Nicolò Scalacci - Publications

Affiliations: 
2013-2017 Institute of Pharmaceutical Science King's College London, London, UK 

10 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Touitou M, Manetti F, Ribeiro CM, Pavan FR, Scalacci N, Zrebna K, Begum N, Semenya D, Gupta A, Bhakta S, McHugh TD, Senderowitz H, Kyriazi M, Castagnolo D. Improving the Potency of -Aryl-2,5-dimethylpyrroles against Multidrug-Resistant and Intracellular Mycobacteria. Acs Medicinal Chemistry Letters. 11: 638-644. PMID 32435364 DOI: 10.1021/Acsmedchemlett.9B00515  0.622
2017 Lauder K, Toscani A, Scalacci N, Castagnolo D. Synthesis and Reactivity of Propargylamines in Organic Chemistry. Chemical Reviews. 117: 14091-14200. PMID 29166000 DOI: 10.1021/Acs.Chemrev.7B00343  0.577
2017 Scalacci N, Black GW, Mattedi G, Brown NL, Turner NJ, Castagnolo D. Unveiling the Biocatalytic Aromatizing Activity of Monoamine Oxidases MAO-N and 6-HDNO: Development of Chemoenzymatic Cascades for the Synthesis of Pyrroles Acs Catalysis. 7: 1295-1300. DOI: 10.1021/Acscatal.6B03081  0.632
2016 Scalacci N, Brown AK, Pavan FR, Ribeiro CM, Manetti F, Bhakta S, Maitra A, Smith DL, Petricci E, Castagnolo D. Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis. European Journal of Medicinal Chemistry. 127: 147-158. PMID 28039773 DOI: 10.1016/J.Ejmech.2016.12.042  0.691
2016 Bhakta S, Scalacci N, Maitra A, Brown AK, Dasugari S, Evangelopoulos D, McHugh TD, Mortazavi PN, Twist A, Petricci E, Manetti F, Castagnolo D. Design and synthesis of 1-((1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethyl-octa-2,6-dienyl)-ethane-1,2-diamine (SQ109) pyrrole hybrid derivatives: discovery of potent anti-tubercular agents effective against multi-drug resistant mycobacteria. Journal of Medicinal Chemistry. PMID 26907951 DOI: 10.1021/Acs.Jmedchem.6B00031  0.725
2016 Castagnolo D, Scalacci N, Pelloja C, Radi M. Microwave-Assisted Domino Reactions of Propargylamines with Isothiocyanates: Selective Synthesis of 2-Aminothiazoles and 2-Amino-4-methylenethiazolines Synlett. 27: 1883-1887. DOI: 10.1055/S-0035-1561985  0.628
2016 Tassini S, Castagnolo D, Scalacci N, Kissova M, Armijos-Rivera JI, Giagnorio F, Maga G, Costantino G, Crespan E, Radi M. A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes Medchemcomm. 7: 484-494. DOI: 10.1039/C5Md00462D  0.608
2016 Vincetti P, Brianza A, Scalacci N, Costantino G, Castagnolo D, Radi M. A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides Tetrahedron Letters. 57: 1464-1467. DOI: 10.1016/J.Tetlet.2016.02.068  0.708
2015 Magri A, Reilly R, Scalacci N, Radi M, Hunter M, Ripoll M, Patel AH, Castagnolo D. Rethinking the old antiviral drug moroxydine: Discovery of novel analogues as anti-hepatitis C virus (HCV) agents. Bioorganic & Medicinal Chemistry Letters. 25: 5372-6. PMID 26428870 DOI: 10.1016/J.Bmcl.2015.09.029  0.651
2015 Chachignon H, Scalacci N, Petricci E, Castagnolo D. Synthesis of 1,2,3-Substituted Pyrroles from Propargylamines via a One-Pot Tandem Enyne Cross Metathesis-Cyclization Reaction. The Journal of Organic Chemistry. 80: 5287-95. PMID 25897951 DOI: 10.1021/Acs.Joc.5B00222  0.634
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