Pascal Rigollier - Publications

Affiliations: 
1991 Michigan State University, East Lansing, MI 

13 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2014 Bassilana F, Carlson A, DaSilva JA, Grosshans B, Vidal S, Beck V, Wilmeringwetter B, Llamas LA, Showalter TB, Rigollier P, Bourret A, Ramamurthy A, Wu X, Harbinski F, Plonsky S, et al. Target identification for a Hedgehog pathway inhibitor reveals the receptor GPR39. Nature Chemical Biology. 10: 343-9. PMID 24633354 DOI: 10.1038/nchembio.1481  0.88
2010 Boettcher A, Ruedisser S, Erbel P, Vinzenz D, Schiering N, Hassiepen U, Rigollier P, Mayr LM, Woelcke J. Fragment-based screening by biochemical assays: Systematic feasibility studies with trypsin and MMP12. Journal of Biomolecular Screening. 15: 1029-41. PMID 20855559 DOI: 10.1177/1087057110380455  0.88
2010 Qin LY, Cole AG, Metzger A, Brescia MR, Saionz KW, Zhang JJ, Rigollier P, Wareing JR, Gstach H, Zimmermann J, Dolle RE, Baldwin JJ, Henderson I. A facile synthesis of novel 2-amino-6-arylmethyl-7-carboxamido-7,8- dihydropyrimido[5,4-f][1,4]thiazepin-5-ones Tetrahedron Letters. 51: 4486-4489. DOI: 10.1016/j.tetlet.2010.06.070  0.88
2007 Maibaum J, Stutz S, Göschke R, Rigollier P, Yamaguchi Y, Cumin F, Rahuel J, Baum HP, Cohen NC, Schnell CR, Fuhrer W, Gruetter MG, Schilling W, Wood JM. Structural modification of the P2' position of 2,7-dialkyl-substituted 5(S)-amino-4(S)-hydroxy-8-phenyl-octanecarboxamides: the discovery of aliskiren, a potent nonpeptide human renin inhibitor active after once daily dosing in marmosets. Journal of Medicinal Chemistry. 50: 4832-44. PMID 17824680 DOI: 10.1021/jm070316i  0.88
2007 Göschke R, Stutz S, Rasetti V, Cohen NC, Rahuel J, Rigollier P, Baum HP, Forgiarini P, Schnell CR, Wagner T, Gruetter MG, Fuhrer W, Schilling W, Cumin F, Wood JM, et al. Novel 2,7-dialkyl-substituted 5(S)-amino-4(S)-hydroxy-8-phenyl-octanecarboxamide transition state peptidomimetics are potent and orally active inhibitors of human renin. Journal of Medicinal Chemistry. 50: 4818-31. PMID 17824679 DOI: 10.1021/jm070314y  0.88
2005 Jacoby E, Schuffenhauer A, Popov M, Azzaoui K, Havill B, Schopfer U, Engeloch C, Stanek J, Acklin P, Rigollier P, Stoll F, Koch G, Meier P, Orain D, Giger R, et al. Key aspects of the Novartis compound collection enhancement project for the compilation of a comprehensive chemogenomics drug discovery screening collection. Current Topics in Medicinal Chemistry. 5: 397-411. PMID 15892682 DOI: 10.2174/1568026053828376  0.88
2004 Rueeger H, Gerspacher M, Buehlmayer P, Rigollier P, Yamaguchi Y, Schmidlin T, Whitebread S, Nuesslein-Hildesheim B, Nick H, Cricione L. Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 14: 2451-7. PMID 15109631 DOI: 10.1016/j.bmcl.2004.03.014  0.88
2003 Wood JM, Maibaum J, Rahuel J, Grütter MG, Cohen NC, Rasetti V, Rüger H, Göschke R, Stutz S, Fuhrer W, Schilling W, Rigollier P, Yamaguchi Y, Cumin F, Baum HP, et al. Structure-based design of aliskiren, a novel orally effective renin inhibitor. Biochemical and Biophysical Research Communications. 308: 698-705. PMID 12927775 DOI: 10.1016/S0006-291X(03)01451-7  0.88
2000 Rueeger H, Rigollier P, Yamaguchi Y, Schmidlin T, Schilling W, Criscione L, Whitebread S, Chiesi M, Walker MW, Dhanoa D, Islam I, Zhang J, Gluchowski C. Design, synthesis and SAR of a series of 2-substituted 4-amino-quinazoline neuropeptide Y Y5 receptor antagonists. Bioorganic & Medicinal Chemistry Letters. 10: 1175-9. PMID 10866375 DOI: 10.1016/S0960-894X(00)00177-3  0.88
1998 Criscione L, Rigollier P, Batzl-Hartmann C, Rüeger H, Stricker-Krongrad A, Wyss P, Brunner L, Whitebread S, Yamaguchi Y, Gerald C, Heurich RO, Walker MW, Chiesi M, Schilling W, Hofbauer KG, et al. Food intake in free-feeding and energy-deprived lean rats is mediated by the neuropeptide Y5 receptor. The Journal of Clinical Investigation. 102: 2136-45. PMID 9854049 DOI: 10.1172/JCI4188  0.88
1993 Magnus P, Rigollier P, Lacour J, Tobler H. New trialkylsilyl enol ether chemistry: Intramolecular [2 + 2] cyclizations of β-amido triisopropylsilyl enol ethers Journal of the American Chemical Society. 115: 12629-12630.  0.88
1992 Magnus P, Rigollier P. New mild methodology for the synthesis of α-phenylthio and α-phenylseleno ketones Tetrahedron Letters. 33: 6111-6114. DOI: 10.1016/S0040-4039(00)60019-9  0.88
1990 Rigollier P, Young JR, Fowley LA, Stille JR. Regioselective cyclopentane ring formation mediated by titanocene chloride Journal of the American Chemical Society. 112: 9441-9442.  0.88
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