Year |
Citation |
Score |
2020 |
Touitou M, Manetti F, Ribeiro CM, Pavan FR, Scalacci N, Zrebna K, Begum N, Semenya D, Gupta A, Bhakta S, McHugh TD, Senderowitz H, Kyriazi M, Castagnolo D. Improving the Potency of -Aryl-2,5-dimethylpyrroles against Multidrug-Resistant and Intracellular Mycobacteria. Acs Medicinal Chemistry Letters. 11: 638-644. PMID 32435364 DOI: 10.1021/Acsmedchemlett.9B00515 |
0.622 |
|
2017 |
Lauder K, Toscani A, Scalacci N, Castagnolo D. Synthesis and Reactivity of Propargylamines in Organic Chemistry. Chemical Reviews. 117: 14091-14200. PMID 29166000 DOI: 10.1021/Acs.Chemrev.7B00343 |
0.577 |
|
2017 |
Scalacci N, Black GW, Mattedi G, Brown NL, Turner NJ, Castagnolo D. Unveiling the Biocatalytic Aromatizing Activity of Monoamine Oxidases MAO-N and 6-HDNO: Development of Chemoenzymatic Cascades for the Synthesis of Pyrroles Acs Catalysis. 7: 1295-1300. DOI: 10.1021/Acscatal.6B03081 |
0.632 |
|
2016 |
Scalacci N, Brown AK, Pavan FR, Ribeiro CM, Manetti F, Bhakta S, Maitra A, Smith DL, Petricci E, Castagnolo D. Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis. European Journal of Medicinal Chemistry. 127: 147-158. PMID 28039773 DOI: 10.1016/J.Ejmech.2016.12.042 |
0.691 |
|
2016 |
Bhakta S, Scalacci N, Maitra A, Brown AK, Dasugari S, Evangelopoulos D, McHugh TD, Mortazavi PN, Twist A, Petricci E, Manetti F, Castagnolo D. Design and synthesis of 1-((1,5-bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N'-((E)-3,7-dimethyl-octa-2,6-dienyl)-ethane-1,2-diamine (SQ109) pyrrole hybrid derivatives: discovery of potent anti-tubercular agents effective against multi-drug resistant mycobacteria. Journal of Medicinal Chemistry. PMID 26907951 DOI: 10.1021/Acs.Jmedchem.6B00031 |
0.725 |
|
2016 |
Castagnolo D, Scalacci N, Pelloja C, Radi M. Microwave-Assisted Domino Reactions of Propargylamines with Isothiocyanates: Selective Synthesis of 2-Aminothiazoles and 2-Amino-4-methylenethiazolines Synlett. 27: 1883-1887. DOI: 10.1055/S-0035-1561985 |
0.628 |
|
2016 |
Tassini S, Castagnolo D, Scalacci N, Kissova M, Armijos-Rivera JI, Giagnorio F, Maga G, Costantino G, Crespan E, Radi M. A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes Medchemcomm. 7: 484-494. DOI: 10.1039/C5Md00462D |
0.608 |
|
2016 |
Vincetti P, Brianza A, Scalacci N, Costantino G, Castagnolo D, Radi M. A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides Tetrahedron Letters. 57: 1464-1467. DOI: 10.1016/J.Tetlet.2016.02.068 |
0.708 |
|
2015 |
Magri A, Reilly R, Scalacci N, Radi M, Hunter M, Ripoll M, Patel AH, Castagnolo D. Rethinking the old antiviral drug moroxydine: Discovery of novel analogues as anti-hepatitis C virus (HCV) agents. Bioorganic & Medicinal Chemistry Letters. 25: 5372-6. PMID 26428870 DOI: 10.1016/J.Bmcl.2015.09.029 |
0.651 |
|
2015 |
Chachignon H, Scalacci N, Petricci E, Castagnolo D. Synthesis of 1,2,3-Substituted Pyrroles from Propargylamines via a One-Pot Tandem Enyne Cross Metathesis-Cyclization Reaction. The Journal of Organic Chemistry. 80: 5287-95. PMID 25897951 DOI: 10.1021/Acs.Joc.5B00222 |
0.634 |
|
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