Year |
Citation |
Score |
2010 |
Williams DR, Clark MP. ChemInform Abstract: The Macrocyclic Domain of Phorboxazole A. A Stereoselective Synthesis of the C1-C32 Macrolactone. Cheminform. 30: no-no. DOI: 10.1002/chin.199925219 |
0.447 |
|
2010 |
Williams DR, Clark MP, Berliner MA. ChemInform Abstract: Synthetic Studies Toward Phorboxazole A. Stereoselective Synthesis of the C3-C19 and C20-C32 Subunits. Cheminform. 30: no-no. DOI: 10.1002/chin.199925218 |
0.733 |
|
2010 |
WILLIAMS DR, BROOKS DA, MEYER KG, CLARK MP. ChemInform Abstract: Asymmetric Allylation. An Effective Strategy for the Convergent Synthesis of Highly Functionalized Homoallylic Alcohols Cheminform. 30: no-no. DOI: 10.1002/chin.199901261 |
0.764 |
|
2007 |
Clark MP, George KM, Bookland RG, Chen J, Laughlin SK, Thakur KD, Lee W, Davis JR, Cabrera EJ, Brugel TA, VanRens JC, Laufersweiler MJ, Maier JA, Sabat MP, Golebiowski A, et al. Development of new pyrrolopyrimidine-based inhibitors of Janus kinase 3 (JAK3). Bioorganic & Medicinal Chemistry Letters. 17: 1250-3. PMID 17189692 DOI: 10.1016/j.bmcl.2006.12.018 |
0.685 |
|
2006 |
Sabat M, Vanrens JC, Clark MP, Brugel TA, Maier J, Bookland RG, Laufersweiler MJ, Laughlin SK, Golebiowski A, De B, Hsieh LC, Walter RL, Mekel MJ, Janusz MJ. The development of novel C-2, C-8, and N-9 trisubstituted purines as inhibitors of TNF-alpha production. Bioorganic & Medicinal Chemistry Letters. 16: 4360-5. PMID 16750367 DOI: 10.1016/j.bmcl.2006.05.050 |
0.765 |
|
2006 |
Brugel TA, Maier JA, Clark MP, Sabat M, Golebiowski A, Bookland RG, Laufersweiler MJ, Laughlin SK, Vanrens JC, De B, Hsieh LC, Mekel MJ, Janusz MJ. Development of N-2,4-pyrimidine-N-phenyl-N'-phenyl ureas as inhibitors of tumor necrosis factor alpha (TNF-alpha) synthesis. Part 1. Bioorganic & Medicinal Chemistry Letters. 16: 3510-3. PMID 16632356 DOI: 10.1016/j.bmcl.2006.03.095 |
0.744 |
|
2006 |
Maier JA, Brugel TA, Clark MP, Sabat M, Golebiowski A, Bookland RG, Laufersweiler MJ, Laughlin SK, Vanrens JC, De B, Hsieh LC, Brown KK, Juergens K, Walter RL, Janusz MJ. Development of N-2,4-pyrimidine-N-phenyl-N'-alkyl ureas as orally active inhibitors of tumor necrosis factor alpha (TNF-alpha) synthesis. Part 2. Bioorganic & Medicinal Chemistry Letters. 16: 3514-8. PMID 16632350 DOI: 10.1016/j.bmcl.2006.03.096 |
0.746 |
|
2006 |
Brugel TA, Hudlicky T, Clark MP, Golebiowski A, Sabat M, Endoma MAA, Bui V, Adams D, Laufersweiler MJ, Maier JA, Bookland RG, De B. Convergent synthesis of 2,3-bisarylpyrazolones through cyclization of bisacylated pyrazolidines and hydrazines Tetrahedron Letters. 47: 3195-3198. DOI: 10.1016/J.Tetlet.2006.03.063 |
0.731 |
|
2006 |
Brugel TA, Maier JA, Clark MP, Sabat M, Golebiowski A, Bookland RG, Laufersweiler MJ, Laughlin SK, VanRens JC, De B, Hsieh LC, Mekel MJ, Janusz MJ. Corrigendum to "Development of N-2,4-pyrimidine-N-phenyl-N′-phenyl ureas as inhibitors of tumor necrosis factor alpha (TNF-α) synthesis. Part 1" [Bioorg. Med. Chem. Lett. 16 (2006) 3510-3513] (DOI:10.1016/j.bmcl.2006.03.095) Bioorganic and Medicinal Chemistry Letters. 16: 4700. DOI: 10.1016/j.bmcl.2006.06.013 |
0.736 |
|
2005 |
Williams DR, Berliner MA, Stroup BW, Nag PP, Clark MP. Samarium Barbier reactions of alpha-iodomethyloxazoles and thiazoles with aliphatic aldehydes. Organic Letters. 7: 4099-102. PMID 16146361 DOI: 10.1021/Ol051345V |
0.782 |
|
2005 |
Laughlin SK, Clark MP, Djung JF, Golebiowski A, Brugel TA, Sabat M, Bookland RG, Laufersweiler MJ, VanRens JC, Townes JA, De B, Hsieh LC, Xu SC, Walter RL, Mekel MJ, et al. The development of new isoxazolone based inhibitors of tumor necrosis factor-alpha (TNF-alpha) production. Bioorganic & Medicinal Chemistry Letters. 15: 2399-403. PMID 15837333 DOI: 10.1016/j.bmcl.2005.02.066 |
0.742 |
|
2005 |
Golebiowski A, Townes JA, Laufersweiler MJ, Brugel TA, Clark MP, Clark CM, Djung JF, Laughlin SK, Sabat MP, Bookland RG, VanRens JC, De B, Hsieh LC, Janusz MJ, Walter RL, et al. The development of monocyclic pyrazolone based cytokine synthesis inhibitors. Bioorganic & Medicinal Chemistry Letters. 15: 2285-9. PMID 15837310 DOI: 10.1016/j.bmcl.2005.03.007 |
0.743 |
|
2004 |
Townes JA, Golebiowski A, Clark MP, Laufersweiler MJ, Brugel TA, Sabat M, Bookland RG, Laughlin SK, VanRens JC, De B, Hsieh LC, Xu SC, Janusz MJ, Walter RL. The development of new bicyclic pyrazole-based cytokine synthesis inhibitors. Bioorganic & Medicinal Chemistry Letters. 14: 4945-8. PMID 15341957 DOI: 10.1016/j.bmcl.2004.07.024 |
0.748 |
|
2004 |
Williams DR, Kiryanov AA, Emde U, Clark MP, Berliner MA, Reeves JT. Studies of stereocontrolled allylation reactions for the total synthesis of phorboxazole A. Proceedings of the National Academy of Sciences of the United States of America. 101: 12058-63. PMID 15277662 DOI: 10.1073/Pnas.0402477101 |
0.735 |
|
2004 |
Laufersweiler MJ, Brugel TA, Clark MP, Golebiowski A, Bookland RG, Laughlin SK, Sabat MP, Townes JA, VanRens JC, De B, Hsieh LC, Heitmeyer SA, Juergens K, Brown KK, Mekel MJ, et al. The development of novel inhibitors of tumor necrosis factor-alpha (TNF-alpha) production based on substituted [5,5]-bicyclic pyrazolones. Bioorganic & Medicinal Chemistry Letters. 14: 4267-72. PMID 15261284 DOI: 10.1016/j.bmcl.2004.06.001 |
0.739 |
|
2004 |
Clark MP, Laughlin SK, Laufersweiler MJ, Bookland RG, Brugel TA, Golebiowski A, Sabat MP, Townes JA, VanRens JC, Djung JF, Natchus MG, De B, Hsieh LC, Xu SC, Walter RL, et al. Development of orally bioavailable bicyclic pyrazolones as inhibitors of tumor necrosis factor-alpha production. Journal of Medicinal Chemistry. 47: 2724-7. PMID 15139749 DOI: 10.1021/jm049968m |
0.738 |
|
2003 |
Tullis JS, VanRens JC, Natchus MG, Clark MP, De B, Hsieh LC, Janusz MJ. The development of new triazole based inhibitors of tumor necrosis factor-alpha (TNF-alpha) production. Bioorganic & Medicinal Chemistry Letters. 13: 1665-8. PMID 12729637 DOI: 10.1016/S0960-894X(03)00238-5 |
0.356 |
|
2003 |
Williams DR, Kiryanov AA, Emde U, Clark MP, Berliner MA, Reeves JT. Total synthesis of phorboxazole A. Angewandte Chemie (International Ed. in English). 42: 1258-62. PMID 12645057 DOI: 10.1002/anie.200390322 |
0.714 |
|
2001 |
Williams DR, Patnaik S, Clark MP. Total synthesis of cystothiazoles A and C. The Journal of Organic Chemistry. 66: 8463-9. PMID 11735526 DOI: 10.1021/Jo0106905 |
0.681 |
|
2000 |
Williams DR, Clark MP, Emde U, Berliner MA. Synthetic studies toward phorboxazole A. stereoselective synthesis of the C(28)-C(46) side chain fragment. Organic Letters. 2: 3023-6. PMID 10986098 DOI: 10.1021/Ol0063656 |
0.773 |
|
1999 |
Williams DR, Clark MP. The macrocyclic domain of phorboxazole A. A stereoselective synthesis of the C1-C32 macrolactone Tetrahedron Letters. 40: 2291-2294. DOI: 10.1016/S0040-4039(99)00210-5 |
0.456 |
|
1999 |
Williams DR, Clark MP, Berliner MA. Synthetic studies toward Phorboxazole A. Stereoselective synthesis of the C3-C19 and C20-C32 subunits Tetrahedron Letters. 40: 2287-2290. DOI: 10.1016/S0040-4039(99)00209-9 |
0.764 |
|
1998 |
Williams DR, Clark MP. Synthesis of atovaquone Tetrahedron Letters. 39: 7629-7632. DOI: 10.1016/S0040-4039(98)01691-8 |
0.366 |
|
1998 |
Williams DR, Clark MP. Synthesis of atovaquone Tetrahedron Letters. 39: 7629-7632. DOI: 10.1016/S0040-4039(98)01691-8 |
0.458 |
|
1998 |
Williams DR, Brooks DA, Meyer KG, Clark MP. Asymmetric allylation. An effective strategy for the convergent synthesis of highly functionalized homoallylic alcohols Tetrahedron Letters. 39: 7251-7254. DOI: 10.1016/S0040-4039(98)01557-3 |
0.765 |
|
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