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Anthony Mastracchio - Publications

Affiliations: 
2010 Princeton University, Princeton, NJ 
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16 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2019 Mastracchio A, Lai C, Torrent M, Bromberg K, Buchanan FG, Ferguson D, Bontcheva V, Johnson EF, Lasko L, Maag D, Soni N, Shoemaker AR, Penning TD. Investigation of biaryl heterocycles as inhibitors of Wee1 kinase. Bioorganic & Medicinal Chemistry Letters. PMID 31014911 DOI: 10.1016/J.Bmcl.2019.04.017  0.327
2011 Jones SB, Simmons B, Mastracchio A, MacMillan DWC. Collective synthesis of natural products by means of organocascade catalysis Nature. 475: 183-188. PMID 21753848 DOI: 10.1038/Nature10232  0.683
2011 Jones SB, Simmons B, Mastracchio A, MacMillan DWC. Collective, Organocatalytic Syntheses of Natural Products:Strychnos Alkaloids Synfacts. 2011: 1125-1125. DOI: 10.1055/S-0030-1261119  0.634
2010 Mastracchio A, Warkentin AA, Walji AM, MacMillan DW. Direct and enantioselective {alpha}-allylation of ketones via singly occupied molecular orbital (SOMO) catalysis. Proceedings of the National Academy of Sciences of the United States of America. 107: 20648-51. PMID 20921367 DOI: 10.1073/Pnas.1002845107  0.646
2010 Mastracchio A, Warkentin AA, Walji AM, MacMillan DWC. Direct and enantioselective a-allylation of ketones via singly occupied molecular orbital (SOMO) catalysis Proceedings of the National Academy of Sciences of the United States of America. 107: 20648-20651. DOI: 10.1073/pnas.1002845107  0.696
2009 Edmondson SD, Mastracchio A, Cox JM, Eiermann GJ, He H, Lyons KA, Patel RA, Patel SB, Petrov A, Scapin G, Wu JK, Xu S, Zhu B, Thornberry NA, Roy RS, et al. Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors. Bioorganic & Medicinal Chemistry Letters. 19: 4097-101. PMID 19539471 DOI: 10.1016/J.Bmcl.2009.06.011  0.323
2008 Gallant M, Chauret N, Claveau D, Day S, Deschênes D, Dubé D, Huang Z, Lacombe P, Laliberté F, Lévesque JF, Liu S, Macdonald D, Mancini J, Masson P, Mastracchio A, et al. Design, synthesis, and biological evaluation of 8-biarylquinolines: a novel class of PDE4 inhibitors. Bioorganic & Medicinal Chemistry Letters. 18: 1407-12. PMID 18207397 DOI: 10.1016/J.Bmcl.2008.01.004  0.331
2007 Kim D, Kowalchick JE, Edmondson SD, Mastracchio A, Xu J, Eiermann GJ, Leiting B, Wu JK, Pryor KD, Patel RA, He H, Lyons KA, Thornberry NA, Weber AE. Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: close analogs of JANUVIA (sitagliptin phosphate). Bioorganic & Medicinal Chemistry Letters. 17: 3373-7. PMID 17434732 DOI: 10.1016/J.Bmcl.2007.03.098  0.332
2007 Beeson TD, Mastracchio A, Hong JB, Ashton K, MacMillan DWC. Enantioselective organocatalysis using SOMO activation Science. 316: 582-585. PMID 17395791 DOI: 10.1055/S-2007-968564  0.668
2006 Edmondson SD, Mastracchio A, Mathvink RJ, He J, Harper B, Park YJ, Beconi M, Di Salvo J, Eiermann GJ, He H, Leiting B, Leone JF, Levorse DA, Lyons K, Patel RA, et al. (2S,3S)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-N,N-dimethyl-4-oxo-2-(4-[1,2,4]triazolo[1,5-a]-pyridin-6-ylphenyl)butanamide: a selective alpha-amino amide dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes. Journal of Medicinal Chemistry. 49: 3614-27. PMID 16759103 DOI: 10.1021/Jm060015T  0.312
2006 Xu J, Wei L, Mathvink R, Edmondson SD, Mastracchio A, Eiermann GJ, He H, Leone JF, Leiting B, Lyons KA, Marsilio F, Patel RA, Petrov A, Wu JK, Thornberry NA, et al. Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitors. Bioorganic & Medicinal Chemistry Letters. 16: 1346-9. PMID 16332437 DOI: 10.1016/J.Bmcl.2005.11.052  0.342
2006 Conlon DA, Drahus-Paone A, Ho GJ, Pipik B, Helmy R, McNamara JM, Shi YJ, Williams JM, Macdonald D, Deschênes D, Gallant M, Mastracchio A, Roy B, Scheigetz J. Process development and large-scale synthesis of a PDE4 inhibitor Organic Process Research and Development. 10: 36-45. DOI: 10.1021/Op050116L  0.401
2005 Macdonald D, Mastracchio A, Perrier H, Dubé D, Gallant M, Lacombe P, Deschênes D, Roy B, Scheigetz J, Bateman K, Li C, Trimble LA, Day S, Chauret N, Nicoll-Griffith DA, et al. Discovery of a substituted 8-arylquinoline series of PDE4 inhibitors: structure-activity relationship, optimization, and identification of a highly potent, well tolerated, PDE4 inhibitor. Bioorganic & Medicinal Chemistry Letters. 15: 5241-6. PMID 16168647 DOI: 10.1016/J.Bmcl.2005.08.036  0.324
2005 Edmondson SD, Mastracchio A, Duffy JL, Eiermann GJ, He H, Ita I, Leiting B, Leone JF, Lyons KA, Makarewicz AM, Patel RA, Petrov A, Wu JK, Thornberry NA, Weber AE. Discovery of potent and selective orally bioavailable beta-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors. Bioorganic & Medicinal Chemistry Letters. 15: 3048-52. PMID 15908206 DOI: 10.1016/J.Bmcl.2005.04.028  0.357
2004 Mastracchio A, Parmee ER, Leiting B, Marsilio F, Patel R, Thornberry NA, Weber AE, Edmondson SD. Heterocycle fused cyclohexylglycine derivatives as novel dipeptidyl peptidase-IV inhibitors Heterocycles. 62: 203-206. DOI: 10.3987/Com-03-S(P)50  0.337
2000 Edmondson SD, Mastracchio A, Parmee ER. Palladium-catalyzed coupling of vinylogous amides with aryl halides: applications to the synthesis of heterocycles Organic Letters. 2: 1109-12. PMID 10804566  0.316
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