Guillaume Bernadat - Publications

2009-2010 ICSN CNRS, Paris, Île-de-France, France 

42 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 N'Tamon AD, Okpekon AT, Bony NF, Bernadat G, Gallard JF, Kouamé T, Séon-Méniel B, Leblanc K, Rharrabti S, Mouray E, Grellier P, Ake M, Amin NC, Champy P, Beniddir MA, et al. Streamlined targeting of Amaryllidaceae alkaloids from the bulbs of Crinum scillifolium using spectrometric and taxonomically-informed scoring metabolite annotations. Phytochemistry. 179: 112485. PMID 32861139 DOI: 10.1016/J.Phytochem.2020.112485  0.335
2020 Cauchie G, N'Nang EO, van der Hooft JJJ, Le Pogam P, Bernadat G, Gallard JF, Kumulungui B, Champy P, Poupon E, Beniddir MA. Phenylpropane as an Alternative Dearomatizing Unit of Indoles: Discovery of Inaequalisines A and B Using Substructure-Informed Molecular Networking. Organic Letters. PMID 32686942 DOI: 10.1021/Acs.Orglett.0C02153  0.306
2020 Khelifi I, Pecnard S, Bernadat G, Bignon J, Levaique H, Dubois J, Provot O, Alami M. Synthesis and Anticancer Properties of Oxazepines Related to Azaisoerianin and IsoCoQuines. Chemmedchem. 15: 1571-1578. PMID 32485077 DOI: 10.1002/Cmdc.202000197  0.308
2020 Varlet T, Gelis C, Retailleau P, Bernadat G, Neuville L, Masson G. Redox-Divergent Chiral Phosphoric Acid-Catalyzed Enantioselective Formal Quinone Diels-Alder Reactions. Angewandte Chemie (International Ed. in English). PMID 32112662 DOI: 10.1002/Anie.202000838  0.412
2020 Alcover CF, Bernadat G, Kabran FA, Le Pogam P, Leblanc K, Fox Ramos AE, Gallard JF, Mouray E, Grellier P, Poupon E, Beniddir MA. Molecular Networking Reveals Serpentinine-Related Bisindole Alkaloids from , a Previously Well-Investigated Species. Journal of Natural Products. PMID 32091210 DOI: 10.1021/Acs.Jnatprod.9B01247  0.319
2020 Tonali N, Correia I, Lesma J, Bernadat G, Ongeri S, Lequin O. Introducing sequential aza-amino acids units induces repeated β-turns and helical conformations in peptides. Organic & Biomolecular Chemistry. PMID 32091060 DOI: 10.1039/C9Ob02654A  0.32
2020 Varlet T, Gelis C, Retailleau P, Bernadat G, Neuville L, Masson G. Redox‐Divergent Chiral Phosphoric Acid‐Catalyzed Enantioselective Formal Quinone Diels–Alder Reactions Angewandte Chemie. DOI: 10.1002/Ange.202000838  0.364
2019 Pinet A, Nguyen TL, Bernadat G, Figadère B, Ferrié L. Synthesis of 3,5-Disubstituted 1,2-Dioxolanes through the Use of Acetoxy Peroxyacetals. Organic Letters. PMID 31184910 DOI: 10.1021/Acs.Orglett.9B01616  0.391
2019 Jarrige L, Glavač D, Levitre G, Retailleau P, Bernadat G, Neuville L, Masson G. Chiral phosphoric acid-catalyzed enantioselective construction of structurally diverse benzothiazolopyrimidines. Chemical Science. 10: 3765-3769. PMID 31015920 DOI: 10.1039/C8Sc05581E  0.393
2019 Duong TH, Beniddir MA, Boustie J, Nguyen KP, Chavasiri W, Bernadat G, Le Pogam P. DP4-Assisted Structure Elucidation of Isodemethylchodatin, a New Norlichexanthone Derivative Meager in H-Atoms, from the Lichen . Molecules (Basel, Switzerland). 24. PMID 31003403 DOI: 10.3390/Molecules24081527  0.313
2018 Otogo N'Nang E, Bernadat G, Mouray E, Kumulungui B, Grellier P, Poupon E, Champy P, Beniddir MA. Theionbrunonines A and B: Dimeric Vobasine Alkaloids Tethered by a Thioether Bridge from Mostuea brunonis. Organic Letters. 20: 6596-6600. PMID 30303382 DOI: 10.1021/Acs.Orglett.8B02961  0.31
2018 Merad J, Lalli C, Bernadat G, Maury J, Masson G. Frontispiece: Enantioselective Brønsted Acid Catalysis as a Tool for the Synthesis of Natural Products and Pharmaceuticals Chemistry - a European Journal. 24. DOI: 10.1002/Chem.201881662  0.355
2017 Naret T, Bignon J, Bernadat G, Benchekroun M, Levaique H, Lenoir C, Dubois J, Pruvost A, Saller F, Borgel D, Manoury B, Leblais V, Darrigrand R, Apcher S, Brion JD, et al. A fluorine scan of a tubulin polymerization inhibitor isocombretastatin A-4: Design, synthesis, molecular modelling, and biological evaluation. European Journal of Medicinal Chemistry. 143: 473-490. PMID 29202409 DOI: 10.1016/J.Ejmech.2017.11.055  0.329
2017 Merad J, Lalli C, Bernadat G, Maury J, Masson G. Enantioselective Brønsted Acid Catalysis as a Tool for the Synthesis of Natural Products and Pharmaceuticals. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28981209 DOI: 10.1002/Chem.201703556  0.415
2017 Lachkar D, Denizot N, Bernadat G, Ahamada K, Beniddir MA, Dumontet V, Gallard JF, Guillot R, Leblanc K, N'nang EO, Turpin V, Kouklovsky C, Poupon E, Evanno L, Vincent G. Unified biomimetic assembly of voacalgine A and bipleiophylline via divergent oxidative couplings. Nature Chemistry. 9: 793-798. PMID 28754932 DOI: 10.1038/Nchem.2735  0.362
2017 Mamone M, Gonçalves RSB, Blanchard F, Bernadat G, Ongeri S, Milcent T, Crousse B. N-Difluoromethyl-triazole as a constrained scaffold in peptidomimetics Chemical Communications. 53: 5024-5027. PMID 28429026 DOI: 10.1039/C7Cc01298E  0.327
2017 Fox Ramos AE, Alcover C, Evanno L, Maciuk A, Litaudon M, Duplais C, Bernadat G, Gallard JF, Jullian JC, Mouray E, Grellier P, Loiseau PM, Pomel S, Poupon E, Champy P, et al. Revisiting Previously Investigated Plants: A Molecular Networking-Based Study of Geissospermum laeve. Journal of Natural Products. 80: 1007-1014. PMID 28282127 DOI: 10.1021/Acs.Jnatprod.6B01013  0.317
2017 Khelifi I, Naret T, Renko D, Hamze A, Bernadat G, Bignon J, Lenoir C, Dubois J, Brion JD, Provot O, Alami M. Design, synthesis and anticancer properties of IsoCombretaQuinolines as potent tubulin assembly inhibitors. European Journal of Medicinal Chemistry. 127: 1025-1034. PMID 28166995 DOI: 10.1016/J.Ejmech.2016.11.012  0.358
2017 Dumoulin A, Bernadat G, Masson G. Enantioselective three-component amination of enecarbamates enables the synthesis of structurally complex small molecules. The Journal of Organic Chemistry. PMID 28092703 DOI: 10.1021/Acs.Joc.6B03093  0.418
2016 Pautus S, Alami M, Adam F, Bernadat G, Lawrence DA, De Carvalho A, Ferry G, Rupin A, Hamze A, Champy P, Bonneau N, Gloanec P, Peglion JL, Brion JD, Bianchini EP, et al. Characterization of the Annonaceous acetogenin, annonacinone, a natural product inhibitor of plasminogen activator inhibitor-1. Scientific Reports. 6: 36462. PMID 27876785 DOI: 10.1038/Srep36462  0.301
2016 Vallerotto S, Douaron GL, Bernadat G, Ferrié L, Figadère B. 6-endo-dig Cycloisomerization of N-Propargyl Aminoquinoxalines: A New Route to 1,4,8-Triazaphenanthrenes Synthesis. 48: 3232-3240. DOI: 10.1055/S-0035-1562443  0.351
2015 AL-Shuaeeb RA, Galvani G, Bernadat G, Brion JD, Alami M, Messaoudi S. Diversity-oriented synthesis of fused thioglycosyl benzo[e][1,4]oxathiepin-5-ones and benzo[f][1,4]thiazepin-5(2H)-ones by a sequence of palladium-catalyzed glycosyl thiol arylation and deprotection-lactonization reactions. Organic & Biomolecular Chemistry. 13: 10904-16. PMID 26369372 DOI: 10.1039/C5Ob01603G  0.368
2015 Pous J, Courant T, Bernadat G, Iorga BI, Blanchard F, Masson G. Regio-, Diastereo-, and Enantioselective Nitroso-Diels-Alder Reaction of 1,3-Diene-1-carbamates Catalyzed by Chiral Phosphoric Acids. Journal of the American Chemical Society. 137: 11950-3. PMID 26355670 DOI: 10.1021/Jacs.5B08515  0.582
2015 Soussi MA, Provot O, Bernadat G, Bignon J, Desravines D, Dubois J, Brion JD, Messaoudi S, Alami M. IsoCombretaQuinazolines: Potent Cytotoxic Agents with Antitubulin Activity. Chemmedchem. 10: 1392-402. PMID 26076053 DOI: 10.1002/Cmdc.201500069  0.348
2015 List B, Höfler D, Pous J, Courant T, Bernadat G, Iorga BI, Blanchard F, Masson G. Phosphoric Acid-Catalyzed Asymmetric Nitroso-Diels–Alder Reaction Synfacts. 11: 1212-1212. DOI: 10.1055/S-0035-1560719  0.561
2015 Skiredj A, Beniddir MA, Joseph D, Bernadat G, Evanno L, Poupon E. Harnessing the Intrinsic Reactivity within the Aplysinopsin Series for the Synthesis of Intricate Dimers: Natural from Start to Finish Synthesis (Germany). 47: 2367-2376. DOI: 10.1055/S-0034-1381032  0.378
2015 Vahdati L, Fanelli R, Bernadat G, Correia I, Lequin O, Ongeri S, Piarulli U. Synthesis and conformational studies of a stable peptidomimetic β-hairpin based on a bifunctional diketopiperazine turn inducer New Journal of Chemistry. 39: 3250-3258. DOI: 10.1039/C4Nj01437E  0.312
2014 Amara Z, Bernadat G, Venot PE, Retailleau P, Troufflard C, Drège E, Le Bideau F, Joseph D. Thermodynamic epimeric equilibration and crystallisation-induced dynamic resolution of lobelanine, norlobelanine and related analogues. Organic & Biomolecular Chemistry. 12: 9797-810. PMID 25320963 DOI: 10.1039/C4Ob01787K  0.383
2014 Tréguier B, Lawson M, Bernadat G, Bignon J, Dubois J, Brion JD, Alami M, Hamze A. Synthesis of a 3-(α-styryl)benzo[b]-thiophene library via bromocyclization of alkynes and palladium-catalyzed to sylhydrazones cross-couplings: evaluation as antitubulin agents. Acs Combinatorial Science. 16: 702-10. PMID 25229390 DOI: 10.1021/Co500115B  0.4
2014 Skiredj A, Beniddir MA, Joseph D, Leblanc K, Bernadat G, Evanno L, Poupon E. A unified bioinspired "aplysinopsin cascade": total synthesis of (±)-tubastrindole B and related biosynthetic congeners. Organic Letters. 16: 4980-3. PMID 25222547 DOI: 10.1021/Ol502177M  0.306
2014 Skiredj A, Beniddir MA, Joseph D, Leblanc K, Bernadat G, Evanno L, Poupon E. Spontaneous biomimetic formation of (±)-dictazole B under irradiation with artificial sunlight. Angewandte Chemie (International Ed. in English). 53: 6419-24. PMID 24817607 DOI: 10.1002/Anie.201403454  0.318
2014 Soussi MA, Provot O, Bernadat G, Bignon J, Wdzieczak-Bakala J, Desravines D, Dubois J, Brion JD, Messaoudi S, Alami M. Discovery of azaisoerianin derivatives as potential antitumors agents. European Journal of Medicinal Chemistry. 78: 178-89. PMID 24681982 DOI: 10.1016/J.Ejmech.2014.03.032  0.323
2014 Bernadat G, Masson G. Enamide derivatives: Versatile building blocks for highly functionalized α,β-substituted amines Synlett. 25. DOI: 10.1055/S-0034-1379166  0.334
2014 Ferrié L, Ferhi S, Bernadat G, Figadère B. Toward the Total Synthesis of Klaivanolide: Complete Reinterpretation of Its Originally Assigned Structure European Journal of Organic Chemistry. 2014: 6183-6189. DOI: 10.1002/Ejoc.201402741  0.332
2013 Gonçalves RS, Dos Santos M, Bernadat G, Bonnet-Delpon D, Crousse B. A one-pot synthesis of 3-trifluoromethyl-2-isoxazolines from trifluoromethyl aldoxime. Beilstein Journal of Organic Chemistry. 9: 2387-94. PMID 24367404 DOI: 10.3762/Bjoc.9.275  0.33
2013 Bordessa A, Keita M, Maréchal X, Formicola L, Lagarde N, Rodrigo J, Bernadat G, Bauvais C, Soulier JL, Dufau L, Milcent T, Crousse B, Reboud-Ravaux M, Ongeri S. α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome. European Journal of Medicinal Chemistry. 70: 505-24. PMID 24185380 DOI: 10.1016/J.Ejmech.2013.09.059  0.338
2013 Bernadat G, Supuran CT, Iorga BI. Carbonic anhydrase binding site parameterization in OPLS-AA force field. Bioorganic & Medicinal Chemistry. 21: 1427-30. PMID 23182217 DOI: 10.1016/J.Bmc.2012.10.040  0.49
2013 Aziz J, Brachet E, Hamze A, Peyrat JF, Bernadat G, Morvan E, Bignon J, Wdzieczak-Bakala J, Desravines D, Dubois J, Tueni M, Yassine A, Brion JD, Alami M. Synthesis, biological evaluation, and structure-activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors. Organic & Biomolecular Chemistry. 11: 430-42. PMID 23047722 DOI: 10.1039/C2Ob26253C  0.384
2013 Lewin G, Bernadat G, Aubert G, Cresteil T. Semisynthesis of (+)- and (-)-goniomitine from (-)- and (+)-vincadifformine Tetrahedron. 69: 1622-1627. DOI: 10.1016/J.Tet.2012.11.084  0.315
2011 Lalli C, Brioche J, Bernadat G, Masson G. Catalytic enantioselective cycloaddition with chiral lewis bases Current Organic Chemistry. 15: 4108-4127. DOI: 10.2174/138527211798109178  0.345
2009 Wu YC, Bernadat G, Masson G, Couturier C, Schlama T, Zhu J. Synthetic studies on (-)-lemonomycin: an efficient asymmetric synthesis of lemonomycinone amide. The Journal of Organic Chemistry. 74: 2046-52. PMID 19196163 DOI: 10.1021/Jo8027449  0.422
2009 Wu Y-, Bernadat G, Masson G, Couturier C, Schlama T, Zhu J. Synthesis of Lemonomycinone Amide Synfacts. 2009: 1070-1070. DOI: 10.1055/S-0029-1217863  0.349
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