| Year |
Citation |
Score |
| 2024 |
Banoo R, Nuthakki VK, Wadje BN, Sharma A, Bharate SB. Design, synthesis, and pharmacological evaluation of indole-piperidine amides as Blood-brain barrier permeable dual cholinesterase and β-secretase inhibitors. European Journal of Medicinal Chemistry. 266: 116131. PMID 38215587 DOI: 10.1016/j.ejmech.2024.116131 |
0.7 |
|
| 2023 |
Sharma M, Sharma A, Thakur S, Nuthakki VK, Jamwal A, Nandi U, Jadhav HR, Bharate SB. Discovery of blood-brain barrier permeable and orally bioavailable caffeine-based amide derivatives as acetylcholinesterase inhibitors. Bioorganic Chemistry. 139: 106719. PMID 37473478 DOI: 10.1016/j.bioorg.2023.106719 |
0.779 |
|
| 2023 |
Sharma A, Bharate SB. Synthesis and Biological Evaluation of Coumarin Triazoles as Dual Inhibitors of Cholinesterases and β-Secretase. Acs Omega. 8: 11161-11176. PMID 37008108 DOI: 10.1021/acsomega.2c07993 |
0.657 |
|
| 2023 |
Nuthakki VK, Choudhary S, Reddy CN, Bhatt S, Jamwal A, Jotshi A, Raghuvanshi R, Sharma A, Thakur S, Jadhav HR, Bharate SS, Nandi U, Kumar A, Bharate SB. Design, Synthesis, and Pharmacological Evaluation of Embelin-Aryl/alkyl Amine Hybrids as Orally Bioavailable Blood-Brain Barrier Permeable Multitargeted Agents with Therapeutic Potential in Alzheimer's Disease: Discovery of SB-1448. Acs Chemical Neuroscience. 14: 1193-1219. PMID 36812360 DOI: 10.1021/acschemneuro.3c00030 |
0.726 |
|
| 2022 |
Sharma M, Sharma A, Nuthakki VK, Bhatt S, Nandi U, Bharate SB. Design, synthesis, and structure-activity relationship of caffeine-based triazoles as dual AChE and BACE-1 inhibitors. Drug Development Research. PMID 36161804 DOI: 10.1002/ddr.21998 |
0.798 |
|
| 2022 |
Sharma A, Nuthakki VK, Gairola S, Singh B, Bharate SB. A Coumarin-donepezil Hybrid as a Blood-brain Barrier Permeable Dual Cholinesterase Inhibitor: Isolation, Synthetic Modifications and Biological Evaluation of Natural Coumarins. Chemmedchem. PMID 35892288 DOI: 10.1002/cmdc.202200300 |
0.798 |
|
| 2021 |
Ali M, Gupta M, Wani A, Sharma A, Abdullaha M, Kour D, Choudhary S, Bharate SB, Singh G, Kumar A. IIIM-941, a Stilbene Derivative Inhibits NLRP3 Inflammasome Activation by Inducing Autophagy. Frontiers in Pharmacology. 12: 695712. PMID 34248643 DOI: 10.3389/fphar.2021.695712 |
0.653 |
|
| 2021 |
Wani A, Al Rihani SB, Sharma A, Weadick B, Govindarajan R, Khan SU, Sharma PR, Dogra A, Nandi U, Reddy CN, Bharate SS, Singh G, Bharate SB, Vishwakarma RA, Kaddoumi A, et al. Crocetin promotes clearance of amyloid-β by inducing autophagy via the STK11/LKB1-mediated AMPK pathway. Autophagy. PMID 33404280 DOI: 10.1080/15548627.2021.1872187 |
0.572 |
|
| 2020 |
Sharma V, Sharma A, Bharate SB. Natural Products in Mitigation of SARS CoV Infections. Current Medicinal Chemistry. PMID 33109028 DOI: 10.2174/0929867327666201027153940 |
0.456 |
|
| 2019 |
Derf A, Sharma A, Bharate SB, Chaudhuri B. Corrigendum to "Aegeline, a natural product from the plant Aegle marmelos, mimics the yeast SNARE protein Sec22p in suppressing α-synuclein and Bax toxicity in yeast" [Bioorg. Med. Chem. Lett. 29 (2019) 454-460]. Bioorganic & Medicinal Chemistry Letters. PMID 31281017 DOI: 10.1016/j.bmcl.2019.06.053 |
0.447 |
|
| 2019 |
Nuthakki VK, Mudududdla R, Sharma A, Kumar A, Bharate SB. Synthesis and biological evaluation of indoloquinoline alkaloid cryptolepine and its bromo-derivative as dual cholinesterase inhibitors. Bioorganic Chemistry. 90: 103062. PMID 31220673 DOI: 10.1016/j.bioorg.2019.103062 |
0.77 |
|
| 2019 |
Nuthakki VK, Sharma A, Kumar A, Bharate SB. Identification of embelin, a 3-undecyl-1,4-benzoquinone from Embelia ribes as a multitargeted anti-Alzheimer agent. Drug Development Research. PMID 31050027 DOI: 10.1002/ddr.21544 |
0.795 |
|
| 2018 |
Kumar V, Bhurta D, Sharma A, Kumar P, Bharate SB, Vishwakarma RA, Bharate SS. Impurity profiling of anticancer preclinical candidate, IIIM-290. Journal of Pharmaceutical and Biomedical Analysis. 166: 1-5. PMID 30590350 DOI: 10.1016/J.Jpba.2018.12.027 |
0.705 |
|
| 2018 |
Derf A, Sharma A, Bharate SB, Chaudhuri B. Aegeline, a natural product from the plant Aegle marmelos, mimics the yeast SNARE protein Sec22p in suppressing α-synuclein and Bax toxicity in yeast. Bioorganic & Medicinal Chemistry Letters. PMID 30579794 DOI: 10.1016/j.bmcl.2018.12.028 |
0.633 |
|
| 2016 |
Sharma M, Areendran G, Raj K, Sharma A, Joshi PK. Multitemporal analysis of forest fragmentation in Hindu Kush Himalaya-a case study from Khangchendzonga Biosphere Reserve, Sikkim, India. Environmental Monitoring and Assessment. 188: 596. PMID 27687183 DOI: 10.1007/s10661-016-5577-8 |
0.404 |
|
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