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Eranthie Weerapana, Ph.D. - Publications

2010- Chemistry Boston College, Newton, MA, United States 

92 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Perez M, Bak DW, Bergholtz SE, Crooks DR, Arimilli BS, Yang Y, Weerapana E, Linehan WM, Meier JL. Heterogeneous adaptation of cysteine reactivity to a covalent oncometabolite. The Journal of Biological Chemistry. PMID 32820045 DOI: 10.1074/jbc.AC120.014993  0.76
2020 Peeler JC, Falco JA, Kelemen RE, Abo M, Chartier BV, Edinger LC, Chen J, Chatterjee A, Weerapana E. Generation of Recombinant Mammalian Selenoproteins through Genetic Code Expansion with Photocaged Selenocysteine. Acs Chemical Biology. PMID 32330002 DOI: 10.1021/acschembio.0c00147  1
2020 Italia JS, Peeler JC, Hillenbrand CM, Latour C, Weerapana E, Chatterjee A. Genetically encoded protein sulfation in mammalian cells. Nature Chemical Biology. 16: 379-382. PMID 32198493 DOI: 10.1038/s41589-020-0493-1  0.4
2020 Salinger AJ, Dubuke ML, Carmona-Rivera C, Maurais AJ, Shaffer SA, Weerapana E, Thompson PR, Kaplan MJ. Technical comment on "Synovial fibroblast-neutrophil interactions promote pathogenic adaptive immunity in rheumatoid arthritis". Science Immunology. 5. PMID 32005680 DOI: 10.1126/sciimmunol.aax5672  0.48
2020 Bechtel TJ, Li C, Kisty EA, Maurais AJ, Weerapana E. Profiling cysteine reactivity and oxidation in the endoplasmic reticulum. Acs Chemical Biology. PMID 31899610 DOI: 10.1021/acschembio.9b01014  0.8
2019 Sun B, Chang HH, Salinger A, Tomita B, Bawadekar M, Holmes CL, Shelef MA, Weerapana E, Thompson PR, Ho IC. Reciprocal regulation of Th2 and Th17 cells by PAD2-mediated citrullination. Jci Insight. 4. PMID 31723060 DOI: 10.1172/jci.insight.129687  0.32
2019 Peeler JC, Weerapana E. Chemical Biology Approaches to Interrogate the Selenoproteome. Accounts of Chemical Research. PMID 31523956 DOI: 10.1021/acs.accounts.9b00379  0.4
2019 Hoffman KS, Vargas-Rodriguez O, Bak DW, Mukai T, Woodward LK, Weerapana E, Söll D, Reynolds NM. A cysteinyl-tRNA synthetase variant confers resistance against selenite toxicity and decreases selenocysteine misincorporation. The Journal of Biological Chemistry. PMID 31296657 DOI: 10.1074/jbc.RA119.008219  0.76
2019 Mondal S, Gong X, Zhang X, Salinger AJ, Zheng L, Sen S, Weerapana E, Zhang X, Thompson P. Halogen Bonding Increases the Potency and Isozyme-selectivity of Protein Arginine Deiminase 1 Inhibitors. Angewandte Chemie (International Ed. in English). PMID 31276611 DOI: 10.1002/anie.201906334  0.48
2019 Sorvillo N, Mizurini D, Coxon C, Martinod K, Tilvawala R, Cherpokova D, Salinger AJ, Seward RJ, Staudinger C, Weerapana E, Shapiro NI, Costello CE, Thompson P, Wagner DD. Plasma Peptidylarginine Deiminase IV Promotes VWF-Platelet String Formation and Accelerates Thrombosis after Vessel Injury. Circulation Research. PMID 31248335 DOI: 10.1161/CIRCRESAHA.118.314571  0.48
2019 Zheng L, Nagar M, Maurais AJ, Slade DJ, Parelkar SS, Coonrod SA, Weerapana E, Thompson PR. Calcium Regulates the Nuclear Localization of Protein Arginine Deiminase 2. Biochemistry. PMID 31243954 DOI: 10.1021/acs.biochem.9b00225  0.48
2019 Libiad M, Vitvitsky V, Bostelaar T, Bak DW, Lee HJ, Sakamoto N, Fearon ER, Lyssiotis CA, Weerapana E, Banerjee R. Hydrogen sulfide perturbs mitochondrial bioenergetics and triggers metabolic reprogramming in colon cells. The Journal of Biological Chemistry. PMID 31213529 DOI: 10.1074/jbc.RA119.009442  0.76
2019 Morimoto K, Cole KS, Kourelis J, Witt CH, Brown D, Krahn D, Stegmann M, Kaschani F, Kaiser M, Burton J, Mohammed S, Yamaguchi-Shinozaki K, Weerapana E, van der Hoorn RAL. Triazine probes targeting ascorbate peroxidases in plants. Plant Physiology. PMID 31138623 DOI: 10.1104/pp.19.00481  1
2019 Llabani E, Hicklin RW, Lee HY, Motika SE, Crawford LA, Weerapana E, Hergenrother PJ. Diverse compounds from pleuromutilin lead to a thioredoxin inhibitor and inducer of ferroptosis. Nature Chemistry. PMID 31086302 DOI: 10.1038/s41557-019-0261-6  0.32
2019 Bak DW, Weerapana E. Interrogation of Functional Mitochondrial Cysteine Residues by Quantitative Mass Spectrometry. Methods in Molecular Biology (Clifton, N.J.). 1967: 211-227. PMID 31069773 DOI: 10.1007/978-1-4939-9187-7_13  0.76
2019 Sen S, Mondal S, Zheng L, Salinger AJ, Fast W, Weerapana E, Thompson PR. Development of a Suicide Inhibition Based Protein Labeling (SIBLing) Strategy for Nicotinamide N-methyltransferase. Acs Chemical Biology. PMID 30933557 DOI: 10.1021/acschembio.9b00211  0.48
2019 Italia JS, Addy PS, Erickson SB, Peeler JC, Weerapana E, Chatterjee A. Mutually orthogonal nonsense-suppression systems and conjugation chemistries for precise protein labeling at up to three distinct sites. Journal of the American Chemical Society. PMID 30909694 DOI: 10.1021/jacs.8b12954  0.4
2019 Kulkarni RA, Bak DW, Wei D, Bergholtz SE, Briney CA, Shrimp JH, Alpsoy A, Thorpe AL, Bavari AE, Crooks DR, Levy M, Florens L, Washburn MP, Frizzell N, Dykhuizen EC, ... Weerapana E, et al. A chemoproteomic portrait of the oncometabolite fumarate. Nature Chemical Biology. PMID 30718813 DOI: 10.1038/s41589-018-0217-y  0.76
2018 Bak DW, Bechtel TJ, Falco JA, Weerapana E. Cysteine reactivity across the subcellular universe. Current Opinion in Chemical Biology. 48: 96-105. PMID 30508703 DOI: 10.1016/j.cbpa.2018.11.002  0.76
2018 Gao J, Yang F, Che J, Han Y, Wang Y, Chen N, Bak DW, Lai S, Xie X, Weerapana E, Wang C. Selenium-Encoded Isotopic Signature Targeted Profiling. Acs Central Science. 4: 960-970. PMID 30159393 DOI: 10.1021/acscentsci.8b00112  0.8
2018 Nemmara VV, Tilvawala R, Salinger AJ, Miller L, Nguyen SH, Weerapana E, Thompson PR. Citrullination Inactivates Nicotinamide-N-methyltransferase. Acs Chemical Biology. PMID 30044909 DOI: 10.1021/acschembio.8b00578  0.48
2018 Bak DW, Gao J, Wang C, Weerapana E. A Quantitative Chemoproteomic Platform to Monitor Selenocysteine Reactivity within a Complex Proteome. Cell Chemical Biology. PMID 29983274 DOI: 10.1016/j.chembiol.2018.05.017  0.8
2018 Lentz CS, Sheldon JR, Crawford LA, Cooper R, Garland M, Amieva MR, Weerapana E, Skaar EP, Bogyo M. Identification of a S. aureus virulence factor by activity-based protein profiling (ABPP). Nature Chemical Biology. PMID 29769740 DOI: 10.1038/s41589-018-0060-1  0.32
2018 Tilvawala R, Nguyen SH, Maurais AJ, Nemmara VV, Nagar M, Salinger AJ, Nagpal S, Weerapana E, Thompson PR. The Rheumatoid Arthritis-Associated Citrullinome. Cell Chemical Biology. PMID 29628436 DOI: 10.1016/j.chembiol.2018.03.002  0.48
2018 Cole KS, Grandjean JMD, Chen K, Witt CH, O'Day J, Shoulders MD, Wiseman RL, Weerapana E. Characterization of an A-Site Selective Protein Disulfide Isomerase A1 Inhibitor. Biochemistry. PMID 29521097 DOI: 10.1021/acs.biochem.8b00178  0.4
2018 Nemmara VJ, Subramanian V, Muth A, Mondal S, Salinger AJ, Maurais AJ, Tilvawala R, Weerapana E, Thompson PR. The Development of Benzimidazole-Based Clickable Probes for the Efficient Labeling of Cellular Protein Arginine Deiminases (PADs). Acs Chemical Biology. PMID 29341591 DOI: 10.1021/acschembio.7b00957  0.48
2017 Abo M, Li C, Weerapana E. Isotopically-Labeled Iodoacetamide-Alkyne Probes for Quantitative Cysteine-Reactivity Profiling. Molecular Pharmaceutics. PMID 29172527 DOI: 10.1021/acs.molpharmaceut.7b00832  1
2017 Abo M, Li C, Weerapana E. Isotopically-Labeled Iodoacetamide-Alkyne Probes for Quantitative Cysteine-Reactivity Profiling. Molecular Pharmaceutics. PMID 29172527 DOI: 10.1021/acs.molpharmaceut.7b00832  1
2017 Gorelenkova Miller O, Cole KS, Emerson CC, Allimuthu D, Golczak M, Stewart PL, Weerapana E, Adams DJ, Mieyal JJ. Novel chloroacetamido compound CWR-J02 is an anti-inflammatory glutaredoxin-1 inhibitor. Plos One. 12: e0187991. PMID 29155853 DOI: 10.1371/journal.pone.0187991  1
2017 Abo M, Weerapana E. Chemical Probes for Redox Signaling and Oxidative Stress. Antioxidants & Redox Signaling. PMID 29132214 DOI: 10.1089/ars.2017.7408  1
2017 Lawson AP, Bak DW, Shannon DA, Long MJC, Vijaykumar T, Yu R, Oualid FE, Weerapana E, Hedstrom L. Identification of deubiquitinase targets of isothiocyanates using SILAC-assisted quantitative mass spectrometry. Oncotarget. 8: 51296-51316. PMID 28881649 DOI: 10.18632/oncotarget.17261  0.76
2017 Sun B, Dwivedi N, Bechtel TJ, Paulsen JL, Muth A, Bawadekar M, Li G, Thompson PR, Shelef MA, Schiffer CA, Weerapana E, Ho IC. Citrullination of NF-κB p65 promotes its nuclear localization and TLR-induced expression of IL-1β and TNFα. Science Immunology. 2. PMID 28783661 DOI: 10.1126/sciimmunol.aal3062  0.56
2017 Quinti L, Dayalan Naidu S, Träger U, Chen X, Kegel-Gleason K, Llères D, Connolly C, Chopra V, Low C, Moniot S, Sapp E, Tousley AR, Vodicka P, Van Kanegan MJ, Kaltenbach LS, ... ... Weerapana E, et al. KEAP1-modifying small molecule reveals muted NRF2 signaling responses in neural stem cells from Huntington's disease patients. Proceedings of the National Academy of Sciences of the United States of America. PMID 28533375 DOI: 10.1073/pnas.1614943114  0.32
2017 Lawson AP, Bak DW, Shannon DA, Long MJC, Vijaykumar T, Yu R, El Oualid F, Weerapana E, Hedstrom L. Identification of deubiquitinase targets of isothiocyanates using SILAC-assisted quantitative mass spectrometry. Oncotarget. PMID 28472782 DOI: 10.18632/oncotarget.17261  0.76
2017 Casas-Selves M, Zhang A, Dowling JE, Hallen S, Kawatkar A, Pace NJ, Denz C, Pontz T, Garahdaghi F, Cao Q, Sabirsh A, Thakur K, O'Connell N, Hu J, Cornella-Taracido I, ... Weerapana E, et al. Target deconvolution efforts on Wnt pathway screen reveal dual modulation of oxidative phosphorylation and SERCA2. Chemmedchem. PMID 28371485 DOI: 10.1002/cmdc.201700028  0.36
2017 Bak DW, Pizzagalli MD, Weerapana E. Identifying Functional Cysteine Residues in the Mitochondria. Acs Chemical Biology. PMID 28157297 DOI: 10.1021/acschembio.6b01074  0.76
2017 Bechtel TJ, Weerapana E. From structure to redox: the diverse functional roles of disulfides and implications in disease. Proteomics. PMID 28044432 DOI: 10.1002/pmic.201600391  0.56
2016 Abo M, Bak DW, Weerapana E. Optimization of Caged Electrophiles for Improved Monitoring of Cysteine Reactivity in Living Cells. Chembiochem : a European Journal of Chemical Biology. PMID 27813293 DOI: 10.1002/cbic.201600524  1
2016 Martell J, Seo Y, Bak DW, Kingsley SF, Tissenbaum HA, Weerapana E. Global Cysteine-Reactivity Profiling during Impaired Insulin/IGF-1 Signaling in C. elegans Identifies Uncharacterized Mediators of Longevity. Cell Chemical Biology. PMID 27499530 DOI: 10.1016/j.chembiol.2016.06.015  1
2016 Hatzios SK, Abel S, Martell J, Hubbard T, Sasabe J, Munera D, Clark L, Bachovchin DA, Qadri F, Ryan ET, Davis BM, Weerapana E, Waldor MK. Erratum: Chemoproteomic profiling of host and pathogen enzymes active in cholera. Nature Chemical Biology. 12: 466. PMID 27191648 DOI: 10.1038/nchembio0616-466  0.52
2016 Louie SM, Grossman EA, Crawford LA, Ding L, Camarda R, Huffman TR, Miyamoto DK, Goga A, Weerapana E, Nomura DK. GSTP1 Is a Driver of Triple-Negative Breast Cancer Cell Metabolism and Pathogenicity. Cell Chemical Biology. PMID 27185638 DOI: 10.1016/j.chembiol.2016.03.017  1
2016 Crawford LA, Weerapana E. A tyrosine-reactive irreversible inhibitor for glutathione S-transferase Pi (GSTP1). Molecular Biosystems. PMID 27113843 DOI: 10.1039/c6mb00250a  1
2016 Sanman LE, Qian Y, Eisele NA, Ng TM, van der Linden WA, Monack DM, Weerapana E, Bogyo M. Disruption of glycolytic flux is a signal for inflammasome signaling and pyroptotic cell death. Elife. 5. PMID 27011353 DOI: 10.7554/eLife.13663  1
2016 Hatzios SK, Abel S, Martell J, Hubbard T, Sasabe J, Munera D, Clark L, Bachovchin DA, Qadri F, Ryan ET, Davis BM, Weerapana E, Waldor MK. Chemoproteomic profiling of host and pathogen enzymes active in cholera. Nature Chemical Biology. PMID 26900865 DOI: 10.1038/nchembio.2025  1
2015 Saghatelian A, Nomura DK, Weerapena E. Editorial overview: Omics: The maturation of chemical biology. Current Opinion in Chemical Biology. PMID 26739665 DOI: 10.1016/j.cbpa.2015.12.005  0.92
2015 Lawson AP, Long MJ, Coffey RT, Qian Y, Weerapana E, El Oualid F, Hedstrom L. Naturally occurring isothiocyanates exert anticancer effects by inhibiting deubiquitinating enzymes. Cancer Research. PMID 26542215 DOI: 10.1158/0008-5472.CAN-15-1544  1
2015 Clancy KW, Weerapana E, Thompson PR. Detection and identification of protein citrullination in complex biological systems. Current Opinion in Chemical Biology. 30: 1-6. PMID 26517730 DOI: 10.1016/j.cbpa.2015.10.014  1
2015 Lewallen DM, Bicker KL, Subramanian V, Clancy KW, Slade DJ, Martell J, Dreyton CJ, Sokolove J, Weerapana E, Thompson PR. Chemical Proteomic Platform To Identify Citrullinated Proteins. Acs Chemical Biology. PMID 26360112 DOI: 10.1021/acschembio.5b00438  1
2015 Abo M, Weerapana E. A Caged Electrophilic Probe for Global Analysis of Cysteine Reactivity in Living Cells. Journal of the American Chemical Society. 137: 7087-90. PMID 26020833 DOI: 10.1021/jacs.5b04350  1
2015 Bak DW, Weerapana E. Cysteine-mediated redox signalling in the mitochondria. Molecular Biosystems. 11: 678-97. PMID 25519845 DOI: 10.1039/c4mb00571f  1
2015 Shannon DA, Weerapana E. Covalent protein modification: the current landscape of residue-specific electrophiles. Current Opinion in Chemical Biology. 24: 18-26. PMID 25461720 DOI: 10.1016/j.cbpa.2014.10.021  1
2014 Couvertier SM, Zhou Y, Weerapana E. Chemical-proteomic strategies to investigate cysteine posttranslational modifications. Biochimica Et Biophysica Acta. 1844: 2315-2330. PMID 25291386 DOI: 10.1016/j.bbapap.2014.09.024  1
2014 Pace NJ, Weerapana E. Zinc-binding cysteines: diverse functions and structural motifs. Biomolecules. 4: 419-34. PMID 24970223 DOI: 10.3390/biom4020419  1
2014 Shannon DA, Banerjee R, Webster ER, Bak DW, Wang C, Weerapana E. Investigating the proteome reactivity and selectivity of aryl halides. Journal of the American Chemical Society. 136: 3330-3. PMID 24548313 DOI: 10.1021/ja4116204  1
2014 Zhuang J, Kuo CH, Chou LY, Liu DY, Weerapana E, Tsung CK. Optimized metal-organic-framework nanospheres for drug delivery: evaluation of small-molecule encapsulation. Acs Nano. 8: 2812-9. PMID 24506773 DOI: 10.1021/nn406590q  1
2014 Martell J, Weerapana E. Applications of copper-catalyzed click chemistry in activity-based protein profiling. Molecules (Basel, Switzerland). 19: 1378-93. PMID 24473203 DOI: 10.3390/molecules19021378  1
2014 Wang C, Weerapana E, Blewett MM, Cravatt BF. A chemoproteomic platform to quantitatively map targets of lipid-derived electrophiles. Nature Methods. 11: 79-85. PMID 24292485 DOI: 10.1038/nmeth.2759  1
2014 Pace NJ, Weerapana E. A competitive chemical-proteomic platform to identify zinc-binding cysteines. Acs Chemical Biology. 9: 258-65. PMID 24111988 DOI: 10.1021/cb400622q  1
2014 Shannon DA, Weerapana E. Orphan PTMs: Rare, yet functionally important modifications of cysteine. Biopolymers. 101: 156-64. PMID 23564220 DOI: 10.1002/bip.22252  1
2014 Couvertier SM, Weerapana E. Cysteine-reactive chemical probes based on a modular 4-aminopiperidine scaffold Medchemcomm. 5: 358-362. DOI: 10.1039/c3md00289f  1
2014 Tamburini F, Kelly T, Weerapana E, Byers JA. Paper to Plastics: An Interdisciplinary Summer Outreach Project in Sustainability Journal of Chemical Education. 91: 1574-1579. DOI: 10.1021/ed400892t  1
2013 Schwaid AG, Shannon DA, Ma J, Slavoff SA, Levin JZ, Weerapana E, Saghatelian A. Chemoproteomic discovery of cysteine-containing human short open reading frames. Journal of the American Chemical Society. 135: 16750-3. PMID 24152191 DOI: 10.1021/ja406606j  1
2013 Child MA, Hall CI, Beck JR, Ofori LO, Albrow VE, Garland M, Bowyer PW, Bradley PJ, Powers JC, Boothroyd JC, Weerapana E, Bogyo M. Small-molecule inhibition of a depalmitoylase enhances Toxoplasma host-cell invasion. Nature Chemical Biology. 9: 651-6. PMID 23934245 DOI: 10.1038/nchembio.1315  1
2013 Lee BC, Péterfi Z, Hoffmann FW, Moore RE, Kaya A, Avanesov A, Tarrago L, Zhou Y, Weerapana E, Fomenko DE, Hoffmann PR, Gladyshev VN. MsrB1 and MICALs regulate actin assembly and macrophage function via reversible stereoselective methionine oxidation. Molecular Cell. 51: 397-404. PMID 23911929 DOI: 10.1016/j.molcel.2013.06.019  1
2013 Qian Y, Martell J, Pace NJ, Ballard TE, Johnson DS, Weerapana E. An isotopically tagged azobenzene-based cleavable linker for quantitative proteomics. Chembiochem : a European Journal of Chemical Biology. 14: 1410-4. PMID 23861326 DOI: 10.1002/cbic.201300396  1
2013 Gu C, Shannon DA, Colby T, Wang Z, Shabab M, Kumari S, Villamor JG, McLaughlin CJ, Weerapana E, Kaiser M, Cravatt BF, van der Hoorn RA. Chemical proteomics with sulfonyl fluoride probes reveals selective labeling of functional tyrosines in glutathione transferases. Chemistry & Biology. 20: 541-8. PMID 23601643 DOI: 10.1016/j.chembiol.2013.01.016  1
2013 Deng X, Weerapana E, Ulanovskaya O, Sun F, Liang H, Ji Q, Ye Y, Fu Y, Zhou L, Li J, Zhang H, Wang C, Alvarez S, Hicks LM, Lan L, et al. Proteome-wide quantification and characterization of oxidation-sensitive cysteines in pathogenic bacteria. Cell Host & Microbe. 13: 358-70. PMID 23498960 DOI: 10.1016/j.chom.2013.02.004  1
2013 Banerjee R, Pace NJ, Brown DR, Weerapana E. 1,3,5-Triazine as a modular scaffold for covalent inhibitors with streamlined target identification. Journal of the American Chemical Society. 135: 2497-500. PMID 23379904 DOI: 10.1021/ja400427e  1
2013 Pace NJ, Weerapana E. Diverse functional roles of reactive cysteines. Acs Chemical Biology. 8: 283-96. PMID 23163700 DOI: 10.1021/cb3005269  1
2013 Ramya TN, Weerapana E, Cravatt BF, Paulson JC. Glycoproteomics enabled by tagging sialic acid- or galactose-terminated glycans. Glycobiology. 23: 211-21. PMID 23070960 DOI: 10.1093/glycob/cws144  1
2013 Banerjee R, Brown DR, Weerapana E. Recent developments in the synthesis of bioactive 2,4,6-trisubstituted 1,3,5-triazines Synlett. 24: 1599-1605. DOI: 10.1055/s-0033-1339284  1
2012 Shannon DA, Gu C, McLaughlin CJ, Kaiser M, van der Hoorn RA, Weerapana E. Sulfonyl fluoride analogues as activity-based probes for serine proteases. Chembiochem : a European Journal of Chemical Biology. 13: 2327-30. PMID 23008217 DOI: 10.1002/cbic.201200531  1
2012 Pace NJ, Pimental DR, Weerapana E. An inhibitor of glutathione S-transferase omega 1 that selectively targets apoptotic cells. Angewandte Chemie (International Ed. in English). 51: 8365-8. PMID 22777685 DOI: 10.1002/anie.201203730  1
2012 Tarrago L, Kaya A, Weerapana E, Marino SM, Gladyshev VN. Methionine sulfoxide reductases preferentially reduce unfolded oxidized proteins and protect cells from oxidative protein unfolding. The Journal of Biological Chemistry. 287: 24448-59. PMID 22628550 DOI: 10.1074/jbc.M112.374520  1
2011 Hall CI, Reese ML, Weerapana E, Child MA, Bowyer PW, Albrow VE, Haraldsen JD, Phillips MR, Sandoval ED, Ward GE, Cravatt BF, Boothroyd JC, Bogyo M. Chemical genetic screen identifies Toxoplasma DJ-1 as a regulator of parasite secretion, attachment, and invasion. Proceedings of the National Academy of Sciences of the United States of America. 108: 10568-73. PMID 21670272 DOI: 10.1073/pnas.1105622108  1
2011 Bachovchin DA, Zuhl AM, Speers AE, Wolfe MR, Weerapana E, Brown SJ, Rosen H, Cravatt BF. Discovery and optimization of sulfonyl acrylonitriles as selective, covalent inhibitors of protein phosphatase methylesterase-1. Journal of Medicinal Chemistry. 54: 5229-36. PMID 21639134 DOI: 10.1021/jm200502u  1
2011 Ahn K, Smith SE, Liimatta MB, Beidler D, Sadagopan N, Dudley DT, Young T, Wren P, Zhang Y, Swaney S, Van Becelaere K, Blankman JL, Nomura DK, Bhattachar SN, Stiff C, ... ... Weerapana E, et al. Mechanistic and pharmacological characterization of PF-04457845: a highly potent and selective fatty acid amide hydrolase inhibitor that reduces inflammatory and noninflammatory pain. The Journal of Pharmacology and Experimental Therapeutics. 338: 114-24. PMID 21505060 DOI: 10.1124/jpet.111.180257  1
2010 Weerapana E, Wang C, Simon GM, Richter F, Khare S, Dillon MB, Bachovchin DA, Mowen K, Baker D, Cravatt BF. Quantitative reactivity profiling predicts functional cysteines in proteomes. Nature. 468: 790-5. PMID 21085121 DOI: 10.1038/nature09472  1
2010 Wurdak H, Zhu S, Min KH, Aimone L, Lairson LL, Watson J, Chopiuk G, Demas J, Charette B, Halder R, Weerapana E, Cravatt BF, Cline HT, Peters EC, Zhang J, et al. A small molecule accelerates neuronal differentiation in the adult rat. Proceedings of the National Academy of Sciences of the United States of America. 107: 16542-7. PMID 20823227 DOI: 10.1073/pnas.1010300107  1
2010 Johnson DS, Weerapana E, Cravatt BF. Strategies for discovering and derisking covalent, irreversible enzyme inhibitors. Future Medicinal Chemistry. 2: 949-64. PMID 20640225 DOI: 10.4155/fmc.10.21  1
2010 Ramya TN, Weerapana E, Liao L, Zeng Y, Tateno H, Liao L, Yates JR, Cravatt BF, Paulson JC. In situ trans ligands of CD22 identified by glycan-protein photocross-linking-enabled proteomics. Molecular & Cellular Proteomics : McP. 9: 1339-51. PMID 20172905 DOI: 10.1074/mcp.M900461-MCP200  1
2009 Ahn K, Johnson DS, Mileni M, Beidler D, Long JZ, McKinney MK, Weerapana E, Sadagopan N, Liimatta M, Smith SE, Lazerwith S, Stiff C, Kamtekar S, Bhattacharya K, Zhang Y, et al. Discovery and characterization of a highly selective FAAH inhibitor that reduces inflammatory pain. Chemistry & Biology. 16: 411-20. PMID 19389627 DOI: 10.1016/j.chembiol.2009.02.013  1
2008 Weerapana E, Simon GM, Cravatt BF. Disparate proteome reactivity profiles of carbon electrophiles. Nature Chemical Biology. 4: 405-7. PMID 18488014 DOI: 10.1038/nchembio.91  1
2007 Chen MM, Weerapana E, Ciepichal E, Stupak J, Reid CW, Swiezewska E, Imperiali B. Polyisoprenol specificity in the Campylobacter jejuni N-linked glycosylation pathway. Biochemistry. 46: 14342-8. PMID 18034500 DOI: 10.1021/bi701956x  1
2007 Weerapana E, Speers AE, Cravatt BF. Tandem orthogonal proteolysis-activity-based protein profiling (TOP-ABPP)--a general method for mapping sites of probe modification in proteomes. Nature Protocols. 2: 1414-25. PMID 17545978 DOI: 10.1038/nprot.2007.194  1
2007 Hanson SR, Hsu TL, Weerapana E, Kishikawa K, Simon GM, Cravatt BF, Wong CH. Tailored glycoproteomics and glycan site mapping using saccharide-selective bioorthogonal probes. Journal of the American Chemical Society. 129: 7266-7. PMID 17506567 DOI: 10.1021/ja0724083  1
2006 Glover KJ, Weerapana E, Chen MM, Imperiali B. Direct biochemical evidence for the utilization of UDP-bacillosamine by PglC, an essential glycosyl-1-phosphate transferase in the Campylobacter jejuni N-linked glycosylation pathway. Biochemistry. 45: 5343-50. PMID 16618123 DOI: 10.1021/bi0602056  1
2006 Weerapana E, Imperiali B. Asparagine-linked protein glycosylation: from eukaryotic to prokaryotic systems. Glycobiology. 16: 91R-101R. PMID 16510493 DOI: 10.1093/glycob/cwj099  1
2005 Glover KJ, Weerapana E, Numao S, Imperiali B. Chemoenzymatic synthesis of glycopeptides with PglB, a bacterial oligosaccharyl transferase from Campylobacter jejuni. Chemistry & Biology. 12: 1311-5. PMID 16356848 DOI: 10.1016/j.chembiol.2005.10.004  1
2005 Weerapana E, Glover KJ, Chen MM, Imperiali B. Investigating bacterial N-linked glycosylation: synthesis and glycosyl acceptor activity of the undecaprenyl pyrophosphate-linked bacillosamine. Journal of the American Chemical Society. 127: 13766-7. PMID 16201778 DOI: 10.1021/ja054265v  1
2005 Glover KJ, Weerapana E, Imperiali B. In vitro assembly of the undecaprenylpyrophosphate-linked heptasaccharide for prokaryotic N-linked glycosylation. Proceedings of the National Academy of Sciences of the United States of America. 102: 14255-9. PMID 16186480 DOI: 10.1073/pnas.0507311102  1
2003 Weerapana E, Imperiali B. Peptides to peptidomimetics: towards the design and synthesis of bioavailable inhibitors of oligosaccharyl transferase. Organic & Biomolecular Chemistry. 1: 93-9. PMID 12929394 DOI: 10.1039/b209342a  1
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