Year |
Citation |
Score |
2018 |
Sieber JD, Rodriguez S, Frutos R, Buono F, Zhang Y, Li N, Qu B, Premasiri A, Li Z, Han ZS, Xu Y, Byrne D, Haddad N, Lorenz J, Grinberg N, ... ... Mulder J, et al. Development of a Scalable, Chromatography-Free Synthesis of t-Bu-SMS-Phos and Application to the Synthesis of an Important Chiral CF3-Alcohol Derivative in High Enantioselectivity Using Rh-Catalyzed Asymmetric Hydrogenation. The Journal of Organic Chemistry. PMID 29323903 DOI: 10.1021/Acs.Joc.7B03022 |
0.462 |
|
2017 |
Mulder JA, Gao J, Fandrick KR, Zeng X, Desrosiers J, Patel ND, Li Z, Rodriguez S, Lorenz JC, Wang J, Ma S, Fandrick DR, Grinberg N, Lee H, Bosanac T, et al. Early Development Scale-Up of a Structurally-Challenging 5-Lipoxygenase Activating Protein (FLAP) Inhibitor Organic Process Research & Development. 21: 1427-1434. DOI: 10.1021/Acs.Oprd.7B00202 |
0.374 |
|
2016 |
Frutos RP, Tampone TG, Mulder JA, Rodriguez S, Yee NK, Yang B, Senanayake CH. Development of a Practical Process for the Synthesis of PDE4 Inhibitors Organic Process Research & Development. 20: 982-988. DOI: 10.1021/Acs.Oprd.6B00104 |
0.351 |
|
2016 |
Patel ND, Zhang Y, Gao J, Sidhu K, Lorenz JC, Fandrick KR, Mulder JA, Herbage MA, Li Z, Ma S, Lee H, Grinberg N, Song JJ, Busacca CA, Yee NK, et al. Development of an Efficient Synthesis of (2-Aminopyrimidin-5-yl) Boronic Acid Organic Process Research and Development. 20: 95-99. DOI: 10.1021/Acs.Oprd.5B00360 |
0.392 |
|
2015 |
Fandrick KR, Mulder JA, Patel ND, Gao J, Konrad M, Archer E, Buono FG, Duran A, Schmid R, Daeubler J, Desrosiers JN, Zeng X, Rodriguez S, Ma S, Qu B, et al. Development of an asymmetric synthesis of a chiral quaternary FLAP inhibitor. The Journal of Organic Chemistry. 80: 1651-60. PMID 25562342 DOI: 10.1021/Jo502550H |
0.466 |
|
2015 |
Snieckus V, Tsai A, Fandrick DR, Sanyal S, Kaloko J, Mulder JA, Wang Y, Wu L, Lee H, Roschangar F, Hoffmann M, Senanayake CH. Selective Synthesis of 3- or 5-Substituted Aminopyrazoles Synfacts. 11: 919-919. DOI: 10.1055/S-0035-1560156 |
0.392 |
|
2014 |
Zeng X, Gao JJ, Song JJ, Ma S, Desrosiers JN, Mulder JA, Rodriguez S, Herbage MA, Haddad N, Qu B, Fandrick KR, Grinberg N, Lee H, Wei X, Yee NK, et al. Remarkable enhancement of enantioselectivity in the asymmetric conjugate addition of dimethylzinc to (Z)-nitroalkenes with a catalytic [(MeCN)₄Cu]PF₆-Hoveyda ligand complex. Angewandte Chemie (International Ed. in English). 53: 12153-7. PMID 25225113 DOI: 10.1002/Anie.201406247 |
0.398 |
|
2014 |
Fandrick KR, Patel ND, Mulder JA, Gao J, Konrad M, Archer E, Buono FG, Duran A, Schmid R, Daeubler J, Fandrick DR, Ma S, Grinberg N, Lee H, Busacca CA, et al. Addressing the configuration stability of lithiated secondary benzylic carbamates for the development of a noncryogenic stereospecific boronate rearrangement. Organic Letters. 16: 4360-3. PMID 25153850 DOI: 10.1021/Ol502060C |
0.376 |
|
2013 |
Frutos RP, Wei X, Patel ND, Tampone TG, Mulder JA, Busacca CA, Senanayake CH. One-pot synthesis of 2,5-disubstituted pyrimidines from nitriles. The Journal of Organic Chemistry. 78: 5800-3. PMID 23656541 DOI: 10.1021/Jo400720P |
0.403 |
|
2013 |
Mulder JA, Frutos RP, Patel ND, Qu B, Sun X, Tampone TG, Gao J, Sarvestani M, Eriksson MC, Haddad N, Shen S, Song JJ, Senanayake CH. Development of a safe and economical synthesis of methyl 6-chloro-5-(trifluoromethyl)nicotinate: Trifluoromethylation on kilogram scale Organic Process Research and Development. 17: 940-945. DOI: 10.1021/Op400061W |
0.333 |
|
2011 |
Frutos RP, Tampone T, Mulder JA, Xu Y, Reeves D, Wang X-, Zhang L, Krishnamurthy D, Senanayake CH. A Boronic Acid Catalyzed Route to Imidazoles. Synthesis ofLFA-1 Antagonists Synfacts. 2011: 603-603. DOI: 10.1055/S-0030-1260450 |
0.395 |
|
2011 |
Frutos RP, Tampone T, Mulder JA, Xu Y, Reeves D, Wang XJ, Zhang L, Krishnamurthy D, Senanayake CH. A new and practical boronic acid catalyzed intramolecular cyclodehydration of ureas for the synthesis of LFA-1 antagonists Tetrahedron Letters. 52: 2465-2467. DOI: 10.1016/J.Tetlet.2011.03.007 |
0.408 |
|
2008 |
Evans DA, Kvaernø L, Dunn TB, Beauchemin A, Raymer B, Mulder JA, Olhava EJ, Juhl M, Kagechika K, Favor DA. Total synthesis of (+)-azaspiracid-1. An exhibition of the intricacies of complex molecule synthesis. Journal of the American Chemical Society. 130: 16295-309. PMID 19006391 DOI: 10.1021/Ja804659N |
0.459 |
|
2007 |
Evans DA, Dunn TB, Kvaernø L, Beauchemin A, Raymer B, Olhava EJ, Mulder JA, Juhl M, Kagechika K, Favor DA. Total synthesis of (+)-azaspiracid-1. Part II: synthesis of the EFGHI sulfone and completion of the synthesis. Angewandte Chemie (International Ed. in English). 46: 4698-703. PMID 17546578 DOI: 10.1002/Anie.200701520 |
0.383 |
|
2007 |
Evans DA, Kvaernø L, Mulder JA, Raymer B, Dunn TB, Beauchemin A, Olhava EJ, Juhl M, Kagechika K. Total synthesis of (+)-azaspiracid-1. Part I: Synthesis of the fully elaborated ABCD aldehyde. Angewandte Chemie (International Ed. in English). 46: 4693-7. PMID 17546577 DOI: 10.1002/Anie.200701515 |
0.343 |
|
2007 |
Evans DA, Dunn TB, Kværnø L, Beauchemin A, Raymer B, Olhava EJ, Mulder JA, Juhl M, Kagechika K, Favor DA. Synthesis of (+)-Azaspiracid-1 Synfacts. 2007: 1117-1117. DOI: 10.1055/S-2007-991211 |
0.409 |
|
2006 |
Kurtz KCM, Frederick MO, Lambeth RH, Mulder JA, Tracey MR, Hsung RP. Synthesis of chiral allenes from ynamides through a highly stereoselective Saucy-Marbet rearrangement Tetrahedron. 62: 3928-3938. DOI: 10.1016/J.Tet.2005.11.087 |
0.791 |
|
2005 |
Xiong H, Tracey MR, Grebe T, Mulder JA, Hsung RP. Practical synthesis of novel chiral allenamides: (R)-4-phenyl-3-(1,2- propadienyl)oxazolidin-2-one Organic Syntheses. 81. DOI: 10.1002/0471264229.Os081.16 |
0.75 |
|
2004 |
Tracey MR, Zhang Y, Frederick MO, Mulder JA, Hsung RP. Sonogashira cross-couplings of ynamides. Syntheses of urethane- and sulfonamide-terminated conjugated phenylacetylenic systems. Organic Letters. 6: 2209-12. PMID 15200322 DOI: 10.1021/Ol0493251 |
0.762 |
|
2003 |
Frederick MO, Hsung RP, Lambeth RH, Mulder JA, Tracey MR. Highly stereoselective Saucy-Marbet rearrangement using chiral ynamides. Synthesis of highly substituted chiral homoallenyl alcohols. Organic Letters. 5: 2663-6. PMID 12868884 DOI: 10.1021/Ol030061C |
0.79 |
|
2003 |
Mulder JA, Kurtz KC, Hsung RP, Coverdale H, Frederick MO, Shen L, Zificsak CA. Highly stereoselective synthesis of novel alpha-haloenamides via a mild and efficient hydrohalogenation of ynamides. Organic Letters. 5: 1547-50. PMID 12713320 DOI: 10.1021/Ol0300266 |
0.737 |
|
2003 |
Frederick MO, Mulder JA, Tracey MR, Hsung RP, Huang J, Kurtz KC, Shen L, Douglas CJ. A copper-catalyzed C-N bond formation involving sp-hybridized carbons. A direct entry to chiral ynamides via N-alkynylation of amides. Journal of the American Chemical Society. 125: 2368-9. PMID 12603105 DOI: 10.1021/Ja021304J |
0.707 |
|
2003 |
Mulder JA, Kurtz KCM, Hsung RP. In search of an atom-economical synthesis of chiral ynamides Synlett. 1379-1390. DOI: 10.1055/S-2003-40817 |
0.579 |
|
2002 |
Huang J, Xiong H, Hsung RP, Rameshkumar C, Mulder JA, Grebe TP. The first successful base-promoted isomerization of propargyl amides to chiral ynamides. Applications in ring-closing metathesis of ene-ynamides and tandem RCM of diene-ynamides. Organic Letters. 4: 2417-20. PMID 12098261 DOI: 10.1021/Ol020097P |
0.699 |
|
2002 |
Mulder JA, Hsung RP, Frederick MO, Tracey MR, Zificsak CA. The first stereoselective Ficini-Claisen rearrangement using chiral ynamides. Organic Letters. 4: 1383-6. PMID 11950368 DOI: 10.1021/Ol020037J |
0.774 |
|
2002 |
Blankespoor RL, DeVries T, Hansen E, Kallemeyn JM, Klooster AM, Mulder JA, Smart RP, Vander Griend DA. Photochemical synthesis of aldehydes in the solid phase. The Journal of Organic Chemistry. 67: 2677-81. PMID 11950316 DOI: 10.1021/Jo025508U |
0.332 |
|
2001 |
Zificsak CA, Mulder JA, Hsung RP, Rameshkumar C, Wei LL. Recent advances in the chemistry of ynamines and ynamides Tetrahedron. 57: 7575-7606. DOI: 10.1016/S0040-4020(01)00681-0 |
0.724 |
|
2001 |
Wei LL, Mulder JA, Xiong H, Zificsak CA, Douglas CJ, Hsung RP. Efficient preparations of novel ynamides and allenamides Tetrahedron. 57: 459-466. DOI: 10.1016/S0040-4020(00)01014-0 |
0.769 |
|
2000 |
Xiong H, Hsung RP, Wei LL, Berry CR, Mulder JA, Stockwell B. The first regioselective alpha-deprotonation and functionalization of allenamides. An application in intramolecular Pauson-Khand-type cycloadditions. Organic Letters. 2: 2869-71. PMID 10964386 DOI: 10.1021/Ol000181+ |
0.735 |
|
2000 |
Zhu XY, Boiadjiev V, Mulder JA, Hsung RP, Major RC. Molecular assemblies on silicon surfaces via Si-O linkages Langmuir. 16: 6766-6772. DOI: 10.1021/La9915264 |
0.507 |
|
1999 |
Degen SJ, Mueller KL, Shen HC, Mulder JA, Golding GM, Wei LL, Zificsak CA, Neeno-Eckwall A, Hsung RP. Synthesis of dihydroxanthone derivatives and evaluation of their inhibitory activity against acetylcholinesterase: unique structural analogs of tacrine based on the BCD-ring of arisugacin. Bioorganic & Medicinal Chemistry Letters. 9: 973-8. PMID 10230623 DOI: 10.1016/S0960-894X(99)00115-8 |
0.753 |
|
1999 |
Zhu XY, Mulder JA, Hsung RP, Bergerson WF, Gasser A, Nguyen A. Integrating organic molecules to silicon surfaces Materials Research Society Symposium - Proceedings. 576: 177-182. DOI: 10.1557/Proc-576-177 |
0.467 |
|
1999 |
Kiely JD, Houston JE, Mulder JA, Hsung RP, Zhu XY. Adhesion, deformation and friction for self-assembled monolayers on Au and Si surfaces Tribology Letters. 7: 103-107. DOI: 10.1023/A:1019109117742 |
0.463 |
|
1999 |
Wei LL, Hsung RP, Xiong H, Mulder JA, Nkansah NT. First stereoselective inverse demand [4 + 2] cycloaddition reactions of novel chiral allenamides with heterodienes. Preparation of highly functionalized 2-arylpyranyl heterocycles Organic Letters. 1: 2145-2148. DOI: 10.1021/Ol990345Q |
0.742 |
|
1999 |
Hsung RP, Zificsak CA, Wei LL, Douglas CJ, Xiong H, Mulder JA. Lewis acid promoted hetero [2 + 2] cycloaddition reactions of aldehydes with 10-propynyl-9(10h)-acridone. A highly stereoselective synthesis of acrylic acid derivatives and 1,3-dienes using an electron deficient variant of ynamine Organic Letters. 1: 1237-1240. DOI: 10.1021/Ol990211C |
0.786 |
|
1999 |
Hsung RP, Wei LL, Sklenicka HM, Douglas CJ, McLaughlin MJ, Mulder JA, Yao LJ. Formal cycloaddition reactions of vinylogous amides with α,β-Unsaturated iminiums. A strategy for constructing piperidinyl heterocycles Organic Letters. 1: 509-512. DOI: 10.1021/Ol990107V |
0.764 |
|
1999 |
Bergerson WF, Mulder JA, Hsung RP, Zhu XY. Assembly of organic molecules on silicon surfaces via the Si-N linkage Journal of the American Chemical Society. 121: 454-455. DOI: 10.1021/Ja9832966 |
0.476 |
|
1998 |
Granum KA, Merkel G, Mulder JA, Debbins SA, Hsung RP. Reactivity of hindered 1,1-dimethylbutadienes towards α, β- unsaturated enones Tetrahedron Letters. 39: 9597-9600. DOI: 10.1016/S0040-4039(98)02333-8 |
0.562 |
|
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