Year |
Citation |
Score |
2024 |
Glennon RA, Dukat M. 1-(2,5-Dimethoxy-4-iodophenyl)-2-aminopropane (DOI): From an Obscure to Pivotal Member of the DOX Family of Serotonergic Psychedelic Agents - A Review. Acs Pharmacology & Translational Science. 7: 1722-1745. PMID 38898956 DOI: 10.1021/acsptsci.4c00157 |
0.419 |
|
2023 |
Hemanth P, Nistala P, Nguyen VT, Eltit JM, Glennon RA, Dukat M. Binding and functional structure-activity similarities of 4-substituted 2,5-dimethoxyphenyl isopropylamine analogues at 5-HT and 5-HT serotonin receptors. Frontiers in Pharmacology. 14: 1101290. PMID 36762110 DOI: 10.3389/fphar.2023.1101290 |
0.426 |
|
2021 |
Alwassil OI, Abdrakhmanova GR, Dukat M. Computational analysis of non-competitive antagonist arylguanidine-α7 nAChR complexes. Journal of Molecular Graphics & Modelling. 107: 107943. PMID 34058639 DOI: 10.1016/j.jmgm.2021.107943 |
0.712 |
|
2021 |
Alwassil OI, Khatri S, Schulte MK, Aripaka SS, Mikkelsen JD, Dukat M. NH- and N-Substituted Phenylguanidines as α7 Nicotinic Acetylcholine (nACh) Receptor Antagonists: Structure-Activity Relationship Studies. Acs Chemical Neuroscience. PMID 34043311 DOI: 10.1021/acschemneuro.1c00212 |
0.72 |
|
2021 |
de la Fuente Revenga M, Shah UH, Nassehi N, Jaster AM, Hemanth P, Sierra S, Dukat M, González-Maeso J. Psychedelic-like Properties of Quipazine and Its Structural Analogues in Mice. Acs Chemical Neuroscience. 12: 831-844. PMID 33400504 DOI: 10.1021/acschemneuro.0c00291 |
0.301 |
|
2020 |
Abdelkhalek AS, Musayev FN, Iyer KA, Hemanth P, Safo MK, Dukat M. X-Ray Crystal Structure of a 2-Amino-3,4-dihydroquinazoline 5-HT Serotonin Receptor Antagonist and Related Analogs. Journal of Molecular Structure. 1202. PMID 32616964 DOI: 10.1016/j.molstruc.2019.127276 |
0.756 |
|
2019 |
Iyer KA, Alix K, Eltit JM, Solis E, Pan X, Argade MD, Khatri S, De Felice LJ, Sweet DH, Schulte MK, Dukat M. Multi-modal antidepressant-like action of 6- and 7-chloro-2-aminodihydroquinazolines in the mouse tail suspension test. Psychopharmacology. PMID 30805668 DOI: 10.1007/S00213-019-05203-5 |
0.616 |
|
2019 |
Shah UH, Gaitonde SA, Moreno JL, Glennon RA, Dukat M, González-Maeso J. A revised pharmacophore model for 5-HT2A receptor antagonists derived from the atypical antipsychotic agent risperidone. Acs Chemical Neuroscience. PMID 30609893 DOI: 10.1021/Acschemneuro.8B00637 |
0.459 |
|
2018 |
Abdelkhalek AS, Alley GS, Alwassil OI, Khatri S, Mosier PD, Nyce HL, White MM, Schulte MK, Dukat M. "Methylene Bridge" to 5-HT3 Receptor Antagonists: Conformationally-Constrained Phenylguanidines". Acs Chemical Neuroscience. PMID 30375852 DOI: 10.1021/Acschemneuro.8B00431 |
0.764 |
|
2018 |
Dukat M, Jain AD, German N, Ferrara-Pontoriero R, Huang Y, Ma Y, Schulte MK, Glennon RA. des-Formylflustrabromine (dFBr): A Structure-Activity Study on its Ability to Potentiate the Action of Acetylcholine at α4β2 Nicotinic Acetylcholine Receptors. Acs Chemical Neuroscience. PMID 30028943 DOI: 10.1021/Acschemneuro.8B00156 |
0.354 |
|
2017 |
Pan X, Iyer KA, Liu H, Sweet DH, Dukat M. A new chemotype inhibitor for the human organic cation transporter 3 (hOCT3). Bioorganic & Medicinal Chemistry Letters. PMID 28811134 DOI: 10.1016/J.Bmcl.2017.08.008 |
0.715 |
|
2017 |
Sguazzini E, Schmidt HR, Iyer KA, Kruse AC, Dukat M. Reevaluation of fenpropimorph as a σ receptor ligand: Structure-affinity relationship studies at human σ1 receptors. Bioorganic & Medicinal Chemistry Letters. 27: 2912-2919. PMID 28495085 DOI: 10.1016/j.bmcl.2017.04.088 |
0.734 |
|
2016 |
Glennon RA, Dukat M. Structure-Activity Relationships of Synthetic Cathinones. Current Topics in Behavioral Neurosciences. PMID 27830576 DOI: 10.1007/7854_2016_41 |
0.304 |
|
2016 |
Alix K, Khatri S, Mosier PD, Casterlow S, Yan D, Nyce HL, White MM, Schulte MK, Dukat M. Super-agonist, full agonist, partial agonist and antagonist actions of arylguanidines at h5-HT3A receptors. Acs Chemical Neuroscience. PMID 27533595 DOI: 10.1021/Acschemneuro.6B00196 |
0.456 |
|
2016 |
Younkin J, Gaitonde SA, Ellaithy A, Vekariya RH, Baki L, Moreno JL, Shah S, Drossopoulos P, Hideshima KS, Eltit JM, González-Maeso J, Logothetis DE, Dukat M, Glennon RA. Reformulating a Pharmacophore for 5-HT2A Serotonin Receptor Antagonists. Acs Chemical Neuroscience. PMID 27385190 DOI: 10.1021/Acschemneuro.6B00162 |
0.454 |
|
2014 |
Rao BK, Samanta D, Joshi S, Basu K, Baldwin SD, Jha A, Dukat M, Glennon RA, Jena P. Receptor-ligand interaction at 5-HT3 serotonin receptors: a cluster approach. The Journal of Physical Chemistry. A. 118: 8471-6. PMID 24878072 DOI: 10.1021/Jp5017906 |
0.391 |
|
2013 |
Dukat M, Alix K, Worsham J, Khatri S, Schulte MK. 2-Amino-6-chloro-3,4-dihydroquinazoline: A novel 5-HT3 receptor antagonist with antidepressant character. Bioorganic & Medicinal Chemistry Letters. 23: 5945-8. PMID 24035337 DOI: 10.1016/J.Bmcl.2013.08.072 |
0.482 |
|
2012 |
Rahman AA, Daoud MK, Dukat M, Herrick-Davis K, Purohit A, Teitler M, do Amaral AT, Malvezzi A, Glennon RA. Corrigendum to “Conformationally-restricted analogues and partition coefficients of the 5-HT3 serotonin receptor ligands meta-Chlorophenylbiguanide (mCPBG) and meta-Chlorophenylguanidine (mCPG)” [Bioorg. Med. Chem. Lett. 15 (2005) 3434–3438] Bioorganic & Medicinal Chemistry Letters. 22: 6526. DOI: 10.1016/J.Bmcl.2012.08.076 |
0.35 |
|
2011 |
German N, Kim JS, Jain A, Dukat M, Pandya A, Ma Y, Weltzin M, Schulte MK, Glennon RA. Deconstruction of the α4β2 nicotinic acetylcholine receptor positive allosteric modulator desformylflustrabromine Journal of Medicinal Chemistry. 54: 7259-7267. PMID 21905680 DOI: 10.1021/Jm200834X |
0.358 |
|
2011 |
Klein MT, Dukat M, Glennon RA, Teitler M. Toward selective drug development for the human 5-hydroxytryptamine 1E receptor: a comparison of 5-hydroxytryptamine 1E and 1F receptor structure-affinity relationships. The Journal of Pharmacology and Experimental Therapeutics. 337: 860-7. PMID 21422162 DOI: 10.1124/Jpet.111.179606 |
0.496 |
|
2010 |
Glennon RA, Siripurapu U, Roth BL, Kolanos R, Bondarev ML, Sikazwe D, Lee M, Dukat M. The medicinal chemistry of 5-HT6 receptor ligands with a focus on arylsulfonyltryptamine analogs. Current Topics in Medicinal Chemistry. 10: 579-95. PMID 20166945 DOI: 10.2174/156802610791111542 |
0.516 |
|
2010 |
Glennon RA, Lee M, Rangisetty JB, Dukat M, Roth BL, Savage JE, McBride A, Rauser L, Hufeisen S, Lee DKH. ChemInform Abstract: 2-Substituted Tryptamines: Agents with Selectivity for 5-HT6 Serotonin Receptors. Cheminform. 31: no-no. DOI: 10.1002/CHIN.200023120 |
0.423 |
|
2010 |
HONG S, DUKAT M, TEITLER M, HERRICK-DAVIS K, MCCALLUM K, KAMBOJ R, GLENNON RA. ChemInform Abstract: Binding of 5-Arylalkyloxytryptamines at Human 5-HT1Dβ Serotonin Receptors. Cheminform. 27: no-no. DOI: 10.1002/CHIN.199621126 |
0.395 |
|
2010 |
DUKAT M, DAMAJ MI, GLASSCO W, DUMAS D, MAY EL, MARTIN BR, GLENNON RA. ChemInform Abstract: Epibatidine: A Very High Affinity Nicotine-Receptor Ligand. Cheminform. 26: no-no. DOI: 10.1002/chin.199513270 |
0.317 |
|
2008 |
Dukat M, Mosier PD, Kolanos R, Roth BL, Glennon RA. Binding of serotonin and N1-benzenesulfonyltryptamine-related analogs at human 5-HT6 serotonin receptors: receptor modeling studies. Journal of Medicinal Chemistry. 51: 603-11. PMID 18201064 DOI: 10.1021/Jm070910S |
0.464 |
|
2007 |
Dukat M, Glennon RA, Young S. MD-354: What is it good for? Cns Drug Reviews. 13: 1-20. PMID 17461887 DOI: 10.1111/J.1527-3458.2007.00002.X |
0.445 |
|
2006 |
Kolanos R, Dukat M, Roth BL, Glennon RA. Interaction of N1-unsubstituted and N1-benzenesulfonyltryptamines at h5-HT6 receptors. Bioorganic & Medicinal Chemistry Letters. 16: 5832-5. PMID 16945532 DOI: 10.1016/J.Bmcl.2006.08.068 |
0.43 |
|
2006 |
Sikazwe D, Bondarev ML, Dukat M, Rangisetty JB, Roth BL, Glennon RA. Binding of sulfonyl-containing arylalkylamines at human 5-HT6 serotonin receptors. Journal of Medicinal Chemistry. 49: 5217-25. PMID 16913710 DOI: 10.1021/Jm060469Q |
0.482 |
|
2006 |
Ragab HM, Kim JS, Dukat M, Navarro H, Glennon RA. Aryloxyethylamines: Binding at α7 nicotinic acetylcholine receptors Bioorganic and Medicinal Chemistry Letters. 16: 4283-4286. PMID 16765047 DOI: 10.1016/J.Bmcl.2006.05.080 |
0.338 |
|
2006 |
Siripurapu U, Kolanos R, Dukat M, Roth BL, Glennon RA. Binding of methoxy-substituted N1-benzenesulfonylindole analogs at human 5-HT6 serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 16: 3793-6. PMID 16709453 DOI: 10.1016/J.Bmcl.2006.04.094 |
0.47 |
|
2005 |
Pullagurla M, Siripurapu U, Kolanos R, Bondarev ML, Dukat M, Setola V, Roth BL, Glennon RA. Binding of amine-substituted N1-benzenesulfonylindoles at human 5-HT6 serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 15: 5298-302. PMID 16183286 DOI: 10.1016/J.Bmcl.2005.08.059 |
0.457 |
|
2005 |
Abate C, Kolanos R, Dukat M, Setola V, Roth BL, Glennon RA. Interaction of chiral MS-245 analogs at h5-HT6 receptors. Bioorganic & Medicinal Chemistry Letters. 15: 3510-3. PMID 15990303 DOI: 10.1016/J.Bmcl.2005.05.092 |
0.392 |
|
2005 |
Setola V, Dukat M, Glennon RA, Roth BL. Molecular determinants for the interaction of the valvulopathic anorexigen norfenfluramine with the 5-HT2B receptor. Molecular Pharmacology. 68: 20-33. PMID 15831837 DOI: 10.1124/Mol.104.009266 |
0.407 |
|
2005 |
Kolanos R, Siripurapu U, Pullagurla M, Riaz M, Setola V, Roth BL, Dukat M, Glennon RA. Binding of isotryptamines and indenes at h5-HT6 serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 15: 1987-91. PMID 15808453 DOI: 10.1016/J.Bmcl.2005.02.070 |
0.366 |
|
2005 |
Lee M, Rangisetty JB, Pullagurla MR, Dukat M, Setola V, Roth BL, Glennon RA. 1-(1-Naphthyl)piperazine as a novel template for 5-HT6 serotonin receptor ligands. Bioorganic & Medicinal Chemistry Letters. 15: 1707-11. PMID 15745826 DOI: 10.1016/J.Bmcl.2005.01.031 |
0.443 |
|
2005 |
Pullagurla M, Dukat M, Roth BL, Setola V, Glennon RA. 5-Azatryptamine analogs as h5-HT6 serotonin receptor ligands Medicinal Chemistry Research. 14: 1-18. DOI: 10.1007/S00044-004-0121-8 |
0.452 |
|
2005 |
Lee M, Rangisetty JB, Pullagurla MR, Dukat M, Setola V, Roth BL, Glennon RA. 1-(1-Naphthyl)piperazine as a Novel Template for 5-HT6 Serotonin Receptor Ligands. Cheminform. 36. DOI: 10.1002/CHIN.200529171 |
0.42 |
|
2004 |
Prisinzano T, Dukat M, Law H, Slassi A, MacLean N, DeLannoy I, Glennon RA. 2-(Anilino)imidazolines and 2-(benzyl)imidazoline derivatives as h5-HT 1D serotonin receptor ligands Bioorganic and Medicinal Chemistry Letters. 14: 4697-4699. PMID 15324890 DOI: 10.1016/J.Bmcl.2004.06.085 |
0.406 |
|
2004 |
Shelton KL, Dukat M, Allan AM. Effect of 5-HT3 receptor over-expression on the discriminative stimulus effects of ethanol. Alcoholism, Clinical and Experimental Research. 28: 1161-71. PMID 15318114 DOI: 10.1097/01.ALC.0000138687.27452.E2 |
0.362 |
|
2004 |
Dukat M, Taroua M, Dahdouh A, Siripurapu U, Damaj MI, Martin BR, Glennon RA. (+/-)8-Amino-5,6,7,8-tetrahydroisoquinolines as novel antinociceptive agents. Bioorganic & Medicinal Chemistry Letters. 14: 3651-4. PMID 15203136 DOI: 10.1016/J.Bmcl.2004.05.020 |
0.316 |
|
2004 |
Dukat M, Smith C, Herrick-Davis K, Teitler M, Glennon RA. Binding of tryptamine analogs at h5-HT1E receptors: A structure-affinity investigation Bioorganic and Medicinal Chemistry. 12: 2545-2552. PMID 15110837 DOI: 10.1016/J.Bmc.2004.03.026 |
0.451 |
|
2004 |
Chang-Fong J, Rangisetty JB, Dukat M, Setola V, Raffay T, Roth B, Glennon RA. 1,2,3,4-Tetrahydrocarbazoles as 5-HT6 serotonin receptor ligands Bioorganic and Medicinal Chemistry Letters. 14: 1961-1964. PMID 15050637 DOI: 10.1016/J.Bmcl.2004.01.071 |
0.438 |
|
2004 |
Glennon RA, Dukat M, Liao L. Musings on alpha4beta2 nicotinic acetylcholine (nACh) receptor pharmacophore models. Current Topics in Medicinal Chemistry. 4: 631-44. PMID 14965299 DOI: 10.2174/1568026043451122 |
0.335 |
|
2004 |
Dogruer D, Lee M, Dukat M, Damaj MI, Martin BR, Glennon RA. 3-(4-Aminobutyn-1-yl)pyridines: binding at alpha 4 beta 2 nicotinic cholinergic receptors. Bioorganic & Medicinal Chemistry Letters. 14: 523-6. PMID 14698195 DOI: 10.1016/J.Bmcl.2003.10.033 |
0.34 |
|
2004 |
Dukat M. 5-HT3 Serotonin Receptor Agonists: A Pharmacophoric Journey Current Medicinal Chemistry-Central Nervous System Agents. 4: 77-94. DOI: 10.2174/1568015043356995 |
0.433 |
|
2004 |
Chang-Fong J, Rangisetty JB, Dukat M, Setola V, Raffay T, Roth B, Glennon RA. 1,2,3,4-Tetrahydrocarbazoles as 5-HT6 Serotonin Receptor Ligands. Cheminform. 35. DOI: 10.1002/CHIN.200431116 |
0.411 |
|
2004 |
Pullagurla MR, Dukat M, Setola V, Roth B, Glennon RA. N1-Benzenesulfonylgramine (I) and N1-Benzenesulfonylskatole (II): Novel 5-HT6 Receptor Ligand Templates. Cheminform. 35. DOI: 10.1002/chin.200401186 |
0.368 |
|
2003 |
Simsek R, Chang-Fong J, Lee M, Dukat M, Imad Damaj M, Martin BR, Glennon RA. Quaternary ammonium 3-(aminoethoxy)pyridines as antinociceptive agents. Bioorganic & Medicinal Chemistry Letters. 13: 2917-20. PMID 14611857 DOI: 10.1016/S0960-894X(03)00585-7 |
0.32 |
|
2003 |
Glennon RA, Daoud MK, Dukat MS, Teitler M, Herrick-Davis K, Purohit A, Syed H. Arylguanidine and arylbiguanide binding at 5-HT3 serotonin receptors: A QSAR study Bioorganic and Medicinal Chemistry. 11: 4449-4454. PMID 13129581 DOI: 10.1016/S0968-0896(03)00488-7 |
0.471 |
|
2003 |
Pullagurla MR, Dukat M, Setola V, Roth B, Glennon RA. N1-benzenesulfonylgramine and N1-benzenesulfonylskatole: novel 5-HT6 receptor ligand templates. Bioorganic & Medicinal Chemistry Letters. 13: 3355-9. PMID 12951125 DOI: 10.1016/S0960-894X(03)00612-7 |
0.408 |
|
2003 |
Khorana N, Smith C, Herrick-Davis K, Purohit A, Teitler M, Grella B, Dukat M, Glennon RA. Binding of tetrahydrocarboline derivatives at human 5-HT5A receptors. Journal of Medicinal Chemistry. 46: 3930-7. PMID 12930153 DOI: 10.1021/Jm030080S |
0.42 |
|
2003 |
Rahman AA, Daoud MK, Dukat M, Herrick-Davis K, Purohit A, Teitler M, do Amaral AT, Malvezzi A, Glennon RA. Conformationally-restricted analogues and partition coefficients of the 5-HT3 serotonin receptor ligands meta-chlorophenylbiguanide (mCPBG) and meta-chlorophenylguanidine (mCPG). Bioorganic & Medicinal Chemistry Letters. 13: 1119-23. PMID 12643925 DOI: 10.1016/S0960-894X(03)00044-1 |
0.35 |
|
2002 |
Ferretti G, Dukat M, Giannella M, Piergentili A, Pigini M, Quaglia W, Damaj MI, Martin BR, Glennon RA. Homoazanicotine: a structure-affinity study for nicotinic acetylcholine (nACh) receptor binding. Journal of Medicinal Chemistry. 45: 4724-31. PMID 12361399 DOI: 10.1021/Jm020188S |
0.368 |
|
2002 |
Glennon RA, Metwally K, Dukat M, Ismaiel AM, De los Angeles J, Herndon J, Teitler M, Khorana N. Ketanserin and spiperone as templates for novel serotonin 5-HT(2A) antagonists. Current Topics in Medicinal Chemistry. 2: 539-58. PMID 12052193 DOI: 10.2174/1568026023393787 |
0.422 |
|
2002 |
Chang-Fong J, Addo J, Dukat M, Smith C, Mitchell NA, Herrick-Davis K, Teitler M, Glennon RA. Evaluation of isotryptamine derivatives at 5-HT(2) serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 12: 155-8. PMID 11755343 DOI: 10.1016/S0960-894X(01)00713-2 |
0.432 |
|
2001 |
Rangisetty JB, Dukat M, Dowd CS, Herrick-Davis K, DuPre A, Gadepalli S, Teitler M, Kelley CR, Sharif NA, Glennon RA. 1-[2-methoxy-5-(3-phenylpropyl)]-2-aminopropane unexpectedly shows 5-HT(2A) serotonin receptor affinity and antagonist character. Journal of Medicinal Chemistry. 44: 3283-91. PMID 11563927 DOI: 10.1021/Jm0100739 |
0.432 |
|
2001 |
Dukat M, Choi YN, Teitler M, Du Pre A, Herrick-Davis K, Smith C, Glennon RA. The binding of arylguanidines at 5-HT(3) serotonin receptors: a structure-affinity investigation. Bioorganic & Medicinal Chemistry Letters. 11: 1599-603. PMID 11412989 DOI: 10.1016/S0960-894X(01)00291-8 |
0.457 |
|
2001 |
Prisinzano T, Law H, Dukat M, Slassi A, MaClean N, Demchyshyn L, Glennon RA. Imidazoline-modified benzylimidazolines as h5-HT(1D/1B) serotonergic ligands. Bioorganic & Medicinal Chemistry. 9: 613-9. PMID 11310595 DOI: 10.1016/S0968-0896(00)00275-3 |
0.351 |
|
2001 |
Tsai Y, Dukat M, Slassi A, MacLean N, Demchyshyn L, Savage JE, Roth BL, Hufesein S, Lee M, Glennon RA. ChemInform Abstract: N1-(Benzenesulfonyl)tryptamines as Novel 5-HT6 Antagonists. Cheminform. 32: no-no. DOI: 10.1002/CHIN.200103235 |
0.369 |
|
2000 |
Tsai Y, Dukat M, Slassi A, MacLean N, Demchyshyn L, Savage JE, Roth BL, Hufesein S, Lee M, Glennon RA. N1-(Benzenesulfonyl)tryptamines as novel 5-HT6 antagonists. Bioorganic & Medicinal Chemistry Letters. 10: 2295-9. PMID 11055342 DOI: 10.1016/S0960-894X(00)00453-4 |
0.423 |
|
2000 |
Glennon RA, Dukat M, Grella B, Hong SS, Costantino L, Teitler M, Smith C, Egan C, Davis K, Mattson MV. Binding of β-carbolines and related agents at serotonin (5-HT2 and 5- HT(1A)), dopamine (D2) and benzodiazepine receptors Drug and Alcohol Dependence. 60: 121-132. PMID 10940539 DOI: 10.1016/S0376-8716(99)00148-9 |
0.438 |
|
2000 |
Dukat M, Young R, Darmani NN, Ahmed B, Glennon RA. The 5-HT3 agent N-(3-chlorophenyl)guanidine (MD-354) serves as a discriminative stimulus in rats and displays partial agonist character in a shrew emesis assay Psychopharmacology. 150: 200-207. PMID 10907673 DOI: 10.1007/S002130000410 |
0.4 |
|
2000 |
Glennon RA, Lee M, Rangisetty JB, Dukat M, Roth BL, Savage JE, McBride A, Rauser L, Hufeisen S, Lee DK. 2-Substituted tryptamines: agents with selectivity for 5-HT(6) serotonin receptors. Journal of Medicinal Chemistry. 43: 1011-8. PMID 10715164 DOI: 10.1021/Jm990550B |
0.427 |
|
2000 |
Glennon RA, Dukat M. Central nicotinic receptor ligands and pharmacophores Pharmacochemistry Library. 31: 103-114. DOI: 10.1016/S0031-6865(99)00022-9 |
0.371 |
|
1999 |
Flammia D, Dukat M, Damaj MI, Martin B, Glennon RA. Lobeline: Structure-affinity investigation of nicotinic acetylcholinergic receptor binding Journal of Medicinal Chemistry. 42: 3726-3731. PMID 10479304 DOI: 10.1021/Jm990286M |
0.307 |
|
1999 |
Gyermek L, Sun X, Nguyen N, Dukat M. Is there a functional response-overlap between 5-HT3 and nicotinic ion channel receptors? Annals of the New York Academy of Sciences. 861: 255-7. PMID 9928275 DOI: 10.1111/J.1749-6632.1998.TB10209.X |
0.312 |
|
1999 |
Cheng YX, Dukat M, Dowd M, Fiedler W, Martin B, Damaj MI, Glennon RA. Synthesis and binding of 6,7,8,9-tetrahydro-5H-pyrido[3,4-d]azepine and related ring-opened analogs at central nicotinic receptors European Journal of Medicinal Chemistry. 34: 177-190. DOI: 10.1016/S0223-5234(99)80051-8 |
0.33 |
|
1999 |
Dukat M, Dowd M, Damaj MI, Martin B, El-Zahabi MA, Glennon RA. Synthesis, receptor binding and QSAR studies on 6-substituted nicotine derivatives as cholinergic ligands European Journal of Medicinal Chemistry. 34: 31-40. DOI: 10.1016/S0223-5234(99)80038-5 |
0.32 |
|
1998 |
Metwally KA, Dukat M, Egan CT, Smith C, DuPre A, Gauthier CB, Herrick-Davis K, Teitler M, Glennon RA. Spiperone: Influence of spiro ring substituents on 5-HT(2A) serotonin receptor binding Journal of Medicinal Chemistry. 41: 5084-5093. PMID 9836624 DOI: 10.1021/Jm980452A |
0.476 |
|
1998 |
Law H, Dukat M, Teitler M, Lee DKH, Mazzocco L, Kamboj R, Rampersad V, Prisinzano T, Glennon RA. Benzylimidazolines as h5-HT(1B/1D) serotonin receptor ligands: A structure-affinity investigation Journal of Medicinal Chemistry. 41: 2243-2251. PMID 9632357 DOI: 10.1021/Jm970513P |
0.406 |
|
1997 |
Ismaiel AM, Dukat M, Law H, Kamboj R, Fan E, Lee DKH, Mazzocco L, Buekschkens D, Teitler M, Pierson ME, Glennon RA. 2-(1-naphthyloxy)ethylamines with enhanced affinity for human 5-HT(1Dβ) (h5-HT(1B)) serotonin receptors Journal of Medicinal Chemistry. 40: 4415-4419. PMID 9435911 DOI: 10.1021/Jm970507T |
0.45 |
|
1996 |
Dukat M, Abdel-Rahman AA, Ismaiel AM, Ingher S, Teitler M, Gyermek L, Glennon RA. Structure-activity relationships for the binding of arylpiperazines and arylbiguanides at 5-HT3 serotonin receptors Journal of Medicinal Chemistry. 39: 4017-4026. PMID 8831767 DOI: 10.1021/Jm9603936 |
0.445 |
|
1996 |
Glennon RA, Hong SS, Bondarev M, Law H, Dukat M, Rakhit S, Power P, Fan E, Kinneau D, Kamboj R, Teitler M, Herrick-Davis K, Smith C. Binding of O-alkyl derivatives of serotonin at human 5-HT1Dβ receptors Journal of Medicinal Chemistry. 39: 314-322. PMID 8568822 DOI: 10.1021/Jm950498T |
0.428 |
|
1996 |
Imad Damaj M, Glassco W, Dukat M, May EL, Glennon RA, Martin BR. Pharmacology of novel nicotinic analogs Drug Development Research. 38: 177-187. DOI: 10.1002/(Sici)1098-2299(199607/08)38:3/4<177::Aid-Ddr6>3.0.Co;2-J |
0.317 |
|
1994 |
Glennon RA, Hong SS, Dukat M, Teitler M, Davis K. 5-(Nonyloxy)tryptamine: A novel high-affinity 5-HTIDβ serotonin receptor agonist Journal of Medicinal Chemistry. 37: 2828-2830. PMID 8071931 DOI: 10.1021/Jm00044A001 |
0.439 |
|
1994 |
Glennon RA, Dukat M, El-Bermawy M, Law H, De Los Angeles J, Teitler M, King A, Herrick-Davis K. Influence of amine substituents on 5-HT2A versus 5-HT2C binding of phenylalkyl- and indolylalkylamines Journal of Medicinal Chemistry. 37: 1929-1935. PMID 8027974 DOI: 10.1021/Jm00039A004 |
0.425 |
|
1992 |
Glennon RA, Dukat M. Serotonin receptors and their ligands: a lack of selective agents. Pharmacology, Biochemistry, and Behavior. 40: 1009-17. PMID 1816555 DOI: 10.1016/0091-3057(91)90121-H |
0.403 |
|
1992 |
Glennon RA, Young R, Dukat M. 5-HT3 agonist 2-methylserotonin as a training drug in discrimination studies. Pharmacology, Biochemistry, and Behavior. 41: 361-4. PMID 1574526 DOI: 10.1016/0091-3057(92)90111-R |
0.323 |
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1990 |
MISZTAL S, DUKAT M, MOKROSZ JL. ChemInform Abstract: Structure and Spectral Properties of β-Carbolines. Part 3. Synthesis and Stereochemistry of 1,2,3,4,6,7,9,10,15b,15c-Decahydropyrido(1′′,2′′:1′,2′)pyrazino(4′,3′:1,2)pyrido(3,4-b)indoles. Cheminform. 21. DOI: 10.1002/CHIN.199046227 |
0.575 |
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1990 |
Mokrosz JL, Dukat M, Misztal S. Structure and Spectral Properties of β-Carbolines, I:13C-NMR and Mass Spectra of Decahydro-5H-pyrido[1′,2′;5,1]-imidazo[3,4-a]-β-carbolines Archiv Der Pharmazie. 323: 453-457. DOI: 10.1002/ARDP.19903230803 |
0.577 |
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1986 |
MISZTAL S, DUKAT M. ChemInform Abstract: The threo and erythro Products of the Catalytic Hydrogenation of 1-(2-Pyridyl)- 1,2,3,4-tetrahydro-β-carboline. Chemischer Informationsdienst. 17. DOI: 10.1002/CHIN.198605205 |
0.562 |
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