Hartmuth C. Kolb - Publications

Affiliations: 
Eli Lilly and Company, Indianapolis, IN, United States 
Area:
Click chemistry
Website:
http://de.wikipedia.org/wiki/Hartmuth_C._Kolb

91 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2015 Ariza M, Kolb HC, Moechars D, Rombouts F, Andrés JI. Tau Positron Emission Tomography (PET) Imaging: Past, Present, and Future. Journal of Medicinal Chemistry. 58: 4365-82. PMID 25671691 DOI: 10.1021/jm5017544  1
2014 Doss M, Kolb HC, Walsh JC, Mocharla VP, Zhu Z, Haka M, Alpaugh RK, Chen DY, Yu JQ. Biodistribution and radiation dosimetry of the carbonic anhydrase IX imaging agent [(18) F]VM4-037 determined from PET/CT scans in healthy volunteers. Molecular Imaging and Biology : Mib : the Official Publication of the Academy of Molecular Imaging. 16: 739-46. PMID 24696183 DOI: 10.1007/s11307-014-0730-7  1
2014 Su H, Gorodny N, Gomez LF, Gangadharmath UB, Mu F, Chen G, Walsh JC, Szardenings K, Berman DS, Kolb HC, Tamarappoo BK. Atherosclerotic plaque uptake of a novel integrin tracer ¹⁸F-Flotegatide in a mouse model of atherosclerosis. Journal of Nuclear Cardiology : Official Publication of the American Society of Nuclear Cardiology. 21: 553-62. PMID 24627345 DOI: 10.1007/s12350-014-9879-3  1
2014 Walsh JC, Lebedev A, Aten E, Madsen K, Marciano L, Kolb HC. The clinical importance of assessing tumor hypoxia: relationship of tumor hypoxia to prognosis and therapeutic opportunities. Antioxidants & Redox Signaling. 21: 1516-54. PMID 24512032 DOI: 10.1089/ars.2013.5378  1
2014 Chien DT, Szardenings AK, Bahri S, Walsh JC, Mu F, Xia C, Shankle WR, Lerner AJ, Su MY, Elizarov A, Kolb HC. Early clinical PET imaging results with the novel PHF-tau radioligand [F18]-T808. Journal of Alzheimer's Disease : Jad. 38: 171-84. PMID 23948934 DOI: 10.3233/JAD-130098  1
2013 Doss M, Kolb HC, Walsh JC, Mocharla V, Fan H, Chaudhary A, Zhu Z, Alpaugh RK, Lango MN, Yu JQ. Biodistribution and radiation dosimetry of 18F-CP-18, a potential apoptosis imaging agent, as determined from PET/CT scans in healthy volunteers. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 54: 2087-92. PMID 24136934 DOI: 10.2967/jnumed.113.119800  1
2013 Hugenberg V, Riemann B, Hermann S, Schober O, Schäfers M, Szardenings K, Lebedev A, Gangadharmath U, Kolb H, Walsh J, Zhang W, Kopka K, Wagner S. Inverse 1,2,3-triazole-1-yl-ethyl substituted hydroxamates as highly potent matrix metalloproteinase inhibitors: (radio)synthesis, in vitro and first in vivo evaluation. Journal of Medicinal Chemistry. 56: 6858-70. PMID 23899323 DOI: 10.1021/jm4006753  1
2013 Mirfeizi L, Walsh J, Kolb H, Campbell-Verduyn L, Dierckx RA, Feringa BL, Elsinga PH, de Groot T, Sannen I, Bormans G, Celen S. Synthesis of [18F]RGD-K5 by catalyzed [3 + 2] cycloaddition for imaging integrin αvβ3 expression in vivo. Nuclear Medicine and Biology. 40: 710-6. PMID 23706550 DOI: 10.1016/j.nucmedbio.2013.04.003  1
2013 Xia CF, Chen G, Gangadharmath U, Gomez LF, Liang Q, Mu F, Mocharla VP, Su H, Szardenings AK, Walsh JC, Zhao T, Kolb HC. In vitro and in vivo evaluation of the caspase-3 substrate-based radiotracer [(18)F]-CP18 for PET imaging of apoptosis in tumors. Molecular Imaging and Biology : Mib : the Official Publication of the Academy of Molecular Imaging. 15: 748-57. PMID 23689985 DOI: 10.1007/s11307-013-0646-7  1
2013 Su H, Chen G, Gangadharmath U, Gomez LF, Liang Q, Mu F, Mocharla VP, Szardenings AK, Walsh JC, Xia CF, Yu C, Kolb HC. Evaluation of [(18)F]-CP18 as a PET imaging tracer for apoptosis. Molecular Imaging and Biology : Mib : the Official Publication of the Academy of Molecular Imaging. 15: 739-47. PMID 23681757 DOI: 10.1007/s11307-013-0644-9  1
2013 Xia CF, Arteaga J, Chen G, Gangadharmath U, Gomez LF, Kasi D, Lam C, Liang Q, Liu C, Mocharla VP, Mu F, Sinha A, Su H, Szardenings AK, Walsh JC, ... ... Kolb HC, et al. [(18)F]T807, a novel tau positron emission tomography imaging agent for Alzheimer's disease. Alzheimer's & Dementia : the Journal of the Alzheimer's Association. 9: 666-76. PMID 23411393 DOI: 10.1016/j.jalz.2012.11.008  1
2013 Chien DT, Bahri S, Szardenings AK, Walsh JC, Mu F, Su MY, Shankle WR, Elizarov A, Kolb HC. Early clinical PET imaging results with the novel PHF-tau radioligand [F-18]-T807. Journal of Alzheimer's Disease : Jad. 34: 457-68. PMID 23234879 DOI: 10.3233/JAD-122059  1
2013 Mocharla VP, Walsh JC, Padgett HC, Su H, Fueger B, Weber WA, Czernin J, Kolb HC. From in situ to in vivo: an in situ click-chemistry-derived carbonic anhydrase II imaging agent for positron emission tomography. Chemmedchem. 8: 43-8. PMID 23208787 DOI: 10.1002/cmdc.201200466  1
2013 Lebedev A, Miraghaie R, Kotta K, Ball CE, Zhang J, Buchsbaum MS, Kolb HC, Elizarov A. Batch-reactor microfluidic device: first human use of a microfluidically produced PET radiotracer. Lab On a Chip. 13: 136-45. PMID 23135409 DOI: 10.1039/c2lc40853h  1
2012 Yokell DL, Leece AK, Lebedev A, Miraghaie R, Ball CE, Zhang J, Kolb H, Elizarov A, Mahmood U. Microfluidic single vessel production of hypoxia tracer 1H-1-(3-[18F]-fluoro-2-hydroxy-propyl)-2-nitro-imidazole ([18F]-FMISO). Applied Radiation and Isotopes : Including Data, Instrumentation and Methods For Use in Agriculture, Industry and Medicine. 70: 2313-6. PMID 22871433 DOI: 10.1016/j.apradiso.2012.05.022  1
2012 Chen L, Zhang Z, Kolb HC, Walsh JC, Zhang J, Guan Y. ¹⁸F-HX4 hypoxia imaging with PET/CT in head and neck cancer: a comparison with ¹⁸F-FMISO. Nuclear Medicine Communications. 33: 1096-102. PMID 22836736 DOI: 10.1097/MNM.0b013e3283571016  1
2012 Zhang W, Arteaga J, Cashion DK, Chen G, Gangadharmath U, Gomez LF, Kasi D, Lam C, Liang Q, Liu C, Mocharla VP, Mu F, Sinha A, Szardenings AK, Wang E, ... ... Kolb HC, et al. A highly selective and specific PET tracer for imaging of tau pathologies. Journal of Alzheimer's Disease : Jad. 31: 601-12. PMID 22683529 DOI: 10.3233/JAD-2012-120712  1
2012 Hugenberg V, Breyholz HJ, Riemann B, Hermann S, Schober O, Schäfers M, Gangadharmath U, Mocharla V, Kolb H, Walsh J, Zhang W, Kopka K, Wagner S. A new class of highly potent matrix metalloproteinase inhibitors based on triazole-substituted hydroxamates: (radio)synthesis and in vitro and first in vivo evaluation. Journal of Medicinal Chemistry. 55: 4714-27. PMID 22540974 DOI: 10.1021/jm300199g  1
2012 Doss M, Kolb HC, Zhang JJ, Bélanger MJ, Stubbs JB, Stabin MG, Hostetler ED, Alpaugh RK, von Mehren M, Walsh JC, Haka M, Mocharla VP, Yu JQ. Biodistribution and radiation dosimetry of the integrin marker 18F-RGD-K5 determined from whole-body PET/CT in monkeys and humans. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 53: 787-95. PMID 22499613 DOI: 10.2967/jnumed.111.088955  1
2012 Kolb HC, Padgett HC, Zigler S, Patanella J, Mu F, Gangadharmath UB, Mocharla VP, Scott PJH, Walsh JC. Radiosynthesis of 3'-Deoxy-3'-[18F]Fluorothymidine ([18F]FLT) Radiochemical Syntheses: Radiopharmaceuticals For Positron Emission Tomography. 1: 21-30. DOI: 10.1002/9781118140345.ch3  1
2011 Dubois LJ, Lieuwes NG, Janssen MH, Peeters WJ, Windhorst AD, Walsh JC, Kolb HC, Ollers MC, Bussink J, van Dongen GA, van der Kogel A, Lambin P. Preclinical evaluation and validation of [18F]HX4, a promising hypoxia marker for PET imaging. Proceedings of the National Academy of Sciences of the United States of America. 108: 14620-5. PMID 21873245 DOI: 10.1073/pnas.1102526108  1
2011 Elizarov AM, Meinhart C, Miraghaie R, van Dam RM, Huang J, Daridon A, Heath JR, Kolb HC. Flow optimization study of a batch microfluidics PET tracer synthesizing device. Biomedical Microdevices. 13: 231-42. PMID 21072595 DOI: 10.1007/s10544-010-9488-0  1
2011 Bejot R, Elizarov AM, Ball E, Zhang J, Miraghaie R, Kolb HC, Gouverneur V. Batch-mode microfluidic radiosynthesis of N-succinimidyl-4-[ 18F]fluorobenzoate for protein labelling Journal of Labelled Compounds and Radiopharmaceuticals. 54: 117-122. DOI: 10.1002/jlcr.1826  1
2010 Walsh JC, Kolb HC. Applications of click chemistry in radiopharmaceutical development. Chimia. 64: 29-33. PMID 21137680 DOI: 10.2533/chimia.2010.29  1
2010 Doss M, Zhang JJ, Bélanger MJ, Stubbs JB, Hostetler ED, Alpaugh K, Kolb HC, Yu JQ. Biodistribution and radiation dosimetry of the hypoxia marker 18F-HX4 in monkeys and humans determined by using whole-body PET/CT. Nuclear Medicine Communications. 31: 1016-24. PMID 20948452 DOI: 10.1097/MNM.0b013e3283407950  1
2010 van Loon J, Janssen MH, Ollers M, Aerts HJ, Dubois L, Hochstenbag M, Dingemans AM, Lalisang R, Brans B, Windhorst B, van Dongen GA, Kolb H, Zhang J, De Ruysscher D, Lambin P. PET imaging of hypoxia using [18F]HX4: a phase I trial. European Journal of Nuclear Medicine and Molecular Imaging. 37: 1663-8. PMID 20369236 DOI: 10.1007/s00259-010-1437-x  1
2010 Elizarov AM, van Dam RM, Shin YS, Kolb HC, Padgett HC, Stout D, Shu J, Huang J, Daridon A, Heath JR. Design and optimization of coin-shaped microreactor chips for PET radiopharmaceutical synthesis. Journal of Nuclear Medicine : Official Publication, Society of Nuclear Medicine. 51: 282-7. PMID 20124050 DOI: 10.2967/jnumed.109.065946  1
2010 Sanchez-Alavez M, Tabarean IV, Osborn O, Mitsukawa K, Schaefer J, Dubins J, Holmberg KH, Klein I, Klaus J, Gomez LF, Kolb H, Secrest J, Jochems J, Myashiro K, Buckley P, et al. Insulin causes hyperthermia by direct inhibition of warm-sensitive neurons. Diabetes. 59: 43-50. PMID 19846801 DOI: 10.2337/db09-1128  1
2010 Zhang J, Elizarov A, Miraghaie R, Ball E, Kolb H. A system for the radiochemical purification of microfluidics-generated compound Journal of Labelled Compounds and Radiopharmaceuticals. 53: 311-314. DOI: 10.1002/jlcr.1768  1
2010 Kolb HC, Finn MG, Sharpless KB. ChemInform Abstract: Click Chemistry: Diverse Chemical Function from a Few Good Reactions Cheminform. 32: no-no. DOI: 10.1002/chin.200135279  1
2010 KOLB HC, ANDERSSON PG, SHARPLESS KB. ChemInform Abstract: Toward an Understanding of the High Enantioselectivity in the Osmium- Catalyzed Asymmetric Dihydroxylation (AD). Part 1. Kinetics. Cheminform. 25: no-no. DOI: 10.1002/chin.199426078  1
2010 KOLB HC, BENNANI YL, SHARPLESS KB. ChemInform Abstract: Short and Practical Syntheses of (R)-(-)-Carnitine and (R)-(-)-γ- Amino-β-hydroxybutyric Acid (GABOB). Cheminform. 24: no-no. DOI: 10.1002/chin.199321060  1
2010 KOLB HC, SHARPLESS KB. ChemInform Abstract: A Simplified Procedure for the Stereospecific Transformation of 1,2- Diols into Epoxides. Cheminform. 24: no-no. DOI: 10.1002/chin.199313174  1
2010 Sanchez-Alavez M, Tabarean IV, Osborn O, Mitsukawa K, Schaefer J, Dubins J, Holmberg KH, Klein I, Klaus J, Gomez LF, Kolb H, Secrest J, Jochems J, Myashiro K, Buckley P, et al. Insulin causes hyperthermia by direct inhibition of warm-sensitive neurons (Diabetes (2010) 59, (43-50)) Diabetes. 59: 756.  1
2009 Wang Y, Lin WY, Liu K, Lin RJ, Selke M, Kolb HC, Zhang N, Zhao XZ, Phelps ME, Shen CK, Faull KF, Tseng HR. An integrated microfluidic device for large-scale in situ click chemistry screening. Lab On a Chip. 9: 2281-5. PMID 19636457 DOI: 10.1039/b907430a  1
2008 Ley SV, Abad-Somovilla A, Anderson JC, Ayats C, Bänteli R, Beckmann E, Boyer A, Brasca MG, Brice A, Broughton HB, Burke BJ, Cleator E, Craig D, Denholm AA, Denton RM, ... ... Kolb HC, et al. The synthesis of azadirachtin: a potent insect antifeedant. Chemistry (Weinheim An Der Bergstrasse, Germany). 14: 10683-704. PMID 18821532 DOI: 10.1002/chem.200801103  1
2008 Finn MG, Kolb HC, Fokin VV, Sharpless KB. Click chemistry - Definition and aims Progress in Chemistry. 20: 1-4.  1
2007 Van Dam RM, Elizarov AM, Ball CE, Shen CKF, Padgett H, Kolb H, Rolland J, Diener L, Williams D, Edgecombe B, Jeffries J, Stoianova D, Stephen T, Motamedi F, Heath JR. Automated microfluidic-chip-based stand-alone instrument for the synthesis of radiopharmaceuticals on human-dose scales 2007 Nsti Nanotechnology Conference and Trade Show - Nsti Nanotech 2007, Technical Proceedings. 3: 300-303.  1
2006 Wang J, Sui G, Mocharla VP, Lin RJ, Phelps ME, Kolb HC, Tseng HR. Integrated microfluidics for parallel screening of an in situ click chemistry library. Angewandte Chemie (International Ed. in English). 45: 5276-81. PMID 16927322 DOI: 10.1002/anie.200601677  1
2006 Whiting M, Muldoon J, Lin YC, Silverman SM, Lindstrom W, Olson AJ, Kolb HC, Finn MG, Sharpless KB, Elder JH, Fokin VV. Inhibitors of HIV-1 protease by using in situ click chemistry. Angewandte Chemie (International Ed. in English). 45: 1435-9. PMID 16425339 DOI: 10.1002/anie.200502161  1
2006 Elizarov AM, Kolb HC, Van Dam RM, Heath JR, Padgett HC, Huang J, Daridon A. Coin-shaped reactor in microfluidic devices used for radiopharmaceutical synthesis 2006 Nsti Nanotechnology Conference and Trade Show - Nsti Nanotech 2006 Technical Proceedings. 2: 542-545.  1
2005 Lee CC, Sui G, Elizarov A, Shu CJ, Shin YS, Dooley AN, Huang J, Daridon A, Wyatt P, Stout D, Kolb HC, Witte ON, Satyamurthy N, Heath JR, Phelps ME, et al. Multistep synthesis of a radiolabeled imaging probe using integrated microfluidics. Science (New York, N.Y.). 310: 1793-6. PMID 16357255 DOI: 10.1126/science.1118919  1
2005 Radi? Z, Manetsch R, Krasi?ski A, Raushel J, Yamauchi J, Garcia C, Kolb H, Sharpless KB, Taylor P. Molecular basis of interactions of cholinesterases with tight binding inhibitors. Chemico-Biological Interactions. 157: 133-41. PMID 16289416 DOI: 10.1016/j.cbi.2005.10.020  1
2005 Bourne Y, Radi? Z, Kolb HC, Sharpless KB, Taylor P, Marchot P. Structural insights into conformational flexibility at the peripheral site and within the active center gorge of AChE. Chemico-Biological Interactions. 157: 159-65. PMID 16259971 DOI: 10.1016/j.cbi.2005.10.018  1
2005 Krasi?ski A, Radi? Z, Manetsch R, Raushel J, Taylor P, Sharpless KB, Kolb HC. In situ selection of lead compounds by click chemistry: target-guided optimization of acetylcholinesterase inhibitors. Journal of the American Chemical Society. 127: 6686-92. PMID 15869290 DOI: 10.1021/ja043031t  1
2005 Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. "On water": unique reactivity of organic compounds in aqueous suspension. Angewandte Chemie (International Ed. in English). 44: 3275-9. PMID 15844112 DOI: 10.1002/anie.200462883  1
2005 Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. Cover Picture: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. Int. Ed. 21/2005) Angewandte Chemie International Edition. 44: 3157-3157. DOI: 10.1002/anie.200590069  1
2005 Narayan S, Muldoon J, Finn MG, Fokin VV, Kolb HC, Sharpless KB. Titelbild: “On Water”: Unique Reactivity of Organic Compounds in Aqueous Suspension (Angew. Chem. 21/2005) Angewandte Chemie. 117: 3219-3219. DOI: 10.1002/ange.200590069  1
2004 Mocharla VP, Colasson B, Lee LV, Röper S, Sharpless KB, Wong CH, Kolb HC. In situ click chemistry: enzyme-generated inhibitors of carbonic anhydrase II. Angewandte Chemie (International Ed. in English). 44: 116-20. PMID 15599912 DOI: 10.1002/anie.200461580  1
2004 Manetsch R, Krasi?ski A, Radi? Z, Raushel J, Taylor P, Sharpless KB, Kolb HC. In situ click chemistry: enzyme inhibitors made to their own specifications. Journal of the American Chemical Society. 126: 12809-18. PMID 15469276 DOI: 10.1021/ja046382g  1
2004 Bourne Y, Kolb HC, Radi? Z, Sharpless KB, Taylor P, Marchot P. Freeze-frame inhibitor captures acetylcholinesterase in a unique conformation. Proceedings of the National Academy of Sciences of the United States of America. 101: 1449-54. PMID 14757816 DOI: 10.1073/pnas.0308206100  1
2004 Voronkov MV, Gontcharov AV, Wang ZM, Richardson PF, Kolb HC. Efficient solution phase parallel synthesis of norstatine analogs Tetrahedron. 60: 9043-9048. DOI: 10.1016/j.tet.2004.07.085  1
2003 Kolb HC, Sharpless KB. The growing impact of click chemistry on drug discovery. Drug Discovery Today. 8: 1128-37. PMID 14678739 DOI: 10.1016/S1359-6446(03)02933-7  1
2003 Schwardt O, Kolb H, Ernst B. Drug discovery today Current Topics in Medicinal Chemistry. 3: 1-9. PMID 12570684  1
2002 Katritzky AR, Zhang S, Wang M, Kolb HC, Steel PJ. Novel syntheses of polysubstituted pyrroles and oxazoles by 1,3-dipolar cycloaddition reactions of benzotriazole-stabilized nitrile ylides Journal of Heterocyclic Chemistry. 39: 759-765.  1
2001 Kolb HC, Finn MG, Sharpless KB. Click Chemistry: Diverse Chemical Function from a Few Good Reactions. Angewandte Chemie (International Ed. in English). 40: 2004-2021. PMID 11433435 DOI: 10.1002/1521-3773(20010601)40:11<2004::AID-ANIE2004>3.0.CO;2-5  1
2001 Kolb HC, Finn MG, Sharpless KB. Click-Chemie: diverse chemische Funktionalität mit einer Handvoll guter Reaktionen Angewandte Chemie. 113: 2056-2075. DOI: 10.1002/1521-3757(20010601)113:11<2056::AID-ANGE2056>3.0.CO;2-W  1
2001 Voronkov MV, Gontcharov AV, Wang ZM, Kolb HC. Reaction of α,β-dihydroxydihydrocinnamic esters with acetonitrile: A new approach to β-amino-α-hydroxydihydrocinnamic acids Arkivoc. 2001: 160-165.  1
2001 Ernst B, Dragic Z, Marti S, Müller C, Wagner B, Jahnke W, Magnani JL, Norman KE, Oehrlein R, Peters T, Kolb HC. Design and synthesis of E-selectin antagonists Chimia. 55: 268-274.  1
2000 Katritzky AR, Huang TB, Voronkov MV, Wang M, Kolb H. Efficient one-pot synthesis of polysubstituted pyrroles Journal of Organic Chemistry. 65: 8819-8821. PMID 11112611 DOI: 10.1021/jo001160w  1
1998 Hanessian S, Huynh HK, Reddy GV, McNaughton-Smith G, Ernst B, Kolb HC, Magnani J, Sweeley C. Exploration of beta-turn scaffolding motifs as components of sialyl Le(X) mimetics and their relevance to P-selectin. Bioorganic & Medicinal Chemistry Letters. 8: 2803-8. PMID 9873626 DOI: 10.1016/S0960-894X(98)00500-9  1
1997 Nelson DW, Gypser A, Ho PT, Kolb HC, Kondo T, Kwong HL, McGrath DV, Rubin AE, Norrby PO, Gable KP, Sharpless KB. Toward an understanding of the high enantioselectivity in the osmium-catalyzed asymmetric dihydroxylation. 4. Electronic effects in amine-accelerated osmylations Journal of the American Chemical Society. 119: 1840-1858. DOI: 10.1021/ja961464t  1
1997 Hanessian S, Reddy GV, Huynh HK, Jingwen P, Pedatella S, Ernst B, Kolb HC. Design and synthesis of sialyl Le(x) mimetics based on carbocyclic scaffolds derived from (-)-quinic acid Bioorganic and Medicinal Chemistry Letters. 7: 2729-2734. DOI: 10.1016/S0960-894X(97)10077-4  1
1997 Kolb HC. Design and synthesis of a macrocyclic E-selectin antagonist Bioorganic and Medicinal Chemistry Letters. 7: 2629-2634. DOI: 10.1016/S0960-894X(97)10041-5  1
1997 Norcross RD, Von Matt P, Kolb HC, Belluš D. Synthesis of novel cyclobutylphosphonic acids as inhibitors of imidazole glycerol phosphate dehydratase Tetrahedron. 53: 10289-10312. DOI: 10.1016/S0040-4020(97)00682-0  1
1997 Jahnke W, Kolb HC, Blommers MJJ, Magnani JL, Ernst B. Comparison of the bioactive conformations of sialyl Lewis(x) and a potent sialyl Lewis(x) mimic Angewandte Chemie - International Edition in English. 36: 2603-2607.  1
1997 Kolb HC, Ernst B. Development of tools for the design of selectin antagonists Chemistry - a European Journal. 3: 1571-1578.  1
1997 Kolb HC, Ernst B. Recent progress in the glycodrug area Pure and Applied Chemistry. 69: 1879-1884.  1
1994 Norrby PO, Kolb HC, Sharpless KB. Calculations on the reaction of ruthenium tetroxide with olefins using density functional theory (DFT). Implications for the possibility of intermediates in osmium-catalyzed asymmetric dihydroxylation Organometallics. 13: 344-347. DOI: 10.1021/om00013a050  1
1994 Wang Z, Kolb HC, Sharpless KB. Large-Scale and Highly Enantioselective Synthesis of the Taxol C-13 Side Chain through Asymmetric Dihydroxylation The Journal of Organic Chemistry. 59: 5104-5105. DOI: 10.1021/jo00096a072  1
1994 Norrby P, Kolb HC, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation. 2. A Qualitative Molecular Mechanics Approach Journal of the American Chemical Society. 116: 8470-8478. DOI: 10.1021/ja00098a006  1
1994 Kolb HC, Andersson PG, Sharpless KB. Toward an Understanding of the High Enantioselectivity in the Osmium-Catalyzed Asymmetric Dihydroxylation (AD). 1. Kinetics Journal of the American Chemical Society. 116: 1278-1291. DOI: 10.1021/ja00083a014  1
1994 Kolb HC, VanNieuwenhze MS, Sharpless KB. Catalytic Asymmetric Dihydroxylation Chemical Reviews. 94: 2483-2547. DOI: 10.1021/cr00032a009  1
1994 Becker H, Tong Ho P, Kolb HC, Loren S, Norrby PO, Sharpless KB. Comparing two models for the selectivity in the asymmetric dihydroxylation reaction (AD) Tetrahedron Letters. 35: 7315-7318. DOI: 10.1016/0040-4039(94)85302-9  1
1994 Norrby PO, Kolb HC, Sharpless KB. Calculations on the reaction of ruthenium tetraoxide with olefins using density functional theory (DFT). Implications for the possibility of intermediates in the osmium-catalyzed asymmetric dihydroxylation (AD) Organometallics. 13: 344-347.  1
1994 Kolb HC, VanNieuwenhze MS, Sharpless KB. Catalytic asymmetric dihydroxylation Chemical Reviews. 94: 2483-2547.  1
1994 Wang ZM, Kolb HC, Sharpless KB. Large-scale and highly enantioselective synthesis of the taxol C-13 side chain through asymmetric dihydroxylation Journal of Organic Chemistry. 59: 5104-5105.  1
1994 Norrby PO, Kolb HC, Sharpless KB. Toward an understanding of the high enantioselectivity in the osmium-catalyzed asymmetric dihydroxylation. 2. A qualitative molecular mechanics approach Journal of the American Chemical Society. 116: 8470-8478.  1
1994 Kolb HC, Andersson PG, Sharpless KB. Toward an understanding of the high enantioselectivity in the osmium-catalyzed asymmetric dihydroxylation (AD). 1. Kinetics Journal of the American Chemical Society. 116: 1278-1291.  1
1993 Kolb HC, Andersson PG, Bennani YL, Crispino GA, Jeong KS, Kwong HL, Sharpless KB. On "The origin of high enantioselectivity in the dihydroxylation of olefins using osmium tetraoxide and cinchona alkaloid catalysts" Journal of the American Chemical Society. 115: 12226-12227. DOI: 10.1021/ja00078a096  1
1993 Kolb HC, Bennani YL, Sharpless KB. Short and practical syntheses of(R)-(-)-carnitine and (R)-(-)-γ-amino-β-hydroxybutyric acid (GABOB) Tetrahedron: Asymmetry. 4: 133-141. DOI: 10.1016/S0957-4166(00)86023-1  1
1993 Crispino GA, Jeong KS, Kolb HC, Wang ZM, Xu D, Barry Sharpless K. Improved enantioselectivity in asymmetric dihydroxylations of terminal olefins using pyrimidine ligands Journal of Organic Chemistry. 58: 3785-3786.  1
1993 Kolb HC, Andersson PG, Bennani YL, Crispino GA, Jeong KS, Kwong HL, Sharpless KB. On "the origin of high enantioselectivity in the dihydroxylation of olefins using osmium tetraoxide and cinchona alkaloid catalysts" Journal of the American Chemical Society. 115: 12226-12227.  1
1992 Kolb HC, Ley SV, Sheppard RN, Slawin AMZ, Smith SC, Williams DJ, Wood A. Chemistry of insect antifeedants from azadirachta indica (Part 13): On the use of the intramolecular diels-alder reaction for the construction of trans-fused hydrobenzofuran fragments for azadirachtin synthesis Journal of the Chemical Society, Perkin Transactions 1. 2763-2777. DOI: 10.1039/P19920002763  1
1992 Kolb HC, Ley SV, Slawin AMZ, Williams DJ. Chemistry of insect antifeedants from azadirachta indica (Part 12): Use of silicon as a control element in the synthesis of a highly functionalized decalin fragment of azadirachtin Journal of the Chemical Society, Perkin Transactions 1. 2735-2762. DOI: 10.1039/P19920002735  1
1992 Kolb HC, Sharpless KB. A simplified procedure for the stereospecific transformation of 1,2-diols into epoxides Tetrahedron. 48: 10515-10530. DOI: 10.1016/S0040-4020(01)88349-6  1
1991 Kolb HC, Ley SV. Chemistry of insect antifeedants from Azadirachta indica (Part 10): synthesis of a highly functionalised decalin fragment of azadirachtin Tetrahedron Letters. 32: 6187-6190. DOI: 10.1016/0040-4039(91)80785-5  1
1991 Ley SV, Armstrong A, Díez-Martín D, Ford MJ, Grice P, Knight JG, Kolb HC, Madin A, Marby CA, Mukherjee S, Shaw AN, Slawin AMZ, Vile S, White AD, Williams DJ, et al. Total synthesis of the anthelmintic macrolide avermectin B1a Journal of the Chemical Society, Perkin Transactions 1. 667-692.  1
1990 Kolb HC, Martin H, Hoffmann R. A total synthesis of racemic and optically active terrein (trans-4,5-dihydroxy-3-[(E)-1-propenyl]-2-cyclopenten-1-one) Tetrahedron: Asymmetry. 1: 237-250. DOI: 10.1016/S0957-4166(00)86329-6  1
1990 Diez-Martin D, Grice P, Kolb HC, Ley SV, Madin A. Synthesis of a C16-C28 spiroacetal fragment of avermectin B1a and reassignment of some 1H and 13C resonances of avermectin B1a Tetrahedron Letters. 31: 3445-3448. DOI: 10.1016/S0040-4039(00)97418-5  1
1990 Kolb HC, Hoffmann HMR. A ring contraction of 6-alkoxy-2,3-dihydro-6h-pyran-3-ones to polyfunctionalized cyclopentenones Tetrahedron. 46: 5127-5144. DOI: 10.1016/S0040-4020(01)87820-0  1
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