| Year |
Citation |
Score |
| 2020 |
Sreenivasulu K, Chaudhari PS, Achanta S, Sud A, Dahanukar V, Cobley CJ, Llewellyn-Beard F, Bandichhor R. A Novel Synthesis of (R)-3-(t-Butoxycarbonylamino)-4-(2,4,5- trifluorophenyl)butanoic Acid, a Key Intermediate, and the Formal Synthesis of Sitagliptin phosphate. Chemistry, An Asian Journal. PMID 32128989 DOI: 10.1002/Asia.202000092 |
0.325 |
|
| 2018 |
Pachore SS, Ambhaikar NB, Siddaiah V, Khobare SR, Kumar S, Dahanukar VH, Kumar UKS. Successful utilization of
$$\upbeta $$
β
-ketonitrile in Biginelli reaction: synthesis of 5-cyanodihydropyrimidine Journal of Chemical Sciences. 130. DOI: 10.1007/S12039-018-1467-7 |
0.321 |
|
| 2017 |
Metil DS, Sonawane SP, Pachore SS, Mohammad A, Dahanukar VH, McCormack PJ, Reddy CV, Bandichhor R. Synthesis and Optimization of Canagliflozin by Employing Quality by Design (QbD) Principles Organic Process Research & Development. DOI: 10.1021/Acs.Oprd.7B00281 |
0.306 |
|
| 2017 |
Kallam SR, Eda VR, Sen S, Datrika R, Rapolu RK, Khobare S, Gajare V, Banda M, Khan RAR, Singh M, Lloyd M, Kandagatla B, Janagili MB, Tadikonda VP, Vidavalur S, ... ... Dahanukar VH, et al. A diastereoselective synthesis of boceprevir's gem-dimethyl bicyclic [3.1.0] proline intermediate from an insecticide ingredient cis-cypermethric acid Tetrahedron. 73: 4285-4294. DOI: 10.1016/J.Tet.2017.05.080 |
0.327 |
|
| 2015 |
Bernardi L, Fochi M, Carbone R, Martinelli A, Fox ME, Cobley CJ, Kandagatla B, Oruganti S, Dahanukar VH, Carlone A. Organocatalytic Asymmetric Conjugate Additions to Cyclopent-1-enecarbaldehyde: A Critical Assessment of Organocatalytic Approaches towards the Telaprevir Bicyclic Core. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26602867 DOI: 10.1002/Chem.201503352 |
0.306 |
|
| 2015 |
Bollikonda S, Mohanarangam S, Jinna RR, Kandirelli VK, Makthala L, Sen S, Chaplin DA, Lloyd RC, Mahoney T, Dahanukar VH, Oruganti S, Fox ME. An enantioselective formal synthesis of montelukast sodium. The Journal of Organic Chemistry. 80: 3891-901. PMID 25807000 DOI: 10.1021/Acs.Joc.5B00197 |
0.316 |
|
| 2015 |
Gutierrez O, Metil D, Dwivedi N, Gudimalla N, Chandrashekar ER, Dahanukar VH, Bhattacharya A, Bandichhor R, Kozlowski MC. Practical, asymmetric route to sitagliptin and derivatives: development and origin of diastereoselectivity. Organic Letters. 17: 1742-5. PMID 25799267 DOI: 10.1021/Acs.Orglett.5B00520 |
0.331 |
|
| 2014 |
Meruva SB, Mekala R, Raghunadh A, Raghavendra Rao K, Dahanukar VH, Pratap TV, Syam Kumar UK, Dubey PK. Synthesis of tetrahedral diarylheptanoid ent-diospongin A and epimer-diospongin B by employing Julia-Kocienski olefination Tetrahedron Letters. 4739-4741. DOI: 10.1016/J.Tetlet.2014.06.112 |
0.321 |
|
| 2014 |
Babu MS, Raghunadh A, Ramulu K, Dahanukar VH, Syam Kumar UK, Dubey PK. A practical and enantiospecific synthesis of (-)-(R)- and (+)-(S)-piperidin-3-ols Helvetica Chimica Acta. 97: 1507-1515. DOI: 10.1002/Hlca.201400008 |
0.328 |
|
| 2008 |
Shanmugapriya D, Shankar R, Satyanarayana G, Dahanukar VH, Kumar UKS, Vembu N. Aerial oxidation of 2,2-dibromo-1-aryl and heteroaryl ethanones: A facile synthesis of aryl and heteroaryl α-keto amides Synlett. 2945-2950. DOI: 10.1055/S-0028-1087353 |
0.309 |
|
| 2004 |
Zavialov IA, Dahanukar VH, Nguyen H, Orr C, Zhang F, Andrews DR. New and practical method for synthesis of 1- and 1,3-substituted xanthines. Organic Letters. 6: 2237-40. PMID 15200329 DOI: 10.1021/Ol049272N |
0.357 |
|
| 2001 |
Grunewald GL, Dahanukar VH, Criscione KR. Effects of a 3-alkyl-, 4-hydroxy- and/or 8-aromatic-substituent on the phenylethanolamine N-methyltransferase inhibitor potency and alpha2-adrenoceptor affinity of 2,3,4,5-tetrahydro-1H-2-benzazepines. Bioorganic & Medicinal Chemistry. 9: 1957-65. PMID 11504632 DOI: 10.1016/S0968-0896(01)00112-2 |
0.692 |
|
| 1999 |
Grunewald GL, Caldwell TM, Li Q, Dahanukar VH, McNeil B, Criscione KR. Enantiospecific synthesis of 3-fluoromethyl-, 3-hydroxymethyl-, and 3-chloromethyl-1,2,3,4-tetrahydroisoquinolines as selective inhibitors of phenylethanolamine N-methyltransferase versus the alpha(2)-adrenoceptor. Journal of Medicinal Chemistry. 42: 4351-61. PMID 10543879 DOI: 10.1021/Jm990086A |
0.765 |
|
| 1999 |
Grunewald GL, Dahanukar VH, Teoh B, Criscione KR. 3,7-Disubstituted-1,2,3,4-tetrahydroisoquinolines display remarkable potency and selectivity as inhibitors of phenylethanolamine N-methyltransferase versus the alpha2-adrenoceptor. Journal of Medicinal Chemistry. 42: 1982-90. PMID 10354406 DOI: 10.1021/Jm9807252 |
0.745 |
|
| 1999 |
Grunewald GL, Caldwell TM, Dahanukar VH, Jalluri RK, Criscione KR. Comparative molecular field analysis (CoMFA) models of phenylethanolamine N-methyltransferase (PNMT) and the alpha2-adrenoceptor: the development of new, highly selective inhibitors of PNMT. Bioorganic & Medicinal Chemistry Letters. 9: 481-6. PMID 10091706 DOI: 10.1016/S0960-894X(99)00022-0 |
0.67 |
|
| 1999 |
Grunewald GL, Dahanukar VH, Jalluri RK, Criscione KR. Synthesis, biochemical evaluation, and classical and three-dimensional quantitative structure-activity relationship studies of 7-substituted-1,2,3,4-tetrahydroisoquinolines and their relative affinities toward phenylethanolamine N-methyltransferase and the alpha2-adrenoceptor. Journal of Medicinal Chemistry. 42: 118-34. PMID 9888838 DOI: 10.1021/Jm980429P |
0.737 |
|
| 1997 |
Grunewald GL, Dahanukar VH, Caldwell TM, Criscione KR. Examination of the role of the acidic hydrogen in imparting selectivity of 7-(aminosulfonyl)-1,2,3,4-tetrahydroisoquinoline (SK&F 29661) toward inhibition of phenylethanolamine N-methyltransferase vs the alpha 2-adrenoceptor. Journal of Medicinal Chemistry. 40: 3997-4005. PMID 9406590 DOI: 10.1021/Jm960235E |
0.762 |
|
| 1996 |
Dahanukar VH, Rychnovsky SD. General Synthesis of alpha-Acetoxy Ethers from Esters by DIBALH Reduction and Acetylation. The Journal of Organic Chemistry. 61: 8317-8320. PMID 11667826 DOI: 10.1021/Jo961205M |
0.48 |
|
| 1996 |
Grunewald GL, Dahanukar VH, Ching P, Criscione KR. Effect of ring size or an additional heteroatom on the potency and selectivity of bicyclic benzylamine-type inhibitors of phenylethanolamine N-methyltransferase. Journal of Medicinal Chemistry. 39: 3539-46. PMID 8784452 DOI: 10.1021/Jm9508292 |
0.731 |
|
| 1994 |
Grunewald GL, Dahanukar VH. Synthesis of 3-alkyl-8-substituted- and 4-hydroxy-8-substituted-2,3,4,5-tetrahydro-1H-2-benzazepines Journal of Heterocyclic Chemistry. 31: 1609-1617. DOI: 10.1002/Jhet.5570310656 |
0.569 |
|
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