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Michio Kurosu - Publications

Affiliations: 
Pharmaceutical Sciences University of Tennessee Health Science Center, Memphis, TN, United States 
Area:
Microbiology, anticancer drug discovery, Medicinal Chemistry
Website:
https://academic.uthsc.edu/faculty/facepage.php?netID=mkurosu&personnel_id=287119

74 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Mitachi K, Kansal RG, Hevener KE, Gillman CD, Hussain SM, Yun HG, Miranda-Carboni GA, Glazer ES, Clemons WM, Kurosu M. DPAGT1 Inhibitors of Capuramycin Analogues and Their Antimigratory Activities of Solid Tumors. Journal of Medicinal Chemistry. PMID 32886511 DOI: 10.1021/Acs.Jmedchem.0C00545  0.4
2020 Lelovic N, Mitachi K, Yang J, Lemieux MR, Ji Y, Kurosu M. Application of Mycobacterium smegmatis as a surrogate to evaluate drug leads against Mycobacterium tuberculosis. The Journal of Antibiotics. PMID 32472054 DOI: 10.1038/S41429-020-0320-7  0.4
2019 Mitachi K, Yun HG, Gillman CD, Skorupinska-Tudek K, Swiezewska E, Clemons WM, Kurosu M. Substrate Tolerance of Bacterial Glycosyltransferase MurG: Novel Fluorescence-based Assays. Acs Infectious Diseases. PMID 31769280 DOI: 10.1021/Acsinfecdis.9B00242  0.4
2019 Mitachi K, Kurosu SM, Gillman CD, Yun HG, Clemons WM, Kurosu M. A practical synthesis of a novel DPAGT1 inhibitor, aminouridyl phenoxypiperidinbenzyl butanamide (APPB) for in vivo studies. Methodsx. 6: 2305-2321. PMID 31667130 DOI: 10.1016/J.Mex.2019.09.031  0.4
2019 Mitachi K, Kurosu SM, Eslamimehr S, Lemieux MR, Ishizaki Y, Clemons WM, Kurosu M. Semisynthesis of an Anticancer DPAGT1 Inhibitor from a Muraymycin Biosynthetic Intermediate. Organic Letters. 21: 876-879. PMID 30698984 DOI: 10.1021/Acs.Orglett.8B03716  0.4
2018 Lemieux MR, Siricilla S, Mitachi K, Eslamimehr S, Wang Y, Yang D, Pressly JD, Kong Y, Park F, Franzblau SG, Kurosu M. An antimycobacterial pleuromutilin analogue effective against dormant bacilli. Bioorganic & Medicinal Chemistry. PMID 30145051 DOI: 10.1016/J.Bmc.2018.07.034  0.4
2018 Mitachi K, Yun HG, Kurosu SM, Eslamimehr S, Lemieux MR, Klaić L, Clemons WM, Kurosu M. Novel FR-900493 Analogues That Inhibit the Outgrowth ofSpores. Acs Omega. 3: 1726-1739. PMID 29503973 DOI: 10.1021/acsomega.7b01740  0.4
2017 Siricilla S, Mitachi K, Yang J, Eslamimehr S, Lemieux MR, Meibohm B, Ji Y, Kurosu M. A New Combination of a Pleuromutilin Derivative and Doxycycline for Treatment of Multidrug-Resistant Acinetobacter baumannii. Journal of Medicinal Chemistry. PMID 28291943 DOI: 10.1021/Acs.Jmedchem.6B01805  0.4
2016 Yang D, Ding F, Mitachi K, Kurosu M, Lee RE, Kong Y. A Fluorescent Probe for Detecting Mycobacterium tuberculosis and Identifying Genes Critical for Cell Entry. Frontiers in Microbiology. 7: 2021. PMID 28066347 DOI: 10.3389/Fmicb.2016.02021  0.4
2016 Mitachi K, Aleiwi BA, Schneider CM, Siricilla S, Kurosu M. Stereocontrolled Total Synthesis of Muraymycin D1 Having a Dual Mode of Action against Mycobacterium tuberculosis. Journal of the American Chemical Society. PMID 27617631 DOI: 10.1021/Jacs.6B07395  0.4
2016 Mitachi K, Siricilla S, Yang D, Kong Y, Skorupinska-Tudek K, Swiezewska E, Franzblau SG, Kurosu M. Fluorescence-based assay for polyprenyl phosphate-GlcNAc-1-phosphate transferase (WecA) and identification of novel antimycobacterial WecA inhibitors. Analytical Biochemistry. PMID 27530653 DOI: 10.1016/J.Ab.2016.08.008  1
2016 Mitachi K, Gautam LN, Rice JH, Eda K, Wadhwa A, Momotani E, Hlopak JP, Eda S, Kurosu M. Structure determination of lipopeptides from Mycobacterium avium subspecies paratuberculosis and identification of antigenic lipopeptide probes. Analytical Biochemistry. PMID 27114041 DOI: 10.1016/J.Ab.2016.04.001  1
2016 Mitachi K, Kurosu YE, Hazlett BT, Kurosu M. Oxyma-based phosphates for racemization-free peptide segment couplings. Journal of Peptide Science : An Official Publication of the European Peptide Society. 22: 186-91. PMID 26856693 DOI: 10.1002/Psc.2859  1
2015 Mitachi K, Siricilla S, Klaic L, Clemons WM, Kurosu M. Chemoenzymatic syntheses of water-soluble lipid I fluorescent probes. Tetrahedron Letters. 56: 3441-3446. PMID 26190869 DOI: 10.1016/J.Tetlet.2015.01.044  0.4
2015 Siricilla S, Mitachi K, Wan B, Franzblau SG, Kurosu M. Discovery of a capuramycin analog that kills nonreplicating Mycobacterium tuberculosis and its synergistic effects with translocase I inhibitors. The Journal of Antibiotics. 68: 271-8. PMID 25269459 DOI: 10.1038/Ja.2014.133  0.4
2015 Mitachi K, Siricilla S, Klai? L, Clemons WM, Kurosu M. Chemoenzymatic syntheses of water-soluble lipid i fluorescent probes This Letter is dedicated to the memory of Professor Harry H. Wasserman, an inspirational scientist Tetrahedron Letters. 56: 3441-3446. DOI: 10.1016/j.tetlet.2015.01.044  1
2014 Siricilla S, Mitachi K, Skorupinska-Tudek K, Swiezewska E, Kurosu M. Biosynthesis of a water-soluble lipid I analogue and a convenient assay for translocase I. Analytical Biochemistry. 461: 36-45. PMID 24939461 DOI: 10.1016/J.Ab.2014.05.018  0.4
2014 Mitachi K, Mohan P, Siricilla S, Kurosu M. One-pot protection-glycosylation reactions for synthesis of lipid II analogues. Chemistry (Weinheim An Der Bergstrasse, Germany). 20: 4554-8. PMID 24623584 DOI: 10.1002/Chem.201400307  0.4
2014 Siricilla S, Mitachi K, Wan B, Franzblau SG, Kurosu M. Discovery of a capuramycin analog that kills nonreplicating Mycobacterium tuberculosis and its synergistic effects with translocase i inhibitors Journal of Antibiotics. 68: 271-278. DOI: 10.1038/ja.2014.133  1
2014 Siricilla S, Mitachi K, Skorupinska-Tudek K, Swiezewska E, Kurosu M. Biosynthesis of a water-soluble lipid i analogue and a convenient assay for translocase i Analytical Biochemistry. 461: 36-45. DOI: 10.1016/j.ab.2014.05.018  1
2014 Mitachi K, Mohan P, Siricilla S, Kurosu M. One-pot protection-glycosylation reactions for synthesis of lipid II analogues Chemistry - a European Journal. 20: 4554-4558. DOI: 10.1002/chem.201400307  1
2013 Wang Y, Siricilla S, Aleiwi BA, Kurosu M. Improved synthesis of capuramycin and its analogues Chemistry - a European Journal. 19: 13847-13858. PMID 24014478 DOI: 10.1002/Chem.201302389  1
2013 Aleiwi BA, Mitachi K, Kurosu M. Mild and convenient N-formylation protocol in water-containing solvents. Tetrahedron Letters. 54: 2077-2081. PMID 23908559 DOI: 10.1016/J.Tetlet.2013.02.013  0.4
2013 Kurosu M, Siricilla S, Mitachi K. Advances in MRSA drug discovery: where are we and where do we need to be? Expert Opinion On Drug Discovery. 8: 1095-116. PMID 23829425 DOI: 10.1517/17460441.2013.807246  0.4
2013 Kurosu M, Siricilla S, Mitachi K. Advances in MRSA drug discovery: Where are we and where do we need to be? Expert Opinion On Drug Discovery. 8: 1095-1116. DOI: 10.1517/17460441.2013.807246  1
2013 Aleiwi BA, Mitachi K, Kurosu M. Mild and convenient N-formylation protocol in water-containing solvents Tetrahedron Letters. 54: 2077-2081. DOI: 10.1016/j.tetlet.2013.02.013  1
2012 Wang Y, Aleiwi BA, Wang Q, Kurosu M. Selective esterifications of primary alcohols in a water-containing solvent Organic Letters. 14: 4910-4913. PMID 22937741 DOI: 10.1021/Ol3022337  1
2012 Wang Q, Wang Y, Kurosu M. A new oxyma derivative for nonracemizable amide-forming reactions in water Organic Letters. 14: 3372-3375. PMID 22697488 DOI: 10.1021/Ol3013556  1
2012 Aleiwi BA, Schneider CM, Kurosu M. Synthesis of ureidomuraymycidine derivatives for structure-activity relationship studies of muraymycins Journal of Organic Chemistry. 77: 3859-3867. PMID 22458337 DOI: 10.1021/Jo300205B  1
2012 Debnath J, Siricilla S, Wan B, Crick DC, Lenaerts AJ, Franzblau SG, Kurosu M. Discovery of selective menaquinone biosynthesis inhibitors against Mycobacterium tuberculosis. Journal of Medicinal Chemistry. 55: 3739-55. PMID 22449052 DOI: 10.1021/Jm201608G  1
2012 Aleiwi BA, Kurosu M. A reliable Pd-mediated hydrogenolytic deprotection of BOM group of uridine ureido nitrogen Tetrahedron Letters. 53: 3758-3762. DOI: 10.1016/j.tetlet.2012.05.035  1
2012 Wang Y, Kurosu M. A new protecting group and linker for uridine ureido nitrogen Tetrahedron. 68: 4797-4804. DOI: 10.1016/j.tet.2012.03.121  1
2010 Kurosu M, Begari E. Vitamin K2 in electron transport system: Are enzymes involved in vitamin K2 biosynthesis promising drug targets? Molecules. 15: 1531-1553. PMID 20335999 DOI: 10.3390/Molecules15031531  1
2010 Kurosu M, Li K. Mild and selective O-glycosylations of primary alcohols with the thioglucosaminide derivative promoted by N-iodosuccinimide and HBF4-adosrobed on silica gel Heterocycles. 80: 115-123. DOI: 10.3987/COM-09-S(S)24  1
2010 Kurosu M, Begari E. Bacterial protein kinase inhibitors Drug Development Research. 71: 168-187. DOI: 10.1002/Ddr.20362  1
2009 Kurosu M, Li K, Crick DC. Concise synthesis of capuramycin. Organic Letters. 11: 2393-6. PMID 19405507 DOI: 10.1021/Ol900458W  1
2009 Kurosu M, Crick DC. MenA is a promising drug target for developing novel lead molecules to combat Mycobacterium tuberculosis. Medicinal Chemistry (ShāRiqah (United Arab Emirates)). 5: 197-207. PMID 19275719 DOI: 10.2174/157340609787582882  1
2009 Dhiman RK, Mahapatra S, Slayden RA, Boyne ME, Lenaerts A, Hinshaw JC, Angala SK, Chatterjee D, Biswas K, Narayanasamy P, Kurosu M, Crick DC. Menaquinone synthesis is critical for maintaining mycobacterial viability during exponential growth and recovery from non-replicating persistence. Molecular Microbiology. 72: 85-97. PMID 19220750 DOI: 10.1111/J.1365-2958.2009.06625.X  1
2009 Kurosu M, Li K. New chiral derivatizing agents: Convenient determination of absolute configurations of free amino acids By 1H NMR Organic Letters. 11: 911-914. PMID 19170578 DOI: 10.1021/Ol8028719  1
2009 Kurosu M, Li K. Synthetic studies towards the identification of novel capuramycin analogs with mycobactericidal activity Heterocycles. 77: 217-225. DOI: 10.3987/Com-08-S(F)38  1
2009 Kurosu M, Li K. (2,6-Dichloro-4-alkoxyphenyl)-(2,4-dichlorophenyl)methyl trichloroacetimidates: Protection of alcohols and carboxylic acids in solution or on polymer support Synthesis. 3633-3641. DOI: 10.1055/S-0029-1216974  1
2008 Kurosu M, Li K. Highly efficient O-glycosylations with p-tolyl thioribosides and p-TolSOTf Journal of Organic Chemistry. 73: 9767-9770. PMID 18783274 DOI: 10.1021/Jo801408X  1
2008 Kurosu M. Multiple-delayed release formulation approach for the treatment of methicillin-resistant Staphylococcus aureus Expert Opinion On Therapeutic Patents. 18: 1313-1319. DOI: 10.1517/13543776.18.11.1313  1
2007 Kurosu M, Katayama S, Shibuya H, Kitagawa I. A study of the calcium complex of a glucosylceramide, soya-cerebroside II Chemical and Pharmaceutical Bulletin. 55: 1758-1761. PMID 18057755 DOI: 10.1248/Cpb.55.1758  1
2007 Kurosu M, Narayanasamy P, Biswas K, Dhiman R, Crick DC. Discovery of 1,4-dihydroxy-2-naphthoate [corrected] prenyltransferase inhibitors: new drug leads for multidrug-resistant gram-positive pathogens. Journal of Medicinal Chemistry. 50: 3973-5. PMID 17658779 DOI: 10.1021/Jm070638M  1
2007 Kurosu M, Biswas K, Crick DC. Polymer-supported (2,6-dichloro- 4-alkoxyphenyl)(2,4-dichlorophenyl)methanol: a new linker for solid-phase organic synthesis. Organic Letters. 9: 1141-4. PMID 17311394 DOI: 10.1021/Ol070150F  1
2007 Kurosu M, Narayanasamy P, Crick DC. High-throughput synthesis of substituted hydrazine derivatives Heterocycles. 73: 169-175. DOI: 10.3987/Com-07-S(U)14  1
2007 Kurosu M, Narayanasamy P, Crick DC. Synthetic studies toward the generation of uridine-amino alcohol-based small optimized libraries Heterocycles. 72: 339-352. DOI: 10.3987/Com-06-S(K)18  1
2007 Kurosu M, Biswas K, Narayanasamy P, Crick DC. Acid- and base-stable esters: A new protecting group for carboxylic acids Synthesis. 2513-2516. DOI: 10.1055/S-2007-983801  1
2007 Kurosu M, Mahapatra S, Narayanasamy P, Crick DC. Chemoenzymatic synthesis of Park's nucleotide: toward the development of high-throughput screening for MraY inhibitors Tetrahedron Letters. 48: 799-803. DOI: 10.1016/J.Tetlet.2006.11.160  1
2006 Kurosu M, Mowers WA. Small-molecule microarrays: Development of novel linkers and an efficient detection method for bound proteins Bioorganic and Medicinal Chemistry Letters. 16: 3392-3395. PMID 16682190 DOI: 10.1016/J.Bmcl.2006.04.057  1
2006 Kurosu M, Kitagawa I. Ganglioside GM3 derivatives with truncated ceramide moiety: Facial synthesis and inhibitory activity against KB cell growth Journal of Carbohydrate Chemistry. 25: 427-439. DOI: 10.1080/07328300600803518  1
2006 Kurosu M, Crick DC. A novel strategy for oligopeptide synthesis using a polymer-supported ammonium fluoride Tetrahedron Letters. 47: 5325-5328. DOI: 10.1016/J.Tetlet.2006.05.129  1
2006 Kurosu M, Dey SS, Crick DC. Efficient synthesis of tertiary amines from secondary amines Tetrahedron Letters. 47: 4871-4875. DOI: 10.1016/J.Tetlet.2006.05.038  1
2006 Kurosu M. Cr-waste free catalytic carbonyl addition reactions with polymer-immobilized CrF2 Tetrahedron Letters. 47: 3395-3399. DOI: 10.1016/J.Tetlet.2006.03.071  1
2005 Kurosu M, Lorca M. Effect of water on Keck's catalytic asymmetric allylations of aldehydes Synlett. 1109-1112. DOI: 10.1055/S-2005-865202  1
2004 Kurosu M, Lin MH, Kishi Y. Fe/Cr- and Co/Cr-mediated catalytic asymmetric 2-haloallylations of aldehydes. Journal of the American Chemical Society. 126: 12248-9. PMID 15453741 DOI: 10.1021/Ja045557J  1
2004 Kurosu M, Kishi Y. Studies on the total synthesis of batrachotoxin Yuki Gosei Kagaku Kyokaishi/Journal of Synthetic Organic Chemistry. 62: 1205-1217. DOI: 10.5059/Yukigoseikyokaishi.62.1205  1
2004 Kurosu M, Porter JR, Foley MA. An efficient synthesis of indane-derived bis(oxazoline) and its application to hetero Diels-Alder reactions on polymer support Tetrahedron Letters. 45: 145-148. DOI: 10.1016/J.Tetlet.2003.10.097  1
2002 Kurosu M, Lorca M. Catalytic asymmetric allylations of achiral and chiral aldehydes via BINOL-Zr complex Tetrahedron Letters. 43: 1765-1769. DOI: 10.1016/S0040-4039(02)00139-9  1
2001 Kurosu M, Lorca M. Highly diastereofacial anti-aldol reaction: Practical synthesis of optically active anti-2-alkyl-3-hydroxycarboxylic acid ester units Journal of Organic Chemistry. 66: 1205-1209. PMID 11312949 DOI: 10.1021/Jo001293H  1
2001 Lorca M, Kurosu M. An efficient amide-forming reaction using tributyltrichloromethylphosphonium chloride Synthetic Communications. 31: 469-473. DOI: 10.1081/Scc-100000572  1
2001 Lorca M, Kuhn D, Kurosu M. Selective reduction of aldehydes via BINOL-Zr complex Tetrahedron Letters. 42: 6243-6246. DOI: 10.1016/S0040-4039(01)01276-X  1
2001 Lorca M, Kurosu M. A practical synthesis of the lipophilic side chain of the polyoxypeptins Tetrahedron Letters. 42: 2431-2434. DOI: 10.1016/S0040-4039(01)00205-2  1
2000 Kurosu M. Expeditious amide-forming reactions using thiol esters Tetrahedron Letters. 41: 591-594. DOI: 10.1016/S0040-4039(99)02132-2  1
1998 Kurosu M, Kishi Y. A Novel Example for Optical Resolution of Racemic Ketones Originating from Batrachotoxin Synthesis. The Journal of Organic Chemistry. 63: 6100-6101. PMID 11672234 DOI: 10.1021/Jo981416M  1
1998 Kurosu M, Marcin LR, Grinsteiner TJ, Kishi Y. Total synthesis of (±)-batrachotoxin A Journal of the American Chemical Society. 120: 6627-6628. DOI: 10.1021/Ja981258G  1
1998 Kurosu M, Marcin LR, Kishi Y. A useful modification of the Garst-Spencer furan annulation: An improved synthesis of 3,4-substituted furans Tetrahedron Letters. 39: 8929-8932. DOI: 10.1016/S0040-4039(98)02017-6  1
1998 Kurosu M, Kishi Y. Reaction of methylcerium reagent with tertiary amides: Synthesis of saturated and unsaturated ketones from tertiary amides Tetrahedron Letters. 39: 4793-4796. DOI: 10.1016/S0040-4039(98)00959-9  1
1995 Kobayashi M, Wang W, Ohyabu N, Kurosu M, Kitagawa I. Improved total synthesis and structure-activity relationship of arenastatin A, a potent cytotoxic spongean depsipeptide. Chemical & Pharmaceutical Bulletin. 43: 1598-600. PMID 7586087 DOI: 10.1248/Cpb.43.1598  1
1994 Kobayashi M, Aoki S, Gato K, Matsunami K, Kurosu M, Kitagawa I. Marine natural products. XXXIV. Trisindoline, a new antibiotic indole trimer, produced by a bacterium of Vibrio sp. separated from the marine sponge Hyrtios altum. Chemical & Pharmaceutical Bulletin. 42: 2449-51. PMID 7697760 DOI: 10.1248/Cpb.42.2449  1
1994 Kobayashi M, Aoki S, Ohyabu N, Kurosu M, Wang W, Kitagawa I. Arenastatin A, a potent cytotoxic depsipeptide from the okinawan marine sponge Dysidea arenaria Tetrahedron Letters. 35: 7969-7972. DOI: 10.1016/0040-4039(94)80024-3  1
1994 Kobayashi M, Kurosu M, Wang W, Kitagawa I. A total synthesis of arenastatin A, an extremely potent cytotoxic depsipeptide, from the Okinawan marine sponge dysidea arenaria Chemical and Pharmaceutical Bulletin. 42: 2394-2396.  1
1993 Shibuya H, Kurosu M, Minagawa K, Katayama S, Kitagawa I. Sphingolipids and glycerolipids. IV. Syntheses and ionophoretic activities of several analogues of soya-cerebroside II, a calcium ionophoretic sphingoglycolipid isolated from soybean Chemical and Pharmaceutical Bulletin. 41: 1534-1544. DOI: 10.1248/Cpb.41.1534  1
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