Roland J. Pieters - Publications

Affiliations: 
2010 Utrecht University, Utrecht, Netherlands 
Website:
https://www.uu.nl/medewerkers/RJPieters

109 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Lu Z, Liu Z, Li X, Qin X, Hong H, Zhou Z, Pieters RJ, Shi J, Wu Z. Nanobody-Based Bispecific Neutralizer for Shiga Toxin-Producing . Acs Infectious Diseases. PMID 35015516 DOI: 10.1021/acsinfecdis.1c00456  1
2021 Asadpoor M, Ithakisiou GN, van Putten JPM, Pieters RJ, Folkerts G, Braber S. Antimicrobial Activities of Alginate and Chitosan Oligosaccharides Against and Group B . Frontiers in Microbiology. 12: 700605. PMID 34589067 DOI: 10.3389/fmicb.2021.700605  1
2021 Martínez-Alarcón D, Balloy V, Bouchara JP, Pieters RJ, Varrot A. Biochemical and structural studies of target lectin SapL1 from the emerging opportunistic microfungus Scedosporium apiospermum. Scientific Reports. 11: 16109. PMID 34373510 DOI: 10.1038/s41598-021-95008-4  0.01
2021 Zaree P, Torano JS, de Haan CAM, Scheltma RA, Barendregt A, Thijssen V, Yu G, Flesch F, Pieters RJ. The assessment of Pseudomonas aeruginosa lectin LecA binding characteristics of divalent galactosides using multiple techniques. Glycobiology. PMID 34255029 DOI: 10.1093/glycob/cwab074  1
2021 Bosman GP, Oliveira S, Simons PJ, Sastre Torano J, Somsen GW, Knippels LMJ, Haselberg R, Pieters RJ, Garssen J, Knipping K. Limited Lactosylation of Beta-Lactoglobulin from Cow's Milk Exerts Strong Influence on Antigenicity and Degranulation of Mast Cells. Nutrients. 13. PMID 34203636 DOI: 10.3390/nu13062041  0.01
2021 Weiss M, Loi EM, Sterle M, Balsollier C, Tomašič T, Pieters RJ, Gobec M, Anderluh M. New Quinolinone O-GlcNAc Transferase Inhibitors Based on Fragment Growth. Frontiers in Chemistry. 9: 666122. PMID 33937202 DOI: 10.3389/fchem.2021.666122  1
2021 Haksar D, Asadpoor M, Heise T, Shi J, Braber S, Folkerts G, Ballell L, Rodrigues J, Pieters RJ. Fighting by Blocking Its Disease-Causing Toxin. Journal of Medicinal Chemistry. PMID 33909975 DOI: 10.1021/acs.jmedchem.1c00152  1
2021 Balsollier C, Pieters RJ, Anderluh M. Overview of the Assays to Probe -Linked β--Acetylglucosamine Transferase Binding and Activity. Molecules (Basel, Switzerland). 26. PMID 33669256 DOI: 10.3390/molecules26041037  1
2020 Shi J, Sharif S, Balsollier C, Ruijtenbeek R, Pieters RJ, Jongkees SAK. C-terminal tag location hampers in vitro profiling of OGT peptide substrates by mRNA display. Chembiochem : a European Journal of Chemical Biology. PMID 33022805 DOI: 10.1002/cbic.202000624  1
2020 Loi EM, Weiss M, Pajk S, Gobec M, Tomašič T, Pieters RJ, Anderluh M. Intracellular Hydrolysis of Small-Molecule -Linked -Acetylglucosamine Transferase Inhibitors Differs among Cells and Is Not Required for Its Inhibition. Molecules (Basel, Switzerland). 25. PMID 32722493 DOI: 10.3390/molecules25153381  1
2020 Steigenberger B, van den Toorn H, Bijl E, Greisch JF, Räther O, Lubeck M, Pieters RJ, Heck AJR, Scheltema RA. Benefits of Collisional Cross Section Assisted Precursor Selection (caps-PASEF) for Cross-linking Mass Spectrometry. Molecular & Cellular Proteomics : McP. PMID 32694122 DOI: 10.1074/Mcp.Ra120.002094  1
2020 Asadpoor M, Peeters C, Henricks PAJ, Varasteh S, Pieters RJ, Folkerts G, Braber S. Anti-Pathogenic Functions of Non-Digestible Oligosaccharides In Vitro. Nutrients. 12. PMID 32560186 DOI: 10.3390/nu12061789  1
2019 Zhang H, Ippel H, Miller MC, Wong TJ, Griffioen AW, Mayo KH, Pieters RJ. Hybrid ligands with calixarene and thiodigalactoside groups: galectin binding and cytotoxicity. Organic Chemistry Frontiers : An International Journal of Organic Chemistry. 6: 2981-2990. PMID 34912566 DOI: 10.1039/c9qo00810a  1
2019 Haksar D, Quarles van Ufford L, Pieters RJ. A hybrid polymer to target blood group dependence of cholera toxin. Organic & Biomolecular Chemistry. 18: 52-55. PMID 31802094 DOI: 10.1039/c9ob02369k  1
2019 Steigenberger B, Pieters RJ, Heck AJR, Scheltema RA. PhoX: An IMAC-Enrichable Cross-Linking Reagent. Acs Central Science. 5: 1514-1522. PMID 31572778 DOI: 10.1021/Acscentsci.9B00416  1
2019 Mahon CS, Wildsmith GC, Haksar D, de Poel E, Beekman JM, Pieters RJ, Webb ME, Turnbull WB. A 'catch-and-release' receptor for the cholera toxin. Faraday Discussions. PMID 31313796 DOI: 10.1039/c9fd00017h  1
2019 Lu W, Du W, Somovilla VJ, Yu G, Haksar D, de Vries E, Boons GJ, de Vries RP, de Haan CAM, Pieters RJ. Enhanced Inhibition of Influenza A Virus Adhesion by Di- and Trivalent Hemagglutinin Inhibitors. Journal of Medicinal Chemistry. PMID 31251606 DOI: 10.1021/Acs.Jmedchem.9B00303  1
2019 Sharif S, Shi J, Ruijtenbeek R, Pieters RJ. Study of cross talk between phosphatases and OGA on a ZO-3-derived peptide. Amino Acids. PMID 30725225 DOI: 10.1007/s00726-019-02699-1  1
2019 Lu W, Pieters RJ. Carbohydrate-protein interactions and multivalency: implications for the inhibition of influenza A virus infections. Expert Opinion On Drug Discovery. 1-9. PMID 30722704 DOI: 10.1080/17460441.2019.1573813  1
2019 Yu G, Vicini AC, Pieters RJ. Assembling of divalent ligands and their Effect on Divalent Binding to Pseudomonas aeruginosa Lectin LecA. The Journal of Organic Chemistry. PMID 30681333 DOI: 10.1021/acs.joc.8b02727  1
2019 Mukherjee R, van de Kaa M, Garssen J, Pieters RJ, Kraneveld AD, Willemsen LEM. Lactulose synergizes with CpG-ODN to modulate epithelial and immune cells cross talk. Food & Function. PMID 30632580 DOI: 10.1039/c8fo02376j  0.01
2019 Haksar D, de Poel E, Quarles van Ufford LHC, Bhatia S, Haag R, Beekman JM, Pieters RJ. Strong inhibition of cholera toxin B subunit by affordable, polymer-based multivalent inhibitors. Bioconjugate Chemistry. PMID 30629410 DOI: 10.1021/Acs.Bioconjchem.8B00902  1
2018 Nemanichvili N, Tomris I, Turner HL, McBride R, Grant OC, van der Woude R, Aldosari MH, Pieters RJ, Woods RJ, Paulson JC, Boons GJ, Ward AB, Verheije MH, de Vries RP. Fluorescent Trimeric Hemagglutinins Reveal Multivalent Receptor Binding Properties. Journal of Molecular Biology. PMID 30597163 DOI: 10.1016/J.Jmb.2018.12.014  1
2018 Zhang H, Tomašič T, Shi J, Weiss M, Ruijtenbeek R, Anderluh M, Pieters RJ. Inhibition of -GlcNAc transferase (OGT) by peptidic hybrids. Medchemcomm. 9: 883-887. PMID 30108977 DOI: 10.1039/c8md00115d  1
2018 Mena-Barragán T, García-Moreno MI, Sevšek A, Okazaki T, Nanba E, Higaki K, Martin NI, Pieters RJ, Fernández JMG, Mellet CO. Probing the Inhibitor versus Chaperone Properties of sp²-Iminosugars towards Human β-Glucocerebrosidase: A Picomolar Chaperone for Gaucher Disease. Molecules (Basel, Switzerland). 23. PMID 29673163 DOI: 10.3390/Molecules23040927  1
2018 Shi J, Ruijtenbeek R, Pieters RJ. Demystifying O-GlcNAcylation: hints from peptide substrates. Glycobiology. PMID 29635275 DOI: 10.1093/glycob/cwy031  1
2018 Zhang H, Laaf D, Elling L, Pieters RJ. Thiodigalactoside-BSA-Conjugates as High-Potency Inhibitors of Ga-lectin-3: An Outstanding Example of Multivalent Presentation of Small Molecule Inhibitors. Bioconjugate Chemistry. PMID 29474087 DOI: 10.1021/acs.bioconjchem.8b00047  1
2018 van Heugten AJP, de Vries WS, Markesteijn MMA, Pieters RJ, Vromans H. The Role of Excipients in the Stability of Triamcinolone Acetonide in Ointments. Aaps Pharmscitech. 19: 1448-1453. PMID 29450828 DOI: 10.1208/s12249-018-0957-8  1
2018 van Heugten AJP, de Boer W, de Vries WS, Pieters RJ, Vromans H. Topically used corticosteroids: What is the big picture of drug product degradation? European Journal of Pharmaceutical Sciences : Official Journal of the European Federation For Pharmaceutical Sciences. PMID 29407556 DOI: 10.1016/j.ejps.2018.02.001  1
2017 Sevšek A, Sastre Toraño J, Quarles van Ufford L, Moret EE, Pieters RJ, Martin NI. Orthoester functionalized -guanidino derivatives of 1,5-dideoxy-1,5-imino-d-xylitol as pH-responsive inhibitors of β-glucocerebrosidase. Medchemcomm. 8: 2050-2054. PMID 30108721 DOI: 10.1039/C7Md00480J  1
2017 Brittoli A, Fallarini S, Zhang H, Pieters RJ, Lombardi G. "In vitro" studies on galectin-3 in human natural killer cells. Immunology Letters. 194: 4-12. PMID 29248489 DOI: 10.1016/j.imlet.2017.12.004  1
2017 Haataja S, Verma P, Fu O, Papageorgiou A, Pöysti S, Pieters R, Nilsson U, Finne J. Rationally designed chemically modified glycodendrimer ligand analogues inhibit Streptococcus suis adhesin SadP in picomolar concentrations. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29094420 DOI: 10.1002/Chem.201704493  1
2017 Aizpurua-Olaizola O, Sastre Torano J, Pukin A, Fu O, Boons GJ, de Jong GJ, Pieters RJ. Affinity capillary electrophoresis for the assessment of binding affinity of carbohydrate-based cholera toxin inhibitors. Electrophoresis. PMID 28905402 DOI: 10.1002/elps.201700207  1
2017 Shi J, Tomašič T, Sharif S, Brouwer AJ, Anderluh M, Ruijtenbeek R, Pieters RJ. Peptide Microarray Analysis of the Cross-talk Between O-GlcNAcylation and Tyrosine Phosphorylation. Febs Letters. PMID 28580691 DOI: 10.1002/1873-3468.12708  1
2017 Sharif S, Shi J, Mostafa B, Ruijtenbeek R, Pieters RJ. Measuring O-GlcNAc cleavage by OGA and cell lysates on a peptide microarray. Analytical Biochemistry. PMID 28571750 DOI: 10.1016/j.ab.2017.05.027  1
2017 Sevšek A, Šrot L, Rihter J, Čelan M, van Ufford LQ, Moret EE, Martin NI, Pieters RJ. N-Guanidino Derivatives of 1,5-Dideoxy-1,5-imino-d-xylitol are Potent, Selective, and Stable Inhibitors of β-Glucocerebrosidase. Chemmedchem. PMID 28328014 DOI: 10.1002/Cmdc.201700050  1
2016 Sevšek A, Čelan M, Erjavec B, Quarles van Ufford L, Sastre Toraño J, Moret EE, Pieters RJ, Martin NI. Bicyclic isoureas derived from 1-deoxynojirimycin are potent inhibitors of β-glucocerebrosidase. Organic & Biomolecular Chemistry. PMID 27604065 DOI: 10.1039/C6Ob01735E  1
2016 Delaine T, Collins P, Mac Kinnon A, Sharma G, Stegmayr J, Rajput VK, Mandal S, Cumpstey I, Larumbe A, Salameh BA, Kahl-Knutsson B, Van Hattum H, Van Scherpenzeel M, Pieters RJ, Sethi T, et al. Galectin-3-binding glycomimetics that strongly reduce bleomycin-induced lung fibrosis and modulate intracellular glycan recognition. Chembiochem : a European Journal of Chemical Biology. PMID 27356186 DOI: 10.1002/Cbic.201600285  1
2016 Zomer-van Ommen DD, Pukin AV, Fu O, Quarles van Ufford LH, Janssens HM, Beekman JM, Pieters RJ. Functional characterization of cholera toxin inhibitors using human intestinal organoids. Journal of Medicinal Chemistry. PMID 27347611 DOI: 10.1021/acs.jmedchem.6b00770  1
2016 Shi J, Sharif S, Ruijtenbeek R, Pieters RJ. Activity Based High-Throughput Screening for Novel O-GlcNAc Transferase Substrates Using a Dynamic Peptide Microarray. Plos One. 11: e0151085. PMID 26960196 DOI: 10.1371/journal.pone.0151085  1
2016 Broekgaarden M, van Vught R, Oliveira S, Roovers RC, van Bergen en Henegouwen PM, Pieters RJ, Van Gulik TM, Breukink E, Heger M. Site-specific conjugation of single domain antibodies to liposomes enhances photosensitizer uptake and photodynamic therapy efficacy. Nanoscale. 8: 6490-4. PMID 26954515 DOI: 10.1039/c6nr00014b  1
2015 Fu O, Pukin AV, van Ufford HC, Branson TR, Thies-Weesie DM, Turnbull WB, Visser GM, Pieters RJ. Tetra- versus Pentavalent Inhibitors of Cholera Toxin. Chemistryopen. 4: 471-7. PMID 26478842 DOI: 10.1002/open.201500006  1
2015 Fu O, Pukin AV, Quarles van Ufford HC, Kemmink J, de Mol NJ, Pieters RJ. Functionalization of a Rigid Divalent Ligand for LecA, a Bacterial Adhesion Lectin. Chemistryopen. 4: 463-70. PMID 26478841 DOI: 10.1002/open.201402171  1
2015 Pukin AV, Brouwer AJ, Koomen L, Quarles van Ufford HC, Kemmink J, de Mol NJ, Pieters RJ. Thiourea-based spacers in potent divalent inhibitors of Pseudomonas aeruginosa virulence lectin LecA. Organic & Biomolecular Chemistry. 13: 10923-8. PMID 26372329 DOI: 10.1039/c5ob01452b  1
2015 Visini R, Jin X, Bergmann M, Michaud G, Pertici F, Fu O, Pukin A, Branson TR, Thies-Weesie DM, Kemmink J, Gillon E, Imberty A, Stocker A, Darbre T, Pieters RJ, et al. Structural Insight into Multivalent Galactoside Binding to Pseudomonas aeruginosa Lectin LecA. Acs Chemical Biology. PMID 26295304 DOI: 10.1021/Acschembio.5B00302  1
2015 Pukin AV, Brouwer AJ, Koomen L, Quarles Van Ufford HC, Kemmink J, De Mol NJ, Pieters RJ. Thiourea-based spacers in potent divalent inhibitors of Pseudomonas aeruginosa virulence lectin LecA Organic and Biomolecular Chemistry. 13: 10923-10928. DOI: 10.1039/c5ob01452b  1
2014 González-Ortiz G, Bronsoms S, Quarles Van Ufford HC, Halkes SB, Virkola R, Liskamp RM, Beukelman CJ, Pieters RJ, Pérez JF, Martín-Orúe SM. A proteinaceous fraction of wheat bran may interfere in the attachment of enterotoxigenic E. coli K88 (F4+) to porcine epithelial cells. Plos One. 9: e104258. PMID 25119298 DOI: 10.1371/Journal.Pone.0104258  1
2014 van Vught R, Pieters RJ, Breukink E. Site-specific functionalization of proteins and their applications to therapeutic antibodies. Computational and Structural Biotechnology Journal. 9: e201402001. PMID 24757499 DOI: 10.5936/csbj.201402001  1
2014 Wang L, Cummings RD, Smith DF, Huflejt M, Campbell CT, Gildersleeve JC, Gerlach JQ, Kilcoyne M, Joshi L, Serna S, Reichardt NC, Parera Pera N, Pieters RJ, Eng W, Mahal LK. Cross-platform comparison of glycan microarray formats. Glycobiology. 24: 507-17. PMID 24658466 DOI: 10.1093/Glycob/Cwu019  1
2014 González-Ortiz G, Quarles Van Ufford HC, Halkes SB, Cerdà-Cuéllar M, Beukelman CJ, Pieters RJ, Liskamp RM, Pérez JF, Martín-Orue SM. New properties of wheat bran: anti-biofilm activity and interference with bacteria quorum-sensing systems. Environmental Microbiology. 16: 1346-53. PMID 24588934 DOI: 10.1111/1462-2920.12441  1
2014 Van Der Wal S, Fu O, Rontogianni S, Pieters RJ, Liskamp RMJ. Convenient stereoselective synthesis of substituted ureido glycosides using stable 4-chlorophenylcarbamates without the requirement of Lewis acids Synlett. 25: 205-208. DOI: 10.1055/S-0033-1340220  1
2013 Kouki A, Pieters RJ, Nilsson UJ, Loimaranta V, Finne J, Haataja S. Bacterial Adhesion of Streptococcus suis to Host Cells and Its Inhibition by Carbohydrate Ligands. Biology. 2: 918-35. PMID 24833053 DOI: 10.3390/Biology2030918  1
2013 Pieters RJ, Slotved HC, Mortensen HM, Arler L, Finne J, Haataja S, Joosten JA, Branderhorst HM, Krogfelt KA. Use of tetravalent galabiose for inhibition of streptococcus suis serotype 2 infection in a mouse model. Biology. 2: 702-18. PMID 24832804 DOI: 10.3390/Biology2020702  1
2013 Pertici F, de Mol NJ, Kemmink J, Pieters RJ. Optimizing divalent inhibitors of Pseudomonas aeruginosa lectin LecA by using a rigid spacer. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 16923-7. PMID 24307357 DOI: 10.1002/chem.201303463  1
2013 Thomsen LB, Linemann T, Pondman KM, Lichota J, Kim KS, Pieters RJ, Visser GM, Moos T. Uptake and transport of superparamagnetic iron oxide nanoparticles through human brain capillary endothelial cells. Acs Chemical Neuroscience. 4: 1352-60. PMID 23919894 DOI: 10.1021/cn400093z  1
2013 Wittmann V, Pieters RJ. Bridging lectin binding sites by multivalent carbohydrates. Chemical Society Reviews. 42: 4492-503. PMID 23598793 DOI: 10.1039/c3cs60089k  1
2013 Pertici F, Varga N, van Duijn A, Rey-Carrizo M, Bernardi A, Pieters RJ. Efficient synthesis of phenylene-ethynylene rods and their use as rigid spacers in divalent inhibitors. Beilstein Journal of Organic Chemistry. 9: 215-22. PMID 23400701 DOI: 10.3762/bjoc.9.25  1
2013 van Hattum H, Branderhorst HM, Moret EE, Nilsson UJ, Leffler H, Pieters RJ. Tuning the preference of thiodigalactoside- and lactosamine-based ligands to galectin-3 over galectin-1. Journal of Medicinal Chemistry. 56: 1350-4. PMID 23281927 DOI: 10.1021/Jm301677R  1
2013 Bernardi A, Jiménez-Barbero J, Casnati A, De Castro C, Darbre T, Fieschi F, Finne J, Funken H, Jaeger KE, Lahmann M, Lindhorst TK, Marradi M, Messner P, Molinaro A, Murphy PV, ... ... Pieters RJ, et al. Multivalent glycoconjugates as anti-pathogenic agents. Chemical Society Reviews. 42: 4709-27. PMID 23254759 DOI: 10.1039/C2Cs35408J  1
2013 van Hattum H, Martin NI, Ruijtenbeek R, Pieters RJ. Development of a microarray detection method for galectin cancer proteins based on ligand binding. Analytical Biochemistry. 434: 99-104. PMID 23149235 DOI: 10.1016/J.Ab.2012.11.003  1
2013 Kooij R, Branderhorst HM, Bonte S, Wieclawska S, Martin NI, Pieters RJ. Glycosidase inhibition by novel guanidinium and urea iminosugar derivatives Medchemcomm. 4: 387-393. DOI: 10.1039/C2Md20343J  1
2012 van Hattum H, van der Zwaluw K, Visser GM, van Putten J, Ruijtenbeek R, Pieters RJ. Functional assay for shiga-like toxin via detection by antibody capture and multivalent galabiose binding. Bioorganic & Medicinal Chemistry Letters. 22: 7448-50. PMID 23142616 DOI: 10.1016/j.bmcl.2012.10.053  1
2012 van der Kaaden M, Breukink E, Pieters RJ. Synthesis and antifungal properties of papulacandin derivatives. Beilstein Journal of Organic Chemistry. 8: 732-7. PMID 23015820 DOI: 10.3762/bjoc.8.82  1
2012 Arnusch CJ, Pieters RJ, Breukink E. Enhanced membrane pore formation through high-affinity targeted antimicrobial peptides. Plos One. 7: e39768. PMID 22768121 DOI: 10.1371/journal.pone.0039768  1
2012 Chamorro C, Boerman MA, Arnusch CJ, Breukink E, Pieters RJ. Enhancing membrane disruption by targeting and multivalent presentation of antimicrobial peptides. Biochimica Et Biophysica Acta. 1818: 2171-4. PMID 22525599 DOI: 10.1016/j.bbamem.2012.04.004  1
2012 Pertici F, Pieters RJ. Potent divalent inhibitors with rigid glucose click spacers for Pseudomonas aeruginosa lectin LecA. Chemical Communications (Cambridge, England). 48: 4008-10. PMID 22428159 DOI: 10.1039/c2cc30234a  1
2012 Schnaar R, Paulson JC, Macauley MS, Nycholat C, Pfrengle F, Rademacher C, Mahan A, Dionne K, Suscovich T, Alter G, Katoh T, Kiwamoto T, Brummet M, Bochner B, Tiemeyer M, ... ... Pieters R, et al. Program and abstracts for the 2012 Joint Meeting of the Society for Glycobiology & American Society for Matrix Biology Glycobiology. 22: 1518-1650. DOI: 10.1093/Glycob/Cws127  1
2011 Mulder MP, Kruijtzer JA, Breukink EJ, Kemmink J, Pieters RJ, Liskamp RM. Synthesis and evaluation of novel macrocyclic antifungal peptides. Bioorganic & Medicinal Chemistry. 19: 6505-17. PMID 21940175 DOI: 10.1016/J.Bmc.2011.08.034  1
2011 Pieters RJ. Carbohydrate mediated bacterial adhesion. Advances in Experimental Medicine and Biology. 715: 227-40. PMID 21557067 DOI: 10.1007/978-94-007-0940-9_14  0.01
2010 Parera Pera N, Branderhorst HM, Kooij R, Maierhofer C, van der Kaaden M, Liskamp RM, Wittmann V, Ruijtenbeek R, Pieters RJ. Rapid screening of lectins for multivalency effects with a glycodendrimer microarray. Chembiochem : a European Journal of Chemical Biology. 11: 1896-904. PMID 20672284 DOI: 10.1002/Cbic.201000340  1
2010 Pera NP, Kouki A, Haataja S, Branderhorst HM, Liskamp RM, Visser GM, Finne J, Pieters RJ. Detection of pathogenic Streptococcus suis bacteria using magnetic glycoparticles. Organic & Biomolecular Chemistry. 8: 2425-9. PMID 20448902 DOI: 10.1039/C000819B  1
2010 van Scherpenzeel M, van den Berg RJ, Donker-Koopman WE, Liskamp RM, Aerts JM, Overkleeft HS, Pieters RJ. Nanomolar affinity, iminosugar-based chemical probes for specific labeling of lysosomal glucocerebrosidase. Bioorganic & Medicinal Chemistry. 18: 267-73. PMID 19931460 DOI: 10.1016/J.Bmc.2009.10.060  1
2010 Arnusch CJ, Ippel JH, Kooijman H, Spek AL, Liskamp RMJ, Kemmink J, Pieters RJ. Direct structural comparison of a rigid cyclic peptidic scaffold using crystallography and NMR in strained PH polymer gels European Journal of Organic Chemistry. 4501-4507. DOI: 10.1002/Ejoc.201000440  1
2009 Kuil J, Branderhorst HM, Pieters RJ, de Mol NJ, Liskamp RM. ITAM-derived phosphopeptide-containing dendrimers as multivalent ligands for Syk tandem SH2 domain. Organic & Biomolecular Chemistry. 7: 4088-94. PMID 19763316 DOI: 10.1039/B905938E  1
2009 Pieters RJ, Arnusch CJ, Breukink E. Membrane permeabilization by multivalent anti-microbial peptides. Protein and Peptide Letters. 16: 736-42. PMID 19601902 DOI: 10.2174/092986609788681841  1
2009 Bauke Albada H, Arnusch CJ, Branderhorst HM, Verel AM, Janssen WT, Breukink E, de Kruijff B, Pieters RJ, Liskamp RM. Potential scorpionate antibiotics: targeted hydrolysis of lipid II containing model membranes by vancomycin-TACzyme conjugates and modulation of their antibacterial activity by Zn-ions. Bioorganic & Medicinal Chemistry Letters. 19: 3721-4. PMID 19524434 DOI: 10.1016/J.Bmcl.2009.05.064  1
2009 van Scherpenzeel M, Moret EE, Ballell L, Liskamp RM, Nilsson UJ, Leffler H, Pieters RJ. Synthesis and evaluation of new thiodigalactoside-based chemical probes to label galectin-3. Chembiochem : a European Journal of Chemical Biology. 10: 1724-33. PMID 19492387 DOI: 10.1002/Cbic.200900198  1
2009 Pieters RJ. Maximising multivalency effects in protein-carbohydrate interactions. Organic & Biomolecular Chemistry. 7: 2013-25. PMID 19421435 DOI: 10.1039/b901828j  0.01
2009 Sisu C, Baron AJ, Branderhorst HM, Connell SD, Weijers CA, de Vries R, Hayes ED, Pukin AV, Gilbert M, Pieters RJ, Zuilhof H, Visser GM, Turnbull WB. The influence of ligand valency on aggregation mechanisms for inhibiting bacterial toxins. Chembiochem : a European Journal of Chemical Biology. 10: 329-37. PMID 19034953 DOI: 10.1002/Cbic.200800550  1
2008 Arnusch CJ, Bonvin AM, Verel AM, Jansen WT, Liskamp RM, de Kruijff B, Pieters RJ, Breukink E. The vancomycin-nisin(1-12) hybrid restores activity against vancomycin resistant Enterococci. Biochemistry. 47: 12661-3. PMID 18989934 DOI: 10.1021/Bi801597B  1
2008 Branderhorst HM, Ruijtenbeek R, Liskamp RM, Pieters RJ. Multivalent carbohydrate recognition on a glycodendrimer-functionalized flow-through chip. Chembiochem : a European Journal of Chemical Biology. 9: 1836-44. PMID 18604837 DOI: 10.1002/Cbic.200800195  1
2008 Branderhorst HM, Kooij R, Salminen A, Jongeneel LH, Arnusch CJ, Liskamp RM, Finne J, Pieters RJ. Synthesis of multivalent Streptococcus suis adhesion inhibitors by enzymatic cleavage of polygalacturonic acid and 'click' conjugation. Organic & Biomolecular Chemistry. 6: 1425-34. PMID 18385849 DOI: 10.1039/B800283E  1
2008 Pieters RJ, Liskamp RMJ. Multivalent presentation strategies in novel inhibitors of bacterial (toxin) adhesion and synthetic vaccines Anti-Infective Agents in Medicinal Chemistry. 7: 193-200. DOI: 10.2174/187152108784911269  1
2007 Branderhorst HM, Liskamp RM, Visser GM, Pieters RJ. Strong inhibition of cholera toxin binding by galactose dendrimers. Chemical Communications (Cambridge, England). 5043-5. PMID 18049747 DOI: 10.1039/B711070G  1
2007 Arnusch CJ, Branderhorst H, de Kruijff B, Liskamp RM, Breukink E, Pieters RJ. Enhanced membrane pore formation by multimeric/oligomeric antimicrobial peptides. Biochemistry. 46: 13437-42. PMID 17944489 DOI: 10.1021/Bi7015553  1
2007 van Zoelen DJ, Egmond MR, Pieters RJ, Liskamp RM. Synthesis and evaluation of TAC-based inhibitors of papain as mimics of cystatin B. Chembiochem : a European Journal of Chemical Biology. 8: 1950-6. PMID 17886319 DOI: 10.1002/Cbic.200700243  1
2007 Pukin AV, Branderhorst HM, Sisu C, Weijers CA, Gilbert M, Liskamp RM, Visser GM, Zuilhof H, Pieters RJ. Strong inhibition of cholera toxin by multivalent GM1 derivatives. Chembiochem : a European Journal of Chemical Biology. 8: 1500-3. PMID 17625801 DOI: 10.1002/Cbic.200700266  1
2007 Salminen A, Loimaranta V, Joosten JA, Khan AS, Hacker J, Pieters RJ, Finne J. Inhibition of P-fimbriated Escherichia coli adhesion by multivalent galabiose derivatives studied by a live-bacteria application of surface plasmon resonance. The Journal of Antimicrobial Chemotherapy. 60: 495-501. PMID 17623698 DOI: 10.1093/Jac/Dkm251  1
2007 van Scherpenzeel M, van der Pot M, Arnusch CJ, Liskamp RM, Pieters RJ. Detection of galectin-3 by novel peptidic photoprobes. Bioorganic & Medicinal Chemistry Letters. 17: 376-8. PMID 17095228 DOI: 10.1016/J.Bmcl.2006.10.043  1
2007 Pieters RJ. Intervention with bacterial adhesion by multivalent carbohydrates. Medicinal Research Reviews. 27: 796-816. PMID 17022032 DOI: 10.1002/med.20089  0.01
2006 Ballell L, van Scherpenzeel M, Buchalova K, Liskamp RM, Pieters RJ. A new chemical probe for the detection of the cancer-linked galectin-3. Organic & Biomolecular Chemistry. 4: 4387-94. PMID 17102885 DOI: 10.1039/B611050A  1
2006 Pieters RJ. Inhibition and detection of galectins. Chembiochem : a European Journal of Chemical Biology. 7: 721-8. PMID 16566049 DOI: 10.1002/cbic.200600011  0.01
2006 Autar R, Liskamp RM, Pieters RJ. A facile synthesis of the GalNAcbeta1-->4Gal target sequence of respiratory pathogens. Carbohydrate Research. 340: 2436-42. PMID 16111663 DOI: 10.1016/J.Carres.2005.08.001  0.01
2006 Kasyanov V, Isenburg J, Draughn RA, Hazard S, Hodde J, Ozolanta I, Murovska M, Halkes SB, Vrasidas I, Liskamp RM, Pieters RJ, Simionescu D, Markwald RR, Mironov V. Tannic acid mimicking dendrimers as small intestine submucosa stabilizing nanomordants. Biomaterials. 27: 745-51. PMID 16102811 DOI: 10.1016/J.Biomaterials.2005.06.022  1
2005 Rijkers DTS, Esse GWv, Merkx R, Brouwer AJ, Jacobs HJF, Pieters RJ, Liskamp RMJ. Efficient microwave-assisted synthesis of multivalent dendrimeric peptides using cycloaddition reaction (click) chemistry Chemical Communications. 4581-4583. PMID 16158121 DOI: 10.1039/B507975F  1
2005 Benedek O, Khan AS, Schneider G, Nagy G, Autar R, Pieters RJ, Emody L. Identification of laminin-binding motifs of Yersinia pestis plasminogen activator by phage display. International Journal of Medical Microbiology : Ijmm. 295: 87-98. PMID 15969469  1
2005 André S, Arnusch CJ, Kuwabara I, Russwurm R, Kaltner H, Gabius HJ, Pieters RJ. Identification of peptide ligands for malignancy- and growth-regulating galectins using random phage-display and designed combinatorial peptide libraries. Bioorganic & Medicinal Chemistry. 13: 563-73. PMID 15598577 DOI: 10.1016/j.bmc.2004.09.053  1
2005 Ballell L, Alink KJ, Slijper M, Versluis C, Liskamp RM, Pieters RJ. A new chemical probe for proteomics of carbohydrate-binding proteins. Chembiochem : a European Journal of Chemical Biology. 6: 291-5. PMID 15578642 DOI: 10.1002/Cbic.200400209  0.01
2004 Joosten JA, Loimaranta V, Appeldoorn CC, Haataja S, El Maate FA, Liskamp RM, Finne J, Pieters RJ. Inhibition of Streptococcus suis adhesion by dendritic galabiose compounds at low nanomolar concentration. Journal of Medicinal Chemistry. 47: 6499-508. PMID 15588085 DOI: 10.1021/Jm049476+  1
2004 Arnusch CJ, André S, Valentini P, Lensch M, Russwurm R, Siebert HC, Fischer MJ, Gabius HJ, Pieters RJ. Interference of the galactose-dependent binding of lectins by novel pentapeptide ligands. Bioorganic & Medicinal Chemistry Letters. 14: 1437-40. PMID 15006378 DOI: 10.1016/j.bmcl.2004.01.029  1
2004 Autar R, Khan AS, Schad M, Hacker J, Liskamp RM, Pieters RJ. Adhesion inhibition of F1C-fimbriated Escherichia coli and Pseudomonas aeruginosa PAK and PAO by multivalent carbohydrate ligands. Chembiochem : a European Journal of Chemical Biology. 4: 1317-25. PMID 14661274 DOI: 10.1002/Cbic.200300719  0.01
2004 Vrasidas I, André S, Valentini P, Böck C, Lensch M, Kaltner H, Liskamp RM, Gabius HJ, Pieters RJ. Rigidified multivalent lactose molecules and their interactions with mammalian galectins: a route to selective inhibitors. Organic & Biomolecular Chemistry. 1: 803-10. PMID 12929363 DOI: 10.1039/B210923A  0.01
2003 Kopitz J, André S, Reitzenstein CV, Versluis K, Kaltner H, Pieters RJ, Wasano K, Kuwabara I, Liu F, Cantz M, Heck AJR, Gabius HJ. Homodimeric galectin-7 (p53-induced gene 1) is a negative growth regulator for human neuroblastoma cells Oncogene. 22: 6277-6288. PMID 13679866 DOI: 10.1038/Sj.Onc.1206631  1
2002 Halkes SB, Vrasidas I, Rooijer GR, van den Berg AJ, Liskamp RM, Pieters RJ. Synthesis and biological activity of polygalloyl-dendrimers as stable tannic acid mimics. Bioorganic & Medicinal Chemistry Letters. 12: 1567-70. PMID 12039563 DOI: 10.1016/S0960-894X(02)00245-7  0.01
2002 Vrasidas I, Kemmink J, Liskamp RM, Pieters RJ. Synthesis and cholera toxin binding properties of a lactose-2-aminothiazoline conjugate. Organic Letters. 4: 1807-8. PMID 12000304 DOI: 10.1021/Ol025909W  0.04
2001 Pieters RJ, Lutje Spelberg JH, Kellogg RM, Janssen DB. The enantioselectivity of haloalkane dehalogenases Tetrahedron Letters. 42: 469-471. DOI: 10.1016/S0040-4039(00)01947-X  1
1999 Pieters RJ, Fennema M, Kellogg RM, Janssen DB. Design and synthesis of reagents for phage display screening of dehalogenases. Bioorganic & Medicinal Chemistry Letters. 9: 161-6. PMID 10021920 DOI: 10.1016/S0960-894X(98)00697-0  1
1999 Rink R, Lutje Spelberg JH, Pieters RJ, Kingma J, Nardini M, Kellogg RM, Dijkstra BW, Janssen DB. Mutation of tyrosine residues involved in the alkylation half reaction of epoxide hydrolase from Agrobacterium radiobacter AD1 results in improved enantioselectivity [7] Journal of the American Chemical Society. 121: 7417-7418. DOI: 10.1021/Ja990501O  1
1990 Doyle MP, Brandes BD, Kazala AP, Pieters RJ, Jarstfer MB, Watkins LM, Eagle CT. Chiral rhodium(II) carboxamides. A new class of catalysts for enantioselective cyclopropanation reactions Tetrahedron Letters. 31: 6613-6616. DOI: 10.1016/S0040-4039(00)97128-4  1
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