Year |
Citation |
Score |
2020 |
Santra SK, Szpilman AM. Visible-Spectrum Solar-Light-Mediated Benzylic C-H Oxygenation Using 9,10-Dibromoanthracene As an Initiator. The Journal of Organic Chemistry. PMID 33236899 DOI: 10.1021/acs.joc.0c01720 |
1 |
|
2020 |
Arava S, Santra SK, Pathe GK, Kapanaiah R, Szpilman AM. Direct Umpolung Morita-Baylis-Hillman like α-Functionalization of Enones via Enolonium Species. Angewandte Chemie (International Ed. in English). PMID 32394609 DOI: 10.1002/anie.202005286 |
1 |
|
2020 |
More AA, Szpilman AM. Indium(III) Catalyzed Reactions of Vinyl Azides and Indoles. Organic Letters. PMID 32330058 DOI: 10.1021/acs.orglett.0c00919 |
1 |
|
2020 |
More AA, Santra SK, Szpilman AM. Azido-Enolonium Species in C-C and C-N Bond-Forming Coupling Reactions. Organic Letters. PMID 31916772 DOI: 10.1021/acs.orglett.9b03824 |
1 |
|
2019 |
Toledo H, Tumanskii B, Sabirov DS, Kaushansky A, Fridman N, Szpilman AM. First α-deuterium nitroxides; synthesis and EPR study. Organic & Biomolecular Chemistry. PMID 31410426 DOI: 10.1039/c9ob01127g |
1 |
|
2018 |
Arava S, Maksymenko S, Parida KN, Pathe GK, More AM, Lipisa YB, Szpilman AM. A Two-Step Protocol for Umpolung Functionalization of Ketones Via Enolonium Species. Journal of Visualized Experiments : Jove. PMID 30175996 DOI: 10.3791/57916 |
1 |
|
2018 |
Parida KN, Pathe GK, Maksymenko S, Szpilman AM. Cross-coupling of dissimilar ketone enolates via enolonium species to afford non-symmetrical 1,4-diketones. Beilstein Journal of Organic Chemistry. 14: 992-997. PMID 29977370 DOI: 10.3762/bjoc.14.84 |
1 |
|
2018 |
More AA, Pathe GK, Parida KN, Maksymenko S, Lipisa YB, Szpilman AM. α-N-Heteroarylation and α-Azidation of Ketones via Enolonium Species. The Journal of Organic Chemistry. 83: 2442-2447. PMID 29334466 DOI: 10.1021/acs.joc.7b03058 |
1 |
|
2017 |
Maksymenko S, Parida KN, Pathe GK, More AA, Lipisa YB, Szpilman AM. Transition-Metal-Free Intermolecular α-Arylation of Ketones via Enolonium Species. Organic Letters. 19: 6312-6315. PMID 29140710 DOI: 10.1021/acs.orglett.7b03064 |
1 |
|
2017 |
Cohen I, Mishra AK, Parvari G, Edrei R, Dantus M, Eichen Y, Szpilman AM. Sunlight assisted direct amide formation via a charge-transfer complex. Chemical Communications (Cambridge, England). PMID 28841217 DOI: 10.1039/c7cc05300b |
0.4 |
|
2017 |
Arava S, Kumar JN, Maksymenko S, Iron MA, Parida KN, Fristrup P, Szpilman AM. Enolonium Species-Umpoled Enolates. Angewandte Chemie (International Ed. in English). PMID 28128488 DOI: 10.1002/anie.201610274 |
1 |
|
2016 |
Iron MA, Szpilman AM. Mechanism of the Copper/TEMPO Catalyzed Aerobic Oxidation of Alcohols. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27862437 DOI: 10.1002/chem.201604402 |
1 |
|
2016 |
Halperin A, Shadkchan Y, Pisarevsky E, Szpilman AM, Sandovsky H, Osherov N, Benhar I. Novel Water-Soluble Amphotericin B-PEG Conjugates with Low Toxicity and Potent in Vivo Efficacy. Journal of Medicinal Chemistry. 59: 1197-206. PMID 26816333 DOI: 10.1021/acs.jmedchem.5b01862 |
1 |
|
2015 |
Toledo H, Amar M, Bar S, Iron MA, Fridman N, Tumanskii B, Shimon LJ, Botoshansky M, Szpilman AM. Synthesis and stability of cyclic α-hydrogen nitroxides. Organic & Biomolecular Chemistry. 13: 10726-33. PMID 26356203 DOI: 10.1039/c5ob01443c |
1 |
|
2015 |
Amar M, Bar S, Iron MA, Toledo H, Tumanskii B, Shimon LJ, Botoshansky M, Fridman N, Szpilman AM. Design concept for α-hydrogen-substituted nitroxides. Nature Communications. 6: 6070. PMID 25655711 DOI: 10.1038/ncomms7070 |
1 |
|
2015 |
Targel TA, Kumar JN, Shneider OS, Bar S, Fridman N, Maximenko S, Szpilman AM. Oxidative asymmetric umpolung alkylation of Evans' β-ketoimides using dialkylzinc nucleophiles. Organic & Biomolecular Chemistry. 13: 2546-9. PMID 25600653 DOI: 10.1039/c4ob02601b |
1 |
|
2015 |
Shneider OS, Pisarevsky E, Fristrup P, Szpilman AM. Oxidative umpolung α-alkylation of ketones. Organic Letters. 17: 282-5. PMID 25562460 DOI: 10.1021/ol503384c |
1 |
|
2015 |
Shneider OS, Pisarevsky E, Fristrup P, Szpilman AM. Oxidative umpolung α-alkylation of ketones Organic Letters. 17: 282-285. DOI: 10.1021/ol503384c |
1 |
|
2015 |
Avidan-Shlomovich S, Ghosh H, Szpilman AM. Synthetic and Mechanistic Study of the Catalytic Enantioselective Preparation of Primary β-Amino Ketones from Enones and a Fluorinated Gabriel Reagent Acs Catalysis. 5: 336-342. DOI: 10.1021/cs501744e |
1 |
|
2015 |
Bar S, Kumar JN, Amar M, Toledo H, Batrice RJ, Szpilman AM. Catalytic Aerobic Oxidation of Alcohols using Recoverable IAPNO α-Hydrogen Nitroxyl Radicals Chemcatchem. 7: 1129-1134. DOI: 10.1002/cctc.201402985 |
1 |
|
2014 |
Ghosh H, Vavilala R, Szpilman AM. Synthesis of axially chiral 1,8-diarylnaphthalene ligands and application in asymmetric catalysis: An intriguing fluorine effect Tetrahedron Asymmetry. DOI: 10.1016/j.tetasy.2014.12.008 |
1 |
|
2013 |
Toledo H, Pisarevsky E, Abramovich A, Szpilman AM. Organocatalytic oxidation of aldehydes to mixed anhydrides. Chemical Communications (Cambridge, England). 49: 4367-9. PMID 22968566 DOI: 10.1039/c2cc35220f |
1 |
|
2010 |
Szpilman AM, Carreira EM. Probing the biology of natural products: molecular editing by diverted total synthesis. Angewandte Chemie (International Ed. in English). 49: 9592-628. PMID 21077064 DOI: 10.1002/anie.200904761 |
1 |
|
2010 |
Volmer AA, Szpilman AM, Carreira EM. Synthesis and biological evaluation of amphotericin B derivatives. Natural Product Reports. 27: 1329-49. PMID 20556271 DOI: 10.1039/b820743g |
1 |
|
2009 |
Szpilman AM, Cereghetti DM, Manthorpe JM, Wurtz NR, Carreira EM. Synthesis and biophysical studies on 35-deoxy amphotericin B methyl ester. Chemistry (Weinheim An Der Bergstrasse, Germany). 15: 7117-28. PMID 19544513 DOI: 10.1002/chem.200900231 |
1 |
|
2009 |
Szpilman AM, Carreira EM. Beta-glycosidation of sterically hindered alcohols. Organic Letters. 11: 1305-7. PMID 19281135 DOI: 10.1021/ol9000735 |
1 |
|
2008 |
Szpilman AM, Cereghetti DM, Wurtz NR, Manthorpe JM, Carreira EM. Synthesis of 35-deoxy amphotericin B methyl ester: a strategy for molecular editing. Angewandte Chemie (International Ed. in English). 47: 4335-8. PMID 18454441 DOI: 10.1002/anie.200800589 |
1 |
|
2008 |
Szpilman AM, Manthorpe JM, Carreira EM. Synthesis and biological studies of 35-deoxy amphotericin B methyl ester. Angewandte Chemie (International Ed. in English). 47: 4339-42. PMID 18442156 DOI: 10.1002/anie.200800590 |
1 |
|
2005 |
Szpilman AM, Korshin EE, Rozenberg H, Bachi MD. Total syntheses of Yingzhaosu A and of its C(14)-epimer including the first evaluation of their antimalarial and cytotoxic activities. The Journal of Organic Chemistry. 70: 3618-32. PMID 15844999 DOI: 10.1021/jo050074z |
1 |
|
2005 |
Manthorpe JM, Szpilman AM, Carreira EM. Scalable synthesis of a mycosamine donor. Overcoming difficult reactivity in allose systems Synthesis. 3380-3388. DOI: 10.1055/s-2005-918474 |
1 |
|
2003 |
Bachi MD, Korshin EE, Hoos R, Szpilman AM, Ploypradith P, Xie S, Shapiro TA, Posner GH. A short synthesis and biological evaluation of potent and nontoxic antimalarial bridged bicyclic beta-sulfonyl-endoperoxides. Journal of Medicinal Chemistry. 46: 2516-33. PMID 12773055 DOI: 10.1021/jm020584a |
1 |
|
2002 |
Korshin EE, Hoos R, Szpilman AM, Konstantinovski L, Posner GH, Bachi MD. An efficient synthesis of bridged-bicyclic peroxides structurally related to antimalarial yingzhaosu A based on radical co-oxygenation of thiols and monoterpenes Tetrahedron. 58: 2449-2469. DOI: 10.1016/S0040-4020(02)00126-6 |
1 |
|
2001 |
Szpilman AM, Korshin EE, Hoos R, Posner GH, Bachi MD. Iron(II)-induced degradation of antimalarial beta-sulfonyl endoperoxides: evidence for the generation of potentially cytotoxic carbocations. The Journal of Organic Chemistry. 66: 6531-40. PMID 11578201 DOI: 10.1021/jo001265z |
1 |
|
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