Year |
Citation |
Score |
2023 |
Moon P, Zammit C, Shao Q, Boike L, Dovala D, Henning NJ, Knapp M, Spradlin JN, Ward CC, Wolleb H, Fuller D, Blake G, Murphy JP, Wang F, Lu Y, et al. Discovery of Potent Pyrazoline-Based Covalent SARS-CoV-2 Main Protease Inhibitors. Chembiochem : a European Journal of Chemical Biology. e202300116. PMID 37069799 DOI: 10.1002/cbic.202300116 |
0.652 |
|
2023 |
Han H, Gracia AV, Røise JJ, Boike L, Leon K, Schulze-Gahmen U, Stentzel MR, Bajaj T, Chen D, Li IC, He M, Behrouzi K, Khodabakhshi Z, Nomura DK, Mofrad MRK, et al. A covalent inhibitor targeting the papain-like protease from SARS-CoV-2 inhibits viral replication. Rsc Advances. 13: 10636-10641. PMID 37025664 DOI: 10.1039/d3ra00426k |
0.613 |
|
2022 |
Boike L, Henning NJ, Nomura DK. Advances in covalent drug discovery. Nature Reviews. Drug Discovery. PMID 36008483 DOI: 10.1038/s41573-022-00542-z |
0.768 |
|
2022 |
Maza JC, García-Almedina DM, Boike LE, Hamlish NX, Nomura DK, Francis MB. Tyrosinase-Mediated Synthesis of Nanobody-Cell Conjugates. Acs Central Science. 8: 955-962. PMID 35912347 DOI: 10.1021/acscentsci.1c01265 |
0.61 |
|
2022 |
Henning NJ, Boike L, Spradlin JN, Ward CC, Liu G, Zhang E, Belcher BP, Brittain SM, Hesse MJ, Dovala D, McGregor LM, Valdez Misiolek R, Plasschaert LW, Rowlands DJ, Wang F, et al. Deubiquitinase-targeting chimeras for targeted protein stabilization. Nature Chemical Biology. PMID 35210618 DOI: 10.1038/s41589-022-00971-2 |
0.605 |
|
2021 |
Luo M, Spradlin JN, Boike L, Tong B, Brittain SM, McKenna JM, Tallarico JA, Schirle M, Maimone TJ, Nomura DK. Chemoproteomics-enabled discovery of covalent RNF114-based degraders that mimic natural product function. Cell Chemical Biology. PMID 33513350 DOI: 10.1016/j.chembiol.2021.01.005 |
0.733 |
|
2020 |
Boike L, Cioffi AG, Majewski FC, Co J, Henning NJ, Jones MD, Liu G, McKenna JM, Tallarico JA, Schirle M, Nomura DK. Discovery of a Functional Covalent Ligand Targeting an Intrinsically Disordered Cysteine within MYC. Cell Chemical Biology. PMID 32966806 DOI: 10.1016/j.chembiol.2020.09.001 |
0.673 |
|
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