Alex Martin Szpilman - Publications

Affiliations: 
Ariel University, Ariel, Israel 
Area:
Organic Chemistry

48 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Verdhi LK, Fridman N, Szpilman AM. Copper- and Chiral Nitroxide-Catalyzed Oxidative Kinetic Resolution of Axially Chiral -Arylpyrroles. Organic Letters. 24: 5078-5083. PMID 35798692 DOI: 10.1021/acs.orglett.2c01860  0.304
2021 Mishra AK, Parvari G, Santra SK, Bazylevich A, Dorfman O, Rahamim J, Eichen Y, Szpilman AM. Solar and Visible Light Assisted Peptide Coupling. Angewandte Chemie (International Ed. in English). PMID 33621382 DOI: 10.1002/anie.202011510  0.768
2020 Santra SK, Szpilman AM. Visible-Spectrum Solar-Light-Mediated Benzylic C-H Oxygenation Using 9,10-Dibromoanthracene As an Initiator. The Journal of Organic Chemistry. PMID 33236899 DOI: 10.1021/acs.joc.0c01720  0.677
2020 Arava S, Santra SK, Pathe GK, Kapanaiah R, Szpilman AM. Direct Umpolung Morita-Baylis-Hillman like α-Functionalization of Enones via Enolonium Species. Angewandte Chemie (International Ed. in English). PMID 32394609 DOI: 10.1002/Anie.202005286  0.838
2020 More AA, Szpilman AM. Indium(III) Catalyzed Reactions of Vinyl Azides and Indoles. Organic Letters. PMID 32330058 DOI: 10.1021/Acs.Orglett.0C00919  0.82
2020 More AA, Santra SK, Szpilman AM. Azido-Enolonium Species in C-C and C-N Bond-Forming Coupling Reactions. Organic Letters. PMID 31916772 DOI: 10.1021/Acs.Orglett.9B03824  0.801
2019 Toledo H, Tumanskii B, Sabirov DS, Kaushansky A, Fridman N, Szpilman AM. First α-deuterium nitroxides; synthesis and EPR study. Organic & Biomolecular Chemistry. PMID 31410426 DOI: 10.1039/C9Ob01127G  0.722
2018 Arava S, Maksymenko S, Parida KN, Pathe GK, More AM, Lipisa YB, Szpilman AM. A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species. Journal of Visualized Experiments : Jove. PMID 30175996 DOI: 10.3791/57916  0.806
2018 Parida KN, Pathe GK, Maksymenko S, Szpilman AM. Cross-coupling of dissimilar ketone enolates via enolonium species to afford non-symmetrical 1,4-diketones. Beilstein Journal of Organic Chemistry. 14: 992-997. PMID 29977370 DOI: 10.3762/Bjoc.14.84  0.782
2018 More AA, Pathe GK, Parida KN, Maksymenko S, Lipisa YB, Szpilman AM. α-N-Heteroarylation and α-Azidation of Ketones via Enolonium Species. The Journal of Organic Chemistry. 83: 2442-2447. PMID 29334466 DOI: 10.1021/Acs.Joc.7B03058  0.79
2018 Mishra AK, Parvari G, Cohen I, Fridman N, Eichen Y, Szpilman AM. Amine-tetrachloromethane charge transfer complexes: a structural and computational study Journal of Coordination Chemistry. 71: 2082-2089. DOI: 10.1080/00958972.2018.1498085  0.757
2017 Maksymenko S, Parida KN, Pathe GK, More AA, Lipisa YB, Szpilman AM. Transition-Metal-Free Intermolecular α-Arylation of Ketones via Enolonium Species. Organic Letters. 19: 6312-6315. PMID 29140710 DOI: 10.1021/Acs.Orglett.7B03064  0.789
2017 Cohen I, Mishra AK, Parvari G, Edrei R, Dantus M, Eichen Y, Szpilman AM. Sunlight assisted direct amide formation via a charge-transfer complex. Chemical Communications (Cambridge, England). PMID 28841217 DOI: 10.1039/C7Cc05300B  0.775
2017 Arava S, Kumar JN, Maksymenko S, Iron MA, Parida KN, Fristrup P, Szpilman AM. Enolonium Species-Umpoled Enolates. Angewandte Chemie (International Ed. in English). PMID 28128488 DOI: 10.1002/Anie.201610274  0.785
2016 Iron MA, Szpilman AM. Mechanism of the Copper/TEMPO Catalyzed Aerobic Oxidation of Alcohols. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27862437 DOI: 10.1002/Chem.201604402  0.377
2016 Halperin A, Shadkchan Y, Pisarevsky E, Szpilman AM, Sandovsky H, Osherov N, Benhar I. Novel Water-Soluble Amphotericin B-PEG Conjugates with Low Toxicity and Potent in Vivo Efficacy. Journal of Medicinal Chemistry. 59: 1197-206. PMID 26816333 DOI: 10.1021/Acs.Jmedchem.5B01862  0.752
2015 Toledo H, Amar M, Bar S, Iron MA, Fridman N, Tumanskii B, Shimon LJ, Botoshansky M, Szpilman AM. Synthesis and stability of cyclic α-hydrogen nitroxides. Organic & Biomolecular Chemistry. 13: 10726-33. PMID 26356203 DOI: 10.1039/C5Ob01443C  0.821
2015 Amar M, Bar S, Iron MA, Toledo H, Tumanskii B, Shimon LJ, Botoshansky M, Fridman N, Szpilman AM. Design concept for α-hydrogen-substituted nitroxides. Nature Communications. 6: 6070. PMID 25655711 DOI: 10.1038/Ncomms7070  0.814
2015 Targel TA, Kumar JN, Shneider OS, Bar S, Fridman N, Maximenko S, Szpilman AM. Oxidative asymmetric umpolung alkylation of Evans' β-ketoimides using dialkylzinc nucleophiles. Organic & Biomolecular Chemistry. 13: 2546-9. PMID 25600653 DOI: 10.1039/C4Ob02601B  0.771
2015 Shneider OS, Pisarevsky E, Fristrup P, Szpilman AM. Oxidative umpolung α-alkylation of ketones. Organic Letters. 17: 282-5. PMID 25562460 DOI: 10.1021/Ol503384C  0.818
2015 Shneider OS, Pisarevsky E, Fristrup P, Szpilman AM. Oxidative umpolung α-alkylation of ketones Organic Letters. 17: 282-285. DOI: 10.1021/ol503384c  0.796
2015 Avidan-Shlomovich S, Ghosh H, Szpilman AM. Synthetic and Mechanistic Study of the Catalytic Enantioselective Preparation of Primary β-Amino Ketones from Enones and a Fluorinated Gabriel Reagent Acs Catalysis. 5: 336-342. DOI: 10.1021/Cs501744E  0.795
2015 Bar S, Kumar JN, Amar M, Toledo H, Batrice RJ, Szpilman AM. ChemInform Abstract: Catalytic Aerobic Oxidation of Alcohols Using Recoverable IAPNO α-Hydrogen Nitroxyl Radicals. Cheminform. 46: no-no. DOI: 10.1002/CHIN.201531050  0.806
2015 Bar S, Kumar JN, Amar M, Toledo H, Batrice RJ, Szpilman AM. Catalytic Aerobic Oxidation of Alcohols using Recoverable IAPNO α-Hydrogen Nitroxyl Radicals Chemcatchem. 7: 1129-1134. DOI: 10.1002/Cctc.201402985  0.797
2014 Ghosh H, Vavilala R, Szpilman AM. Synthesis of axially chiral 1,8-diarylnaphthalene ligands and application in asymmetric catalysis: An intriguing fluorine effect Tetrahedron Asymmetry. DOI: 10.1016/J.Tetasy.2014.12.008  0.76
2013 Toledo H, Pisarevsky E, Abramovich A, Szpilman AM. Organocatalytic oxidation of aldehydes to mixed anhydrides. Chemical Communications (Cambridge, England). 49: 4367-9. PMID 22968566 DOI: 10.1039/C2Cc35220F  0.803
2013 Abramovich A, Toledo H, Pisarevsky E, Szpilman AM. ChemInform Abstract: Organocatalytic Oxidative Dimerization of Alcohols to Esters. Cheminform. 44: no-no. DOI: 10.1002/CHIN.201301051  0.779
2012 Szpilman A, Abramovich A, Toledo H, Pisarevsky E. Organocatalytic Oxidative Dimerization of Alcohols to Esters Synlett. 23: 2261-2265. DOI: 10.1055/S-0032-1317018  0.798
2011 Szpilman AM, Carreira EM. ChemInform Abstract: Probing the Biology of Natural Products: Molecular Editing by Diverted Total Synthesis. Cheminform. 42: no-no. DOI: 10.1002/chin.201114256  0.354
2010 Szpilman AM, Carreira EM. Probing the biology of natural products: molecular editing by diverted total synthesis. Angewandte Chemie (International Ed. in English). 49: 9592-628. PMID 21077064 DOI: 10.1002/Anie.200904761  0.445
2010 Volmer AA, Szpilman AM, Carreira EM. Synthesis and biological evaluation of amphotericin B derivatives. Natural Product Reports. 27: 1329-49. PMID 20556271 DOI: 10.1039/B820743G  0.438
2010 Volmer AA, Szpilman AM, Carreira EM. ChemInform Abstract: Synthesis and Biological Evaluation of Amphotericin B Derivatives Cheminform. 41: no-no. DOI: 10.1002/chin.201052259  0.361
2010 Korshin EE, Hoos R, Szpilman AM, Konstantinovski L, Posner GH, Bachi MD. ChemInform Abstract: An Efficient Synthesis of Bridged-Bicyclic Peroxides Structurally Related to Antimalarial Yingzhaosu A Based on Radical Co-Oxygenation of Thiols and Monoterpenes. Cheminform. 33: no-no. DOI: 10.1002/CHIN.200231177  0.619
2010 Szpilman AM, Korshin EE, Hoos R, Posner GH, Bachi MD. ChemInform Abstract: Iron(II)-Induced Degradation of Antimalarial β-Sulfonyl Endoperoxides. Evidence for the Generation of Potentially Cytotoxic Carbocations. Cheminform. 33: no-no. DOI: 10.1002/CHIN.200211144  0.599
2010 Szpilman AM, Carreira EM. Untersuchung der Biologie von Naturstoffen: systematische Strukturvariation durch umgelenkte Totalsynthese Angewandte Chemie. 122: 9786-9823. DOI: 10.1002/Ange.200904761  0.352
2009 Szpilman AM, Cereghetti DM, Manthorpe JM, Wurtz NR, Carreira EM. Synthesis and biophysical studies on 35-deoxy amphotericin B methyl ester. Chemistry (Weinheim An Der Bergstrasse, Germany). 15: 7117-28. PMID 19544513 DOI: 10.1002/Chem.200900231  0.742
2009 Szpilman AM, Carreira EM. Beta-glycosidation of sterically hindered alcohols. Organic Letters. 11: 1305-7. PMID 19281135 DOI: 10.1021/Ol9000735  0.481
2009 Szpilman AM, Carreira EM. ChemInform Abstract: β-Glycosidation of Sterically Hindered Alcohols. Cheminform. 40. DOI: 10.1002/chin.200930200  0.379
2008 Szpilman AM, Cereghetti DM, Wurtz NR, Manthorpe JM, Carreira EM. Synthesis of 35-deoxy amphotericin B methyl ester: a strategy for molecular editing. Angewandte Chemie (International Ed. in English). 47: 4335-8. PMID 18454441 DOI: 10.1002/Anie.200800589  0.74
2008 Szpilman AM, Manthorpe JM, Carreira EM. Synthesis and biological studies of 35-deoxy amphotericin B methyl ester. Angewandte Chemie (International Ed. in English). 47: 4339-42. PMID 18442156 DOI: 10.1002/Anie.200800590  0.742
2008 Szpilman AM, Manthorpe JM, Carreira EM. Synthesis of 35-Deoxy Amphotericin B Methyl Ester Synfacts. 2008: 1245-1245. DOI: 10.1055/S-0028-1087282  0.738
2005 Szpilman AM, Korshin EE, Rozenberg H, Bachi MD. Total syntheses of Yingzhaosu A and of its C(14)-epimer including the first evaluation of their antimalarial and cytotoxic activities. The Journal of Organic Chemistry. 70: 3618-32. PMID 15844999 DOI: 10.1021/Jo050074Z  0.705
2005 Manthorpe JM, Szpilman AM, Carreira EM. Scalable synthesis of a mycosamine donor. Overcoming difficult reactivity in allose systems Synthesis. 3380-3388. DOI: 10.1055/S-2005-918474  0.749
2003 Bachi MD, Korshin EE, Hoos R, Szpilman AM, Ploypradith P, Xie S, Shapiro TA, Posner GH. A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic beta-sulfonyl-endoperoxides. Journal of Medicinal Chemistry. 46: 2516-33. PMID 12773055 DOI: 10.1021/Jm020584A  0.627
2002 Korshin EE, Hoos R, Szpilman AM, Konstantinovski L, Posner GH, Bachi MD. An efficient synthesis of bridged-bicyclic peroxides structurally related to antimalarial yingzhaosu A based on radical co-oxygenation of thiols and monoterpenes Tetrahedron. 58: 2449-2469. DOI: 10.1016/S0040-4020(02)00126-6  0.714
2001 Szpilman AM, Korshin EE, Hoos R, Posner GH, Bachi MD. Iron(II)-induced degradation of antimalarial beta-sulfonyl endoperoxides: evidence for the generation of potentially cytotoxic carbocations. The Journal of Organic Chemistry. 66: 6531-40. PMID 11578201 DOI: 10.1021/Jo001265Z  0.623
2000 Bachi MD, Korshin EE, Hoos R, Szpilman AM. Synthesis and reactions of antimalarial bicyclic peroxides Journal of Heterocyclic Chemistry. 37: 639-646. DOI: 10.1002/Jhet.5570370321  0.706
2000 Bachi MD, Korshin EE, Hoos R, Szpilman AM. ChemInform Abstract: Synthesis and Reactions of Antimalarial Bicyclic Peroxides Cheminform. 31: no-no. DOI: 10.1002/CHIN.200039264  0.687
Show low-probability matches.