselective cleavage of protecting groups: an alternative to conventional deprotection methodologies. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 11014-6. PMID 26121554 DOI: 10.1002/Chem.201501799  0.304
2015 Bilyachenko AN, Dronova MS, Yalymov AI, Lamaty F, Bantreil X, Martinez J, Bizet C, Shul'pina LS, Korlyukov AA, Arkhipov DE, Levitsky MM, Shubina ES, Kirillov AM, Shul'pin GB. Frontispiece: Cage-like Copper(II) Silsesquioxanes: Transmetalation Reactions and Structural, Quantum Chemical, and Catalytic Studies. Chemistry (Weinheim An Der Bergstrasse, Germany). 21. PMID 26017160 DOI: 10.1002/Chem.201582462  0.708
2015 Bilyachenko AN, Dronova MS, Yalymov AI, Lamaty F, Bantreil X, Martinez J, Bizet C, Shul'pina LS, Korlyukov AA, Arkhipov DE, Levitsky MM, Shubina ES, Kirillov AM, Shul'pin GB. Cage-like copper(II) silsesquioxanes: transmetalation reactions and structural, quantum chemical, and catalytic studies. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 8758-70. PMID 25950426 DOI: 10.1002/Chem.201500791  0.788
2015 Dalm SU, Martens JW, Sieuwerts AM, van Deurzen CH, Koelewijn SJ, de Blois E, Maina T, Nock BA, Brunel L, Fehrentz JA, Martinez J, de Jong M, Melis M. In vitro and in vivo application of radiolabeled gastrin-releasing peptide receptor ligands in breast cancer. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 56: 752-7. PMID 25791989 DOI: 10.2967/Jnumed.114.153023  0.712
2015 Ben Haj Salah K, Legrand B, Das S, Martinez J, Inguimbert N. A Straightforward Strategy to Substitute Amide Bonds by 1,2,3 Triazoles in Peptaibols Analogs Using Aibψ[Tz]-Xaa Dipeptides. Biopolymers. PMID 25784277 DOI: 10.1002/Bip.22641  0.737
2015 Fanelli R, Jeanne-Julien L, René A, Martinez J, Cavelier F. Stereoselective synthesis of unsaturated α-amino acids. Amino Acids. 47: 1107-15. PMID 25715756 DOI: 10.1007/S00726-015-1934-0  0.785
2015 Jebors S, Pinese C, Nottelet B, Parra K, Amblard M, Mehdi A, Martinez J, Subra G. Turning peptides in comb silicone polymers. Journal of Peptide Science : An Official Publication of the European Peptide Society. 21: 243-7. PMID 25688748 DOI: 10.1002/Psc.2757  0.717
2015 Grychowska K, Masurier N, Verdié P, Sata?a G, Bojarski AJ, Martinez J, Paw?owski M, Subra G, Zajdel P. Solid-Supported Synthesis and 5-HT7 /5-HT1A Receptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1H)-one. Chemical Biology & Drug Design. PMID 25684690 DOI: 10.1111/Cbdd.12539  0.515
2015 Arama DP, Soualmia F, Lisowski V, Longevial JF, Bosc E, Maillard LT, Martinez J, Masurier N, El Amri C. Pyrido-imidazodiazepinones as a new class of reversible inhibitors of human kallikrein 7. European Journal of Medicinal Chemistry. 93: 202-13. PMID 25682203 DOI: 10.1016/J.Ejmech.2015.02.008  0.785
2015 Jebors S, Ciccione J, Al-Halifa S, Nottelet B, Enjalbal C, M'Kadmi C, Amblard M, Mehdi A, Martinez J, Subra G. A new way to silicone-based peptide polymers. Angewandte Chemie (International Ed. in English). 54: 3778-82. PMID 25650781 DOI: 10.1002/Anie.201411065  0.486
2015 Damian M, Mary S, Maingot M, M'Kadmi C, Gagne D, Leyris JP, Denoyelle S, Gaibelet G, Gavara L, Garcia de Souza Costa M, Perahia D, Trinquet E, Mouillac B, Galandrin S, Galès C, ... ... Martinez J, et al. Ghrelin receptor conformational dynamics regulate the transition from a preassembled to an active receptor:Gq complex. Proceedings of the National Academy of Sciences of the United States of America. 112: 1601-6. PMID 25605885 DOI: 10.1073/Pnas.1414618112  0.783
2015 Blayo AL, Maingot M, Aicher B, M'Kadmi C, Schmidt P, Müller G, Teifel M, Günther E, Gagne D, Denoyelle S, Martinez J, Fehrentz JA. New trisubstituted 1,2,4-triazoles as ghrelin receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 25: 20-4. PMID 25435152 DOI: 10.1016/J.Bmcl.2014.11.031  0.805
2015 Sacco M, Charnay C, Angelis FD, Radoiu M, Lamaty F, Martinez J, Colacino E. Microwave-ultrasound simultaneous irradiation: a hybrid technology applied to ring closing metathesis Rsc Advances. 5: 16878-16885. DOI: 10.1039/C4Ra14938F  0.559
2015 Métro T, Salom-Roig XJ, Reverte M, Martinez J, Lamaty F. Faster and cleaner dynamic kinetic resolution via mechanochemistry Green Chemistry. 17: 204-208. DOI: 10.1039/C4Gc01416B  0.537
2015 Lanzillotto M, Konnert L, Lamaty F, Martinez J, Colacino E. Mechanochemical 1,1′-Carbonyldiimidazole-Mediated Synthesis of Carbamates Acs Sustainable Chemistry & Engineering. 3: 2882-2889. DOI: 10.1021/Acssuschemeng.5B00819  0.601
2015 Mnasri N, Nyalosaso JL, Colacino E, Derrien G, Lamaty F, Martinez J, Zajac J, Charnay C. Copper-Containing Rod-Shaped Nanosized Silica Particles for Microwave-Assisted Synthesis of Triazoles in Aqueous Solution Acs Sustainable Chemistry & Engineering. 3: 2516-2525. DOI: 10.1021/Acssuschemeng.5B00661  0.564
2015 Denoyelle S, Tambutet G, Masurier N, Maillard LT, Martinez J, Lisowski V. Synthesis of Thieno[3,2‐e][1,4]diazepin‐2‐ones: Application of an Uncatalysed Pictet–Spengler Reaction European Journal of Organic Chemistry. 2015: 7146-7153. DOI: 10.1002/Ejoc.201500943  0.356
2015 Mathieu L, Bonnel C, Masurier N, Maillard LT, Martinez J, Lisowski V. Cross-Claisen Condensation of N-Fmoc-Amino Acids – A Short Route to Heterocyclic γ-Amino Acids European Journal of Organic Chemistry. 2015: 2262-2270. DOI: 10.1002/Ejoc.201500012  0.356
2015 Bantreil X, Navals P, Martinez J, Lamaty F. Iron/Caffeine as a Catalytic System for Microwave‐Promoted Benzamide Formation European Journal of Organic Chemistry. 2015: 417-422. DOI: 10.1002/Ejoc.201403173  0.553
2014 Chatalic KL, Franssen GM, van Weerden WM, McBride WJ, Laverman P, de Blois E, Hajjaj B, Brunel L, Goldenberg DM, Fehrentz JA, Martinez J, Boerman OC, de Jong M. Preclinical comparison of Al18F- and 68Ga-labeled gastrin-releasing peptide receptor antagonists for PET imaging of prostate cancer. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 55: 2050-6. PMID 25413139 DOI: 10.2967/Jnumed.114.141143  0.738
2014 Paolantoni D, Rubio-Magnieto J, Cantel S, Martinez J, Dumy P, Surin M, Ulrich S. Probing the importance of π-stacking interactions in DNA-templated self-assembly of bisfunctionalized guanidinium compounds. Chemical Communications (Cambridge, England). 50: 14257-60. PMID 25285342 DOI: 10.1039/C4Cc05706F  0.677
2014 Alvarez R, Molist P, González-Sierra S, Martinez JJ, Nafría JM. The histo structure of galls induced by aphids as a useful taxonomic character: the case of Rectinasus (Hemiptera, Aphididae, Eriosomatinae). Zootaxa. 3861: 487-92. PMID 25283424  0.266
2014 Konnert L, Reneaud B, De Figueiredo RM, Campagne JM, Lamaty F, Martinez J, Colacino E. Mechanochemical preparation of hydantoins from amino esters: Application to the synthesis of the antiepileptic drug phenytoin Journal of Organic Chemistry. 79: 10132-10142. PMID 25279490 DOI: 10.1021/Jo5017629  0.783
2014 Legrand B, André C, Moulat L, Wenger E, Didierjean C, Aubert E, Averlant-Petit MC, Martinez J, Calmes M, Amblard M. Unprecedented chain-length-dependent conformational conversion between 11/9 and 18/16 helix in α/β-hybrid peptides. Angewandte Chemie (International Ed. in English). 53: 13131-5. PMID 25258017 DOI: 10.1002/Anie.201407329  0.581
2014 Martin C, Legrand B, Lebrun A, Berthomieu D, Martinez J, Cavelier F. Silaproline helical mimetics selectively form an all-trans PPII helix. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 14240-4. PMID 25212635 DOI: 10.1002/Chem.201404820  0.29
2014 Holubová M, Nagelová V, Lacinová Z, Haluzík M, Sýkora D, Moulin A, Blayo AL, Fehrentz JA, Martinez J, Stofkova A, Jurčovičová J, Železná B, Maletínská L. Triazole GHS-R1a antagonists JMV4208 and JMV3002 attenuate food intake, body weight, and adipose tissue mass in mice Molecular and Cellular Endocrinology. 393: 120-128. PMID 24953973 DOI: 10.1016/J.Mce.2014.06.003  0.263
2014 Boyer JB, Dedieu A, Armengaud J, Verdié P, Subra G, Martinez J, Enjalbal C. N- and O-acetylation of threonine residues in the context of proteomics. Journal of Proteomics. 108: 369-72. PMID 24937263 DOI: 10.1016/J.Jprot.2014.06.005  0.674
2014 Fleith C, Cantel S, Subra G, Mehdi A, Ciccione J, Martinez J, Enjalbal C. Laser desorption ionization mass spectrometry of peptides on a hybrid CHCA organic-inorganic matrix. The Analyst. 139: 3748-54. PMID 24910856 DOI: 10.1039/C3An01465G  0.287
2014 Konnert L, Lamaty F, Martinez J, Colacino E. Solventless mechanosynthesis of N-protected amino esters. The Journal of Organic Chemistry. 79: 4008-17. PMID 24738762 DOI: 10.1021/Jo500463Y  0.598
2014 Giachi G, Frediani M, Oberhauser W, Lamaty F, Martinez J, Colacino E. Ultrasounds in melted poly(ethylene glycol) promote copper-catalyzed cyanation of aryl halides with K(4)[Fe(CN)(6)]. Chemsuschem. 7: 919-24. PMID 24678012 DOI: 10.1002/Cssc.201300997  0.536
2014 Canale V, Guzik P, Kurczab R, Verdie P, Satała G, Kubica B, Pawłowski M, Martinez J, Subra G, Bojarski AJ, Zajdel P. Solid-supported synthesis, molecular modeling, and biological activity of long-chain arylpiperazine derivatives with cyclic amino acid amide fragments as 5-HT(7) and 5-HT(1A) receptor ligands. European Journal of Medicinal Chemistry. 78: 10-22. PMID 24675176 DOI: 10.1016/J.Ejmech.2014.03.005  0.384
2014 Legrand B, Mathieu L, Lebrun A, Andriamanarivo S, Lisowski V, Masurier N, Zirah S, Kang YK, Martinez J, Maillard LT. Thiazole-based γ-building blocks as reverse-turn mimetic to design a gramicidin S analogue: conformational and biological evaluation. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 6713-20. PMID 24668890 DOI: 10.1002/Chem.201402190  0.611
2014 Gallud A, Vaillant O, Maillard LT, Arama DP, Dubois J, Maynadier M, Lisowski V, Garcia M, Martinez J, Masurier N. Imidazopyridine-fused [1,3]-diazepinones: synthesis and antiproliferative activity. European Journal of Medicinal Chemistry. 75: 382-90. PMID 24561668 DOI: 10.1016/J.Ejmech.2014.01.044  0.787
2014 Charlier L, Louet M, Chaloin L, Fuchs P, Martinez J, Muriaux D, Favard C, Floquet N. Coarse-grained simulations of the HIV-1 matrix protein anchoring: revisiting its assembly on membrane domains. Biophysical Journal. 106: 577-85. PMID 24507598 DOI: 10.1016/J.Bpj.2013.12.019  0.267
2014 Peralta-Ramírez A, Montes de Oca A, Raya AI, Pineda C, López I, Guerrero F, Diez E, Muñoz-Castañeda JR, Martinez J, Almaden Y, Rodríguez M, Aguilera-Tejero E. Vitamin E protection of obesity-enhanced vascular calcification in uremic rats. American Journal of Physiology. Renal Physiology. 306: F422-9. PMID 24370590 DOI: 10.1152/Ajprenal.00355.2013  0.747
2014 Cecchini MM, Charnay C, De Angelis F, Lamaty F, Martinez J, Colacino E. Poly(ethylene glycol)-based ionic liquids: properties and uses as alternative solvents in organic synthesis and catalysis. Chemsuschem. 7: 45-65. PMID 24323519 DOI: 10.1002/Cssc.201300421  0.555
2014 Moulin A, Brunel L, Verdie P, Gavara L, Martinez J, Fehrentz J. Ghrelin Receptor Ligands: Design and Synthesis of Pseudopeptides and Peptidomimetics Current Chemical Biology. 7: 254-270. DOI: 10.2174/2212796807999131128125920  0.627
2014 Bauder C, Martínez J, Salom-Roig XJ. Chiral Sulfoxides as Building Blocks for Enantiopure 1,3-Diol Precursors in the Synthesis of Natural Products Current Organic Synthesis. 10: 885-902. DOI: 10.2174/157017941006140206103254  0.266
2014 Chaubet G, Cazals G, Lebrun A, Martinez J, Parrot I. From Diketopiperazines to Hydantoins: An Unprecedented Rearrangement Synlett. 25: 574-578. DOI: 10.1055/S-0033-1340622  0.334
2014 Cecchini MM, Bendjeriou A, Mnasri N, Charnay C, Angelis FD, Lamaty F, Martinez J, Colacino E. Synthesis of novel multi-cationic PEG-based ionic liquids New Journal of Chemistry. 38: 6133-6138. DOI: 10.1039/C4Nj01208A  0.549
2014 Hamel A, Sacco M, Mnasri N, Lamaty F, Martinez J, Angelis FD, Colacino E, Charnay C. Micelles into Glycerol Solvent: Overcoming Side Reactions of Glycerol. Acs Sustainable Chemistry & Engineering. 2: 1353-1358. DOI: 10.1021/Sc500207R  0.57
2014 Sebih F, Bellahouel S, Rolland M, Derdour A, Martinez J, Rolland V. Diastereospecific synthesis of new 4-substituted l-theanine derivatives Tetrahedron-Asymmetry. 25: 690-696. DOI: 10.1016/J.Tetasy.2014.03.016  0.326
2014 Bantreil X, Kanfar N, Gehin N, Golliard E, Ohlmann P, Martinez J, Lamaty F. Iron-catalyzed benzamide formation. Application to the synthesis of moclobemide Tetrahedron. 70: 5093-5099. DOI: 10.1016/J.Tet.2014.06.001  0.563
2014 Malcor J, Brouillette Y, Graffion J, Spielmann K, Masurier N, Maillard LT, Martinez J, Lisowski V. Synthesis and reactivity of pyrrolo[3,2-d][1,3]oxazine-2,4-dione. Access to new pyrrolo[3,2-e][1,4]diazepine-2,5-diones Tetrahedron. 70: 4631-4639. DOI: 10.1016/J.Tet.2014.05.046  0.338
2014 René A, Martinez J, Cavelier F. N-Substituted Glycines with Functional Side-Chains for Peptoid Synthesis European Journal of Organic Chemistry. 2014: 8142-8147. DOI: 10.1002/Ejoc.201402864  0.384
2013 Jebors S, Cecillon S, Faye C, Enjalbal C, Amblard M, Mehdi A, Subra G, Martinez J. From protected trialkoxysilyl-peptide building blocks to bioorganic-silica hybrid materials. Journal of Materials Chemistry. B. 1: 6510-6515. PMID 32261327 DOI: 10.1039/C3Tb21326A  0.329
2013 Jebors S, Enjalbal C, Amblard M, Mehdi A, Subra G, Martinez J. Bioorganic hybrid OMS by straightforward grafting of trialkoxysilyl peptides. Journal of Materials Chemistry B. 1: 2921-2925. PMID 32260858 DOI: 10.1039/C3Tb20122H  0.314
2013 André C, Legrand B, Moulat L, Wenger E, Didierjean C, Aubert E, Averlant-Petit MC, Martinez J, Amblard M, Calmes M. Mixed oligoureas based on constrained bicyclic and acyclic β-amino acids derivatives: on the significance of the subunit configuration for folding. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 16963-71. PMID 24307359 DOI: 10.1002/Chem.201302829  0.602
2013 Echalier C, Al-Halifa S, Kreiter A, Enjalbal C, Sanchez P, Ronga L, Puget K, Verdié P, Amblard M, Martinez J, Subra G. Heating and microwave assisted SPPS of C-terminal acid peptides on trityl resin: the truth behind the yield. Amino Acids. 45: 1395-403. PMID 24142338 DOI: 10.1007/S00726-013-1604-Z  0.675
2013 Rouhana J, Hoh F, Estaran S, Henriquet C, Boublik Y, Kerkour A, Trouillard R, Martinez J, Pugnière M, Padilla A, Chavanieu A. Fragment-based identification of a locus in the Sec7 domain of Arno for the design of protein-protein interaction inhibitors. Journal of Medicinal Chemistry. 56: 8497-511. PMID 24112024 DOI: 10.1021/Jm4009357  0.788
2013 Maynadier M, Vezenkov LL, Amblard M, Martin V, Gandreuil C, Vaillant O, Gary-Bobo M, Basile I, Hernandez JF, Garcia M, Martinez J. Dipeptide mimic oligomer transporter mediates intracellular delivery of Cathepsin D inhibitors: a potential target for cancer therapy. Journal of Controlled Release : Official Journal of the Controlled Release Society. 171: 251-7. PMID 23899821 DOI: 10.1016/J.Jconrel.2013.07.017  0.776
2013 Bocheva A, Nocheva H, Pavlov N, Todorov P, Calmès M, Martinez J, Naydenova E. Synthesis and analgesic effects of novel β2-tryptophan hexapeptide analogs. Amino Acids. 45: 983-8. PMID 23851698 DOI: 10.1007/S00726-013-1555-4  0.75
2013 Louet M, Karakas E, Perret A, Perahia D, Martinez J, Floquet N. Conformational restriction of G-proteins Coupled Receptors (GPCRs) upon complexation to G-proteins: A putative activation mode of GPCRs? Febs Letters. 587: 2656-2661. PMID 23851072 DOI: 10.1016/J.Febslet.2013.06.052  0.78
2013 Mary S, Fehrentz JA, Damian M, Gaibelet G, Orcel H, Verdié P, Mouillac B, Martinez J, Marie J, Banères JL. Heterodimerization with Its splice variant blocks the ghrelin receptor 1a in a non-signaling conformation: a study with a purified heterodimer assembled into lipid discs. The Journal of Biological Chemistry. 288: 24656-65. PMID 23839942 DOI: 10.1074/Jbc.M113.453423  0.784
2013 Touati-Jallabe Y, Bojnik E, Legrand B, Mauchauffée E, Chung NN, Schiller PW, Benyhe S, Averlant-Petit MC, Martinez J, Hernandez JF. Cyclic enkephalins with a diversely substituted guanidine bridge or a thiourea bridge: synthesis, biological and structural evaluations. Journal of Medicinal Chemistry. 56: 5964-73. PMID 23822516 DOI: 10.1021/Jm4008592  0.749
2013 Zamfirova R, Pavlov N, Todorov P, Mateeva P, Martinez J, Calmès M, Naydenova E. Synthesis and changes in affinity for NOP and opioid receptors of novel hexapeptides containing β(2)-tryptophan analogues. Bioorganic & Medicinal Chemistry Letters. 23: 4052-5. PMID 23768905 DOI: 10.1016/J.Bmcl.2013.05.064  0.756
2013 Chaubet G, Coursindel T, Morelli X, Betzi S, Roche P, Guari Y, Lebrun A, Toupet L, Collette Y, Parrot I, Martinez J. Stereoselective synthesis of original spirolactams displaying promising folded structures. Organic & Biomolecular Chemistry. 11: 4719-26. PMID 23760068 DOI: 10.1039/C3Ob40643A  0.535
2013 Tétreault P, Beaudet N, Perron A, Belleville K, René A, Cavelier F, Martinez J, Stroh T, Jacobi AM, Rose SD, Behlke MA, Sarret P. Spinal NTS2 receptor activation reverses signs of neuropathic pain. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 27: 3741-52. PMID 23756650 DOI: 10.1096/Fj.12-225540  0.773
2013 René A, Vanthuyne N, Martinez J, Cavelier F. (L)-(Trimethylsilyl)alanine synthesis exploiting hydroxypinanone-induced diastereoselective alkylation. Amino Acids. 45: 301-7. PMID 23620077 DOI: 10.1007/S00726-013-1492-2  0.346
2013 Mathieu L, Legrand B, Deng C, Vezenkov L, Wenger E, Didierjean C, Amblard M, Averlant-Petit MC, Masurier N, Lisowski V, Martinez J, Maillard LT. Helical oligomers of thiazole-based γ-amino acids: synthesis and structural studies. Angewandte Chemie (International Ed. in English). 52: 6006-10. PMID 23619818 DOI: 10.1002/Anie.201302106  0.581
2013 Miralles G, Verdié P, Puget K, Maurras A, Martinez J, Subra G. Microwave-mediated reduction of disulfide bridges with supported (tris(2-carboxyethyl)phosphine) as resin-bound reducing agent. Acs Combinatorial Science. 15: 169-173. PMID 23438263 DOI: 10.1021/Co300104K  0.368
2013 Bahi A, Tolle V, Fehrentz JA, Brunel L, Martinez J, Tomasetto CL, Karam SM. Ghrelin knockout mice show decreased voluntary alcohol consumption and reduced ethanol-induced conditioned place preference Peptides. 43: 48-55. PMID 23428971 DOI: 10.1016/J.Peptides.2013.02.008  0.66
2013 Marsouvanidis PJ, Nock BA, Hajjaj B, Fehrentz JA, Brunel L, M'Kadmi C, van der Graaf L, Krenning EP, Maina T, Martinez J, de Jong M. Gastrin releasing peptide receptor-directed radioligands based on a bombesin antagonist: synthesis, (111)in-labeling, and preclinical profile. Journal of Medicinal Chemistry. 56: 2374-84. PMID 23427837 DOI: 10.1021/Jm301692P  0.63
2013 Spina R, Colacino E, Martinez J, Lamaty F. Poly(ethylene glycol) as a reaction matrix in platinum- or gold-catalyzed cycloisomerization: a mechanistic investigation. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 3817-21. PMID 23417756 DOI: 10.1002/Chem.201203800  0.545
2013 Maillard LT, Bertout S, Quinonéro O, Akalin G, Turan-Zitouni G, Fulcrand P, Demirci F, Martinez J, Masurier N. Synthesis and anti-Candida activity of novel 2-hydrazino-1,3-thiazole derivatives. Bioorganic & Medicinal Chemistry Letters. 23: 1803-7. PMID 23403080 DOI: 10.1016/J.Bmcl.2013.01.039  0.781
2013 Spina R, Colacino E, Gabriele B, Salerno G, Martinez J, Lamaty F. Synthesis of pyrrolin-4-ones by Pt-catalyzed cycloisomerization in PEG under microwaves. The Journal of Organic Chemistry. 78: 2698-702. PMID 23374030 DOI: 10.1021/Jo302474R  0.579
2013 Mary S, Fehrentz JA, Damian M, Verdié P, Martinez J, Marie J, Banères JL. How ligands and signalling proteins affect G-protein-coupled receptors' conformational landscape. Biochemical Society Transactions. 41: 144-7. PMID 23356274 DOI: 10.1042/Bst20120267  0.719
2013 Schaeffer M, Langlet F, Lafont C, Molino F, Hodson DJ, Roux T, Lamarque L, Verdié P, Bourrier E, Dehouck B, Banères JL, Martinez J, Méry PF, Marie J, Trinquet E, et al. Rapid sensing of circulating ghrelin by hypothalamic appetite-modifying neurons. Proceedings of the National Academy of Sciences of the United States of America. 110: 1512-7. PMID 23297228 DOI: 10.1073/Pnas.1212137110  0.769
2013 Peuchmaur M, Lacour MA, Sévalle J, Lisowski V, Touati-Jallabe Y, Rodier F, Martinez J, Checler F, Hernandez JF. Further characterization of a putative serine protease contributing to the γ-secretase cleavage of β-amyloid precursor protein. Bioorganic & Medicinal Chemistry. 21: 1018-29. PMID 23294826 DOI: 10.1016/J.Bmc.2012.11.045  0.799
2013 Paramelle D, Miralles G, Subra G, Martinez J. Chemical cross-linkers for protein structure studies by mass spectrometry Proteomics. 13: 438-456. PMID 23255214 DOI: 10.1002/Pmic.201200305  0.32
2013 Henry L, Fabre C, Guiraud I, Bastide S, Fabbro-Peray P, Martinez J, Lavabre-Bertrand T, Meunier L, Stoebner PE. Clinical use of p-proteasome in discriminating metastatic melanoma patients: Comparative study with LDH, MIA and S100B protein International Journal of Cancer. 133: 142-148. PMID 23238767 DOI: 10.1002/Ijc.27991  0.75
2013 Enomoto H, Nottelet B, Halifa SA, Enjalbal C, Dupré M, Tailhades J, Coudane J, Subra G, Martinez J, Amblard M. Synthesis of peptide-grafted comb polypeptides via polymerisation of NCA-peptides. Chemical Communications (Cambridge, England). 49: 409-11. PMID 23187977 DOI: 10.1039/C2Cc37597D  0.635
2013 Cassina V, Torsello A, Tempestini A, Salerno D, Brogioli D, Tamiazzo L, Bresciani E, Martinez J, Fehrentz JA, Verdié P, Omeljaniuk RJ, Possenti R, Rizzi L, Locatelli V, Mantegazza F. Biophysical characterization of a binding site for TLQP-21, a naturally occurring peptide which induces resistance to obesity Biochimica Et Biophysica Acta. 1828: 455-460. PMID 23122777 DOI: 10.1016/J.Bbamem.2012.10.023  0.63
2013 Ronga L, Verdié P, Sanchez P, Enjabal C, Maurras A, Jullian M, Puget K, Martinez J, Subra G. Supported oligomethionine sulfoxide and Ellman's reagent for cysteine bridges formation. Amino Acids. 44: 733-742. PMID 22968665 DOI: 10.1007/S00726-012-1397-5  0.29
2013 Moulin A, Brunel L, Boeglin D, Demange L, Ryan J, M'Kadmi C, Denoyelle S, Martinez J, Fehrentz JA. The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist. Amino Acids. 44: 301-14. PMID 22798076 DOI: 10.1007/S00726-012-1355-2  0.632
2013 Bonnamour J, Métro T, Martinez J, Lamaty F. Environmentally benign peptide synthesis using liquid-assisted ball-milling: application to the synthesis of Leu-enkephalin Green Chemistry. 15: 1116-1120. DOI: 10.1039/C3Gc40302E  0.614
2013 Konnert L, Gauliard A, Lamaty F, Martinez J, Colacino E. Solventless Synthesis of N-Protected Amino Acids in a Ball Mill Acs Sustainable Chemistry & Engineering. 1: 1186-1191. DOI: 10.1021/Sc4001115  0.603
2013 Arama DP, Lisowski V, Scarlata E, Fulcrand P, Maillard LT, Martinez J, Masurier N. An efficient synthesis of pyrido-imidazodiazepinediones Tetrahedron Letters. 54: 1364-1367. DOI: 10.1016/J.Tetlet.2012.12.087  0.801
2013 Zajdel P, Masurier N, Canale V, Verdie P, Amblard M, Pawłowski M, Martinez J, Subra G. The pipecolic linker—an acid-labile handle for derivatization of secondary amines on a solid-support. Part 3 Tetrahedron Letters. 54: 998-1002. DOI: 10.1016/J.Tetlet.2012.12.036  0.289
2013 Jebors S, Enjalbal C, Amblard M, Subra G, Mehdi A, Martinez J. Switchable polymer-grafted mesoporous silica's: from polyesters to polyamides biosilica hybrid materials Tetrahedron. 69: 7670-7674. DOI: 10.1016/J.Tet.2013.05.090  0.289
2013 Martin C, Lebrun A, Martinez J, Cavelier F. Synthesis of homopolypeptides with PPII structure Journal of Polymer Science Part A. 51: 3103-3109. DOI: 10.1002/Pola.26705  0.273
2013 Azua A, Mata JA, Heymes P, Peris E, Lamaty F, Martinez J, Colacino E. Palladium N-Heterocyclic Carbene Catalysts for the Ultrasound-Promoted Suzuki-Miyaura Reaction in Glycerol Advanced Synthesis & Catalysis. 355: 1107-1116. DOI: 10.1002/Adsc.201201047  0.782
2012 Dupré M, Enjalbal C, Cantel S, Martinez J, Megouda N, Hadjersi T, Boukherroub R, Coffinier Y. Investigation of silicon-based nanostructure morphology and chemical termination on laser desorption ionization mass spectrometry performance. Analytical Chemistry. 84: 10637-44. PMID 23163782 DOI: 10.1021/Ac3021104  0.605
2012 Métro TX, Bonnamour J, Reidon T, Sarpoulet J, Martinez J, Lamaty F. Mechanosynthesis of amides in the total absence of organic solvent from reaction to product recovery. Chemical Communications (Cambridge, England). 48: 11781-3. PMID 23108313 DOI: 10.1039/C2Cc36352F  0.593
2012 Declerck V, Colacino E, Bantreil X, Martinez J, Lamaty F. Poly(ethylene glycol) as reaction medium for mild Mizoroki-Heck reaction in a ball-mill. Chemical Communications (Cambridge, England). 48: 11778-80. PMID 23104100 DOI: 10.1039/C2Cc36286D  0.556
2012 Louet M, Charlier L, Martinez J, Floquet N. Dissociation of membrane-anchored heterotrimeric G-protein induced by G(α) subunit binding to GTP. Journal of Chemical Information and Modeling. 52: 3022-3027. PMID 23094679 DOI: 10.1021/Ci3003717  0.277
2012 Spina R, Colacino E, Gabriele B, Salerno G, Martinez J, Lamaty F. Preparation of enantioenriched iodinated pyrrolinones by iodocyclization of α-amino-ynones. Organic & Biomolecular Chemistry. 10: 9085-9. PMID 23086312 DOI: 10.1039/C2Ob26427G  0.588
2012 Legrand B, André C, Wenger E, Didierjean C, Averlant-Petit MC, Martinez J, Calmes M, Amblard M. Robust helix formation in a new family of oligoureas based on a constrained bicyclic building block. Angewandte Chemie (International Ed. in English). 51: 11267-70. PMID 23038643 DOI: 10.1002/Anie.201205842  0.576
2012 Cantel S, Brunel L, Ohara K, Enjalbal C, Martinez J, Vasseur JJ, Smietana M. An innovative strategy for sulfopeptides analysis using MALDI-TOF MS reflectron positive ion mode. Proteomics. 12: 2247-57. PMID 22887944 DOI: 10.1002/Pmic.201100525  0.623
2012 Dupré M, Cantel S, Durand JO, Martinez J, Enjalbal C. Silica nanoparticles pre-spotted onto target plate for laser desorption/ionization mass spectrometry analyses of peptides. Analytica Chimica Acta. 741: 47-57. PMID 22840704 DOI: 10.1016/J.Aca.2012.06.037  0.471
2012 Louet M, Martinez J, Floquet N. GDP Release Preferentially Occurs on the Phosphate Side in Heterotrimeric G-proteins Plos Computational Biology. 8. PMID 22829757 DOI: 10.1371/Journal.Pcbi.1002595  0.255
2012 Pringos E, Crouzin N, Cavalier M, Guiramand J, Cohen-Solal C, Martinez J, Vignes M, Rolland V. Synthesis and characterization of a cyclooctapeptide analogue of ω-agatoxin IVB enhancing the activity of Cav2.1 calcium channels activity in cultured hippocampal neurons. Neurochemistry International. 61: 632-639. PMID 22819793 DOI: 10.1016/J.Neuint.2012.07.009  0.298
2012 Shi X, Betzi S, Lugari A, Opi S, Restouin A, Parrot I, Martinez J, Zimmermann P, Lecine P, Huang M, Arold ST, Collette Y, Morelli X. Structural recognition mechanisms between human Src homology domain 3 (SH3) and ALG-2-interacting protein X (Alix). Febs Letters. 586: 1759-64. PMID 22641034 DOI: 10.1016/J.Febslet.2012.05.017  0.588
2012 Mary S, Damian M, Louet M, Floquet N, Fehrentz JA, Marie J, Martinez J, Banères JL. Ligands and signaling proteins govern the conformational landscape explored by a G protein-coupled receptor. Proceedings of the National Academy of Sciences of the United States of America. 109: 8304-9. PMID 22573814 DOI: 10.1073/Pnas.1119881109  0.726
2012 Masurier N, Aruta R, Gaumet V, Denoyelle S, Moreau E, Lisowski V, Martinez J, Maillard LT. Selective C-acylation of 2-aminoimidazo[1,2-a]pyridine: application to the synthesis of imidazopyridine-fused [1,3]diazepinones. Journal of Organic Chemistry. 77: 3679-3685. PMID 22423645 DOI: 10.1021/Jo300364D  0.316
2012 Nun P, Pérez V, Calmès M, Martinez J, Lamaty F. Preparation of chiral amino esters by asymmetric phase-transfer catalyzed alkylations of Schiff bases in a ball mill. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 3773-9. PMID 22322525 DOI: 10.1002/Chem.201102885  0.58
2012 André C, Legrand B, Deng C, Didierjean C, Pickaert G, Martinez J, Averlant-Petit MC, Amblard M, Calmes M. (S)-ABOC: a rigid bicyclic β-amino acid as turn inducer. Organic Letters. 14: 960-3. PMID 22292802 DOI: 10.1021/Ol203406V  0.592
2012 Dupré M, Coffinier Y, Boukherroub R, Cantel S, Martinez J, Enjalbal C. Laser desorption ionization mass spectrometry of protein tryptic digests on nanostructured silicon plates. Journal of Proteomics. 75: 1973-90. PMID 22282018 DOI: 10.1016/J.Jprot.2011.12.039  0.619
2012 Malcor JD, Payrot N, David M, Faucon A, Abouzid K, Jacquot G, Floquet N, Debarbieux F, Rougon G, Martinez J, Khrestchatisky M, Vlieghe P, Lisowski V. Chemical optimization of new ligands of the low-density lipoprotein receptor as potential vectors for central nervous system targeting. Journal of Medicinal Chemistry. 55: 2227-41. PMID 22257077 DOI: 10.1021/Jm2014919  0.794
2012 Todorov PT, Wesselinova DW, Pavlov ND, Martinez J, Calmes M, Naydenova ED. Cytotoxic activity of new racemic and optically active N-phosphonoalkyl bicyclic β-amino acids against human malignant cell lines. Amino Acids. 43: 1445-50. PMID 22237947 DOI: 10.1007/S00726-012-1217-Y  0.727
2012 Laville L, Charnay C, Lamaty F, Martinez J, Colacino E. Ring-closing metathesis in aqueous micellar medium. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 760-4. PMID 22161970 DOI: 10.1002/Chem.201101985  0.549
2012 Damian M, Marie J, Leyris JP, Fehrentz JA, Verdié P, Martinez J, Banères JL, Mary S. High constitutive activity is an intrinsic feature of ghrelin receptor protein: a study with a functional monomeric GHS-R1a receptor reconstituted in lipid discs. The Journal of Biological Chemistry. 287: 3630-41. PMID 22117076 DOI: 10.1074/Jbc.M111.288324  0.734
2012 Dupré M, Cantel S, Martinez J, Enjalbal C. Occurrence of C-terminal residue exclusion in peptide fragmentation by ESI and MALDI tandem mass spectrometry. Journal of the American Society For Mass Spectrometry. 23: 330-46. PMID 22095165 DOI: 10.1007/S13361-011-0254-1  0.633
2012 Martin C, Vanthuyne N, Miramon H, Martinez J, Cavelier F. Resolution of protected silaproline for a gram scale preparation. Amino Acids. 43: 649-655. PMID 22002795 DOI: 10.1007/S00726-011-1112-Y  0.287
2012 André C, Calmès M, Escale F, Amblard M, Martinez J, Songis O. New 1,3-amino alcohols derived from enantiopure bridgehead β-aminobicyclo[2.2.2]oct-5-ene-2-carboxylic acids. Amino Acids. 43: 415-21. PMID 21968501 DOI: 10.1007/S00726-011-1097-6  0.741
2012 Henri P, Beaumel S, Guezennec A, Poumès C, Stoebner PE, Stasia MJ, Guesnet J, Martinez J, Meunier L. MC1R expression in HaCaT keratinocytes inhibits UVA-induced ROS production via NADPH Oxidase- and cAMP-dependent mechanisms Journal of Cellular Physiology. 227: 2578-2585. PMID 21898403 DOI: 10.1002/Jcp.22996  0.704
2012 Clifford PS, Rodriguez J, Schul D, Hughes S, Kniffin T, Hart N, Eitan S, Brunel L, Fehrentz JA, Martinez J, Wellman PJ. Attenuation of cocaine-induced locomotor sensitization in rats sustaining genetic or pharmacologic antagonism of ghrelin receptors. Addiction Biology. 17: 956-63. PMID 21790898 DOI: 10.1111/J.1369-1600.2011.00339.X  0.769
2012 Moussa A, Meffre P, Martinez J, Rolland V. Chemoenzymatic routes to enantiomerically pure 2-azatyrosine and 2-, 3- and 4-pyridylalanine derivatives. Amino Acids. 42: 1339-1348. PMID 21279396 DOI: 10.1007/S00726-010-0829-3  0.344
2012 Boutard N, Labéguère F, Vidal Y, Lavergne JP, Martinez J. New C-glycosylated α-amino acid synthesis by addition reaction of an amino acid organozinc reagent on carbohydrate-derived aldehydes Synthetic Communications. 42: 1461-1471. DOI: 10.1080/00397911.2010.540698  0.599
2012 Spina R, Colacino E, Gabriele B, Salerno G, Martinez J, Lamaty F. Electrophilic Iodo-Mediated Cyclization in PEG under Microwave Irradiation: Easy Access to Highly Functionalized Furans and Pyrroles Synlett. 23: 1481-1484. DOI: 10.1055/S-0031-1291012  0.575
2012 Géant P, Martínez J, Rocard L, Salom-Roig XJ. A Divergent Synthetic StrategyBased on the Regioselective Reductive Ring-Opening ofa Cyclic 1,2-p-Methoxybenzylidene Acetal Synthesis. 44: 1247-1252. DOI: 10.1055/S-0031-1289746  0.266
2012 Aubin Y, Colacino E, Bouchouk D, Chataigner I, Sánchez MdM, Martinez J, Dewynter G. Unprecedented directed oxidative cross-coupling of sulfahydantoins with aldehydes via a radical sulfonate–sulfinate conversion New Journal of Chemistry. 36: 1560-1563. DOI: 10.1039/C2Nj40294G  0.303
2012 Azua A, Mata JA, Peris E, Lamaty F, Martinez J, Colacino E. Alternative Energy Input for Transfer Hydrogenation using Iridium NHC Based Catalysts in Glycerol as Hydrogen Donor and Solvent Organometallics. 31: 3911-3919. DOI: 10.1021/Om300109E  0.783
2012 Mekki S, Bellahouel S, Vanthuyne N, Rolland M, Derdour A, Martinez J, Vignes M, Rolland V. A focus on the asymmetric synthesis of a novel threo-β-benzyl-β-hydroxy aspartate analogue Tetrahedron-Asymmetry. 23: 94-99. DOI: 10.1016/J.Tetasy.2012.01.004  0.274
2012 Bantreil X, Sidi-Ykhlef M, Aringhieri L, Colacino E, Martinez J, Lamaty F. Comprehensive study on olefin metathesis in PEG as an alternative solvent under microwave irradiation Journal of Catalysis. 294: 113-118. DOI: 10.1016/J.Jcat.2012.07.007  0.559
2012 Colacino E, Martinez J, Lamaty F, Patrikeeva LS, Khemchyan LL, Ananikov VP, Beletskaya IP. PEG as an alternative reaction medium in metal-mediated transformations Coordination Chemistry Reviews. 256: 2893-2920. DOI: 10.1016/J.Ccr.2012.05.027  0.668
2012 Bubenikova S, Stancu IC, Kalinovska L, Schacht E, Lippens E, Declercq H, Cornelissen M, Santin M, Amblard M, Martinez J. Chemoselective cross-linking of alginate with thiol-terminated peptides for tissue engineering applications Carbohydrate Polymers. 88: 1239-1250. DOI: 10.1016/J.Carbpol.2012.01.089  0.683
2012 Todorov PT, Pavlov ND, Shivachev BL, Petrova RN, Martinez J, Naydenova ED, Calmes M. Synthesis of new racemic and optically active N‐phosphonoalkyl bicyclic β‐amino acids via the kabachnik–fields reaction as potential biologically active compounds Heteroatom Chemistry. 23: 123-130. DOI: 10.1002/Hc.20759  0.345
2012 Géant P, Martínez J, Salom‐Roig XJ. A Route to “all-cis” 2-Methyl-6-Substituted Piperidin-3-ol Alkaloids from syn-(2R,1′S)-2-(1-Dibenzylaminomethyl)epoxide: Rapid Total Synthesis of (+)-Deoxocassine European Journal of Organic Chemistry. 2012: 62-65. DOI: 10.1002/Ejoc.201101333  0.349
2012 Bantreil X, Fleith C, Martinez J, Lamaty F. Copper‐Catalyzed Direct Synthesis of Benzamides from Alcohols and Amines Chemcatchem. 4: 1922-1925. DOI: 10.1002/Cctc.201200441  0.591
2011 Pringos E, Vignes M, Martinez J, Rolland V. Peptide Neurotoxins That Affect Voltage-Gated Calcium Channels: A Close-Up on ω-Agatoxins Toxins. 3: 17-42. PMID 22069688 DOI: 10.3390/Toxins3010017  0.259
2011 Lugari A, Breuer S, Coursindel T, Opi S, Restouin A, Shi X, Nazabal A, Torbett BE, Martinez J, Collette Y, Parrot I, Arold ST, Morelli X. A specific protein disorder catalyzer of HIV-1 Nef. Bioorganic & Medicinal Chemistry. 19: 7401-6. PMID 22061824 DOI: 10.1016/J.Bmc.2011.10.051  0.66
2011 Wellman PJ, Clifford PS, Rodriguez J, Hughes S, Eitan S, Brunel L, Fehrentz JA, Martinez J. Pharmacologic antagonism of ghrelin receptors attenuates development of nicotine induced locomotor sensitization in rats. Regulatory Peptides. 172: 77-80. PMID 21903141 DOI: 10.1016/J.Regpep.2011.08.014  0.766
2011 Crouzin N, Ferreira MdJ, Cohen-Solal C, M'Kadmi C, Bernad N, Martinez J, Barbanel G, Vignes M, Guiramand J. α-Tocopherol and α-tocopheryl phosphate interact with the cannabinoid system in the rodent hippocampus Free Radical Biology and Medicine. 51: 1643-1655. PMID 21843633 DOI: 10.1016/J.Freeradbiomed.2011.07.012  0.257
2011 Pirnik Z, Bundziková J, Holubová M, Pýchová M, Fehrentz JA, Martinez J, Železná B, Maletínská L, Kiss A. Ghrelin agonists impact on Fos protein expression in brain areas related to food intake regulation in male C57BL/6 mice. Neurochemistry International. 59: 889-895. PMID 21843570 DOI: 10.1016/J.Neuint.2011.08.001  0.278
2011 Henry L, Le Gallic L, Garcin G, Coux O, Jumez N, Roger P, Lavabre-Bertrand T, Martinez J, Meunier L, Stoebner PE. Proteolytic activity and expression of the 20S proteasome are increased in psoriasis lesional skin British Journal of Dermatology. 165: 311-320. PMID 21740404 DOI: 10.1111/J.1365-2133.2011.10447.X  0.695
2011 Pavlov N, Gilles P, Didierjean C, Wenger E, Naydenova E, Martinez J, Calmès M. Asymmetric synthesis of β2-tryptophan analogues via Friedel-Crafts alkylation of indoles with a chiral nitroacrylate. The Journal of Organic Chemistry. 76: 6116-24. PMID 21671594 DOI: 10.1021/Jo200733T  0.565
2011 Louet M, Perahia D, Martinez J, Floquet N. A concerted mechanism for opening the GDP binding pocket and release of the nucleotide in hetero-trimeric G-proteins. Journal of Molecular Biology. 411: 298-312. PMID 21663745 DOI: 10.1016/J.Jmb.2011.05.034  0.701
2011 Verdié P, Ronga L, Cristau M, Amblard M, Cantel S, Enjalbal C, Puget K, Martinez J, Subra G. Oxyfold: a simple and efficient solid-supported reagent for disulfide bond formation. Chemistry-An Asian Journal. 6: 2382-2389. PMID 21656691 DOI: 10.1002/Asia.201100202  0.305
2011 Tailhades J, Blanquer S, Nottelet B, Coudane J, Subra G, Verdié P, Schacht E, Martinez J, Amblard M. From polyesters to polyamides via O-N acyl migration: an original multi-transfer reaction. Macromolecular Rapid Communications. 32: 876-80. PMID 21604313 DOI: 10.1002/Marc.201100235  0.542
2011 Floquet N, Hernandez JF, Boucher JL, Martinez J. L-arginine binding to human inducible nitric oxide synthase: an antisymmetric funnel route toward isoform-specific inhibitors? Journal of Chemical Information and Modeling. 51: 1325-35. PMID 21574590 DOI: 10.1021/Ci100422V  0.727
2011 Dreyfus C, Larrouy M, Cavelier F, Martinez J, Pignol D, Arnoux P. The crystallographic structure of thermoNicotianamine synthase with a synthetic reaction intermediate highlights the sequential processing mechanism Chemical Communications. 47: 5825-5827. PMID 21487608 DOI: 10.1039/C1Cc10565E  0.526
2011 Dupré M, Cantel S, Verdié P, Martinez J, Enjalbal C. Sequencing Lys-N proteolytic peptides by ESI and MALDI tandem mass spectrometry. Journal of the American Society For Mass Spectrometry. 22: 265-79. PMID 21472586 DOI: 10.1007/S13361-010-0022-7  0.64
2011 Paramelle D, Enjalbal C, Amblard M, Forest E, Heymann M, Cantel S, Geourjon C, Martinez J, Subra G. Solid-Phase Cross-Linking (SPCL): a new tool for protein structure studies. Proteomics. 11: 1277-86. PMID 21319301 DOI: 10.1002/Pmic.201000029  0.793
2011 Touati-Jallabe Y, Chiche L, Hamzé A, Aumelas A, Lisowski V, Berthomieu D, Martinez J, Hernandez JF. Cyclic peptides with a diversely substituted guanidine bridge: solid-phase synthesis and structural analysis. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 2566-70. PMID 21294201 DOI: 10.1002/Chem.201003299  0.728
2011 Baron A, Verdié P, Martinez J, Lamaty F. cis-Apa: a practical linker for the microwave-assisted preparation of cyclic pseudopeptides via RCM cyclative cleavage. The Journal of Organic Chemistry. 76: 766-72. PMID 21214240 DOI: 10.1021/Jo101629V  0.681
2011 Leyris JP, Roux T, Trinquet E, Verdié P, Fehrentz JA, Oueslati N, Douzon S, Bourrier E, Lamarque L, Gagne D, Galleyrand JC, M'kadmi C, Martinez J, Mary S, Banères JL, et al. Homogeneous time-resolved fluorescence-based assay to screen for ligands targeting the growth hormone secretagogue receptor type 1a. Analytical Biochemistry. 408: 253-62. PMID 20937574 DOI: 10.1016/J.Ab.2010.09.030  0.73
2011 Calmes M, Escale F, Didierjean C, Martinez J. Synthesis of enantiopure trans-N-Boc-3-aminobicyclo[2.2.2]octane-2-carboxylic acids and their bicyclic 1,3-amino alcohol derivatives via the [4+2] cycloaddition of 1,3-cyclohexadiene to a chiral β-nitroacrylate. Chirality. 23: 245-9. PMID 20928894 DOI: 10.1002/Chir.20906  0.789
2011 Lenda F, Crouzin N, Cavalier M, Guiramand J, Lanté F, Barbanel G, Cohen-Solal C, Martinez J, Guenoun F, Lamaty F, Vignes M. Synthesis of C5-tetrazole derivatives of 2-amino-adipic acid displaying NMDA glutamate receptor antagonism. Amino Acids. 40: 913-22. PMID 20706748 DOI: 10.1007/S00726-010-0713-1  0.58
2011 Zajdel P, Król J, Grychowska K, Pawlowski M, Subra G, Nomezine G, Martinez J, Satala G, Bojarski AJ, Zhou Z, O'Donnell MJ, Scott WL. Solid-phase synthesis of arylpiperazine derivatives and implementatio of the distributed drug discovery (d3) project in the search for cns agents Molecules. 16: 4104-4121. DOI: 10.3390/Molecules16054104  0.717
2011 Subra G, Mehdi A, Enjalbal C, Amblard M, Brunel L, Corriu R, Martinez J. Functionalised mesoporous silica: a good opportunity for controlled peptide oligomerisation Journal of Materials Chemistry. 21: 6321-6326. DOI: 10.1039/C0Jm04492J  0.65
2011 Nun P, Martin C, Martinez J, Lamaty F. Solvent-free synthesis of hydrazones and their subsequent N-alkylation in a Ball-mill Tetrahedron. 67: 8187-8194. DOI: 10.1016/J.Tet.2011.07.056  0.583
2011 Bibian M, Martinez J, Fehrentz J. Amino acids as building blocks for the synthesis of substituted 1,2,4-triazoles Tetrahedron. 67: 7042-7049. DOI: 10.1016/J.Tet.2011.07.011  0.632
2011 Chaubet G, Maillard LT, Martinez J, Masurier N. A tandem aza-Friedel–Crafts reaction/Hantzsch cyclization: a simple procedure to access polysubstituted 2-amino-1,3-thiazoles Tetrahedron. 67: 4897-4904. DOI: 10.1016/J.Tet.2011.04.090  0.309
2011 Gilles A, Martinez J, Cavelier F. A flexible synthesis of C33-C39 polyketide region of apratoxin: Synthesis of natural and unnatural analogues Comptes Rendus Chimie. 14: 437-440. DOI: 10.1016/J.Crci.2010.09.002  0.327
2011 Baron A, Kreuz C, Gosselin G, Lamaty F, Martinez J, Surleraux D, Pierra C, Clayette P. 37Synthesis and Anti-HIV Activity of d-peptide Analogs as HIV Fusion Inhibitors Antiviral Research. 90. DOI: 10.1016/J.Antiviral.2011.03.023  0.553
2011 Blayo A, Brunel F, Martinez J, Fehrentz J. Synthesis of Various Chiral 1,2,4-Triazole-Containing α-Amino Acids from Aspartic or Glutamic Acids European Journal of Organic Chemistry. 2011: 4293-4297. DOI: 10.1002/Ejoc.201100611  0.644
2011 Coursindel T, Martinez J, Parrot I. Concise Pathway to New Multifunctionalized Constrained Pentacin Derivatives by Means of Two Stereospecific Tandem Reactions European Journal of Organic Chemistry. 2011: 4519-4522. DOI: 10.1002/Ejoc.201100593  0.351
2011 Farran D, Archirel P, Toupet L, Martinez J, Dewynter G. Enantiodivergent transannular rearrangement of 3-isopropyl-1,4- benzodiazepine-2,5-dione by memory of chirality European Journal of Organic Chemistry. 2043-2047. DOI: 10.1002/Ejoc.201100030  0.678
2011 Géant P, Martínez J, Salom‐Roig XJ. Highly Enantioselective Access to α‐Dibenzylamino Ketones from Chiral Nonracemic α‐Bromo α′‐Sulfinyl Ketones by Dynamic Kinetic Resolution: Synthesis of (2R,1′S)‐2‐[1‐(Dibenzylamino)alkyl]oxiranes European Journal of Organic Chemistry. 2011: 1300-1309. DOI: 10.1002/Ejoc.201001403  0.276
2010 Zajdel P, Nomezine G, Masurier N, Amblard M, Pawłowski M, Martinez J, Subra G. A New Highly Versatile Handle for Chemistry on a Solid Support: The Pipecolic Linker Chemistry: a European Journal. 16: 7547-7553. PMID 22865765 DOI: 10.1002/Chem.201201452  0.365
2010 Petiot P, Charnay C, Martinez J, Puttergill L, Galindo F, Lamaty F, Colacino E. Synthesis of a new hydrophilic poly(ethylene glycol)-ionic liquid and its application in peptide synthesis. Chemical Communications (Cambridge, England). 46: 8842-4. PMID 20953493 DOI: 10.1039/C0Cc02402C  0.706
2010 Paramelle D, Subra G, Vezenkov LL, Maynadier M, André C, Enjalbal C, Calmès M, Garcia M, Martinez J, Amblard M. A straightforward approach for cellular-uptake quantification. Angewandte Chemie (International Ed. in English). 49: 8240-3. PMID 20865711 DOI: 10.1002/Anie.201003347  0.266
2010 Vezenkov LL, Maynadier M, Hernandez JF, Averlant-Petit MC, Fabre O, Benedetti E, Garcia M, Martinez J, Amblard M. Noncationic dipeptide mimic oligomers as cell penetrating nonpeptides (CPNP). Bioconjugate Chemistry. 21: 1850-4. PMID 20815388 DOI: 10.1021/Bc1002086  0.774
2010 Zajdel P, Masurier N, Sanchez P, Pawlowski M, Kreiter A, Nomezine G, Enjalbal C, Amblard M, Martinez J, Subra G. Recycling the versatile Pipecolic linker. Journal of Combinatorial Chemistry. 12: 747-53. PMID 20715810 DOI: 10.1021/Cc100099Z  0.656
2010 Henry L, Lavabre-Bertrand T, Douche T, Uttenweiler-Joseph S, Fabbro-Peray P, Monsarrat B, Martinez J, Meunier L, Stoebner PE. Diagnostic value and prognostic significance of plasmatic proteasome level in patients with melanoma Experimental Dermatology. 19: 1054-1059. PMID 20707810 DOI: 10.1111/J.1600-0625.2010.01151.X  0.749
2010 Papazacharias S, Magafa V, Bernad N, Pairas G, Spyroulias GA, Martinez J, Cordopatis P. Synthesis and Biological Evaluation of New CRH Analogues Bioinorganic Chemistry and Applications. 2010: 6652-6657. PMID 20689735 DOI: 10.1155/2010/252348  0.336
2010 Coursindel T, Restouin A, Dewynter G, Martinez J, Collette Y, Parrot I. Stereoselective ring contraction of 2,5-diketopiperazines: An innovative approach to the synthesis of promising bioactive 5-membered scaffolds. Bioorganic Chemistry. 38: 210-217. PMID 20609458 DOI: 10.1016/J.Bioorg.2010.05.002  0.298
2010 Gozé C, Bergé G, M'Kadmi C, Floquet N, Gagne D, Galleyrand JC, Fehrentz JA, Martinez J. Involvement of tryptophan W276 and of two surrounding amino acid residues in the high constitutive activity of the ghrelin receptor GHS-R1a. European Journal of Pharmacology. 643: 153-61. PMID 20599926 DOI: 10.1016/J.Ejphar.2010.06.018  0.725
2010 Schmidt J, Garambois V, Rocheblave L, Martinez J, Pèlegrin A, Cavelier F, Vivès E. Cyclization of peptides through a urea bond: application to the Arg-Gly-Asp tripeptide. Chembiochem. 11: 1083-1092. PMID 20422669 DOI: 10.1002/Cbic.201000062  0.351
2010 Osterstock G, Escobar P, Mitutsova V, Gouty-Colomer LA, Fontanaud P, Molino F, Fehrentz JA, Carmignac D, Martinez J, Guerineau NC, Robinson IC, Mollard P, Méry PF. Ghrelin stimulation of growth hormone-releasing hormone neurons is direct in the arcuate nucleus. Plos One. 5: e9159. PMID 20161791 DOI: 10.1371/Journal.Pone.0009159  0.779
2010 Moulin A, Bibian M, Blayo AL, El Habnouni S, Martinez J, Fehrentz JA. Synthesis of 3,4,5-trisubstituted-1,2,4-triazoles. Chemical Reviews. 110: 1809-27. PMID 20151658 DOI: 10.1021/Cr900107R  0.579
2010 Dalkas GA, Marchand D, Galleyrand J, Martinez J, Spyroulias GA, Cordopatis P, Cavelier F. Study of a lipophilic captopril analogue binding to angiotensin I converting enzyme. Journal of Peptide Science. 16: 91-97. PMID 20014331 DOI: 10.1002/Psc.1201  0.309
2010 Miramon H, Cavelier F, Martinez J, Cottet H. Highly Resolutive Separations of Hardly Soluble Synthetic Polypeptides by Capillary Electrophoresis Analytical Chemistry. 82: 394-399. PMID 19954161 DOI: 10.1021/Ac902211F  0.306
2010 Tailhades J, Gidel MA, Grossi B, Lécaillon J, Brunel L, Subra G, Martinez J, Amblard M. Synthesis of Peptide Alcohols on the Basis of an O–N Acyl‐Transfer Reaction Angewandte Chemie. 49: 117-120. PMID 19950151 DOI: 10.1002/Anie.200904276  0.266
2010 Vlieghe P, Lisowski V, Martinez J, Khrestchatisky M. Synthetic therapeutic peptides: science and market. Drug Discovery Today. 15: 40-56. PMID 19879957 DOI: 10.1016/J.Drudis.2009.10.009  0.588
2010 Floquet N, M'Kadmi C, Perahia D, Gagne D, Bergé G, Marie J, Banères JL, Galleyrand JC, Fehrentz JA, Martinez J. Activation of the ghrelin receptor is described by a privileged collective motion: a model for constitutive and agonist-induced activation of a sub-class A G-protein coupled receptor (GPCR). Journal of Molecular Biology. 395: 769-84. PMID 19782690 DOI: 10.1016/J.Jmb.2009.09.051  0.8
2010 Roussy G, Lemire M, Belleville K, Beaudet N, Martinez J, Sarret P. Targeting the neurotensinergic system to soothe bone cancer pain F1000research. 1. DOI: 10.7490/F1000Research.495.1  0.557
2010 Geneviève R, Lemire M, Belleville K, Beaudet N, Martinez J, Philippe S. Abstract P1-03-08: Targeting Neurotensinergic Receptors for Bone Cancer Pain Relief Cancer Research. 70. DOI: 10.1158/0008-5472.Sabcs10-P1-03-08  0.236
2010 Nun P, Martinez J, Lamaty F. Microwave-Assisted Neat Procedurefor the Petasis Reaction Synthesis. 2010: 2063-2068. DOI: 10.1055/S-0029-1218727  0.573
2010 Coursindel T, Martinez J, Parrot I. Microwave-Assisted Hydantoins Synthesis on Solid Support Journal of Chemical Education. 87: 640-642. DOI: 10.1021/Ed100169F  0.307
2010 Schmidt J, Garambois V, Rocheblave L, Martinez J, Cavelier F, Pelegrin A, Vivès É. R120 Un tétracyclopeptide inhibiteur de la prolifération métastatique Bulletin Du Cancer. 97. DOI: 10.1016/S0007-4551(15)31039-0  0.266
2010 Henry L, Lavabre-Bertrand T, Douché T, Uttenweiler-Joseph S, Fabbro-Peray P, Monsarrat B, Martinez J, Meunier L, Stoebner P. R49: Valeurs diagnostique, pronostique et caractérisation structurale des protéasomes plasmatiques dans le mélanome Bulletin Du Cancer. 97: S34. DOI: 10.1016/S0007-4551(15)30966-8  0.553
2010 Baron A, Martinez J, Lamaty F. Solvent-free synthesis of unsaturated amino esters in a ball-mill Tetrahedron Letters. 51: 6246-6249. DOI: 10.1016/J.Tetlet.2010.09.069  0.591
2010 Bakhrou N, Lamaty F, Martinez J, Colacino E. Ring-closing metathesis in glycerol under microwave activation Tetrahedron Letters. 51: 3935-3937. DOI: 10.1016/J.Tetlet.2010.05.101  0.556
2010 Bibian M, Blayo A, Moulin A, Martinez J, Fehrentz J. Multi-gram scale mercury-free synthesis of optically pure 3,4,5-trisubstituted 1,2,4-triazoles using silver benzoate Tetrahedron Letters. 51: 2660-2663. DOI: 10.1016/J.Tetlet.2010.03.037  0.607
2010 Fécourt F, Lopez G, Lee AVD, Martinez J, Dewynter G. Cyclosulfamide as a chiral auxiliary: application to efficient asymmetric synthesis (alkylation/aldolization) Tetrahedron-Asymmetry. 21: 2361-2366. DOI: 10.1016/J.Tetasy.2010.09.001  0.294
2010 Colacino E, Villebrun L, Martinez J, Lamaty F. PEG3400-Cu2O-CS2CO3: an efficient and recyclable microwave-enhanced catalytic system for ligand-free Ullmann arylation of indole and benzimidazole Tetrahedron. 66: 3730-3735. DOI: 10.1016/J.Tet.2010.03.065  0.561
2010 Blanquer S, Tailhades J, Darcos V, Amblard M, Martinez J, Nottelet B, Coudane J. Easy synthesis and ring‐opening polymerization of 5‐Z‐amino‐δ‐valerolactone: New degradable amino‐functionalized (Co)polyesters Journal of Polymer Science Part A. 48: 5891-5898. DOI: 10.1002/Pola.24400  0.32
2010 Bouazaoui M, Larrouy M, Martinez J, Cavelier F. Efficient synthesis of nicotianamine and non-natural analogues. European Journal of Organic Chemistry. 2010: 6609-6617. DOI: 10.1002/Ejoc.201000920  0.354
2010 PARIS M, POTHION C, MICHALAK C, MARTINEZ J, FEHRENTZ J. ChemInform Abstract: Synthesis of Cyanoketophosphoranes, Precursors of β-Amino-α-keto-esters from UNCAs. Cheminform. 29: no-no. DOI: 10.1002/CHIN.199849249  0.266
2010 PARIS M, FEHRENTZ J, HEITZ A, LOFFET A, MARTINEZ J. ChemInform Abstract: Synthesis of N-Protected γ-Amino-β-keto-esters from Urethane N-Carboxyanhydrides (UNCAs). Cheminform. 28: no-no. DOI: 10.1002/CHIN.199712189  0.266
2010 POTHION C, FEHRENTZ J, AUMELAS A, LOFFET A, MARTINEZ J. ChemInform Abstract: Synthesis of Pyrrolidine-2,4-diones from Urethane N-Carboxyanhydrides ( UNCAs). Cheminform. 27: no-no. DOI: 10.1002/CHIN.199622124  0.266
2010 FEHRENTZ J, POTHION C, CALIFANO J, LOFFET A, MARTINEZ J. ChemInform Abstract: Synthesis of Chiral N-Protected α-Amino Aldehydes by Reduction of N-Protected N-Carboxyanhydrides (UNCAs). Cheminform. 26: no-no. DOI: 10.1002/CHIN.199517039  0.266
2010 FEHRENTZ J, CALIFANO J, AMBLARD M, LOFFET A, MARTINEZ J. ChemInform Abstract: Synthesis of Chiral N-Protected β-Amino Alcohols by the Use of UNCAs. Cheminform. 25: no-no. DOI: 10.1002/CHIN.199423212  0.266
2009 Paramelle D, Cantel S, Enjalbal C, Amblard M, Forest E, Heymann M, Geourjon C, Martinez J, Subra G. A new generation of cross-linkers for selective detection by MALDI MS. Proteomics. 9: 5384-8. PMID 19902427 DOI: 10.1002/Pmic.200900562  0.794
2009 Declerck V, Nun P, Martinez J, Lamaty F. Solvent-free synthesis of peptides. Angewandte Chemie (International Ed. in English). 48: 9318-21. PMID 19882706 DOI: 10.1002/Anie.200903510  0.553
2009 Nehmé R, Perrin C, Guerlavais V, Fehrentz JA, Cottet H, Martinez J, Fabre H. Use of coated capillaries for the electrophoretic separation of stereoisomers of a growth hormone secretagogue. Electrophoresis. 30: 3772-9. PMID 19810026 DOI: 10.1002/Elps.200900093  0.575
2009 Salomé N, Hansson C, Taube M, Gustafsson-Ericson L, Egecioglu E, Karlsson-Lindahl L, Fehrentz JA, Martinez J, Perrissoud D, Dickson SL. On the central mechanism underlying ghrelin's chronic pro-obesity effects in rats: new insights from studies exploiting a potent ghrelin receptor antagonist. Journal of Neuroendocrinology. 21: 777-85. PMID 19703102 DOI: 10.1111/J.1365-2826.2009.01895.X  0.683
2009 Garcin G, Le Gallic L, Stoebner PE, Guezennec A, Guesnet J, Lavabre-Bertrand T, Martinez J, Meunier L. Constitutive expression of mc1r in hacat keratinocytes inhibits basal and uvb-induced tnf-α production Photochemistry and Photobiology. 85: 1440-1450. PMID 19656324 DOI: 10.1111/J.1751-1097.2009.00598.X  0.695
2009 Roussy G, Dansereau MA, Baudisson S, Ezzoubaa F, Belleville K, Beaudet N, Martinez J, Richelson E, Sarret P. Evidence for a role of NTS2 receptors in the modulation of tonic pain sensitivity. Molecular Pain. 5: 38. PMID 19580660 DOI: 10.1186/1744-8069-5-38  0.546
2009 Shenar N, Cantel S, Martinez J, Enjalbal C. Comparison of inert supports in laser desorption/ionization mass spectrometry of peptides: pencil lead, porous silica gel, DIOS-chip and NALDI target. Rapid Communications in Mass Spectrometry. 23: 2371-2379. PMID 19575411 DOI: 10.1002/Rcm.4158  0.295
2009 Zajdel P, Subra G, Verdie P, Gabzdyl E, Bojarski AJ, Duszyńska B, Martinez J, Pawłowski M. Sulfonamides with the N-alkyl-N'-dialkylguanidine moiety as 5-HT7 receptor ligands. Bioorganic & Medicinal Chemistry Letters. 19: 4827-4831. PMID 19560916 DOI: 10.1016/J.Bmcl.2009.06.038  0.312
2009 Zajdel P, Pawlowski M, Martinez J, Subra G. Combinatorial Chemistry on Solid Support in the Search for Central Nervous System Agents Combinatorial Chemistry & High Throughput Screening. 12: 723-739. PMID 19531014 DOI: 10.2174/138620709788923719  0.318
2009 Brouillette Y, Martinez J, Lisowski V. From thienodiazepinediones to thienopyridinones: flexible synthesis of substituted thieno[3,2-e][1,4]diazepinones and 6-aminothieno[3,2-b]pyridinones. Journal of Organic Chemistry. 74: 4975-4981. PMID 19480411 DOI: 10.1021/Jo900627A  0.312
2009 Sevalle J, Ayral E, Hernandez JF, Martinez J, Checler F. Pharmacological evidences for DFK167-sensitive presenilin-independent gamma-secretase-like activity. Journal of Neurochemistry. 110: 275-83. PMID 19457123 DOI: 10.1111/J.1471-4159.2009.06131.X  0.729
2009 Peuchmaur M, Lisowski V, Gandreuil C, Maillard LT, Martinez J, Hernandez JF. Solid-phase synthesis of isocoumarins: a traceless halocyclization approach. The Journal of Organic Chemistry. 74: 4158-65. PMID 19438216 DOI: 10.1021/Jo900281A  0.751
2009 Gilles A, Martinez J, Cavelier F. Supported Synthesis of Oxoapratoxin A Journal of Organic Chemistry. 74: 4298-4304. PMID 19432410 DOI: 10.1021/Jo900583J  0.329
2009 Farran D, Echalier D, Martinez J, Dewynter G. Regioselective and sequential reactivity of activated 2,5-diketopiperazines Journal of Peptide Science. 15: 474-478. PMID 19408248 DOI: 10.1002/Psc.1139  0.688
2009 Bouazaoui M, Mari S, Czernic P, Curie C, Martinez J, Cavelier F. Synthesis and biological activity of nicotianamine and analogues. Advances in Experimental Medicine and Biology. 611: 555-7. PMID 19400311 DOI: 10.1007/978-0-387-73657-0_244  0.738
2009 Touati-Jallabe Y, Hamzé A, Bergé G, Verna C, Lajoix AD, Fulcrand P, Martinez J, Hernandez JF. Solid-phase synthesis of dipeptidic and pseudo-dipeptidic potential NOS inhibitors through a side-chain anchoring approach. Advances in Experimental Medicine and Biology. 611: 133-4. PMID 19400126 DOI: 10.1007/978-0-387-73657-0_59  0.728
2009 Ronga L, Palladino P, Ragone R, Martinez J, Benedetti E, Rossi F, Amblard M. Spectroscopic analysis of synthetic PrP helix2-binding peptide constructs. Advances in Experimental Medicine and Biology. 611: 75-6. PMID 19400100 DOI: 10.1007/978-0-387-73657-0_33  0.735
2009 Brouillette Y, Lisowski V, Martinez J. Thieno[3,2-e]diazepinediones and 3-Thienylimidazolidinediones Syntheses: Regio-Controlled Ring Opening of Thiaisatoic Anhydride by α-Amino Acids Advances in Experimental Medicine and Biology. 611: 9-10. PMID 19400071 DOI: 10.1007/978-0-387-73657-0_4  0.266
2009 Salomé N, Haage D, Perrissoud D, Moulin A, Demange L, Egecioglu E, Fehrentz JA, Martinez J, Dickson SL. Anorexigenic and electrophysiological actions of novel ghrelin receptor (GHS-R1A) antagonists in rats. European Journal of Pharmacology. 612: 167-73. PMID 19356720 DOI: 10.1016/J.Ejphar.2009.03.066  0.78
2009 Couffin-Hoarau AC, Aubertin AM, Boustta M, Schmidt S, Fehrentz JA, Martinez J, Vert M. Peptide-poly(L-lysine citramide) conjugates and their in vitro anti-HIV behavior. Biomacromolecules. 10: 865-76. PMID 19296658 DOI: 10.1021/Bm801376V  0.617
2009 Declerck V, Toupet L, Martinez J, Lamaty F. Selective [3 + 2] Huisgen cycloaddition. Synthesis of trans-disubstituted triazolodiazepines from aza-Baylis-Hillman adducts. The Journal of Organic Chemistry. 74: 2004-7. PMID 19199794 DOI: 10.1021/Jo802533D  0.583
2009 Ayral E, Gloanec P, Bergé G, de Nanteuil G, Mennecier P, Rupin A, Verbeuren TJ, Fulcrand P, Martinez J, Hernandez JF. Design, synthesis, and biological evaluation of 1,5-benzothiazepine-4-one derivatives targeting factor VIIa/tissue factor. Bioorganic & Medicinal Chemistry Letters. 19: 1386-91. PMID 19181521 DOI: 10.1016/J.Bmcl.2009.01.039  0.755
2009 Declerck V, Martinez J, Lamaty F. aza-Baylis-Hillman reaction. Chemical Reviews. 109: 1-48. PMID 19140772 DOI: 10.1021/Cr068057C  0.553
2009 Bélanger S, Bovenzi V, Côté J, Neugebauer W, Amblard M, Martinez J, Lammek B, Savard M, Gobeil F. Structure-activity relationships of novel peptide agonists of the human bradykinin B2 receptor. Peptides. 30: 777-87. PMID 19111586 DOI: 10.1016/J.Peptides.2008.12.003  0.646
2009 Shenar N, Sommerer N, Martinez J, Enjalbal C. Comparison of LID versus CID activation modes in tandem mass spectrometry of peptides. Journal of Mass Spectrometry. 44: 621-632. PMID 19097045 DOI: 10.1002/Jms.1535  0.263
2009 Zajdel P, Subra G, Verdie P, Bojarski AJ, Duszyńska B, Basista K, Obniska J, Martinez J, Pawłowski M. The influence of an ethylene spacer on the 5-HT(1A) and 5-HT(2A) receptor affinity of arylpiperazine derivatives of amides with N-acylated amino acids and 3-differently substituted pyrrolidine-2,5-diones. European Journal of Medicinal Chemistry. 44: 800-808. PMID 18603331 DOI: 10.1016/J.Ejmech.2008.05.021  0.32
2009 Royuela M, Chazalette D, Rivier F, Hugon G, Paniagua R, Guerlavais V, Fehrentz J, Martinez J, Mornet D. Dystrophin and dystrophin-associated protein in muscles and nerves from monkey. European Journal of Histochemistry. 47: 29-38. PMID 12685555 DOI: 10.4081/804  0.235
2009 Condamine E, Chapdeleine G, Demarcy L, Duclos J, Davoust D, Llinares M, Azay J, Martinez J, Chapelle S. Biological activity and three-dimensional structure of an agonist analog of bombesin Journal of Peptide Research. 51: 55-64. PMID 9495592 DOI: 10.1111/J.1399-3011.1998.Tb00417.X  0.327
2009 Galleyrand JC, Lima‐Leite AC, Lallement JC, Lignon MF, Bernad N, Fulcrand P, Martinez J. Synthesis and characterization of a new labeled gastrin ligand, 125I‐BH‐[Leu15]‐gastrin‐(5‐17), on binding to canine fundic mucosal cells and Jurkat cells International Journal of Peptide and Protein Research. 44: 348-356. PMID 7875937 DOI: 10.1111/J.1399-3011.1994.Tb01019.X  0.296
2009 Martinez J, Laur J, Winternitz F. Synthesis of an IgG fragment decapeptide exhibiting phagocytosis stimulating activity of polymorphonuclear leucocytes International Journal of Peptide and Protein Research. 22: 119-124. PMID 6885245 DOI: 10.1111/J.1399-3011.1983.Tb02075.X  0.32
2009 Martinez J, Rodriguez M, Bali J, Laur J. Phenylethylamide derivatives of the C-terminal tetrapeptide of gastrin International Journal of Peptide and Protein Research. 28: 529-535. PMID 3818170 DOI: 10.1111/J.1399-3011.1986.Tb03288.X  0.359
2009 Laur J, Rodriguez M, Aumelas A, Bali J, Martinez J. Synthesis of analogues of the Des‐Phe‐NH2C‐terminal hexapeptide of cholecystokinin showing gastrin antagonist activity International Journal of Peptide and Protein Research. 27: 386-393. PMID 3710694 DOI: 10.1111/J.1399-3011.1986.Tb01032.X  0.356
2009 Aumelas A, Rodriguez M, Heitz A, Castro B, Martinez J. 1H and 13C n.m.r. studies of pseudo-peptide analogues of the C-terminal tetrapeptide of gastrin. International Journal of Peptide and Protein Research. 30: 596-604. PMID 3436696 DOI: 10.1111/J.1399-3011.1987.Tb03370.X  0.315
2009 Rodriguez M, Bali J, Magous R, Castro B, Martinez J. Synthesis of pseudo‐peptide analogues of the C‐terminal tetra‐peptide of gastrin and evaluation of their biological activity on acid secretion International Journal of Peptide and Protein Research. 27: 293-299. PMID 3011690 DOI: 10.1111/J.1399-3011.1986.Tb01823.X  0.349
2009 Briet C, Aumelas A, Martinez J. Synthesis of Z-CCK-27–32-NH2, Z-Tyr(So3-)-Met-Gly-Trp-Met-Asp-NH2, a cholecystokinin receptor antagonist and an inhibitor of gastrin-induced acid secretion International Journal of Peptide and Protein Research. 26: 294-298. PMID 2997059 DOI: 10.1111/J.1399-3011.1985.Tb03207.X  0.361
2009 Aumelas A, Audousset‐Puech M, Heitz A, Bataille D, Martinez J. 1H n.m.r. conformational studies on the C‐terminal octapeptide of oxyntomodulin, a β‐turn locked by a salt bridge International Journal of Peptide and Protein Research. 34: 268-276. PMID 2599765 DOI: 10.1111/J.1399-3011.1989.Tb01574.X  0.337
2009 Rodriguez M, Rolland M, Lignon M, Galas M, Laur J, Aumelas A, Martinez J. Synthesis and biological activities of some cholecystokinin analogues substituted in position 29 by a β-alanine International Journal of Peptide and Protein Research. 34: 394-404. PMID 2482263 DOI: 10.1111/J.1399-3011.1989.Tb00708.X  0.329
2009 Fulcrand P, Rodriguez M, Galas M, Lignon M, Laur J, Aumelas A, Martinez J. 2-Phenylethyl ester and 2-phenylethyl amide derivative analogues of the C-terminal hepta- and octapeptide of cholecystokinin. International Journal of Peptide and Protein Research. 32: 384-395. PMID 2463231 DOI: 10.1111/J.1399-3011.1988.Tb01273.X  0.328
2009 Rodriguez M, Amblard M, Galas M, Lignon M, Aumelas A, Martinez J. Synthesis of cyclic analogues of cholecystokinin highly selective for central receptors. International Journal of Peptide and Protein Research. 35: 441-451. PMID 2376470 DOI: 10.1111/J.1399-3011.1990.Tb00071.X  0.347
2009 Rolland M, Rodriguez M, Lignon M, Galas M, Laur J, Aumelas A, Martinez J. Synthesis and biological activity of 2‐phenylethyl ester analogues of C‐terminal heptapeptide of cholecystokinin modified in Trp 30 region International Journal of Peptide and Protein Research. 38: 181-192. PMID 1723720 DOI: 10.1111/J.1399-3011.1991.Tb01427.X  0.358
2009 Rodriguez M, Heitz A, Martinez J. Carba peptide bond surrogates : different approaches to Gly-ψ(CH2-CH2)-D,L-Xaa pseudo-dipeptide units International Journal of Peptide and Protein Research. 39: 273-277. PMID 1399267 DOI: 10.1111/J.1399-3011.1992.Tb00800.X  0.302
2009 Blanot D, Martinez J, Auger G, Bricas E. Synthesis of analogs of the serum thymic nonapeptide, "facteur thymique serique" (FTS). Part I. International Journal of Peptide and Protein Research. 14: 41-56. PMID 489246 DOI: 10.1111/J.1399-3011.1979.Tb01919.X  0.365
2009 MARTINEZ J, TOLLE JC, BODANSZKY M. SIDE REACTIONS IN PEPTIDE SYNTHESIS International Journal of Peptide and Protein Research. 13: 22-27. DOI: 10.1111/J.1399-3011.1979.Tb01845.X  0.605
2009 Turan-Zitouni G, Özdemir A, Kaplancıklı ZA, Fehrentz J, Martinez J, Chevallet P, Dusart G. Preparation of Some Thiazolyl Hydrazone Derivatives and Evaluation of Their Antibacterial Activities Phosphorus Sulfur and Silicon and the Related Elements. 184: 2613-2623. DOI: 10.1080/10426500802534176  0.61
2009 Colacino E, Benakki H, Guenoun F, Martinez J, Lamaty F. Synthesis of Novel Pyrrolo-[3,2-c]quinolines via Iron-Catalyzed Cross-Coupling Reaction of Grignard Reagents Synthetic Communications. 39: 1583-1591. DOI: 10.1080/00397910802550039  0.568
2009 Martinez J, Bodanszky M. SIDE REACTIONS IN PEPTIDE SYNTHESIS International Journal of Peptide and Protein Research. 12: 277-283. DOI: 10.1055/S-1981-29442  0.54
2009 Nun P, Martinez J, Lamaty F. Solvent-Free Microwave-Assisted Suzuki―Miyaura Coupling Catalyzed by PEPPSI-iPr Synlett. 2009: 1761-1764. DOI: 10.1055/S-0029-1217359  0.548
2009 Bibian M, El-Habnouni S, Martinez J, Fehrentz J. Enantioselective Synthesis of N-Protected α-Amino Acid Hydrazides Synthesis. 2009: 1180-1184. DOI: 10.1055/S-0028-1088013  0.618
2009 Brouillette Y, Sujol G, Martinez J, Lisowski V. Regio-Controlled NucleophilicAttack of 3-Thiaisatoic Anhydride by α-Amino Acids: One-PotSynthesis of 3-(2-Thienyl)imidazolidine-2,4-dione and 3,4-SubstitutedThieno[2,3-e][1,4]diazepine-2,5-dione Analogues Synthesis. 2009: 389-394. DOI: 10.1055/S-0028-1083320  0.332
2009 Jeanson A, Berthon C, Coantic S, Auwer CD, Floquet N, Funke H, Guillaneux D, Hennig C, Martinez J, Moisy P, Petit S, Proux O, Quémeneur E, Solari PL, Subra G. The role of aspartyl-rich pentapeptides in comparative complexation of actinide(IV) and iron(III). Part 1 New Journal of Chemistry. 33: 976-985. DOI: 10.1039/B813523A  0.28
2009 Salom-Roig XJ, Martínez J, Burguete MI, Galindo F, Luis SV, Miranda MA, Morant-Miñana MC, Pérez-Prieto J. Chiral synthetic pseudopeptidic derivatives as triplet excited state quenchers Tetrahedron Letters. 50: 4859-4862. DOI: 10.1016/J.Tetlet.2009.06.047  0.692
2009 Bouchouk D, Colacino E, Toupet L, Aouf N, Martinez J, Dewynter G. Activated sulfahydantoin as Boc-glycine enolate equivalent: highly diastereoselective α-hydroxyalkylation and application to the synthesis of aldopentonate analogues Tetrahedron Letters. 50: 1100-1104. DOI: 10.1016/J.Tetlet.2008.12.070  0.58
2009 Jullian M, Hernandez A, Maurras A, Puget K, Amblard M, Martinez J, Subra G. N-terminus FITC labeling of peptides on solid support: the truth behind the spacer Tetrahedron Letters. 50: 260-263. DOI: 10.1016/J.Tetlet.2008.10.141  0.362
2009 Burguete MI, Fawaz G, Galindo F, Izquierdo MÁ, Luis SV, Martínez J, Salom-Roig XJ. Fluorescence and mass spectrometry studies of the interaction between naproxen and synthetic pseudopeptidic models in organic media Tetrahedron. 65: 7801-7808. DOI: 10.1016/J.Tet.2009.07.031  0.687
2009 Bouazaoui M, Martinez J, Cavelier F. Direct Access to L‐Azetidine‐2‐carboxylic Acid European Journal of Organic Chemistry. 2009: 2729-2732. DOI: 10.1002/Ejoc.200900233  0.332
2009 Brouillette Y, Martinez J, Lisowski V. Chemistry of Ring‐Fused Oxazine‐2,4‐diones European Journal of Organic Chemistry. 2009: 3487-3503. DOI: 10.1002/Ejoc.200801007  0.303
2008 Farran D, Parrot I, Toupet L, Martinez J, Dewynter G. Transannular rearrangement of activated 2,5-diketopiperazines: A key route to original scaffolds Organic and Biomolecular Chemistry. 6: 3989-3996. PMID 18931807 DOI: 10.1039/B810352F  0.668
2008 Heymann M, Paramelle D, Subra G, Forest E, Martinez J, Geourjon C, Deléage G. MSX-3D: a tool to validate 3D protein models using mass spectrometry. Bioinformatics (Oxford, England). 24: 2782-3. PMID 18826958 DOI: 10.1093/Bioinformatics/Btn510  0.771
2008 Verdié P, Subra G, Averland-Petit M, Amblard M, Martinez J. Solid-phase synthesis of 4-methylcarboxy-1,4-benzodiazepine-2,5-diones. Acs Combinatorial Science. 10: 869-874. PMID 18821806 DOI: 10.1021/Cc800085D  0.404
2008 Cavelier F, Marchand D, Martinez J. α,α′‐Disubstituted Amino Acids with Silylated Side Chains as Lipophilic Building Blocks for the Synthesis of Peptaibol Analogues Chemistry & Biodiversity. 5: 1279-1287. PMID 18649314 DOI: 10.1002/Cbdv.200890114  0.337
2008 Shenar N, Martinez J, Enjalbal C. Laser desorption/ionization mass spectrometry on porous silica and alumina for peptide mass fingerprinting. Journal of the American Society For Mass Spectrometry. 19: 632-644. PMID 18356075 DOI: 10.1016/J.Jasms.2008.02.006  0.283
2008 Stoebner PE, Le Gallic L, Berthe ML, Boulle N, Lallemant B, Marque M, Gaspard C, Delfour C, Lavabre-Bertrand T, Martinez J, Meunier L. Decreased expression of thymidine phosphorylase/platelet-derived endothelial cell growth factor in basal cell carcinomas Experimental Dermatology. 17: 908-915. PMID 18341568 DOI: 10.1111/J.1600-0625.2008.00718.X  0.766
2008 Bredeloux P, Cavelier F, Dubuc I, Vivet B, Costentin J, Martinez J. Synthesis and biological effects of c(Lys-Lys-Pro-Tyr-Ile-Leu-Lys-Lys-Pro-Tyr-Ile-Leu) (JMV2012), a new analogue of neurotensin that crosses the blood-brain barrier. Journal of Medicinal Chemistry. 51: 1610-6. PMID 18321036 DOI: 10.1021/Jm700925K  0.798
2008 Moulin A, Demange L, Ryan J, Mousseaux D, Sanchez P, Bergé G, Gagne D, Perrissoud D, Locatelli V, Torsello A, Galleyrand JC, Fehrentz JA, Martinez J. New trisubstituted 1,2,4-triazole derivatives as potent ghrelin receptor antagonists. 3. Synthesis and pharmacological in vitro and in vivo evaluations. Journal of Medicinal Chemistry. 51: 689-93. PMID 18193826 DOI: 10.1021/Jm701292S  0.741
2008 Moulin A, Demange L, Ryan J, M'Kadmi C, Galleyrand JC, Martinez J, Fehrentz JA. Trisubstituted 1,2,4-triazoles as ligands for the ghrelin receptor: on the significance of the orientation and substitution at position 3. Bioorganic & Medicinal Chemistry Letters. 18: 164-8. PMID 18023181 DOI: 10.1016/J.Bmcl.2007.10.113  0.642
2008 Minta E, Kafarski P, Martinez J, Rolland V. Synthesis of cyclooctapeptides: constraints analogues of the peptidic neurotoxin, omega-agatoxine IVB-an experimental point of view. Journal of Peptide Science. 14: 267-277. PMID 17853503 DOI: 10.1002/Psc.919  0.371
2008 Brouillette Y, Verdié P, Martinez J, Lisowski V. Valuable Versatile Reactivityof Thiaisatoic Anhydrides: Expedient Solid­Phase Synthesisof Thieno[1,4]diazepine-2,5-diones Synlett. 2008: 2360-2364. DOI: 10.1055/S-2008-1078210  0.381
2008 Colacino E, André C, Martinez J, Lamaty F. Synthesis of a novel pyrrolo-[3,2-c]quinoline N-oxide by aza-Baylis–Hillman adduct of o-nitrobenzaldehyde Tetrahedron Letters. 49: 4953-4955. DOI: 10.1016/J.Tetlet.2008.05.121  0.592
2008 Lécaillon J, Gilles P, Subra G, Martinez J, Amblard M. Synthesis of cyclic peptides via O–N-acyl migration Tetrahedron Letters. 49: 4674-4676. DOI: 10.1016/J.Tetlet.2008.05.049  0.368
2008 Coursindel T, Farran D, Martinez J, Dewynter G. [15N]-Isotopic labeling: a suitable tool to study the reactivity of bis lactams Tetrahedron Letters. 49: 906-909. DOI: 10.1016/J.Tetlet.2007.11.159  0.657
2008 Songis O, Didierjean C, Martinez J, Calmès M. The iodolactone approach to enantiopure oxiranes of constrained chiral cyclic β-amino acids Tetrahedron-Asymmetry. 19: 2135-2139. DOI: 10.1016/J.Tetasy.2008.09.005  0.785
2008 Cerezo V, Amblard M, Martinez J, Verdié P, Planas M, Feliu L. Solid-phase synthesis of 5-arylhistidines via a microwave-assisted Suzuki–Miyaura cross-coupling Tetrahedron. 64: 10538-10545. DOI: 10.1016/J.Tet.2008.08.077  0.331
2008 Benakki H, Colacino E, André C, Guenoun F, Martinez J, Lamaty F. Microwave-assisted multi-step synthesis of novel pyrrolo-[3,2-c]quinoline derivatives Tetrahedron. 64: 5949-5955. DOI: 10.1016/J.Tet.2008.04.034  0.596
2008 Colacino E, Nun P, Colacino FM, Martinez J, Lamaty F. Solvent-free synthesis of nitrones in a ball-mill Tetrahedron. 64: 5569-5576. DOI: 10.1016/J.Tet.2008.03.091  0.592
2008 Coantic S, Subra G, Martinez J. Microwave-assisted Solid Phase Peptide Synthesis on High Loaded Resins International Journal of Peptide Research and Therapeutics. 14: 143-147. DOI: 10.1007/S10989-008-9123-6  0.281
2008 Marchand D, Martinez J, Cavelier F. Straightforward Synthesis of Chiral Silylated Amino Acids through Hydrosilylation European Journal of Organic Chemistry. 2008: 3107-3112. DOI: 10.1002/Ejoc.200800066  0.353
2008 Songis O, Géant PY, Sautrey G, Martinez J, Calmès M. Asymmetric Diels-Alder Reaction of Aminodienes with a Nonracemic Acrylate Bound to Rink Resin: A Comparison of These Reactions with Their Solution- State Analogues European Journal of Organic Chemistry. 2008: 308-318. DOI: 10.1002/Ejoc.200700677  0.352
2007 Farran D, Toupet L, Martinez J, Dewynter G. Stereocontrolled synthesis of 2,4-diamino-3-hydroxyacids starting from diketopiperazines: A new route for the preparation of statine analogues Organic Letters. 9: 4833-4836. PMID 17939675 DOI: 10.1021/Ol7021593  0.663
2007 Moulin A, Demange L, Bergé G, Gagne D, Ryan J, Mousseaux D, Heitz A, Perrissoud D, Locatelli V, Torsello A, Galleyrand JC, Fehrentz JA, Martinez J. Toward potent ghrelin receptor ligands based on trisubstituted 1,2,4-triazole structure. 2. Synthesis and pharmacological in vitro and in vivo evaluations. Journal of Medicinal Chemistry. 50: 5790-806. PMID 17927165 DOI: 10.1021/Jm0704550  0.733
2007 Dubs P, Bourel-Bonnet L, Subra G, Blanpain A, Melnyk O, Pinel A, Gras-Masse H, Martinez J. Parallel synthesis of a lipopeptide library by hydrazone-based chemical ligation. Acs Combinatorial Science. 9: 973-981. PMID 17896820 DOI: 10.1021/Cc070033B  0.643
2007 Farran D, Parrot I, Martinez J, Dewynter G. Transannular rearrangement of activated lactams: Stereoselective synthesis of substituted pyrrolidine-2,4-diones from diketopiperazines Angewandte Chemie - International Edition. 46: 7488-7490. PMID 17722139 DOI: 10.1002/Anie.200702132  0.669
2007 Villain-Guillot P, Gualtieri M, Bastide L, Roquet F, Martinez J, Amblard M, Pugniere M, Leonetti JP. Structure-activity relationships of phenyl-furanyl-rhodanines as inhibitors of RNA polymerase with antibacterial activity on biofilms. Journal of Medicinal Chemistry. 50: 4195-204. PMID 17665895 DOI: 10.1021/Jm0703183  0.657
2007 Lascoux D, Paramelle D, Subra G, Heymann M, Geourjon C, Martinez J, Forest E. Discrimination and selective enhancement of signals in the MALDI mass spectrum of a protein by combining a matrix-based label for lysine residues with a neutral matrix. Angewandte Chemie (International Ed. in English). 46: 5594-7. PMID 17591739 DOI: 10.1002/Anie.200700811  0.778
2007 Turan-Zitouni G, Fehrentz JA, Chevallet P, Martinez J, Kaplancikli ZA, Ozdemir A, Arslanyolu M, Yildiz MT. Synthesis and antibacterial activity of tert-butyl [1-benzyl-2[(4-aryl-2-thiazolyl)hydrazono]ethyl]carbamate derivatives. Archiv Der Pharmazie. 340: 310-4. PMID 17562564 DOI: 10.1002/Ardp.200600200  0.79
2007 Stoebner PE, Poosti R, Djoukelfit K, Martinez J, Meunier L. Decreased human epidermal antigen-presenting cell activity after ultraviolet A exposure: Dose-response effects and protection by sunscreens British Journal of Dermatology. 156: 1315-1320. PMID 17535231 DOI: 10.1111/J.1365-2133.2007.07895.X  0.698
2007 Moulin A, Ryan J, Martinez J, Fehrentz JA. Recent developments in ghrelin receptor ligands. Chemmedchem. 2: 1242-59. PMID 17520591 DOI: 10.1002/Cmdc.200700015  0.618
2007 Garcin G, Douki T, Stoebner PE, Guesnet J, Guezennec A, Martinez J, Cadet J, Meunier L. Cell surface expression of melanocortin-1 receptor on HaCaT keratinocytes and α-melanocortin stimulation do not affect the formation and repair of UVB-induced DNA photoproducts Photochemical and Photobiological Sciences. 6: 585-593. PMID 17487313 DOI: 10.1039/B615656H  0.743
2007 Demange L, Boeglin D, Moulin A, Mousseaux D, Ryan J, Bergé G, Gagne D, Heitz A, Perrissoud D, Locatelli V, Torsello A, Galleyrand JC, Fehrentz JA, Martinez J. Synthesis and pharmacological in vitro and in vivo evaluations of novel triazole derivatives as ligands of the ghrelin receptor. 1. Journal of Medicinal Chemistry. 50: 1939-57. PMID 17375904 DOI: 10.1021/Jm070024H  0.738
2007 Verdié P, Subra G, Feliu L, Sanchez P, Bergé G, Garcin G, Martinez J. On-line synthesis of pseudopeptide library incorporating a benzodiazepinone turn mimic: biological evaluation on MC1 receptors. Acs Combinatorial Science. 9: 254-262. PMID 17348731 DOI: 10.1021/Cc060054Q  0.372
2007 Brouillette Y, Lisowski V, Fulcrand P, Martinez J. Reactivity study of 1H-thieno[3,2-d][1,3]oxazine-2,4-dione toward the synthesis of bicyclic 3,4-dihydro-1H-thieno[3,2-e][1,4]diazepine-2,5-dione analogues. Journal of Organic Chemistry. 72: 2662-2665. PMID 17323999 DOI: 10.1021/Jo0622882  0.322
2007 Zajdel P, Subra G, Bojarski AJ, DuszyÅ„ska B, TatarczyÅ„ska E, Nikiforuk A, Chojnacka-Wójcik E, PawÅ‚owski M, Martinez J. Novel class of arylpiperazines containing N-acylated amino acids: their synthesis, 5-HT1A, 5-HT2A receptor affinity, and in vivo pharmacological evaluation. Bioorganic & Medicinal Chemistry. 15: 2907-19. PMID 17321139 DOI: 10.1016/J.Bmc.2007.02.018  0.613
2007 Mouls L, Aubagnac J, Martinez J, Enjalbal C. Low Energy Peptide Fragmentations in an ESI-Q-Tof Type Mass Spectrometer Journal of Proteome Research. 6: 1378-1391. PMID 17311442 DOI: 10.1021/Pr060574O  0.287
2007 Declerck V, Allouchi H, Martinez J, Lamaty F. 2-Trimethylsilylethanesulfonyl (SES) versus tosyl (Ts) protecting group in the preparation of nitrogen-containing five-membered rings. A novel route for the synthesis of substituted pyrrolines and pyrrolidines. The Journal of Organic Chemistry. 72: 1518-21. PMID 17288397 DOI: 10.1021/Jo062239P  0.583
2007 Nachman RJ, Fehrentz JA, Martinez J, Kaczmarek K, Zabrocki J, Coast GM. A C-terminal aldehyde analog of the insect kinins inhibits diuresis in the housefly. Peptides. 28: 146-52. PMID 17134792 DOI: 10.1016/J.Peptides.2006.09.017  0.6
2007 Moulin A, Martinez J, Fehrentz JA. Synthesis of peptide aldehydes. Journal of Peptide Science : An Official Publication of the European Peptide Society. 13: 1-15. PMID 16998827 DOI: 10.1002/Psc.787  0.622
2007 Boukallaba K, Elachqar A, Hallaoui AE, Alami A, Hajji SE, Labriti B, Atmani A, Bali BE, Lachkar M, Allouchi H, Martinez J, Rolland V. Synthesis of α-Heterocyclic α-Aminophosphonates, 1 Part II: Morpholine, Piperidine, Pyrrolidine, Tetrahydrofurylmethylamine, N-Benzyl-N-Methylamine, and Aniline Derivatives Phosphorus Sulfur and Silicon and the Related Elements. 182: 1045-1052. DOI: 10.1080/10426500601093739  0.299
2007 Moulin A, Garcia S, Martinez J, Fehrentz J. Synthesis of Substituted Imidazo[1,5-a]pyridines Starting from N-2-Pyridylmethylamides Using Lawesson’s Reagent and Mercury(II) Acetate Synthesis. 2007: 2667-2673. DOI: 10.1055/S-2007-983852  0.632
2007 Colacino E, Daïch L, Martinez J, Lamaty F. Microwave-Assisted Copper-Catalyzed Sonogashira Reaction in PEG Solvent Synlett. 2007: 1279-1283. DOI: 10.1055/S-2007-980337  0.55
2007 Colacino E, Lamaty F, Martinez J, Parrot I. Microwave-assisted solid-phase synthesis of hydantoin derivatives Tetrahedron Letters. 48: 5317-5320. DOI: 10.1016/J.Tetlet.2007.05.084  0.614
2007 Raynal N, Averlant-Petit M, Bergé G, Didierjean C, Marraud M, Duru C, Martinez J, Amblard M. Molecular modeling study for a novel structured oligomer subunit selection: the example of 2-aminomethyl-phenyl-acetic acid Tetrahedron Letters. 48: 1787-1790. DOI: 10.1016/J.Tetlet.2007.01.032  0.573
2007 Lenda F, Guenoun F, Martinez J, Lamaty F. Synthesis of new tetrazole and triazole substituted pyroglutamic acid and proline derivatives Tetrahedron Letters. 48: 805-808. DOI: 10.1016/J.Tetlet.2006.11.163  0.597
2007 Calmès M, Escale F, Didierjean C, Cazals G, Martinez J. Asymmetric Diels–Alder reaction using a new chiral β-nitroacrylate for enantiopure trans-β-norbornane amino acid preparation Tetrahedron-Asymmetry. 18: 2491-2496. DOI: 10.1016/J.Tetasy.2007.10.001  0.791
2007 Brouillette Y, Lisowski V, Guillon J, Massip S, Martinez J. Efficient one-pot microwave-assisted synthesis of 3-(thien-3-yl)imidazolidine-2,4-dione analogs Tetrahedron. 63: 7538-7544. DOI: 10.1016/J.Tet.2007.05.057  0.321
2007 Szlosek-Pinaud M, Diaz P, Martinez J, Lamaty F. Efficient synthetic approach to heterocycles possessing the 3,3-disubstituted-2,3-dihydrobenzofuran skeleton via diverse palladium-catalyzed tandem reactions Tetrahedron. 63: 3340-3349. DOI: 10.1016/J.Tet.2007.02.035  0.607
2007 Colacino E, Martinez J, Lamaty F. Preparation of NHC–ruthenium complexes and their catalytic activity in metathesis reaction Coordination Chemistry Reviews. 251: 726-764. DOI: 10.1016/J.Ccr.2006.07.017  0.571
2007 Verdié P, Subra G, Chevallet P, Amblard M, Martinez J. Solid Phase Synthesis of a Hydroxypyrrolidine Derivative and its Use in Solid Phase Peptide Synthesis as Constrained Statine Mimic International Journal of Peptide Research and Therapeutics. 13: 337-343. DOI: 10.1007/S10989-007-9088-X  0.393
2007 Zajdel P, Subra G, Pawłowski M, Martinez J. Solid‐Phase Synthesis of Aryl‐Alkylamine Derivatives Using Protected Aminoalcohol Building Blocks on SynPhaseTM Lanterns Qsar & Combinatorial Science. 26: 215-219. DOI: 10.1002/Qsar.200620036  0.347
2007 Subra G, Amblard M, Verdié P, Komesli S, Dutartre P, Durand P, Renaut P, Martinez J. Synthesis and TGF-β Receptor Binding Inhibition of Multibranched Compounds Qsar & Combinatorial Science. 26: 496-510. DOI: 10.1002/Qsar.200520134  0.277
2007 Songis O, Didierjean C, Laurent C, Martinez J, Calmès M. Asymmetric diels-alder cycloaddition of 1-aminocyclohexadiene to chiral acrylate : Synthesis of enantiopure bridgehead-aminobicyclo[2.2.2]octane-2-carboxylic acid derivatives European Journal of Organic Chemistry. 2007: 3166-3172. DOI: 10.1002/Ejoc.200700236  0.794
2007 Declerck V, Ribière P, Nédellec Y, Allouchi H, Martinez J, Lamaty F. A Microwave‐Assisted Heck Reaction in Poly(ethylene glycol) for the Synthesis of Benzazepines European Journal of Organic Chemistry. 2007: 201-208. DOI: 10.1002/Ejoc.200600680  0.594
2006 Buisson M, Rivail L, Hernandez JF, Jamin M, Martinez J, Ruigrok RW, Burmeister WP. Kinetics, inhibition and oligomerization of Epstein-Barr virus protease. Febs Letters. 580: 6570-8. PMID 17118362 DOI: 10.1016/J.Febslet.2006.11.006  0.783
2006 Mouls L, Subra G, Aubagnac J, Martinez J, Enjalbal C. Tandem mass spectrometry of amidated peptides Journal of Mass Spectrometry. 41: 1470-1483. PMID 17072914 DOI: 10.1002/Jms.1118  0.351
2006 Amblard M, Fehrentz JA, Martinez J, Subra G. Methods and protocols of modern solid phase Peptide synthesis. Molecular Biotechnology. 33: 239-54. PMID 16946453 DOI: 10.1385/Mb:33:3:239  0.625
2006 Cissé MA, Gandreuil C, Hernandez JF, Martinez J, Checler F, Vincent B. Design and characterization of a novel cellular prion-derived quenched fluorimetric substrate of alpha-secretase. Biochemical and Biophysical Research Communications. 347: 254-60. PMID 16806063 DOI: 10.1016/J.Bbrc.2006.06.065  0.743
2006 Pujals S, Fernandez-Carneado J, Kogan MJ, Martinez J, Cavelier F, Giralt E. Replacement of a Proline with Silaproline Causes a 20-Fold Increase in the Cellular Uptake of a Pro-Rich Peptide Journal of the American Chemical Society. 128: 8479-8483. PMID 16802813 DOI: 10.1021/Ja060036C  0.5
2006 Cavelier F, Marchand D, Mbassi P, Martinez J, Marraud M. Conformational studies of proline‐, thiaproline‐ and dimethylsilaproline‐containing diketopiperazines Journal of Peptide Science. 12: 621-625. PMID 16786506 DOI: 10.1002/Psc.767  0.313
2006 Ribière P, Declerck V, Martinez J, Lamaty F. 2-(Trimethylsilyl)ethanesulfonyl (or SES) group in amine protection and activation. Chemical Reviews. 106: 2249-69. PMID 16771449 DOI: 10.1021/Cr0300587  0.553
2006 Zajdel P, Subra G, Bojarski AJ, Duszyńska B, Pawłowski M, Martinez J. Arylpiperazines with N-acylated amino acids as 5-HT1A receptor ligands Bioorganic & Medicinal Chemistry Letters. 16: 3406-3410. PMID 16677812 DOI: 10.1016/J.Bmcl.2006.04.035  0.346
2006 Ganneau C, Moulin A, Demange L, Martinez J, Fehrentz JA. The epimerization of peptide aldehydes--a systematic study. Journal of Peptide Science : An Official Publication of the European Peptide Society. 12: 497-501. PMID 16625681 DOI: 10.1002/Psc.751  0.618
2006 Mousseaux D, Le Gallic L, Ryan J, Oiry C, Gagne D, Fehrentz JA, Galleyrand JC, Martinez J. Regulation of ERK1/2 activity by ghrelin-activated growth hormone secretagogue receptor 1A involves a PLC/PKCvarepsilon pathway. British Journal of Pharmacology. 148: 350-65. PMID 16582936 DOI: 10.1038/Sj.Bjp.0706727  0.736
2006 Ibarz G, Oiry C, Carnazzi E, Crespy P, Escrieut C, Fourmy D, Galleyrand JC, Gagne D, Martinez J. Cholecystokinin 1 receptor modulates the MEKK1-induced c-Jun trans-activation: structural requirements of the receptor. British Journal of Pharmacology. 147: 951-8. PMID 16491099 DOI: 10.1038/Sj.Bjp.0706690  0.628
2006 Feliu L, Font D, Soley R, Tailhades J, Martinez J, Amblard M. Microwave-enhanced solid phase synthesis of 1,4,8-triazaspiro[4.5]decan-2-ones Arkivoc. 2007: 65-72. DOI: 10.3998/Ark.5550190.0008.406  0.312
2006 Boukallaba K, Elachqar A, Hallaoui AE, Alami A, Hajji SE, Labriti B, Martinez J, Rolland V. Synthesis of New α-Heterocyclic α-Aminophosphonates Phosphorus Sulfur and Silicon and the Related Elements. 181: 819-823. DOI: 10.1080/10426500500272046  0.279
2006 Bouifraden S, Lavergne J, Martinez J, Viallefont P. Synthesis of New Glycopeptides from the α-D-Allofuranos-3-Spiropropiolactone Synthetic Communications. 27: 3909-3916. DOI: 10.1080/00397919708005914  0.313
2006 Nara S, Martinez J, Wermuth C, Parrot I. Palladium-catalysed cross-coupling reactions on pyridazine moieties Synlett. 2006: 3185-3204. DOI: 10.1055/S-2006-951528  0.287
2006 Declerck V, Martinez J, Lamaty F. Microwave-Assisted Copper-Catalyzed Heck Reaction in PEG Solvent Synlett. 2006: 3029-3032. DOI: 10.1055/S-2006-951523  0.556
2006 Moulin A, Martinez J, Fehrentz J. Convenient two-step preparation of [1,2,4]triazolo[4,3-a]pyridines from 2-hydrazinopyridine and carboxylic acids Tetrahedron Letters. 47: 7591-7594. DOI: 10.1016/J.Tetlet.2006.08.075  0.64
2006 Ribière P, Declerck V, Nédellec Y, Yadav-Bhatnagar N, Martinez J, Lamaty F. Synthesis of novel poly(ethylene glycol) supported benzazepines: the crucial role of PEG on the selectivity of an intramolecular Heck reaction Tetrahedron. 62: 10456-10466. DOI: 10.1016/J.Tet.2006.08.009  0.565
2006 Sévalle J, Eyral E, Hernandez J, Martinez J, Checler F. P3-238: Design of new fluorimetric substrates and new inhibitors of gamma-secretase and presenilinase activities Alzheimers & Dementia. 2. DOI: 10.1016/J.Jalz.2006.05.1507  0.266
2005 Sarret P, Esdaile MJ, Perron A, Martinez J, Stroh T, Beaudet A. Potent spinal analgesia elicited through stimulation of NTS2 neurotensin receptors. The Journal of Neuroscience : the Official Journal of the Society For Neuroscience. 25: 8188-96. PMID 16148226 DOI: 10.1523/Jneurosci.0810-05.2005  0.782
2005 Amblard M, Fehrentz JA, Martinez J, Subra G. Fundamentals of modern peptide synthesis. Methods in Molecular Biology (Clifton, N.J.). 298: 3-24. PMID 15897611 DOI: 10.1385/1-59259-877-3:003  0.624
2005 Enjalbal C, Ribière P, Lamaty F, Yadav-Bhatnagar N, Martinez J, Aubagnac JL. MALDI-TOF MS analysis of soluble PEG based multi-step synthetic reaction mixtures with automated detection of reaction failure. Journal of the American Society For Mass Spectrometry. 16: 670-8. PMID 15862768 DOI: 10.1016/J.Jasms.2005.01.020  0.557
2005 Zajdel P, Subra G, Bojarski AJ, Duszyńska B, Pawłowski M, Martinez J. Parallel solid-phase synthesis and characterization of new sulfonamide and carboxamide proline derivatives as potential CNS agents Bioorganic & Medicinal Chemistry. 13: 3029-3035. PMID 15781412 DOI: 10.1016/J.Bmc.2005.01.060  0.291
2005 Morel C, Ibarz G, Oiry C, Carnazzi E, Bergé G, Gagne D, Galleyrand JC, Martinez J. Cross-interactions of two p38 mitogen-activated protein (MAP) kinase inhibitors and two cholecystokinin (CCK) receptor antagonists with the CCK1 receptor and p38 MAP kinase. The Journal of Biological Chemistry. 280: 21384-93. PMID 15772081 DOI: 10.1074/Jbc.M408851200  0.617
2005 Lefranc-Jullien S, Lisowski V, Hernandez JF, Martinez J, Checler F. Design and characterization of a new cell-permeant inhibitor of the beta-secretase BACE1. British Journal of Pharmacology. 145: 228-35. PMID 15753947 DOI: 10.1038/Sj.Bjp.0706183  0.746
2005 Archer-Lahlou E, Escrieut C, Clerc P, Martinez J, Moroder L, Logsdon C, Kopin A, Seva C, Dufresne M, Pradayrol L, Maigret B, Fourmy D. Molecular mechanism underlying partial and full agonism mediated by the human cholecystokinin-1 receptor. The Journal of Biological Chemistry. 280: 10664-74. PMID 15632187 DOI: 10.1074/Jbc.M409451200  0.735
2005 Hamzé A, Gandreuil C, Lisowski V, Andureu F, Fulcrand P, Martinez J, Hernandez JF. Solid phase synthesis of mono- or disubstituted arginine containing peptides from an isothiocitrulline precursor Tetrahedron Letters. 46: 7349-7353. DOI: 10.1016/J.Tetlet.2005.08.120  0.645
2005 Amblard M, Raynal N, Averlant-Petit MC, Didierjean C, Calmès M, Fabre O, Aubry A, Marraud M, Martinez J. Structural elucidation of the β-turn inducing (S)-[3-amino-4-oxo-2,3- dihydro-5H-benzo[b][1,4]thiazepin-5-yl] acetic acid (DBT) motif Tetrahedron Letters. 46: 3733-3735. DOI: 10.1016/J.Tetlet.2005.03.134  0.784
2005 Minta E, Boutonnet C, Boutard N, Martinez J, Rolland V. Easy saponification by metal silanolates: application in SPPS and in (S)-5-hydroxynorvaline preparation Tetrahedron Letters. 46: 1795-1797. DOI: 10.1016/J.Tetlet.2005.01.115  0.333
2005 Calmès M, Didierjean C, Martinez J, Songis O. (R)-(4-(Benzyloxycarbonylphenyl)-3-hydroxy-4,4-dimethyl-2-pyrrolidinone) acrylate derivative as a chiral dienophile for the synthesis of enantiopure 2-aminocyclohexane carboxylic acids Tetrahedron-Asymmetry. 16: 2173-2178. DOI: 10.1016/J.Tetasy.2005.05.024  0.592
2005 Calmès M, Akkari R, Barthes N, Escale F, Martinez J. Asymmetric Baylis–Hillman reactions using (R)-4-(3-hydroxy-4,4-dimethyl-2-oxopyrrolidin-1-yl) benzoic acid acrylate derivatives in solution and on solid support Tetrahedron-Asymmetry. 16: 2179-2185. DOI: 10.1016/J.Tetasy.2005.05.016  0.334
2005 Sélambarom J, Smadja J, Thomas O, Parrot I, Martinez J, Pavia AA. A Novel Route to Pseudoproline (ΨH,HPro)-Containing Dipeptides Building Blocks International Journal of Peptide Research and Therapeutics. 11: 267-270. DOI: 10.1007/S10989-005-8114-0  0.574
2005 Lenda F, Guenoun F, Tazi B, larbi NB, Allouchi H, Martinez J, Lamaty F. Synthesis of New Tetrazole‐Substituted Pyroaminoadipic and Pipecolic Acid Derivatives European Journal of Organic Chemistry. 2005: 326-333. DOI: 10.1002/Ejoc.200400328  0.602
2004 Hamzé A, Martinez J, Hernandez JF. Solid-phase synthesis of arginine-containing peptides and fluorogenic substrates using a side-chain anchoring approach. The Journal of Organic Chemistry. 69: 8394-402. PMID 15549812 DOI: 10.1021/Jo048792T  0.75
2004 Declerck V, Ribière P, Martinez J, Lamaty F. Sequential aza-Baylis-Hillman/ring closing metathesis/aromatization as a novel route for the synthesis of substituted pyrroles. The Journal of Organic Chemistry. 69: 8372-81. PMID 15549809 DOI: 10.1021/Jo048519R  0.586
2004 Cantel S, Heitz A, Martinez J, Fehrentz JA. Synthesis of chiral alpha-amino aldehydes linked by their amine function to solid support. Journal of Peptide Science : An Official Publication of the European Peptide Society. 10: 531-4. PMID 15473261 DOI: 10.1002/Psc.605  0.627
2004 Giovannoni J, Didierjean C, Durand P, Marraud M, Aubry A, Renaut P, Martinez J, Amblard M. Synthesis and structure of symmetrical bicyclic hexapeptides bridged by metathesis reaction. Organic Letters. 6: 3449-52. PMID 15387520 DOI: 10.1021/Ol0487940  0.666
2004 Zajdel P, Bojarski AJ, Bugno R, Jurczyk S, Kołaczkowski M, Nowak M, Subra G, Martinez J, Pawłowski M. A study on application of impregnated synthetic peptide TLC stationary phases for the screening of 5-HT1A ligands. Part 2. Biomedical Chromatography. 18: 542-549. PMID 15386518 DOI: 10.1002/Bmc.354  0.354
2004 Zajdel P, Subra G, Bojarski AJ, Duszyńska B, Pawłowski M, Martinez J. A new class of arylpiperazine derivatives: the library synthesis on SynPhase lanterns and biological evaluation on serotonin 5-HT(1A) and 5-HT(2A) receptors. Acs Combinatorial Science. 6: 761-767. PMID 15360211 DOI: 10.1021/Cc049970Z  0.36
2004 Enjalbal C, Roggero R, Cerdan R, Martinez J, Vial H, Aubagnac JL. Automated monitoring of phosphatidylcholine biosyntheses in Plasmodium falciparum by electrospray ionization mass spectrometry through stable isotope labeling experiments. Analytical Chemistry. 76: 4515-21. PMID 15283596 DOI: 10.1021/Ac049759+  0.705
2004 Ribière P, Enjalbal C, Aubagnac JL, Yadav-Bhatnagar N, Martinez J, Lamaty F. Preparation of poly(ethylene glycol) sulfonamide: synthesis of N-supported beta-aminoesters via the aza-Baylis-Hillman reaction. Journal of Combinatorial Chemistry. 6: 464-7. PMID 15244405 DOI: 10.1021/Cc049966N  0.553
2004 Cantel S, Desgranges S, Martinez J, Fehrentz JA. Saponification of esters of chiral alpha-amino acids anchored through their amine function on solid support. Journal of Peptide Science : An Official Publication of the European Peptide Society. 10: 326-8. PMID 15214436 DOI: 10.1002/Psc.561  0.622
2004 Cavelier F, Marchand D, Martinez J, Sagan S. Biological activity of silylated amino acid containing substance P analogues Journal of Peptide Research. 63: 290-296. PMID 15049841 DOI: 10.1111/J.1399-3011.2004.00145.X  0.352
2004 Aubagnac J, Enjalbal C, Martinez J, Sanchez P, Subra G. Automated vs manual profiling of peptide libraries by mass spectrometry. Methods of Molecular Biology. 251: 377-385. PMID 14704459 DOI: 10.1385/1-59259-742-4:377  0.266
2004 Lenda F, Guenoun F, Tazi B, larbi NB, Martinez J, Lamaty F, Allouchi H. A new key intermediate in the synthesis of 6-oxo­piperidine-2-carboxyl­ate derivatives Acta Crystallographica Section E: Crystallographic Communications. 60. DOI: 10.1107/S1600536804011626  0.565
2004 Cantel S, Martinez J, Fehrentz J. Synthesis of chiral α-amino-diazoketones on solid support: An access to β-homologated amino acid derivatives Synlett. 2004: 2791-2793. DOI: 10.1055/S-2004-835639  0.631
2004 Lenda F, Guenoun F, Tazi B, larbi NB, Martinez J, Lamaty F. Synthesis of new triazole substituted pyroaminoadipic and pipecolic acid derivatives Tetrahedron Letters. 45: 8905-8907. DOI: 10.1016/J.Tetlet.2004.09.166  0.613
2004 Mouls L, Subra G, Enjalbal C, Martinez J, Aubagnac J-. O–N-Acyl migration in N-terminal serine-containing peptides: mass spectrometric elucidation and subsequent development of site-directed acylation protocols Tetrahedron Letters. 45: 1173-1178. DOI: 10.1016/J.Tetlet.2003.12.008  0.319
2004 Akkari R, Calmès M, Escale F, Iapichella J, Rolland M, Martinez J. (R)- or (S)-4-(3-hydroxy-4,4-dimethyl-2-oxopyrrolidin-1-yl)benzoic acid as a new chiral auxiliary for solid phase asymmetric Diels-Alder reactions Tetrahedron-Asymmetry. 15: 2515-2525. DOI: 10.1016/J.Tetasy.2004.06.012  0.35
2004 Wehbe J, Rolland V, Fruchier A, Roumestant M, Martinez J. Enantioselective synthesis of new 4-substituted glutamic acid derivatives Tetrahedron-Asymmetry. 15: 851-858. DOI: 10.1016/J.Tetasy.2004.01.006  0.308
2004 Ribière P, Yadav-Bhatnagar N, Martinez J, Lamaty F. Microwave-assisted aza-Baylis-Hillman Reaction. Preparation of Poly(ethylene Glycol) Supported α-methylene-β-Aminoester Qsar & Combinatorial Science. 23: 911-914. DOI: 10.1002/Qsar.200420041  0.58
2004 Feliu L, Martinez J, Amblard M. Synthesis of an 8-benzyl-4-(p-substituted-benzyl)-1,4,8-triazaspiro[4.5]decan-2-one library on synphase TMLanterns Qsar & Combinatorial Science. 23: 56-60. DOI: 10.1002/Qsar.200320007  0.364
2004 Akkari R, Calmès M, Martinez J. Toward Diels−Alder Reactions on a Solid Support Using Polymer Bound N‐Substituted 3‐Hydroxy‐4,4‐dimethyl‐2‐pyrrolidinone Acrylate Derivatives European Journal of Organic Chemistry. 2004: 2441-2450. DOI: 10.1002/Ejoc.200400019  0.344
2004 Filip SV, Lejeune V, Vors J, Martinez J, Cavelier F. Peptide Bond Formation Using Polymer‐Bound BOP European Journal of Organic Chemistry. 2004: 1936-1939. DOI: 10.1002/Ejoc.200300798  0.341
2004 Rolland-Fulcrand V, Rolland M, Roumestant ML, Martinez J. Chemoenzymatic synthesis of enantiomerically pure (2S,3R,4S)-4- hydroxyisoleucine, an insulinotropic amino acid isolated from fenugreek seeds European Journal of Organic Chemistry. 873-877. DOI: 10.1002/Ejoc.200300434  0.545
2004 Ghanem N, Martinez J, Stien D. Quaternary Ammonium-Supported Scavenger Reagents for Acids and Electrophiles European Journal of Organic Chemistry. 2004: 84-89. DOI: 10.1002/Ejoc.200300403  0.299
2003 Nachman RJ, Coast GM, Douat C, Fehrentz JA, Kaczmarek K, Zabrocki J, Pryor NW, Martinez J. A C-terminal aldehyde insect kinin analog enhances inhibition of weight gain and induces significant mortality in Helicoverpa zea larvae. Peptides. 24: 1615-21. PMID 14706541 DOI: 10.1016/J.Peptides.2003.06.008  0.784
2003 Royuela M, Chazalette D, Hugon G, Paniagua R, Guerlavais V, Fehrentz JA, Martinez J, Labbe J-, Rivier F, Mornet D. Formation of multiple complexes between beta-dystroglycan and dystrophin family products Journal of Muscle Research and Cell Motility. 24: 387-397. PMID 14677641 DOI: 10.1023/A:1027309822007  0.235
2003 Huck J, Roumestant ML, Martinez J. From beta-N-tert-butyloxycarbonyl N-carboxyanhydrides to beta-aminoacid derivatives. The Journal of Peptide Research : Official Journal of the American Peptide Society. 62: 233-7. PMID 14632925 DOI: 10.1046/J.1399-3011.2003.00080.X  0.32
2003 Boeglin D, Cantel S, Heitz A, Martinez J, Fehrentz JA. Solution and solid-supported synthesis of 3,4,5-trisubstituted 1,2,4-triazole-based peptidomimetics. Organic Letters. 5: 4465-8. PMID 14602026 DOI: 10.1021/Ol035778E  0.647
2003 Petit A, Pasini A, Alves Da Costa C, Ayral E, Hernandez JF, Dumanchin-Njock C, Phiel CJ, Marambaud P, Wilk S, Farzan M, Fulcrand P, Martinez J, Andrau D, Checler F. JLK isocoumarin inhibitors: selective gamma-secretase inhibitors that do not interfere with notch pathway in vitro or in vivo. Journal of Neuroscience Research. 74: 370-7. PMID 14598313 DOI: 10.1002/Jnr.10747  0.773
2003 Hamzé A, Hernandez JF, Fulcrand P, Martinez J. Synthesis of various 3-substituted 1,2,4-oxadiazole-containing chiral beta 3- and alpha-amino acids from Fmoc-protected aspartic acid. The Journal of Organic Chemistry. 68: 7316-21. PMID 12968881 DOI: 10.1021/Jo0345953  0.772
2003 Wehbe J, Kassem T, Rolland V, Rolland M, Tabcheh M, Roumestant M, Martinez J. Optically pure β-substituted β-hydroxy aspartates as glutamate transporter blockers Organic and Biomolecular Chemistry. 1: 1938-1942. PMID 12945776 DOI: 10.1039/B212538B  0.292
2003 Claramunt RM, Sanz D, Torralba MP, Elguero J, Sanchez P, Enjalbal C, Martinez J, Aubagnac J. Electrospray mass spectrometry of 2-aminotroponimines and 2-aminotropones European Journal of Mass Spectrometry. 9: 403-407. PMID 12939491 DOI: 10.1255/Ejms.560  0.234
2003 Zajdel P, Bojarski AJ, Byrtus H, Chłoń-Rzepa G, Obniska J, Chevallet P, Martinez J, Pawłowski M. Preliminary study on application of impregnated synthetic peptide TLC stationary phases for the pre-screening of 5-HT1A ligands Biomedical Chromatography. 17: 312-317. PMID 12884396 DOI: 10.1002/Bmc.224  0.379
2003 Feliu L, Subra G, Martinez J, Amblard M. Spiroimidazolidinone library derivatives on SynPhase lanterns. Acs Combinatorial Science. 5: 356-361. PMID 12857102 DOI: 10.1021/Cc020111P  0.357
2003 Andrau D, Dumanchin-Njock C, Ayral E, Vizzavona J, Farzan M, Boisbrun M, Fulcrand P, Hernandez JF, Martinez J, Lefranc-Jullien S, Checler F. BACE1- and BACE2-expressing human cells: characterization of beta-amyloid precursor protein-derived catabolites, design of a novel fluorimetric assay, and identification of new in vitro inhibitors. The Journal of Biological Chemistry. 278: 25859-66. PMID 12736275 DOI: 10.1074/Jbc.M302622200  0.744
2003 Galés C, Poirot M, Taillefer J, Maigret B, Martinez J, Moroder L, Escrieut C, Pradayrol L, Fourmy D, Silvente-Poirot S. Identification of tyrosine 189 and asparagine 358 of the cholecystokinin 2 receptor in direct interaction with the crucial C-terminal amide of cholecystokinin by molecular modeling, site-directed mutagenesis, and structure/affinity studies Molecular Pharmacology. 63: 973-982. PMID 12695525 DOI: 10.1124/Mol.63.5.973  0.627
2003 Guerlavais V, Boeglin D, Mousseaux D, Oiry C, Heitz A, Deghenghi R, Locatelli V, Torsello A, Ghé C, Catapano F, Muccioli G, Galleyrand JC, Fehrentz JA, Martinez J. New active series of growth hormone secretagogues. Journal of Medicinal Chemistry. 46: 1191-203. PMID 12646029 DOI: 10.1021/Jm020985Q  0.612
2003 Enjalbal C, Maux D, Combarieu R, Martinez J, Aubagnac J. Imaging combinatorial libraries by mass spectrometry: from peptide to organic-supported syntheses. Acs Combinatorial Science. 5: 102-109. PMID 12625699 DOI: 10.1021/Cc0200484  0.3
2003 Enjalbal C, Lamaty F, Ribière P, Varray S, Suberchicot E, Yadav-Bhatnagar N, Martinez J, Aubagnac J. Characterization of Soluble Polymer Supported Organic Molecules by Mass Spectrometry Mrs Proceedings. 804. DOI: 10.1557/Proc-804-Jj5.2  0.557
2003 Enjalbal C, Maux D, Combarieu R, Martinez J, Aubagnac J. Imaging polymer supported organic molecules by mass spectrometry Application in combinatorial chemistry Mrs Proceedings. 804. DOI: 10.1557/Proc-804-Jj10.2  0.295
2003 Raynal N, Amblard M, Martinez J, Rolland M. [2‐(tert­‐Butyl­carbonyl­methylamino)phenyl]­acetic acid Acta Crystallographica Section E: Crystallographic Communications. 59. DOI: 10.1107/S1600536802021074  0.245
2003 Wehbe J, Rolland V, Martinez J, Rolland M. An intermediate in a new synthesis approach to β-substituted β-hydroxyaspartame Acta Crystallographica Section C: Crystal Structure Communications. 59. DOI: 10.1107/S0108270103014057  0.524
2003 Huck J, Duru C, Roumestant ML, Martinez J. Parallel Synthesis of New β-Amino Esters via Conjugate Nucleophilic Additions­ Synthesis. 2003: 2165-2168. DOI: 10.1055/S-2003-42084  0.32
2003 Varray S, Lazaro R, Martinez J, Lamaty F. New Soluble-Polymer Bound Ruthenium Carbene Catalysts: Synthesis, Characterization, and Application to Ring-Closing Metathesis Organometallics. 22: 2426-2435. DOI: 10.1021/Om021007N  0.555
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