Year |
Citation |
Score |
2020 |
N'Tamon AD, Okpekon AT, Bony NF, Bernadat G, Gallard JF, Kouamé T, Séon-Méniel B, Leblanc K, Rharrabti S, Mouray E, Grellier P, Ake M, Amin NC, Champy P, Beniddir MA, et al. Streamlined targeting of Amaryllidaceae alkaloids from the bulbs of Crinum scillifolium using spectrometric and taxonomically-informed scoring metabolite annotations. Phytochemistry. 179: 112485. PMID 32861139 DOI: 10.1016/J.Phytochem.2020.112485 |
0.335 |
|
2020 |
Cauchie G, N'Nang EO, van der Hooft JJJ, Le Pogam P, Bernadat G, Gallard JF, Kumulungui B, Champy P, Poupon E, Beniddir MA. Phenylpropane as an Alternative Dearomatizing Unit of Indoles: Discovery of Inaequalisines A and B Using Substructure-Informed Molecular Networking. Organic Letters. PMID 32686942 DOI: 10.1021/Acs.Orglett.0C02153 |
0.306 |
|
2020 |
Khelifi I, Pecnard S, Bernadat G, Bignon J, Levaique H, Dubois J, Provot O, Alami M. Synthesis and Anticancer Properties of Oxazepines Related to Azaisoerianin and IsoCoQuines. Chemmedchem. 15: 1571-1578. PMID 32485077 DOI: 10.1002/Cmdc.202000197 |
0.308 |
|
2020 |
Varlet T, Gelis C, Retailleau P, Bernadat G, Neuville L, Masson G. Redox-Divergent Chiral Phosphoric Acid-Catalyzed Enantioselective Formal Quinone Diels-Alder Reactions. Angewandte Chemie (International Ed. in English). PMID 32112662 DOI: 10.1002/Anie.202000838 |
0.412 |
|
2020 |
Alcover CF, Bernadat G, Kabran FA, Le Pogam P, Leblanc K, Fox Ramos AE, Gallard JF, Mouray E, Grellier P, Poupon E, Beniddir MA. Molecular Networking Reveals Serpentinine-Related Bisindole Alkaloids from , a Previously Well-Investigated Species. Journal of Natural Products. PMID 32091210 DOI: 10.1021/Acs.Jnatprod.9B01247 |
0.319 |
|
2020 |
Tonali N, Correia I, Lesma J, Bernadat G, Ongeri S, Lequin O. Introducing sequential aza-amino acids units induces repeated β-turns and helical conformations in peptides. Organic & Biomolecular Chemistry. PMID 32091060 DOI: 10.1039/C9Ob02654A |
0.32 |
|
2020 |
Varlet T, Gelis C, Retailleau P, Bernadat G, Neuville L, Masson G. Redox‐Divergent Chiral Phosphoric Acid‐Catalyzed Enantioselective Formal Quinone Diels–Alder Reactions Angewandte Chemie. DOI: 10.1002/Ange.202000838 |
0.364 |
|
2019 |
Pinet A, Nguyen TL, Bernadat G, Figadère B, Ferrié L. Synthesis of 3,5-Disubstituted 1,2-Dioxolanes through the Use of Acetoxy Peroxyacetals. Organic Letters. PMID 31184910 DOI: 10.1021/Acs.Orglett.9B01616 |
0.391 |
|
2019 |
Jarrige L, Glavač D, Levitre G, Retailleau P, Bernadat G, Neuville L, Masson G. Chiral phosphoric acid-catalyzed enantioselective construction of structurally diverse benzothiazolopyrimidines. Chemical Science. 10: 3765-3769. PMID 31015920 DOI: 10.1039/C8Sc05581E |
0.393 |
|
2019 |
Duong TH, Beniddir MA, Boustie J, Nguyen KP, Chavasiri W, Bernadat G, Le Pogam P. DP4-Assisted Structure Elucidation of Isodemethylchodatin, a New Norlichexanthone Derivative Meager in H-Atoms, from the Lichen . Molecules (Basel, Switzerland). 24. PMID 31003403 DOI: 10.3390/Molecules24081527 |
0.313 |
|
2018 |
Otogo N'Nang E, Bernadat G, Mouray E, Kumulungui B, Grellier P, Poupon E, Champy P, Beniddir MA. Theionbrunonines A and B: Dimeric Vobasine Alkaloids Tethered by a Thioether Bridge from Mostuea brunonis. Organic Letters. 20: 6596-6600. PMID 30303382 DOI: 10.1021/Acs.Orglett.8B02961 |
0.31 |
|
2018 |
Merad J, Lalli C, Bernadat G, Maury J, Masson G. Frontispiece: Enantioselective Brønsted Acid Catalysis as a Tool for the Synthesis of Natural Products and Pharmaceuticals Chemistry - a European Journal. 24. DOI: 10.1002/Chem.201881662 |
0.355 |
|
2017 |
Naret T, Bignon J, Bernadat G, Benchekroun M, Levaique H, Lenoir C, Dubois J, Pruvost A, Saller F, Borgel D, Manoury B, Leblais V, Darrigrand R, Apcher S, Brion JD, et al. A fluorine scan of a tubulin polymerization inhibitor isocombretastatin A-4: Design, synthesis, molecular modelling, and biological evaluation. European Journal of Medicinal Chemistry. 143: 473-490. PMID 29202409 DOI: 10.1016/J.Ejmech.2017.11.055 |
0.329 |
|
2017 |
Merad J, Lalli C, Bernadat G, Maury J, Masson G. Enantioselective Brønsted Acid Catalysis as a Tool for the Synthesis of Natural Products and Pharmaceuticals. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28981209 DOI: 10.1002/Chem.201703556 |
0.415 |
|
2017 |
Lachkar D, Denizot N, Bernadat G, Ahamada K, Beniddir MA, Dumontet V, Gallard JF, Guillot R, Leblanc K, N'nang EO, Turpin V, Kouklovsky C, Poupon E, Evanno L, Vincent G. Unified biomimetic assembly of voacalgine A and bipleiophylline via divergent oxidative couplings. Nature Chemistry. 9: 793-798. PMID 28754932 DOI: 10.1038/Nchem.2735 |
0.362 |
|
2017 |
Mamone M, Gonçalves RSB, Blanchard F, Bernadat G, Ongeri S, Milcent T, Crousse B. N-Difluoromethyl-triazole as a constrained scaffold in peptidomimetics Chemical Communications. 53: 5024-5027. PMID 28429026 DOI: 10.1039/C7Cc01298E |
0.327 |
|
2017 |
Fox Ramos AE, Alcover C, Evanno L, Maciuk A, Litaudon M, Duplais C, Bernadat G, Gallard JF, Jullian JC, Mouray E, Grellier P, Loiseau PM, Pomel S, Poupon E, Champy P, et al. Revisiting Previously Investigated Plants: A Molecular Networking-Based Study of Geissospermum laeve. Journal of Natural Products. 80: 1007-1014. PMID 28282127 DOI: 10.1021/Acs.Jnatprod.6B01013 |
0.317 |
|
2017 |
Khelifi I, Naret T, Renko D, Hamze A, Bernadat G, Bignon J, Lenoir C, Dubois J, Brion JD, Provot O, Alami M. Design, synthesis and anticancer properties of IsoCombretaQuinolines as potent tubulin assembly inhibitors. European Journal of Medicinal Chemistry. 127: 1025-1034. PMID 28166995 DOI: 10.1016/J.Ejmech.2016.11.012 |
0.358 |
|
2017 |
Dumoulin A, Bernadat G, Masson G. Enantioselective three-component amination of enecarbamates enables the synthesis of structurally complex small molecules. The Journal of Organic Chemistry. PMID 28092703 DOI: 10.1021/Acs.Joc.6B03093 |
0.418 |
|
2016 |
Pautus S, Alami M, Adam F, Bernadat G, Lawrence DA, De Carvalho A, Ferry G, Rupin A, Hamze A, Champy P, Bonneau N, Gloanec P, Peglion JL, Brion JD, Bianchini EP, et al. Characterization of the Annonaceous acetogenin, annonacinone, a natural product inhibitor of plasminogen activator inhibitor-1. Scientific Reports. 6: 36462. PMID 27876785 DOI: 10.1038/Srep36462 |
0.301 |
|
2016 |
Vallerotto S, Douaron GL, Bernadat G, Ferrié L, Figadère B. 6-endo-dig Cycloisomerization of N-Propargyl Aminoquinoxalines: A New Route to 1,4,8-Triazaphenanthrenes Synthesis. 48: 3232-3240. DOI: 10.1055/S-0035-1562443 |
0.351 |
|
2015 |
AL-Shuaeeb RA, Galvani G, Bernadat G, Brion JD, Alami M, Messaoudi S. Diversity-oriented synthesis of fused thioglycosyl benzo[e][1,4]oxathiepin-5-ones and benzo[f][1,4]thiazepin-5(2H)-ones by a sequence of palladium-catalyzed glycosyl thiol arylation and deprotection-lactonization reactions. Organic & Biomolecular Chemistry. 13: 10904-16. PMID 26369372 DOI: 10.1039/C5Ob01603G |
0.368 |
|
2015 |
Pous J, Courant T, Bernadat G, Iorga BI, Blanchard F, Masson G. Regio-, Diastereo-, and Enantioselective Nitroso-Diels-Alder Reaction of 1,3-Diene-1-carbamates Catalyzed by Chiral Phosphoric Acids. Journal of the American Chemical Society. 137: 11950-3. PMID 26355670 DOI: 10.1021/Jacs.5B08515 |
0.582 |
|
2015 |
Soussi MA, Provot O, Bernadat G, Bignon J, Desravines D, Dubois J, Brion JD, Messaoudi S, Alami M. IsoCombretaQuinazolines: Potent Cytotoxic Agents with Antitubulin Activity. Chemmedchem. 10: 1392-402. PMID 26076053 DOI: 10.1002/Cmdc.201500069 |
0.348 |
|
2015 |
List B, Höfler D, Pous J, Courant T, Bernadat G, Iorga BI, Blanchard F, Masson G. Phosphoric Acid-Catalyzed Asymmetric Nitroso-Diels–Alder Reaction Synfacts. 11: 1212-1212. DOI: 10.1055/S-0035-1560719 |
0.561 |
|
2015 |
Skiredj A, Beniddir MA, Joseph D, Bernadat G, Evanno L, Poupon E. Harnessing the Intrinsic Reactivity within the Aplysinopsin Series for the Synthesis of Intricate Dimers: Natural from Start to Finish Synthesis (Germany). 47: 2367-2376. DOI: 10.1055/S-0034-1381032 |
0.378 |
|
2015 |
Vahdati L, Fanelli R, Bernadat G, Correia I, Lequin O, Ongeri S, Piarulli U. Synthesis and conformational studies of a stable peptidomimetic β-hairpin based on a bifunctional diketopiperazine turn inducer New Journal of Chemistry. 39: 3250-3258. DOI: 10.1039/C4Nj01437E |
0.312 |
|
2014 |
Amara Z, Bernadat G, Venot PE, Retailleau P, Troufflard C, Drège E, Le Bideau F, Joseph D. Thermodynamic epimeric equilibration and crystallisation-induced dynamic resolution of lobelanine, norlobelanine and related analogues. Organic & Biomolecular Chemistry. 12: 9797-810. PMID 25320963 DOI: 10.1039/C4Ob01787K |
0.383 |
|
2014 |
Tréguier B, Lawson M, Bernadat G, Bignon J, Dubois J, Brion JD, Alami M, Hamze A. Synthesis of a 3-(α-styryl)benzo[b]-thiophene library via bromocyclization of alkynes and palladium-catalyzed to sylhydrazones cross-couplings: evaluation as antitubulin agents. Acs Combinatorial Science. 16: 702-10. PMID 25229390 DOI: 10.1021/Co500115B |
0.4 |
|
2014 |
Skiredj A, Beniddir MA, Joseph D, Leblanc K, Bernadat G, Evanno L, Poupon E. A unified bioinspired "aplysinopsin cascade": total synthesis of (±)-tubastrindole B and related biosynthetic congeners. Organic Letters. 16: 4980-3. PMID 25222547 DOI: 10.1021/Ol502177M |
0.306 |
|
2014 |
Skiredj A, Beniddir MA, Joseph D, Leblanc K, Bernadat G, Evanno L, Poupon E. Spontaneous biomimetic formation of (±)-dictazole B under irradiation with artificial sunlight. Angewandte Chemie (International Ed. in English). 53: 6419-24. PMID 24817607 DOI: 10.1002/Anie.201403454 |
0.318 |
|
2014 |
Soussi MA, Provot O, Bernadat G, Bignon J, Wdzieczak-Bakala J, Desravines D, Dubois J, Brion JD, Messaoudi S, Alami M. Discovery of azaisoerianin derivatives as potential antitumors agents. European Journal of Medicinal Chemistry. 78: 178-89. PMID 24681982 DOI: 10.1016/J.Ejmech.2014.03.032 |
0.323 |
|
2014 |
Bernadat G, Masson G. Enamide derivatives: Versatile building blocks for highly functionalized α,β-substituted amines Synlett. 25. DOI: 10.1055/S-0034-1379166 |
0.334 |
|
2014 |
Ferrié L, Ferhi S, Bernadat G, Figadère B. Toward the Total Synthesis of Klaivanolide: Complete Reinterpretation of Its Originally Assigned Structure European Journal of Organic Chemistry. 2014: 6183-6189. DOI: 10.1002/Ejoc.201402741 |
0.332 |
|
2013 |
Gonçalves RS, Dos Santos M, Bernadat G, Bonnet-Delpon D, Crousse B. A one-pot synthesis of 3-trifluoromethyl-2-isoxazolines from trifluoromethyl aldoxime. Beilstein Journal of Organic Chemistry. 9: 2387-94. PMID 24367404 DOI: 10.3762/Bjoc.9.275 |
0.33 |
|
2013 |
Bordessa A, Keita M, Maréchal X, Formicola L, Lagarde N, Rodrigo J, Bernadat G, Bauvais C, Soulier JL, Dufau L, Milcent T, Crousse B, Reboud-Ravaux M, Ongeri S. α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome. European Journal of Medicinal Chemistry. 70: 505-24. PMID 24185380 DOI: 10.1016/J.Ejmech.2013.09.059 |
0.338 |
|
2013 |
Bernadat G, Supuran CT, Iorga BI. Carbonic anhydrase binding site parameterization in OPLS-AA force field. Bioorganic & Medicinal Chemistry. 21: 1427-30. PMID 23182217 DOI: 10.1016/J.Bmc.2012.10.040 |
0.49 |
|
2013 |
Aziz J, Brachet E, Hamze A, Peyrat JF, Bernadat G, Morvan E, Bignon J, Wdzieczak-Bakala J, Desravines D, Dubois J, Tueni M, Yassine A, Brion JD, Alami M. Synthesis, biological evaluation, and structure-activity relationships of tri- and tetrasubstituted olefins related to isocombretastatin A-4 as new tubulin inhibitors. Organic & Biomolecular Chemistry. 11: 430-42. PMID 23047722 DOI: 10.1039/C2Ob26253C |
0.384 |
|
2013 |
Lewin G, Bernadat G, Aubert G, Cresteil T. Semisynthesis of (+)- and (-)-goniomitine from (-)- and (+)-vincadifformine Tetrahedron. 69: 1622-1627. DOI: 10.1016/J.Tet.2012.11.084 |
0.315 |
|
2011 |
Lalli C, Brioche J, Bernadat G, Masson G. Catalytic enantioselective cycloaddition with chiral lewis bases Current Organic Chemistry. 15: 4108-4127. DOI: 10.2174/138527211798109178 |
0.345 |
|
2009 |
Wu YC, Bernadat G, Masson G, Couturier C, Schlama T, Zhu J. Synthetic studies on (-)-lemonomycin: an efficient asymmetric synthesis of lemonomycinone amide. The Journal of Organic Chemistry. 74: 2046-52. PMID 19196163 DOI: 10.1021/Jo8027449 |
0.422 |
|
2009 |
Wu Y-, Bernadat G, Masson G, Couturier C, Schlama T, Zhu J. Synthesis of Lemonomycinone Amide Synfacts. 2009: 1070-1070. DOI: 10.1055/S-0029-1217863 |
0.349 |
|
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