Valery V. Fokin - Publications

2000-2015 Chemistry Scripps Research Institute, La Jolla, La Jolla, CA, United States 
 2015- University of Southern California, Los Angeles, CA, United States 
New Reactivity, Catalysis, Organic Synthesis, and Macromolecules

121 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2019 Kovarik Z, Hrvat NM, Kalisiak J, Katalinić M, Sit RK, Zorbaz T, Radić Z, Fokin VV, Sharpless KB, Taylor P. Counteracting tabun inhibition by reactivation by pyridinium aldoximes that interact with active center gorge mutants of acetylcholinesterase. Toxicology and Applied Pharmacology. PMID 30978400 DOI: 10.1016/j.taap.2019.04.007  0.96
2018 Kovarik Z, Kalisiak J, Hrvat NM, Katalinić M, Zorbaz T, Žunec S, Green C, Radić Z, Fokin VV, Sharpless KB, Taylor P. Reversal of tabun toxicity, enabled by a triazole annulated oxime library-reactivators of acetylcholinesterase. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 30458057 DOI: 10.1002/chem.201805051  0.96
2018 Sit R, Kovarik Z, Macek-Hrvat N, Zunec S, Green C, Fokin V, Sharpless KB, Radic' Z, Taylor P. Pharmacology, pharmacokinetics and tissue disposition of zwitterionic hydoxyiminoacetamido alkylamines as reactivating antidotes for organophosphate exposure. The Journal of Pharmacology and Experimental Therapeutics. PMID 30190337 DOI: 10.1124/jpet.118.249383  0.96
2017 Kim WJ, Korthals K, Li S, Le C, Kalisiak J, Sharpless KB, Fokin VV, Miyamoto Y, Eckmann L. Click chemistry-facilitated structural diversification of nitrothiazoles, nitrofurans and nitropyrroles enhances antimicrobial activity against Giardia lamblia. Antimicrobial Agents and Chemotherapy. PMID 28396548 DOI: 10.1128/AAC.02397-16  0.96
2015 Arunrungvichian K, Boonyarat C, Fokin VV, Taylor P, Vajragupta O. Cognitive Improvements in a Mouse Model with Substituted 1,2,3-Triazole Agonists for Nicotinic Acetylcholine Receptors. Acs Chemical Neuroscience. PMID 25978789 DOI: 10.1021/acschemneuro.5b00059  0.44
2015 Arunrungvichian K, Fokin VV, Vajragupta O, Taylor P. Selectivity Optimization of Substituted 1,2,3-Triazoles as α7 Nicotinic Acetylcholine Receptor Agonists. Acs Chemical Neuroscience. PMID 25932897 DOI: 10.1021/acschemneuro.5b00058  0.44
2015 Kovarik Z, Ma?ek Hrvat N, Katalini? M, Sit RK, Paradyse A, Žunec S, Musilek K, Fokin VV, Taylor P, Radi? Z. Catalytic Soman Scavenging by the Y337A/F338A Acetylcholinesterase Mutant Assisted with Novel Site-Directed Aldoximes. Chemical Research in Toxicology. 28: 1036-44. PMID 25835984 DOI: 10.1021/acs.chemrestox.5b00060  1
2015 Voitovich YV, Shegravina ES, Sitnikov NS, Faerman VI, Fokin VV, Schmalz HG, Combes S, Allegro D, Barbier P, Beletskaya IP, Svirshchevskaya EV, Fedorov AY. Synthesis and biological evaluation of furanoallocolchicinoids. Journal of Medicinal Chemistry. 58: 692-704. PMID 25496412 DOI: 10.1021/jm501678w  1
2014 Dong J, Sharpless KB, Kwisnek L, Oakdale JS, Fokin VV. SuFEx-based synthesis of polysulfates. Angewandte Chemie (International Ed. in English). 53: 9466-70. PMID 25100330 DOI: 10.1002/anie.201403758  1
2014 Oakdale JS, Sit RK, Fokin VV. Ruthenium-catalyzed cycloadditions of 1-haloalkynes with nitrile oxides and organic azides: synthesis of 4-haloisoxazoles and 5-halotriazoles. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 11101-10. PMID 25059647 DOI: 10.1002/chem.201402559  1
2014 Rillahan CD, Macauley MS, Schwartz E, He Y, McBride R, Arlian BM, Rangarajan J, Fokin VV, Paulson JC. Disubstituted Sialic Acid Ligands Targeting Siglecs CD33 and CD22 Associated with Myeloid Leukaemias and B Cell Lymphomas. Chemical Science (Royal Society of Chemistry : 2010). 5: 2398-2406. PMID 24921038 DOI: 10.1039/C4SC00451E  1
2014 Kwok SW, Zhang L, Grimster NP, Fokin VV. Catalytic asymmetric transannulation of NH-1,2,3-triazoles with olefins. Angewandte Chemie (International Ed. in English). 53: 3452-6. PMID 24677710 DOI: 10.1002/anie.201306706  1
2014 Sit RK, Fokin VV, Amitai G, Sharpless KB, Taylor P, Radić Z. Imidazole aldoximes effective in assisting butyrylcholinesterase catalysis of organophosphate detoxification. Journal of Medicinal Chemistry. 57: 1378-89. PMID 24571195 DOI: 10.1021/jm401650z  1
2014 Chuprakov S, Worrell BT, Selander N, Sit RK, Fokin VV. Stereoselective 1,3-insertions of rhodium(II) azavinyl carbenes. Journal of the American Chemical Society. 136: 195-202. PMID 24295389 DOI: 10.1021/ja408185c  1
2014 Nyuchev AV, Schegravin KV, Lopatin MA, Fokin VV, Beletskaya IP, Fedorov AY. Synthesis of fluorescent boron difluoride complexes of 3-acyl-4-hydroxy-coumarins Synthesis (Germany). 46: 3239-3248. DOI: 10.1055/s-0034-1379020  1
2013 Oakdale JS, Fokin VV, Umezaki S, Fukuyama T. Preparation of 1,5-Disubstituted 1,2,3-Triazoles via Ruthenium-catalyzed Azide Alkyne Cycloaddition. Organic Syntheses; An Annual Publication of Satisfactory Methods For the Preparation of Organic Chemicals. 90: 96-104. PMID 25253916 DOI: 10.15227/orgsyn.090.0096  1
2013 Worrell BT, Ellery SP, Fokin VV. Copper(I)-catalyzed cycloaddition of bismuth(III) acetylides with organic azides: synthesis of stable triazole anion equivalents. Angewandte Chemie (International Ed. in English). 52: 13037-41. PMID 24130150 DOI: 10.1002/anie.201306192  1
2013 Miyamoto Y, Kalisiak J, Korthals K, Lauwaet T, Cheung DY, Lozano R, Cobo ER, Upcroft P, Upcroft JA, Berg DE, Gillin FD, Fokin VV, Sharpless KB, Eckmann L. Expanded therapeutic potential in activity space of next-generation 5-nitroimidazole antimicrobials with broad structural diversity. Proceedings of the National Academy of Sciences of the United States of America. 110: 17564-9. PMID 24101497 DOI: 10.1073/pnas.1302664110  1
2013 Rillahan CD, Schwartz E, Rademacher C, McBride R, Rangarajan J, Fokin VV, Paulson JC. On-chip synthesis and screening of a sialoside library yields a high affinity ligand for Siglec-7. Acs Chemical Biology. 8: 1417-22. PMID 23597400 DOI: 10.1021/cb400125w  1
2013 Sanphanya K, Wattanapitayakul SK, Phowichit S, Fokin VV, Vajragupta O. Novel VEGFR-2 kinase inhibitors identified by the back-to-front approach. Bioorganic & Medicinal Chemistry Letters. 23: 2962-7. PMID 23562241 DOI: 10.1016/j.bmcl.2013.03.042  1
2013 Worrell BT, Malik JA, Fokin VV. Direct evidence of a dinuclear copper intermediate in Cu(I)-catalyzed azide-alkyne cycloadditions. Science (New York, N.Y.). 340: 457-60. PMID 23558174 DOI: 10.1126/science.1229506  1
2013 Chuprakov S, Kwok SW, Fokin VV. Transannulation of 1-sulfonyl-1,2,3-triazoles with heterocumulenes. Journal of the American Chemical Society. 135: 4652-5. PMID 23477345 DOI: 10.1021/ja400350c  1
2013 Zibinsky M, Fokin VV. Sulfonyl-1,2,3-triazoles: convenient synthones for heterocyclic compounds. Angewandte Chemie (International Ed. in English). 52: 1507-10. PMID 23255432 DOI: 10.1002/anie.201206388  1
2013 Radi? Z, Sit RK, Garcia E, Zhang L, Berend S, Kovarik Z, Amitai G, Fokin VV, Barry Sharpless K, Taylor P. Mechanism of interaction of novel uncharged, centrally active reactivators with OP-hAChE conjugates. Chemico-Biological Interactions. 203: 67-71. PMID 22975155 DOI: 10.1016/j.cbi.2012.08.014  1
2013 Kovarik Z, Ma?ek N, Sit RK, Radi? Z, Fokin VV, Barry Sharpless K, Taylor P. Centrally acting oximes in reactivation of tabun-phosphoramidated AChE. Chemico-Biological Interactions. 203: 77-80. PMID 22960624 DOI: 10.1016/j.cbi.2012.08.019  1
2013 Malysheva YB, Buchvalova SY, Svirshchevskaya EV, Fokin VV, Fedorov AY. Negishi cross-coupling reaction as a route to isocombretastatins Synlett. 24: 1772-1776. DOI: 10.1055/s-0033-1339334  1
2013 Fraser BH, Hamilton S, Krause-Heuer AM, Wright PJ, Greguric I, Tucker SP, Draffan AG, Fokin VV, Sharpless KB. Synthesis of 1,4-triazole linked zanamivir dimers as highly potent inhibitors of influenza A and B Medchemcomm. 4: 383-386. DOI: 10.1039/c2md20300f  1
2012 Selander N, Worrell BT, Fokin VV. Ring expansion and rearrangements of rhodium(II) azavinyl carbenes. Angewandte Chemie (International Ed. in English). 51: 13054-7. PMID 23161725 DOI: 10.1002/anie.201207820  1
2012 Worrell BT, Hein JE, Fokin VV. Halogen exchange (Halex) reaction of 5-iodo-1,2,3-triazoles: synthesis and applications of 5-fluorotriazoles. Angewandte Chemie (International Ed. in English). 51: 11791-4. PMID 23059856 DOI: 10.1002/anie.201204979  1
2012 Rillahan CD, Schwartz E, McBride R, Fokin VV, Paulson JC. Click and pick: identification of sialoside analogues for siglec-based cell targeting. Angewandte Chemie (International Ed. in English). 51: 11014-8. PMID 23038623 DOI: 10.1002/anie.201205831  1
2012 Selander N, Worrell BT, Chuprakov S, Velaparthi S, Fokin VV. Arylation of rhodium(II) azavinyl carbenes with boronic acids. Journal of the American Chemical Society. 134: 14670-3. PMID 22913576 DOI: 10.1021/ja3062453  1
2012 Yamauchi JG, Gomez K, Grimster N, Dufouil M, Nemecz A, Fotsing JR, Ho KY, Talley TT, Sharpless KB, Fokin VV, Taylor P. Synthesis of selective agonists for the α7 nicotinic acetylcholine receptor with in situ click-chemistry on acetylcholine-binding protein templates. Molecular Pharmacology. 82: 687-99. PMID 22784805 DOI: 10.1124/mol.112.080291  1
2012 Jiaranaikulwanitch J, Govitrapong P, Fokin VV, Vajragupta O. From BACE1 inhibitor to multifunctionality of tryptoline and tryptamine triazole derivatives for Alzheimer's disease. Molecules (Basel, Switzerland). 17: 8312-33. PMID 22781443 DOI: 10.3390/molecules17078312  1
2012 Sanphanya K, Wattanapitayakul SK, Prangsaengtong O, Jo M, Koizumi K, Shibahara N, Priprem A, Fokin VV, Vajragupta O. Synthesis and evaluation of 1-(substituted)-3-prop-2-ynylureas as antiangiogenic agents. Bioorganic & Medicinal Chemistry Letters. 22: 3001-5. PMID 22414612 DOI: 10.1016/j.bmcl.2012.02.029  1
2012 Grimster NP, Stump B, Fotsing JR, Weide T, Talley TT, Yamauchi JG, Nemecz Á, Kim C, Ho KY, Sharpless KB, Taylor P, Fokin VV. Generation of candidate ligands for nicotinic acetylcholine receptors via in situ click chemistry with a soluble acetylcholine binding protein template. Journal of the American Chemical Society. 134: 6732-40. PMID 22394239 DOI: 10.1021/ja3001858  1
2012 Radi? Z, Sit RK, Kovarik Z, Berend S, Garcia E, Zhang L, Amitai G, Green C, Radi? B, Fokin VV, Sharpless KB, Taylor P. Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases. The Journal of Biological Chemistry. 287: 11798-809. PMID 22343626 DOI: 10.1074/jbc.M111.333732  1
2012 Selander N, Fokin VV. Rhodium(II)-catalyzed asymmetric sulfur(VI) reduction of diazo sulfonylamidines. Journal of the American Chemical Society. 134: 2477-80. PMID 22233190 DOI: 10.1021/ja210180q  1
2012 Hein JE, Krasnova LB, Iwasaki M, Fokin VV. Cu-catalyzed azide-alkyne cycloaddition: Preparation of tris((1-benzyl-1h-1,2,3-triazolyl)methyl)amine Organic Syntheses. 88: 238-246. DOI: 10.15227/orgsyn.088.0238  1
2012 Radi? Z, Sit RK, Kovarik Z, Berend S, Garcia E, Zhang L, Amitai G, Green C, Radi? B, Fokin VV, Sharpless KB, Taylor P. Refinement of structural leads for centrally acting oxime reactivators of phosphylated cholinesterases (Journal of Biological Chemistry (2012) 287, (11798-11809)) Journal of Biological Chemistry. 287: 19337. DOI: 10.1074/jbc.A111.333732  1
2012 Liu PN, Li J, Su FH, Ju KD, Zhang L, Shi C, Sung HHY, Williams ID, Fokin VV, Lin Z, Jia G. Selective formation of 1,4-disubstituted triazoles from ruthenium-catalyzed cycloaddition of terminal alkynes and organic azides: Scope and reaction mechanism Organometallics. 31: 4904-4915. DOI: 10.1021/om300513w  1
2012 Fokin VV, Matyjaszewski K. CuAAC: The Quintessential Click Reaction Organic Chemistry - Breakthroughs and Perspectives. 247-277. DOI: 10.1002/9783527664801.ch7  1
2011 Zibinsky M, Fokin VV. Reactivity of N-(1,2,4-triazolyl)-substituted 1,2,3-triazoles. Organic Letters. 13: 4870-2. PMID 21848347 DOI: 10.1021/ol201949h  1
2011 Culhane JC, Fokin VV. Synthesis and reactivity of sulfamoyl azides and 1-sulfamoyl-1,2,3-triazoles. Organic Letters. 13: 4578-80. PMID 21812453 DOI: 10.1021/ol201705k  1
2011 Cochran R, Kalisiak J, Küçükkilinç T, Radic Z, Garcia E, Zhang L, Ho KY, Amitai G, Kovarik Z, Fokin VV, Sharpless KB, Taylor P. Oxime-assisted acetylcholinesterase catalytic scavengers of organophosphates that resist aging. The Journal of Biological Chemistry. 286: 29718-24. PMID 21730071 DOI: 10.1074/jbc.M111.264739  1
2011 Chuprakov S, Malik JA, Zibinsky M, Fokin VV. Catalytic asymmetric C-H insertions of rhodium(II) azavinyl carbenes. Journal of the American Chemical Society. 133: 10352-5. PMID 21619004 DOI: 10.1021/ja202969z  1
2011 Sit RK, Radi? Z, Gerardi V, Zhang L, Garcia E, Katalini? M, Amitai G, Kovarik Z, Fokin VV, Sharpless KB, Taylor P. New structural scaffolds for centrally acting oxime reactivators of phosphylated cholinesterases. The Journal of Biological Chemistry. 286: 19422-30. PMID 21464125 DOI: 10.1074/jbc.M111.230656  1
2011 Gastaminza P, Pitram SM, Dreux M, Krasnova LB, Whitten-Bauer C, Dong J, Chung J, Fokin VV, Sharpless KB, Chisari FV. Antiviral stilbene 1,2-diamines prevent initiation of hepatitis C virus RNA replication at the outset of infection. Journal of Virology. 85: 5513-23. PMID 21430055 DOI: 10.1128/JVI.02116-10  1
2011 Schwartz E, Breitenkamp K, Fokin VV. Synthesis and postpolymerization functionalization of poly(5-iodo-1,2,3- triazole)s Macromolecules. 44: 4735-4741. DOI: 10.1021/ma2005469  1
2010 Krasnova LB, Hein JE, Fokin VV. Synthesis of 7-aza-5-deazapurine analogues via copper(I)-catalyzed hydroamination of alkynes and 1-iodoalkynes. The Journal of Organic Chemistry. 75: 8662-5. PMID 21105687 DOI: 10.1021/jo1016376  1
2010 Jiaranaikulwanitch J, Boonyarat C, Fokin VV, Vajragupta O. Triazolyl tryptoline derivatives as β-secretase inhibitors. Bioorganic & Medicinal Chemistry Letters. 20: 6572-6. PMID 20943389 DOI: 10.1016/j.bmcl.2010.09.043  1
2010 Raushel J, Fokin VV. Efficient synthesis of 1-sulfonyl-1,2,3-triazoles. Organic Letters. 12: 4952-5. PMID 20931987 DOI: 10.1021/ol102087r  1
2010 Kwok SW, Fotsing JR, Fraser RJ, Rodionov VO, Fokin VV. Transition-metal-free catalytic synthesis of 1,5-diaryl-1,2,3-triazoles. Organic Letters. 12: 4217-9. PMID 20825167 DOI: 10.1021/ol101568d  1
2010 Weide T, Saldanha SA, Minond D, Spicer TP, Fotsing JR, Spaargaren M, Frère JM, Bebrone C, Sharpless KB, Hodder PS, Fokin VV. NH-1,2,3-Triazole-based Inhibitors of the VIM-2 Metallo-β-Lactamase: Synthesis and Structure-Activity Studies. Acs Medicinal Chemistry Letters. 1: 150-154. PMID 20625539 DOI: 10.1021/ml900022q  1
2010 Radi? Z, Kalisiak J, Fokin VV, Sharpless KB, Taylor P. Interaction kinetics of oximes with native, phosphylated and aged human acetylcholinesterase. Chemico-Biological Interactions. 187: 163-6. PMID 20412789 DOI: 10.1016/j.cbi.2010.04.014  1
2010 Hein JE, Fokin VV. Copper-catalyzed azide-alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(I) acetylides. Chemical Society Reviews. 39: 1302-15. PMID 20309487 DOI: 10.1039/b904091a  1
2010 Finn MG, Fokin VV. Click chemistry: function follows form. Chemical Society Reviews. 39: 1231-2. PMID 20309482 DOI: 10.1039/c003740k  1
2010 Grimster N, Zhang L, Fokin VV. Synthesis and reactivity of rhodium(II) N-triflyl azavinyl carbenes. Journal of the American Chemical Society. 132: 2510-1. PMID 20131915 DOI: 10.1021/ja910187s  1
2010 Cravotto G, Fokin VV, Garella D, Binello A, Boffa L, Barge A. Ultrasound-promoted copper-catalyzed azide-alkyne cycloaddition. Journal of Combinatorial Chemistry. 12: 13-5. PMID 19904971 DOI: 10.1021/cc900150d  1
2010 Lewis DG, Krasnova LB, Skinner PJ, Fokin VV. Conductive dendrimers obtained by click chemistry Proceedings of Spie - the International Society For Optical Engineering. 7755. DOI: 10.1117/12.860879  1
2010 Fokin VV. New Reactions of Copper Acetylides: Catalytic Dipolar Cycloadditions and Beyond Catalyzed Carbon-Heteroatom Bond Formation. 199-222. DOI: 10.1002/9783527633388.ch7  1
2009 Chuprakov S, Kwok SW, Zhang L, Lercher L, Fokin VV. Rhodium-catalyzed enantioselective cyclopropanation of olefins with N-sulfonyl 1,2,3-triazoles. Journal of the American Chemical Society. 131: 18034-5. PMID 19928917 DOI: 10.1021/ja908075u  1
2009 Hein JE, Tripp JC, Krasnova LB, Sharpless KB, Fokin VV. Copper(I)-catalyzed cycloaddition of organic azides and 1-iodoalkynes. Angewandte Chemie (International Ed. in English). 48: 8018-21. PMID 19774581 DOI: 10.1002/anie.200903558  1
2009 Minond D, Saldanha SA, Subramaniam P, Spaargaren M, Spicer T, Fotsing JR, Weide T, Fokin VV, Sharpless KB, Galleni M, Bebrone C, Lassaux P, Hodder P. Inhibitors of VIM-2 by screening pharmacologically active and click-chemistry compound libraries. Bioorganic & Medicinal Chemistry. 17: 5027-37. PMID 19553129 DOI: 10.1016/j.bmc.2009.05.070  1
2009 Valdez CA, Tripp JC, Miyamoto Y, Kalisiak J, Hruz P, Andersen YS, Brown SE, Kangas K, Arzu LV, Davids BJ, Gillin FD, Upcroft JA, Upcroft P, Fokin VV, Smith DK, et al. Synthesis and electrochemistry of 2-ethenyl and 2-ethanyl derivatives of 5-nitroimidazole and antimicrobial activity against Giardia lamblia. Journal of Medicinal Chemistry. 52: 4038-53. PMID 19480409 DOI: 10.1021/jm900356n  1
2009 Agnew HD, Rohde RD, Millward SW, Nag A, Yeo WS, Hein JE, Pitram SM, Tariq AA, Burns VM, Krom RJ, Fokin VV, Sharpless KB, Heath JR. Iterative in situ click chemistry creates antibody-like protein-capture agents. Angewandte Chemie (International Ed. in English). 48: 4944-8. PMID 19301344 DOI: 10.1002/anie.200900488  1
2009 Chanda A, Fokin VV. Organic synthesis "on water". Chemical Reviews. 109: 725-48. PMID 19209944 DOI: 10.1021/cr800448q  1
2009 Kalisiak J, Trauger SA, Kalisiak E, Morita H, Fokin VV, Adams MW, Sharpless KB, Siuzdak G. Identification of a new endogenous metabolite and the characterization of its protein interactions through an immobilization approach. Journal of the American Chemical Society. 131: 378-86. PMID 19055353 DOI: 10.1021/ja808172n  1
2008 Kwok SW, Hein JE, Fokin VV, Sharpless KB. REGIOSELECTIVE SYNTHESIS OF EITHER 1H- OR 2H-1,2,3- TRIAZOLES VIA MICHAEL ADDITION TO α,ß-UNSATURATED KETONES. Heterocycles. 76: 1141-1154. PMID 19802363 DOI: 10.3987/COM-08-S(N)73  1
2008 Horneff T, Chuprakov S, Chernyak N, Gevorgyan V, Fokin VV. Rhodium-catalyzed transannulation of 1,2,3-triazoles with nitriles. Journal of the American Chemical Society. 130: 14972-4. PMID 18855475 DOI: 10.1021/ja805079v  1
2008 Grecian S, Fokin VV. Ruthenium-catalyzed cycloaddition of nitrile oxides and alkynes: practical synthesis of isoxazoles. Angewandte Chemie (International Ed. in English). 47: 8285-7. PMID 18814156 DOI: 10.1002/anie.200801920  1
2008 Raushel J, Pitram SM, Fokin VV. Efficient synthesis of sulfonyl azides from sulfonamides. Organic Letters. 10: 3385-8. PMID 18630918 DOI: 10.1021/ol8011088  1
2008 Kalisiak J, Sharpless KB, Fokin VV. Efficient synthesis of 2-substituted-1,2,3-triazoles. Organic Letters. 10: 3171-4. PMID 18597477 DOI: 10.1021/ol8006748  1
2008 Boren BC, Narayan S, Rasmussen LK, Zhang L, Zhao H, Lin Z, Jia G, Fokin VV. Ruthenium-catalyzed azide-alkyne cycloaddition: scope and mechanism. Journal of the American Chemical Society. 130: 8923-30. PMID 18570425 DOI: 10.1021/ja0749993  1
2008 Yoo EJ, Ahlquist M, Bae I, Sharpless KB, Fokin VV, Chang S. Mechanistic studies on the Cu-catalyzed three-component reactions of sulfonyl azides, 1-alkynes and amines, alcohols, or water: dichotomy via a common pathway. The Journal of Organic Chemistry. 73: 5520-8. PMID 18557650 DOI: 10.1021/jo800733p  1
2008 Boren BC, Narayan S, Rasmussen LK, Zhang L, Zhao H, Lin Z, Jia G, Fokin VV. Ruthenium-catalyzed azide-alkyne cycloaddition: Scope and mechanism (Journal of the American Chemical Society (2008) 130, (8923-8930)) Journal of the American Chemical Society. 130: 14900. DOI: 10.1021/ja805956e  1
2008 Finn MG, Kolb HC, Fokin VV, Sharpless KB. Click chemistry - Definition and aims Progress in Chemistry. 20: 1-4.  1
2007 Fokin VV. Click imaging of biochemical processes in living systems. Acs Chemical Biology. 2: 775-8. PMID 18154263 DOI: 10.1021/cb700254v  1
2007 Rasmussen LK, Boren BC, Fokin VV. Ruthenium-catalyzed cycloaddition of aryl azides and alkynes. Organic Letters. 9: 5337-9. PMID 18052070 DOI: 10.1021/ol701912s  1
2007 Rodionov VO, Presolski SI, Díaz DD, Fokin VV, Finn MG. Ligand-accelerated Cu-catalyzed azide-alkyne cycloaddition: a mechanistic report. Journal of the American Chemical Society. 129: 12705-12. PMID 17914817 DOI: 10.1021/ja072679d  1
2007 Yoo EJ, Ahlquist M, Kim SH, Bae I, Fokin VV, Sharpless KB, Chang S. Copper-catalyzed synthesis of N-sulfonyl-1,2,3-triazoles: controlling selectivity. Angewandte Chemie (International Ed. in English). 46: 1730-3. PMID 17397087 DOI: 10.1002/anie.200604241  1
2007 Hawker CJ, Fokin VV, Finn MG, Sharpless KB. Bringing efficiency to materials synthesis: The philosophy of click chemistry Australian Journal of Chemistry. 60: 381-383. DOI: 10.1071/CH07107  1
2007 Ahlquist M, Fokin VV. Enhanced reactivity of dinuclear copper(I) acetylides in dipolar cycloadditions Organometallics. 26: 4389-4391. DOI: 10.1021/om700669v  1
2007 Chan TR, Fokin VV. Polymer-supported copper(I) catalysts for the experimentally simplified azide-alkyne cycloaddition Qsar and Combinatorial Science. 26: 1274-1279. DOI: 10.1002/qsar.200740131  1
2007 Liu Y, Díaz DD, Accurso AA, Sharpless KB, Fokin VV, Finn MG. Click chemistry in materials synthesis. III. Metal-adhesive polymers from Cu(I)-catalyzed azide-alkyne cycloaddition Journal of Polymer Science, Part a: Polymer Chemistry. 45: 5182-5189. DOI: 10.1002/pola.22262  1
2007 Vestberg R, Malkoch M, Kade M, Wu P, Fokin VV, Sharpless KB, Drockenmuller E, Hawker CJ. Role of architecture and molecular weight in the formation of tailor-made ultrathin multilayers using dendritic macromolecules and click chemistry Journal of Polymer Science, Part a: Polymer Chemistry. 45: 2835-2846. DOI: 10.1002/pola.22178  1
2007 Narayan S, Fokin VV, Sharpless KB. Chemistry 'On Water'-Organic Synthesis in Aqueous Suspension Organic Reactions in Water: Principles, Strategies and Applications. 350-365. DOI: 10.1002/9780470988817.ch11  1
2007 Fokin VV. Kitchen microwaves - Not for the lab [3] Education in Chemistry. 44: 137.  1
2007 Wu P, Fokin VV. Catalytic azide-alkyne cycloaddition: Reactivity and applications Aldrichimica Acta. 40: 7-17.  1
2006 Whiting M, Tripp JC, Lin YC, Lindstrom W, Olson AJ, Elder JH, Sharpless KB, Fokin VV. Rapid discovery and structure-activity profiling of novel inhibitors of human immunodeficiency virus type 1 protease enabled by the copper(I)-catalyzed synthesis of 1,2,3-triazoles and their further functionalization. Journal of Medicinal Chemistry. 49: 7697-710. PMID 17181152 DOI: 10.1021/jm060754+  1
2006 Whiting M, Fokin VV. Copper-catalyzed reaction cascade: direct conversion of alkynes into N-sulfonylazetidin-2-imines. Angewandte Chemie (International Ed. in English). 45: 3157-61. PMID 16570331 DOI: 10.1002/anie.200503936  1
2006 Cassidy MP, Raushel J, Fokin VV. Practical synthesis of amides from in situ generated copper(I) acetylides and sulfonyl azides. Angewandte Chemie (International Ed. in English). 45: 3154-7. PMID 16570330 DOI: 10.1002/anie.200503805  1
2006 Whiting M, Muldoon J, Lin YC, Silverman SM, Lindstrom W, Olson AJ, Kolb HC, Finn MG, Sharpless KB, Elder JH, Fokin VV. Inhibitors of HIV-1 protease by using in situ click chemistry. Angewandte Chemie (International Ed. in English). 45: 1435-9. PMID 16425339 DOI: 10.1002/anie.200502161  1
2006 Wu P, Hilgraf R, Fokin VV. Osmium-catalyzed olefin dihydroxylation and aminohydroxylation in the second catalytic cycle Advanced Synthesis and Catalysis. 348: 1079-1085. DOI: 10.1002/adsc.200505252  1
2006 Fokin VV, Wu P. Epoxides and Aziridines in Click Chemistry Aziridines and Epoxides in Organic Synthesis. 443-477. DOI: 10.1002/3527607862.ch12  1
2006 Bae I, Han H, Chang S, Cho SH, Yoo EJ, Cassidy MP, Raushel J, Fokin VV, Whiting M, Kellogg RM. Multicomponent reactions with ketene imine intermediates formed from the reaction of sulfonyl azides with acetylenes Chemtracts. 19: 31-37.  1
2005 Wu P, Malkoch M, Hunt JN, Vestberg R, Kaltgrad E, Finn MG, Fokin VV, Sharpless KB, Hawker CJ. Multivalent, bifunctional dendrimers prepared by click chemistry. Chemical Communications (Cambridge, England). 5775-7. PMID 16307142 DOI: 10.1039/b512021g  1
2005 Zhang L, Chen X, Xue P, Sun HH, Williams ID, Sharpless KB, Fokin VV, Jia G. Ruthenium-catalyzed cycloaddition of alkynes and organic azides. Journal of the American Chemical Society. 127: 15998-9. PMID 16287266 DOI: 10.1021/ja054114s  1
2005 Feldman AK, Colasson B, Sharpless KB, Fokin VV. The allylic azide rearrangement: achieving selectivity. Journal of the American Chemical Society. 127: 13444-5. PMID 16190677 DOI: 10.1021/ja050622q  1
2005 Hansen TV, Wu P, Fokin VV. One-pot copper(I)-catalyzed synthesis of 3,5-disubstituted isoxazoles. The Journal of Organic Chemistry. 70: 7761-4. PMID 16149810 DOI: 10.1021/jo050163b  1
2005 Petasis NA, Akritopoulou-Zanze I, Fokin VV, Bernasconi G, Keledjian R, Yang R, Uddin J, Nagulapalli KC, Serhan CN. Design, synthesis and bioactions of novel stable mimetics of lipoxins and aspirin-triggered lipoxins. Prostaglandins, Leukotrienes, and Essential Fatty Acids. 73: 301-21. PMID 16098719 DOI: 10.1016/j.plefa.2005.05.020  1
2005 Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. "On water": unique reactivity of organic compounds in aqueous suspension. Angewandte Chemie (International Ed. in English). 44: 3275-9. PMID 15844112 DOI: 10.1002/anie.200462883  1
2005 Rodionov VO, Fokin VV, Finn MG. Mechanism of the ligand-free CuI-catalyzed azide-alkyne cycloaddition reaction. Angewandte Chemie (International Ed. in English). 44: 2210-5. PMID 15693051 DOI: 10.1002/anie.200461496  1
2005 Himo F, Lovell T, Hilgraf R, Rostovtsev VV, Noodleman L, Sharpless KB, Fokin VV. Copper(I)-catalyzed synthesis of azoles. DFT study predicts unprecedented reactivity and intermediates. Journal of the American Chemical Society. 127: 210-6. PMID 15631470 DOI: 10.1021/ja0471525  1
2005 Loren JC, Krasiński A, Fokin VV, Sharpless KB. NH-1,2,3-triazoles from azidomethyl pivalate and carbamates: Base-labile N-protecting groups Synlett. 2847-2850. DOI: 10.1055/s-2005-918944  1
2005 Malkoch M, Schleicher K, Drockenmuller E, Hawker CJ, Russell TP, Wu P, Fokin VV. Structurally diverse dendritic libraries: A highly efficient functionalization approach using click chemistry Macromolecules. 38: 3663-3678. DOI: 10.1021/ma047657f  1
2005 Meng JC, Fokin VV, Finn MG. Kinetic resolution by copper-catalyzed azide-alkyne cycloaddition Tetrahedron Letters. 46: 4543-4546. DOI: 10.1016/j.tetlet.2005.05.019  1
2004 Feldman AK, Colasson B, Fokin VV. One-pot synthesis of 1,4-disubstituted 1,2,3-triazoles from in situ generated azides. Organic Letters. 6: 3897-9. PMID 15496058 DOI: 10.1021/ol048859z  1
2004 Chan TR, Hilgraf R, Sharpless KB, Fokin VV. Polytriazoles as copper(I)-stabilizing ligands in catalysis. Organic Letters. 6: 2853-5. PMID 15330631 DOI: 10.1021/ol0493094  1
2004 Lewis WG, Magallon FG, Fokin VV, Finn MG. Discovery and characterization of catalysts for azide-alkyne cycloaddition by fluorescence quenching. Journal of the American Chemical Society. 126: 9152-3. PMID 15281783 DOI: 10.1021/ja048425z  0.88
2004 Wu P, Feldman AK, Nugent AK, Hawker CJ, Scheel A, Voit B, Pyun J, Fréchet JM, Sharpless KB, Fokin VV. Efficiency and fidelity in a click-chemistry route to triazole dendrimers by the copper(i)-catalyzed ligation of azides and alkynes. Angewandte Chemie (International Ed. in English). 43: 3928-32. PMID 15274216 DOI: 10.1002/anie.200454078  1
2004 Krasi?ski A, Fokin VV, Sharpless KB. Direct synthesis of 1,5-disubstituted-4-magnesio-1,2,3-triazoles, revisited. Organic Letters. 6: 1237-40. PMID 15070306 DOI: 10.1021/ol0499203  1
2003 Brik A, Muldoon J, Lin YC, Elder JH, Goodsell DS, Olson AJ, Fokin VV, Sharpless KB, Wong CH. Rapid diversity-oriented synthesis in microtiter plates for in situ screening of HIV protease inhibitors. Chembiochem : a European Journal of Chemical Biology. 4: 1246-8. PMID 14613121 DOI: 10.1002/cbic.200300724  1
2003 Lee LV, Mitchell ML, Huang SJ, Fokin VV, Sharpless KB, Wong CH. A potent and highly selective inhibitor of human alpha-1,3-fucosyltransferase via click chemistry. Journal of the American Chemical Society. 125: 9588-9. PMID 12904015 DOI: 10.1021/ja0302836  1
2003 Wang Q, Chan TR, Hilgraf R, Fokin VV, Sharpless KB, Finn MG. Bioconjugation by copper(I)-catalyzed azide-alkyne [3 + 2] cycloaddition. Journal of the American Chemical Society. 125: 3192-3. PMID 12630856 DOI: 10.1021/ja021381e  1
2002 Andersson MA, Epple R, Fokin VV, Sharpless KB. A new approach to osmium-catalyzed asymmetric dihydroxylation and aminohydroxylation of olefins. Angewandte Chemie (International Ed. in English). 41: 472-5. PMID 12491382 DOI: 10.1002/1521-3773(20020201)41:3<472::AID-ANIE472>3.0.CO;2-7  1
2002 Rostovtsev VV, Green LG, Fokin VV, Sharpless KB. A stepwise huisgen cycloaddition process: copper(I)-catalyzed regioselective "ligation" of azides and terminal alkynes. Angewandte Chemie (International Ed. in English). 41: 2596-9. PMID 12203546 DOI: 10.1002/1521-3773(20020715)41:14<2596::AID-ANIE2596>3.0.CO;2-4  1
2001 Fokin VV, Sharpless KB. A Practical and Highly Efficient Aminohydroxylation of Unsaturated Carboxylic Acids We thank the National Institute of General Medical Sciences, the National Institutes of Health (GM 28384), National Science Foundation (CHE-9985553), and the W. M. Keck Foundation for financial support. We are also grateful to Prof. M. G. Finn, Dr. Wallace Pringle, and Dr. A. Erik Rubin for many helpful discussions. Angewandte Chemie (International Ed. in English). 40: 3455-3457. PMID 11592169 DOI: 10.1002/1521-3773(20010917)40:18<3455::AID-ANIE3455>3.0.CO;2-I  0.96
1999 Levy BD, Fokin VV, Clark JM, Wakelam MJ, Petasis NA, Serhan CN. Polyisoprenyl phosphate (PIPP) signaling regulates phospholipase D activity: a 'stop' signaling switch for aspirin-triggered lipoxin A4. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 13: 903-11. PMID 10224233  1
1999 Gewirtz AT, Fokin VV, Petasis NA, Serhan CN, Madara JL. LXA4, aspirin-triggered 15-epi-LXA4, and their analogs selectively downregulate PMN azurophilic degranulation. The American Journal of Physiology. 276: C988-94. PMID 10199831  1
1998 Maddox JF, Colgan SP, Clish CB, Petasis NA, Fokin VV, Serhan CN. Lipoxin B4 regulates human monocyte/neutrophil adherence and motility: design of stable lipoxin B4 analogs with increased biologic activity. Faseb Journal : Official Publication of the Federation of American Societies For Experimental Biology. 12: 487-94. PMID 9535221  1
1997 Maddox JF, Hachicha M, Takano T, Petasis NA, Fokin VV, Serhan CN. Lipoxin A4 stable analogs are potent mimetics that stimulate human monocytes and THP-1 cells via a G-protein-linked lipoxin A4 receptor. The Journal of Biological Chemistry. 272: 6972-8. PMID 9054386 DOI: 10.1074/jbc.272.11.6972  1
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