Alex Martin Szpilman - Publications

Ariel University, Ariel, Israel 
Organic Chemistry

33 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Santra SK, Szpilman AM. Visible-Spectrum Solar-Light-Mediated Benzylic C-H Oxygenation Using 9,10-Dibromoanthracene As an Initiator. The Journal of Organic Chemistry. PMID 33236899 DOI: 10.1021/acs.joc.0c01720  1
2020 Arava S, Santra SK, Pathe GK, Kapanaiah R, Szpilman AM. Direct Umpolung Morita-Baylis-Hillman like α-Functionalization of Enones via Enolonium Species. Angewandte Chemie (International Ed. in English). PMID 32394609 DOI: 10.1002/anie.202005286  1
2020 More AA, Szpilman AM. Indium(III) Catalyzed Reactions of Vinyl Azides and Indoles. Organic Letters. PMID 32330058 DOI: 10.1021/acs.orglett.0c00919  1
2020 More AA, Santra SK, Szpilman AM. Azido-Enolonium Species in C-C and C-N Bond-Forming Coupling Reactions. Organic Letters. PMID 31916772 DOI: 10.1021/acs.orglett.9b03824  1
2019 Toledo H, Tumanskii B, Sabirov DS, Kaushansky A, Fridman N, Szpilman AM. First α-deuterium nitroxides; synthesis and EPR study. Organic & Biomolecular Chemistry. PMID 31410426 DOI: 10.1039/c9ob01127g  1
2018 Arava S, Maksymenko S, Parida KN, Pathe GK, More AM, Lipisa YB, Szpilman AM. A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species. Journal of Visualized Experiments : Jove. PMID 30175996 DOI: 10.3791/57916  1
2018 Parida KN, Pathe GK, Maksymenko S, Szpilman AM. Cross-coupling of dissimilar ketone enolates via enolonium species to afford non-symmetrical 1,4-diketones. Beilstein Journal of Organic Chemistry. 14: 992-997. PMID 29977370 DOI: 10.3762/bjoc.14.84  1
2018 More AA, Pathe GK, Parida KN, Maksymenko S, Lipisa YB, Szpilman AM. α-N-Heteroarylation and α-Azidation of Ketones via Enolonium Species. The Journal of Organic Chemistry. 83: 2442-2447. PMID 29334466 DOI: 10.1021/acs.joc.7b03058  1
2017 Maksymenko S, Parida KN, Pathe GK, More AA, Lipisa YB, Szpilman AM. Transition-Metal-Free Intermolecular α-Arylation of Ketones via Enolonium Species. Organic Letters. 19: 6312-6315. PMID 29140710 DOI: 10.1021/acs.orglett.7b03064  1
2017 Cohen I, Mishra AK, Parvari G, Edrei R, Dantus M, Eichen Y, Szpilman AM. Sunlight assisted direct amide formation via a charge-transfer complex. Chemical Communications (Cambridge, England). PMID 28841217 DOI: 10.1039/c7cc05300b  0.4
2017 Arava S, Kumar JN, Maksymenko S, Iron MA, Parida KN, Fristrup P, Szpilman AM. Enolonium Species-Umpoled Enolates. Angewandte Chemie (International Ed. in English). PMID 28128488 DOI: 10.1002/anie.201610274  1
2016 Iron MA, Szpilman AM. Mechanism of the Copper/TEMPO Catalyzed Aerobic Oxidation of Alcohols. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27862437 DOI: 10.1002/chem.201604402  1
2016 Halperin A, Shadkchan Y, Pisarevsky E, Szpilman AM, Sandovsky H, Osherov N, Benhar I. Novel Water-Soluble Amphotericin B-PEG Conjugates with Low Toxicity and Potent in Vivo Efficacy. Journal of Medicinal Chemistry. 59: 1197-206. PMID 26816333 DOI: 10.1021/acs.jmedchem.5b01862  1
2015 Toledo H, Amar M, Bar S, Iron MA, Fridman N, Tumanskii B, Shimon LJ, Botoshansky M, Szpilman AM. Synthesis and stability of cyclic α-hydrogen nitroxides. Organic & Biomolecular Chemistry. 13: 10726-33. PMID 26356203 DOI: 10.1039/c5ob01443c  1
2015 Amar M, Bar S, Iron MA, Toledo H, Tumanskii B, Shimon LJ, Botoshansky M, Fridman N, Szpilman AM. Design concept for α-hydrogen-substituted nitroxides. Nature Communications. 6: 6070. PMID 25655711 DOI: 10.1038/ncomms7070  1
2015 Targel TA, Kumar JN, Shneider OS, Bar S, Fridman N, Maximenko S, Szpilman AM. Oxidative asymmetric umpolung alkylation of Evans' β-ketoimides using dialkylzinc nucleophiles. Organic & Biomolecular Chemistry. 13: 2546-9. PMID 25600653 DOI: 10.1039/c4ob02601b  1
2015 Shneider OS, Pisarevsky E, Fristrup P, Szpilman AM. Oxidative umpolung α-alkylation of ketones. Organic Letters. 17: 282-5. PMID 25562460 DOI: 10.1021/ol503384c  1
2015 Shneider OS, Pisarevsky E, Fristrup P, Szpilman AM. Oxidative umpolung α-alkylation of ketones Organic Letters. 17: 282-285. DOI: 10.1021/ol503384c  1
2015 Avidan-Shlomovich S, Ghosh H, Szpilman AM. Synthetic and Mechanistic Study of the Catalytic Enantioselective Preparation of Primary β-Amino Ketones from Enones and a Fluorinated Gabriel Reagent Acs Catalysis. 5: 336-342. DOI: 10.1021/cs501744e  1
2015 Bar S, Kumar JN, Amar M, Toledo H, Batrice RJ, Szpilman AM. Catalytic Aerobic Oxidation of Alcohols using Recoverable IAPNO α-Hydrogen Nitroxyl Radicals Chemcatchem. 7: 1129-1134. DOI: 10.1002/cctc.201402985  1
2014 Ghosh H, Vavilala R, Szpilman AM. Synthesis of axially chiral 1,8-diarylnaphthalene ligands and application in asymmetric catalysis: An intriguing fluorine effect Tetrahedron Asymmetry. DOI: 10.1016/j.tetasy.2014.12.008  1
2013 Toledo H, Pisarevsky E, Abramovich A, Szpilman AM. Organocatalytic oxidation of aldehydes to mixed anhydrides. Chemical Communications (Cambridge, England). 49: 4367-9. PMID 22968566 DOI: 10.1039/c2cc35220f  1
2010 Szpilman AM, Carreira EM. Probing the biology of natural products: molecular editing by diverted total synthesis. Angewandte Chemie (International Ed. in English). 49: 9592-628. PMID 21077064 DOI: 10.1002/anie.200904761  1
2010 Volmer AA, Szpilman AM, Carreira EM. Synthesis and biological evaluation of amphotericin B derivatives. Natural Product Reports. 27: 1329-49. PMID 20556271 DOI: 10.1039/b820743g  1
2009 Szpilman AM, Cereghetti DM, Manthorpe JM, Wurtz NR, Carreira EM. Synthesis and biophysical studies on 35-deoxy amphotericin B methyl ester. Chemistry (Weinheim An Der Bergstrasse, Germany). 15: 7117-28. PMID 19544513 DOI: 10.1002/chem.200900231  1
2009 Szpilman AM, Carreira EM. Beta-glycosidation of sterically hindered alcohols. Organic Letters. 11: 1305-7. PMID 19281135 DOI: 10.1021/ol9000735  1
2008 Szpilman AM, Cereghetti DM, Wurtz NR, Manthorpe JM, Carreira EM. Synthesis of 35-deoxy amphotericin B methyl ester: a strategy for molecular editing. Angewandte Chemie (International Ed. in English). 47: 4335-8. PMID 18454441 DOI: 10.1002/anie.200800589  1
2008 Szpilman AM, Manthorpe JM, Carreira EM. Synthesis and biological studies of 35-deoxy amphotericin B methyl ester. Angewandte Chemie (International Ed. in English). 47: 4339-42. PMID 18442156 DOI: 10.1002/anie.200800590  1
2005 Szpilman AM, Korshin EE, Rozenberg H, Bachi MD. Total syntheses of Yingzhaosu A and of its C(14)-epimer including the first evaluation of their antimalarial and cytotoxic activities. The Journal of Organic Chemistry. 70: 3618-32. PMID 15844999 DOI: 10.1021/jo050074z  1
2005 Manthorpe JM, Szpilman AM, Carreira EM. Scalable synthesis of a mycosamine donor. Overcoming difficult reactivity in allose systems Synthesis. 3380-3388. DOI: 10.1055/s-2005-918474  1
2003 Bachi MD, Korshin EE, Hoos R, Szpilman AM, Ploypradith P, Xie S, Shapiro TA, Posner GH. A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic beta-sulfonyl-endoperoxides. Journal of Medicinal Chemistry. 46: 2516-33. PMID 12773055 DOI: 10.1021/jm020584a  1
2002 Korshin EE, Hoos R, Szpilman AM, Konstantinovski L, Posner GH, Bachi MD. An efficient synthesis of bridged-bicyclic peroxides structurally related to antimalarial yingzhaosu A based on radical co-oxygenation of thiols and monoterpenes Tetrahedron. 58: 2449-2469. DOI: 10.1016/S0040-4020(02)00126-6  1
2001 Szpilman AM, Korshin EE, Hoos R, Posner GH, Bachi MD. Iron(II)-induced degradation of antimalarial beta-sulfonyl endoperoxides: evidence for the generation of potentially cytotoxic carbocations. The Journal of Organic Chemistry. 66: 6531-40. PMID 11578201 DOI: 10.1021/jo001265z  1
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