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Year Citation  Score
2020 Fischer NH, Nielsen DS, Palmer D, Meldal M, Diness F. C-Terminal lactamization of peptides. Chemical Communications (Cambridge, England). PMID 33367306 DOI: 10.1039/d0cc06018f  0.714
2020 Wang Y, Oliveira MT, Madsen D, Thompson A, Meldal M, Diness F. Dihydroquinazolinones via A3-Type Reactions of N-Carbamoyliminium Ions. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32790088 DOI: 10.1002/Chem.202003117  0.795
2020 Madsen D, Jørgensen FP, Palmer D, Roux M, Olsen JV, Bols M, Schoffelen S, Diness F, Meldal M. Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12. Acs Combinatorial Science. PMID 32027120 DOI: 10.1021/Acscombsci.9B00197  0.807
2019 Jorgesen FP, Madsen D, Meldal M, Olsen JV, Petersen M, Granhøj J, Bols M. Synthesis of Shld derivatives, their binding the Destabilizing Domain and influence on protein accumulation in transgenic plants. Journal of Medicinal Chemistry. PMID 31059249 DOI: 10.1021/Acs.Jmedchem.9B00497  0.635
2019 Jacobsen CBB, Nielsen DS, Meldal M, Diness F. Azotides as Modular Peptide-Based Ligands for Asymmetric Lewis Acid Catalysis. The Journal of Organic Chemistry. PMID 31033291 DOI: 10.1021/Acs.Joc.9B00732  0.718
2019 Kofoed C, Riesenberg S, Šmolíková J, Meldal M, Schoffelen S. Semisynthesis of an Active Enzyme by Quantitative Click Ligation. Bioconjugate Chemistry. 30: 1169-1174. PMID 30883092 DOI: 10.1021/Acs.Bioconjchem.9B00110  0.787
2019 Hu H, Kofoed C, Li M, Gonçalves JPL, Hansen J, Wolfram M, Hansen AK, Friis Hansen CH, Diness F, Schoffelen S, Meldal M. Computational Evolution of Threonine-Rich β-Hairpin Peptides Mimicking Specificity and Affinity of Antibodies. Acs Central Science. 5: 259-269. PMID 30834314 DOI: 10.1021/Acscentsci.8B00614  0.78
2018 Embaby AM, Lelieveldt LPWM, Diness F, Meldal M. Metallo-Organozymes with Specific Proteolytic Activity. Chemistry: a European Journal. 24: 17424-17428. PMID 30146681 DOI: 10.1002/Chem.201803666  0.733
2018 Hu H, Nikitin SV, Berthelsen AB, Diness F, Schoffelen S, Meldal M. Sustainable Flow Synthesis of Encoded Beads for Combinatorial Chemistry and Chemical Biology. Acs Combinatorial Science. PMID 29969235 DOI: 10.1021/Acscombsci.8B00052  0.688
2018 Gonçalves JPL, Palmer D, Meldal M. MC4R Agonists: Structural Overview on Antiobesity Therapeutics. Trends in Pharmacological Sciences. 39: 402-423. PMID 29478721 DOI: 10.1016/J.Tips.2018.01.004  0.322
2018 Embaby AM, Schoffelen S, Kofoed C, Meldal M, Diness F. Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification Angewandte Chemie. 57: 8022-8026. PMID 29469231 DOI: 10.1002/Anie.201712589  0.773
2018 Fowkes MM, Meldal MP, Vincent TL, Lim NH. Screening for selective aggrecanase substrates to detect early proteolytic events in cartilage degradation Osteoarthritis and Cartilage. 26. DOI: 10.1016/J.Joca.2018.02.888  0.752
2018 Embaby AM, Schoffelen S, Kofoed C, Meldal M, Diness F. Inside Back Cover: Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification (Angew. Chem. Int. Ed. 27/2018) Angewandte Chemie. 57: 8831-8831. DOI: 10.1002/Anie.201805102  0.759
2018 Embaby AM, Schoffelen S, Kofoed C, Meldal M, Diness F. Innenrücktitelbild: Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification (Angew. Chem. 27/2018) Angewandte Chemie. 130: 8463-8463. DOI: 10.1002/Ange.201805102  0.759
2017 Palmer D, Gonçalves JPL, Hansen LV, Wu B, Hald H, Schoffelen S, Diness F, Le Quement ST, Nielsen TE, Meldal M. Click Chemistry-Mediated Synthesis of Selective Melanocortin Receptor-4 Agonists. Journal of Medicinal Chemistry. PMID 28972753 DOI: 10.1021/Acs.Jmedchem.7B00353  0.705
2017 Wang Y, Madsen AØ, Diness F, Meldal M. Diversity oriented syntheses by combining CuAAC and stereoselective INCIC reactions with peptides. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28833706 DOI: 10.1002/Chem.201702900  0.735
2017 Jacobsen CB, Meldal M, Diness F. Mechanism and Scope of Base‐Controlled Catalyst‐Free N‐Arylation of Amines with Unactivated Fluorobenzenes Chemistry: a European Journal. 23: 846-851. PMID 27739610 DOI: 10.1002/Chem.201604098  0.714
2016 Meldal M, Schoffelen S. Recent advances in covalent, site-specific protein immobilization. F1000research. 5: 2303. PMID 27785356 DOI: 10.12688/F1000Research.9002.1  0.319
2016 Nikitin S, Palmer D, Meldal M, Diness F. Comparative studies of adhesion peptides based on l- or d-amino acids Journal of Peptide Science. 22: 642-646. PMID 27580849 DOI: 10.1002/Psc.2913  0.739
2016 Li M, Hoeck C, Schoffelen S, Gotfredsen CH, Meldal M. Specific Electrostatic Molecular Recognition in Water. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27073143 DOI: 10.1002/Chem.201600231  0.348
2016 Hansen J, Diness F, Meldal M. C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles. Organic & Biomolecular Chemistry. 14: 3238-45. PMID 26924021 DOI: 10.1039/C6Ob00213G  0.752
2016 Ødum ASR, Østergaard S, Nørby I, Meldal M, Olesen K. Novel Application of Peptidyl-Lys Metallopeptidase as a C-Terminal Processing Protease. Protein and Peptide Letters. 23: 396-403. PMID 26845767 DOI: 10.2174/0929866523666160204123702  0.399
2016 Vutti S, Schoffelen S, Bolinsson J, Buch-Månson N, Bovet N, Nygård J, Martinez KL, Meldal M. Click Chemistry Mediated Functionalization of Vertical Nanowires for Biological Applications. Chemistry (Weinheim An Der Bergstrasse, Germany). 22: 496-500. PMID 26601641 DOI: 10.1002/Chem.201504540  0.373
2015 Vutti S, Buch-Månson N, Schoffelen S, Bovet N, Martinez KL, Meldal M. Covalent and stable CuAAC modification of silicon surfaces for control of cell adhesion. Chembiochem : a European Journal of Chemical Biology. 16: 782-91. PMID 25737226 DOI: 10.1002/Cbic.201402629  0.321
2015 Diness F, Meldal M. Fmox: A Base‐Labile Aldehyde Protecting Group European Journal of Organic Chemistry. 2015: 1433-1436. DOI: 10.1002/Ejoc.201403643  0.696
2011 Meldal M, Wu B, Diness F, Michael R, Hagel G. Metabolically stable cellular adhesion to inert surfaces. Chembiochem : a European Journal of Chemical Biology. 12: 2463-70. PMID 21928441 DOI: 10.1002/Cbic.201100382  0.723
2011 Pedersen JW, Bennett EP, Schjoldager KT, Meldal M, Holmér AP, Blixt O, Cló E, Levery SB, Clausen H, Wandall HH. Lectin domains of polypeptide GalNAc transferases exhibit glycopeptide binding specificity. The Journal of Biological Chemistry. 286: 32684-96. PMID 21768105 DOI: 10.1074/Jbc.M111.273722  0.758
2011 Jahn MR, Andreasen HB, Fütterer S, Nawroth T, Schünemann V, Kolb U, Hofmeister W, Muñoz M, Bock K, Meldal M, Langguth P. A comparative study of the physicochemical properties of iron isomaltoside 1000 (Monofer), a new intravenous iron preparation and its clinical implications. European Journal of Pharmaceutics and Biopharmaceutics : Official Journal of Arbeitsgemeinschaft FüR Pharmazeutische Verfahrenstechnik E.V. 78: 480-91. PMID 21439379 DOI: 10.1016/J.Ejpb.2011.03.016  0.555
2010 Meldal M, Tornøe CW, Nielsen TE, Diness F, Le Quement ST, Christensen CA, Jensen JF, Worm-Leonhard K, Groth T, Bouakaz L, Wu B, Hagel G, Keinicke L. Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity. Biopolymers. 94: 161-82. PMID 20225304 DOI: 10.1002/Bip.21344  0.803
2010 Diness F, Meldal M. Amino acid derived 1,4-dialkyl substituted imidazolones. Biopolymers. 94: 236-241. PMID 20225297 DOI: 10.1002/Bip.21359  0.719
2010 Quement STl, Petersen R, Meldal M, Nielsen TE. N-acyliminium intermediates in solid-phase synthesis Biopolymers. 94: 242-256. PMID 20225296 DOI: 10.1002/Bip.21358  0.356
2009 Diness F, Meldal M. Imidazolones in Diastereoselective Cyclization Reactions and CuII‐Catalysed Cross‐Coupling Reactions Chemistry: a European Journal. 15: 7044-7047. PMID 19544506 DOI: 10.1002/Chem.200900633  0.683
2009 Meldal M, Holm CB, Bojesen G, Jakobsen MH, Holm A. Multiple column peptide synthesis, Part 2 (1, 2). International Journal of Peptide and Protein Research. 41: 250-260. PMID 8463049 DOI: 10.1111/J.1399-3011.1993.Tb00333.X  0.463
2009 Breddam K, Widmer F, Meldal M. Amidation of growth hormone releasing factor (1-29) by serine carboxypeptidase catalysed transpeptidation. International Journal of Peptide and Protein Research. 37: 153-160. PMID 2019477 DOI: 10.1111/J.1399-3011.1991.Tb00096.X  0.423
2009 Karup G, Meldal M, Nielsen PE, Buchardt O. 9-Acridinylpeptides and 9-acridinyl-4-nitrophenylsulfonylpeptides. Synthesis, binding to DNA, and photoinduced DNA cleavage. International Journal of Peptide and Protein Research. 32: 331-343. DOI: 10.1111/J.1399-3011.1988.Tb01268.X  0.404
2008 Meldal M, Tornøe CW. Cu-catalyzed azide-alkyne cycloaddition. Chemical Reviews. 108: 2952-3015. PMID 18698735 DOI: 10.1021/Cr0783479  0.774
2008 Lanfranco MF, Loayza-Muro R, Clark D, Núñez R, Zavaleta AI, Jimenez M, Meldal M, Coombs GH, Mottram JC, Izidoro M, Juliano MA, Juliano L, Arévalo J. Expression and substrate specificity of a recombinant cysteine proteinase B of Leishmania braziliensis. Molecular and Biochemical Parasitology. 161: 91-100. PMID 18639590 DOI: 10.1016/J.Molbiopara.2008.06.005  0.349
2008 Quement STL, Nielsen TE, Meldal M. Divergent pathway for the solid-phase conversion of aromatic acetylenes to carboxylic acids, alpha-ketocarboxylic acids, and methyl ketones. Acs Combinatorial Science. 10: 546-556. PMID 18588350 DOI: 10.1021/Cc8000037  0.343
2008 Quement STL, Nielsen TE, Meldal M. Solid-Phase Synthesis of Aryl-Substituted Thienoindolizines: Sequential Pictet−Spengler, Bromination and Suzuki Cross-Coupling Reactions of Thiophenes Acs Combinatorial Science. 10: 447-455. PMID 18386932 DOI: 10.1021/Cc700199N  0.374
2008 Worm-Leonhard K, Meldal M. Green Catalysts: Solid‐Phase Peptide Carbene Ligands in Aqueous Transition‐Metal Catalysis European Journal of Organic Chemistry. 2008: 5244-5253. DOI: 10.1002/Ejoc.200800633  0.343
2008 Jensen JF, Worm-Leonhard K, Meldal M. Optically active (peptido-carbene)palladium complexes: Towards true solid-phase combinatorial libraries of transition metal catalysts European Journal of Organic Chemistry. 3785-3797. DOI: 10.1002/Ejoc.200800234  0.392
2007 Quement STL, Nielsen TE, Meldal M. Scaffold diversity through intramolecular cascade reactions of solid-supported cyclic N-acyliminium intermediates. Acs Combinatorial Science. 9: 1060-1072. PMID 17994787 DOI: 10.1021/Cc700097K  0.36
2007 Alves FM, Hirata IY, Gouvea IE, Alves MF, Meldal M, Brömme D, Juliano L, Juliano MA. Controlled peptide solvation in portion-mixing libraries of FRET peptides: improved specificity determination for Dengue 2 virus NS2B-NS3 protease and human cathepsin S. Journal of Combinatorial Chemistry. 9: 627-34. PMID 17563123 DOI: 10.1021/Cc070042K  0.39
2007 Nielsen TE, Quement STL, Meldal M. Solid-phase synthesis of carboxylic and oxamic acids via OsO4/NaIO4/HMTA-mediated oxidative cleavage of acetylenic peptides. Organic Letters. 9: 2469-2472. PMID 17518476 DOI: 10.1021/Ol070693P  0.442
2007 Christensen CA, Meldal M. Solid-phase synthesis of a peptide-based P,S-ligand system designed for generation of combinatorial catalyst libraries. Journal of Combinatorial Chemistry. 9: 79-85. PMID 17206835 DOI: 10.1021/Cc0600627  0.437
2007 Reenberg T, Nyberg N, Duus JØ, van Dongen JLJ, Meldal M. Specific Recognition of Disaccharides in Water by an Artificial Bicyclic Carbohydrate Receptor (Eur. J. Org. Chem. 30/2007) European Journal of Organic Chemistry. 2007: 4971-4971. DOI: 10.1002/Ejoc.200790079  0.583
2007 Reenberg T, Nyberg N, Duus J, Van Dongen JLJ, Meldal M. Specific recognition of disaccharides in water by an artificial bicyclic carbohydrate receptor European Journal of Organic Chemistry. 5003-5009. DOI: 10.1002/Ejoc.200700518  0.588
2006 Diness F, Beyer J, Meldal M. Solid‐Phase Synthesis of Tetrahydro‐β‐carbolines and Tetrahydroisoquinolines by Stereoselective Intramolecular N‐Carbamyliminium Pictet–Spengler Reactions Chemistry: a European Journal. 12: 8056-8066. PMID 16881029 DOI: 10.1002/Chem.200600138  0.741
2006 Nielsen TE, Le Quement S, Meldal M. Solid-phase synthesis of bicyclic dipeptide mimetics by intramolecular cyclization of alcohols, thiols, amines, and amides with N-acyliminium intermediates. Organic Letters. 7: 3601-4. PMID 16092829 DOI: 10.1021/ol050871j  0.352
2005 Nielsen TE, Meldal M. Solid-Phase Synthesis of Pyrroloisoquinolines via the Intramolecular N-Acyliminium Pictet−Spengler Reaction Acs Combinatorial Science. 7: 599-610. PMID 16004504 DOI: 10.1021/Cc050008A  0.427
2005 Nielsen TE, Meldal M. Highly Efficient Solid-Phase Oxidative Cleavage of Olefins by OsO4−NaIO4 in the Intramolecular N-Acyliminium Pictet−Spengler Reaction Organic Letters. 7: 2695-2698. PMID 15957924 DOI: 10.1021/Ol050870R  0.419
2005 Christensen CA, Meldal M. Efficient solid-phase synthesis of peptide-based phosphine ligands: towards combinatorial libraries of selective transition metal catalysts. Chemistry (Weinheim An Der Bergstrasse, Germany). 11: 4121-31. PMID 15861474 DOI: 10.1002/Chem.200500105  0.434
2005 Benito JM, Christensen CA, Meldal M. Versatile solid-phase synthesis of peptide-derived 2-oxazolines. Application in the synthesis of ligands for asymmetric catalysis. Organic Letters. 7: 581-4. PMID 15704899 DOI: 10.1021/Ol047675H  0.455
2005 Fieber W, Kragelund BB, Meldal M, Poulsen FM. Reversible dimerization of acid-denatured ACBP controlled by helix A4. Biochemistry. 44: 1375-84. PMID 15683223 DOI: 10.1021/Bi0481949  0.328
2005 Nielsen TE, Quement SL, Meldal M. Solid-phase synthesis of biarylalanines via Suzuki cross-coupling and intramolecular N-acyliminium Pictet–Spengler reactions Tetrahedron Letters. 46: 7959-7962. DOI: 10.1016/J.Tetlet.2005.09.080  0.393
2005 Vázquez-Campos S, Hilaire PMS, Damgaard D, Meldal M. GAG Mimetic Libraries: Sulphated Peptide as Heparin‐like Glycosaminoglycan Mimics in Their Interaction with FGF‐1 Qsar & Combinatorial Science. 24: 923-942. DOI: 10.1002/Qsar.200420100  0.438
2005 Minkwitz R, Meldal M. Application of a photolabile backbone amide linker for cleavage of internal amides in the synthesis towards melanocortin subtype-4 agonists Qsar & Combinatorial Science. 24: 343-353. DOI: 10.1002/Qsar.200420050  0.374
2004 Roice M, Christensen SF, Meldal M. ULTRAMINE: a high-capacity polyethylene-imine-based polymer and its application as a scavenger resin. Chemistry: a European Journal. 10: 4407-4415. PMID 15378618 DOI: 10.1002/Chem.200400314  0.326
2004 Juliano MA, Brooks DR, Selzer PM, Pandolfo HL, Judice WA, Juliano L, Meldal M, Sanderson SJ, Mottram JC, Coombs GH. Differences in substrate specificities between cysteine protease CPB isoforms of Leishmania mexicana are mediated by a few amino acid changes. European Journal of Biochemistry / Febs. 271: 3704-14. PMID 15355348 DOI: 10.1111/J.1432-1033.2004.04311.X  0.364
2004 Meldal M. 'One bead two compound libraries' for detecting chemical and biochemical conversions. Current Opinion in Chemical Biology. 8: 238-244. PMID 15183321 DOI: 10.1016/J.Cbpa.2004.04.007  0.325
2004 Nielsen TE, Meldal M. Solid-Phase Intramolecular N-Acyliminium Pictet−Spengler Reactions as Crossroads to Scaffold Diversity Journal of Organic Chemistry. 69: 3765-3773. PMID 15153007 DOI: 10.1021/Jo049918P  0.405
2004 Tornøe CW, Sanderson SJ, Mottram JC, Coombs GH, Meldal M. Combinatorial library of peptidotriazoles: identification of [1,2,3]-triazole inhibitors against a recombinant Leishmania mexicana cysteine protease. Journal of Combinatorial Chemistry. 6: 312-24. PMID 15132590 DOI: 10.1021/Cc020085V  0.811
2004 and AP, Meldal M. α-Keto Amide Peptides: A Synthetic Strategy to Resin-Bound Peptide Isosteres for Protease Inhibitor Screening on Solid Support Acs Combinatorial Science. 6: 181-195. PMID 15002966 DOI: 10.1021/Cc030107T  0.462
2004 Roice M, Johannsen I, Meldal M. High Capacity Poly(ethylene glycol) Based Amino Polymers for Peptide and Organic Synthesis Qsar & Combinatorial Science. 23: 662-673. DOI: 10.1002/Qsar.200420021  0.449
2004 Diness F, Beyer J, Meldal M. Synthesis of 3‐Boc‐(1,3)‐oxazinane‐Protected Amino Aldehydes from Amino Acids and Their Conversion into Urea Precursors. Novel Building Blocks for Combinatorial Synthesis Qsar & Combinatorial Science. 23: 130-144. DOI: 10.1002/Qsar.200320012  0.73
2004 Benito JM, Meldal M. Bicyclic Organo‐Peptides as Selective Carbohydrate Receptors: Design, Solid‐phase Synthesis, and on‐bead Binding Capability Qsar & Combinatorial Science. 23: 117-129. DOI: 10.1002/Qsar.200320011  0.403
2004 Christensen C, Tornøe CW, Meldal M. Pyrazines on Solid Support from Peptides by Periodinane Oxidation of Threonine Side‐Chains. A Quantitative Chemical Transformation (QCT) for Combinatorial Chemistry Qsar & Combinatorial Science. 23: 109-116. DOI: 10.1002/Qsar.200320009  0.388
2003 Nielsen TE, Diness F, Meldal M. The Pictet-Spengler reaction in solid-phase combinatorial chemistry. Current Opinion in Drug Discovery & Development. 6: 801-14. PMID 14758752  0.69
2003 Willert M, Benito JM, Meldal M. Solid-phase combinatorial library of norstatine-type isosters by the nitroaldol reaction. Acs Combinatorial Science. 5: 91-101. PMID 12625698 DOI: 10.1021/Cc0100722  0.41
2003 Bondebjerg J, Grunnet M, Jespersen T, Meldal M. Solid-phase synthesis and biological activity of a thioether analogue of conotoxin G1. Chembiochem : a European Journal of Chemical Biology. 4: 186-94. PMID 12616632 DOI: 10.1002/Cbic.200390030  0.4
2003 Halkes KM, Hilaire PMS, Crocker PR, Meldal M. Glycopeptides as oligosaccharide mimics: high affinity sialopeptide ligands for sialoadhesin from combinatorial libraries. Acs Combinatorial Science. 5: 18-27. PMID 12523830 DOI: 10.1021/Cc0200641  0.347
2003 Christensen C, Schiødt CB, Foged NT, Meldal M. Solid Phase Combinatorial Library of 1,3‐Azole Containing Peptides for the Discovery of Matrix Metallo Proteinase Inhibitors Qsar & Combinatorial Science. 22: 754-766. DOI: 10.1002/Qsar.200320006  0.356
2003 Christensen C, Groth T, Schiødt CB, Foged NT, Meldal M. Automated Sorting of Beads from a “One-Bead-Two-Compounds” Combinatorial Library of Metalloproteinase Inhibitors Qsar & Combinatorial Science. 22: 737-744. DOI: 10.1002/Qsar.200320005  0.588
2002 Gad M, Werdelin O, Meldal M, Komba S, Jensen T. Characterization of T cell hybridomas raised against a glycopeptide containing the tumor-associated T antigen, (βGal (1-3) αGalNAc-O/Ser) Glycoconjugate Journal. 19: 59-65. PMID 12652081 DOI: 10.1023/A:1022537031617  0.333
2002 Meldal M. The one-bead two-compound assay for solid phase screening of combinatorial libraries. Biopolymers. 66: 93-100. PMID 12325159 DOI: 10.1002/Bip.10229  0.361
2002 Bondebjerg J, Xiang Z, Bauzo RM, Haskell-Luevano C, Meldal M. A solid-phase approach to mouse melanocortin receptor agonists derived from a novel thioether cyclized peptidomimetic scaffold. Journal of the American Chemical Society. 124: 11046-55. PMID 12224952 DOI: 10.1021/Ja0123913  0.345
2002 Miranda LP, Lubell WD, Halkes KM, Groth T, Grøtli M, Rademann J, Gotfredsen CH, Meldal M. SPOCC-194, a new high functional group density PEG-based resin for solid-phase organic synthesis. Journal of Combinatorial Chemistry. 4: 523-9. PMID 12217026 DOI: 10.1021/Cc020030T  0.602
2002 St Hilaire PM, Alves LC, Herrera F, Renil M, Sanderson SJ, Mottram JC, Coombs GH, Juliano MA, Juliano L, Arevalo J, Meldal M. Solid-phase library synthesis, screening, and selection of tight-binding reduced peptide bond inhibitors of a recombinant Leishmania mexicana cysteine protease B. Journal of Medicinal Chemistry. 45: 1971-82. PMID 11985465 DOI: 10.1021/Jm0110901  0.339
2002 Tornøe CW, Christensen C, Meldal M. Peptidotriazoles on solid phase: [1,2,3]-triazoles by regiospecific copper(i)-catalyzed 1,3-dipolar cycloadditions of terminal alkynes to azides. The Journal of Organic Chemistry. 67: 3057-64. PMID 11975567 DOI: 10.1021/Jo011148J  0.813
2002 Campos SV, Miranda LP, Meldal M. Preparation of novel O-sulfated amino acid building blocks with improved acid stability for Fmoc-based solid-phase peptide synthesis Journal of the Chemical Society-Perkin Transactions 1. 682-686. DOI: 10.1039/B107320F  0.459
2002 Tornøe CW, Meldal M. EXPO3000—a new expandable polymer for synthesis and enzymatic assays Tetrahedron Letters. 43: 6409-6411. DOI: 10.1016/S0040-4039(02)01369-2  0.302
2001 Miranda LP, Meldal M. Unichemo Protection: A Concept for Chemical Synthesis This work was supported by the Danish National Research Foundation. Angewandte Chemie. 40: 3655-3657. PMID 11592212 DOI: 10.1002/1521-3773(20011001)40:19<3655::Aid-Anie3655>3.0.Co;2-K  0.339
2001 Halkes KM, Gotfredsen CH, Grøtli M, Miranda LP, Duus JO, Meldal M. Solid-phase glycosylation of peptide templates and on-bead MAS-NMR analysis: perspectives for glycopeptide libraries. Chemistry (Weinheim An Der Bergstrasse, Germany). 7: 3584-91. PMID 11560330 DOI: 10.1002/1521-3765(20010817)7:16<3584::Aid-Chem3584>3.0.Co;2-Z  0.646
2001 Groth T, Grøtli M, Meldal M. Diffusion of Reagents in Macrobeads Acs Combinatorial Science. 3: 461-468. PMID 11549364 DOI: 10.1021/Cc000106Q  0.509
2001 Graven A, St Hilaire PM, Sanderson SJ, Mottram JC, Coombs GH, Meldal M. Combinatorial library of peptide isosters based on Diels-Alder reactions: identification of novel inhibitors against a recombinant cysteine protease from Leishmania mexicana. Journal of Combinatorial Chemistry. 3: 441-52. PMID 11549362 DOI: 10.1021/Cc0001102  0.417
2001 Alves LC, Judice WA, St Hilaire PM, Meldal M, Sanderson SJ, Mottram JC, Coombs GH, Juliano L, Juliano MA. Substrate specificity of recombinant cysteine proteinase, CPB, of Leishmania mexicana. Molecular and Biochemical Parasitology. 116: 1-9. PMID 11463460 DOI: 10.1016/S0166-6851(01)00290-0  0.397
2001 Papanikos A, Rademann J, Meldal M. α-Ketocarbonyl Peptides: A General Approach to Reactive Resin-Bound Intermediates in the Synthesis of Peptide Isosteres for Protease Inhibitor Screening on Solid Support Journal of the American Chemical Society. 123: 2176-2181. PMID 11456862 DOI: 10.1021/Ja003690F  0.44
2001 Schiodt CB, Buchardt J, Terp GE, Christensen U, Brink M, Larsen YB, Meldal M, Foged NT. Phosphinic peptide inhibitors of macrophage metalloelastase (MMP-12). Selectivity and mechanism of binding. Current Medicinal Chemistry. 8: 967-976. PMID 11375764 DOI: 10.2174/0929867013372670  0.745
2001 Alves LC, St Hilaire PM, Meldal M, Sanderson SJ, Mottram JC, Coombs GH, Juliano L, Juliano MA. Identification of peptides inhibitory to recombinant cysteine proteinase, CPB, of Leishmania mexicana. Molecular and Biochemical Parasitology. 114: 81-8. PMID 11356516 DOI: 10.1016/S0166-6851(01)00239-0  0.347
2001 and TG, Meldal M. N-Terminal Peptide Aldehydes as Electrophiles in Combinatorial Solid Phase Synthesis of Novel Peptide Isosteres1,† Acs Combinatorial Science. 3: 45-63. PMID 11148063 DOI: 10.1021/cc000058  0.437
2001 Groth T, Meldal M. Synthesis of aldehyde building blocks protected as acid labile N-Boc N,O-acetals: toward combinatorial solid phase synthesis of novel peptide isosteres. Acs Combinatorial Science. 3: 34-44. PMID 11148062 DOI: 10.1021/Cc000057H  0.624
2001 Grøtli M, Rademan J, Groth T, Lubell WD, Miranda LP, Meldal M. Surfactant Mediated Cationic and Anionic Suspension Polymerization of PEG-Based Resins in Silicon Oil: Beaded SPOCC 1500 and POEPOP 1500 Acs Combinatorial Science. 3: 28-33. PMID 11148061 DOI: 10.1021/Cc000053C  0.53
2001 Graven A, Meldal M. Peptido-organic Diels–Alder reactions on hydrophilic resin: scope for combinatorial chemistry Journal of the Chemical Society-Perkin Transactions 1. 3198-3203. DOI: 10.1039/B103765J  0.418
2001 Miranda LP, Meldal M. Unichemo Protection: A Concept for Chemical Synthesis** Angewandte Chemie. 113: 3767-3769. DOI: 10.1002/1521-3757(20011001)113:19<3767::Aid-Ange3767>3.0.Co;2-Q  0.353
2000 St Hilaire PM, Alves LC, Sanderson SJ, Mottram JC, Juliano MA, Juliano L, Coombs GH, Meldal M. The substrate specificity of a recombinant cysteine protease from Leishmania mexicana: application of a combinatorial peptide library approach. Chembiochem : a European Journal of Chemical Biology. 1: 115-22. PMID 11828405 DOI: 10.1002/1439-7633(20000818)1:2<115::Aid-Cbic115>3.0.Co;2-8  0.304
2000 Tornøe CW, Davis P, Porreca F, Meldal M. Alpha-azido acids for direct use in solid-phase peptide synthesis. Journal of Peptide Science : An Official Publication of the European Peptide Society. 6: 594-602. PMID 11192239 DOI: 10.1002/1099-1387(200012)6:12<594::Aid-Psc276>3.0.Co;2-X  0.423
2000 Komba S, Werdelin O, Jensen T, Meldal M. Synthesis of tumor associated sialyl-T-glycopeptides and their immunogenicity. Journal of Peptide Science. 6: 585-593. PMID 11192238 DOI: 10.1002/1099-1387(200012)6:12<585::Aid-Psc274>3.0.Co;2-0  0.363
2000 Buchardt J, Schiødt CB, Krog-Jensen ‡C, Delaissé §J, Foged aNT, Meldal M. Solid phase combinatorial library of phosphinic peptides for discovery of matrix metalloproteinase inhibitors. Acs Combinatorial Science. 2: 624-638. PMID 11138549 DOI: 10.1021/Cc000031Q  0.775
2000 Tornøe CW, Sengeløv H, Meldal M. Solid-phase Synthesis of Chemotactic Peptides Using α-Azido Acids Journal of Peptide Science. 6: 314-320. PMID 10946996 DOI: 10.1002/1099-1387(200007)6:7<314::Aid-Psc255>3.0.Co;2-E  0.441
2000 Almeida PC, Oliveira V, Chagas JR, Meldal M, Juliano MA, Juliano L. Hydrolysis by cathepsin B of fluorescent peptides derived from human prorenin. Hypertension (Dallas, Tex. : 1979). 35: 1278-83. PMID 10856277 DOI: 10.1161/01.Hyp.35.6.1278  0.335
2000 Hilaire PMS, Meldal M. Glycopeptide and Oligosaccharide Libraries Angewandte Chemie. 39: 1162-1179. PMID 10767009 DOI: 10.1002/(Sici)1521-3773(20000403)39:7<1162::Aid-Anie1162>3.0.Co;2-6  0.346
2000 Grøtli M, Gotfredsen CH, Rademann J, Buchardt J, Clark AJ, Duus JO, Meldal M. Physical properties of poly(ethylene glycol) (PEG)-based resins for combinatorial solid phase organic chemistry: a comparison of PEG-cross-linked and PEG-grafted resins. Journal of Combinatorial Chemistry. 2: 108-19. PMID 10757090 DOI: 10.1021/Cc990048C  0.771
2000 St Hilaire PM, Willert M, Juliano MA, Juliano L, Meldal M. Fluorescence-quenched solid phase combinatorial libraries in the characterization of cysteine protease substrate specificity. Journal of Combinatorial Chemistry. 1: 509-23. PMID 10748728 DOI: 10.1021/Cc990031U  0.381
2000 Stennicke HR, Renatus M, Meldal M, Salvesen GS. Internally quenched fluorescent peptide substrates disclose the subsite preferences of human caspases 1, 3, 6, 7 and 8. Biochemical Journal. 350: 563-568. DOI: 10.1042/Bj3500563  0.36
2000 Groth T, Grøtli M, Lubell WD, Miranda LP, Meldal M. HYDRA: A novel hydroxy and amine functionalised resin synthesised by reductive amination of PEG aldehyde and a polyamine Journal of the Chemical Society-Perkin Transactions 1. 4258-4264. DOI: 10.1039/B007141M  0.591
2000 Buchardt J, Meldal M. Novel methodology for the solid-phase synthesis of phosphinic peptides Journal of the Chemical Society-Perkin Transactions 1. 3306-3310. DOI: 10.1039/B003848M  0.808
2000 Graven A, Grøtli M, Meldal M. Towards peptide isostere libraries: aqueous aldol reactions on hydrophilic solid supports Journal of the Chemical Society-Perkin Transactions 1. 955-962. DOI: 10.1039/A909246C  0.418
2000 Halkes KM, Hilaire PMS, Jansson AM, Gotfredsen CH, Meldal M. Synthesis and application of sialic acid-containing building blocks for glycopeptide libraries. Establishing glycosylation conditions Journal of the Chemical Society-Perkin Transactions 1. 2127-2133. DOI: 10.1039/A908321I  0.399
2000 Gotfredsen CH, Grøtli M, Willert M, Meldal M, Duus JØ. Single-bead structure elucidation. Requirements for analysis of combinatorial solid-phase libraries by Nanoprobe MAS-NMR spectroscopy Journal of the Chemical Society-Perkin Transactions 1. 1167-1171. DOI: 10.1039/A906835J  0.633
1999 Duus JØ, Hilaire PMS, Meldal M, Bock K. Carbohydrate chemistry: synthetic and structural challenges towards the end of the 20th century Pure and Applied Chemistry. 71: 755-765. DOI: 10.1351/Pac199971050755  0.573
1999 Hilaire PMS, Cipolla L, Franco A, Tedebark U, Tilly DA, Meldal M. Synthesis of T-antigen-containing glycopeptides as potential cancer vaccines Journal of the Chemical Society-Perkin Transactions 1. 3559-3564. DOI: 10.1039/A908270K  0.451
1999 Mehta S, Meldal M, Duus JØ, Bock K. Evaluation of the effect of glycosylation on the enzymic hydrolysis of peptides Journal of the Chemical Society-Perkin Transactions 1. 1445-1452. DOI: 10.1039/A901492F  0.655
1999 Komba S, Meldal M, Werdelin O, Jensen T, Bock K. Convenient synthesis of Thr and Ser carrying the tumor associated sialyl-(2→3)-T antigen as building blocks for solid-phase glycopeptide synthesis Journal of the Chemical Society-Perkin Transactions 1. 415-420. DOI: 10.1039/A809524H  0.39
1999 Rademann J, Grøtli M, Meldal M, Bock K. SPOCC: A resin for solid-phase organic chemistry and enzymatic reactions on solid phase Journal of the American Chemical Society. 121: 5459-5466. DOI: 10.1021/Ja984355I  0.67
1999 Tornøe CW, Sonke T, Maes I, Schoemaker HE, Meldal M. Enzymatic and chiral HPLC resolution of α-azido acids and amides Tetrahedron Asymmetry. 11: 1239-1248. DOI: 10.1016/S0957-4166(00)00043-4  0.38
1999 Krog-Jensen C, Christensen MK, Meldal M. Preparation of an unprotected phosphotyrosine building block and its application in solid-phase synthesis of phosphopeptides Letters in Peptide Science. 6: 193-197. DOI: 10.1007/Bf02443506  0.449
1999 Buchardt J, Ferreras M, Krog-Jensen C, Delaissé J, Foged NT, Meldal M. Phosphinic Peptide Matrix Metalloproteinase‐9 Inhibitors by Solid‐Phase Synthesis Using a Building Block Approach Chemistry: a European Journal. 5: 2877-2884. DOI: 10.1002/(Sici)1521-3765(19991001)5:10<2877::Aid-Chem2877>3.0.Co;2-Z  0.795
1999 Rademann J, Meldal M, Bock K. Solid-phase synthesis of peptide isosters by nucleophilic reactions with N-terminal peptide aldehydes on a polar support tailored for solid-phase organic chemistry Chemistry - a European Journal. 5: 1218-1225. DOI: 10.1002/(Sici)1521-3765(19990401)5:4<1218::Aid-Chem1218>3.0.Co;2-X  0.683
1998 Westphal V, Spetzler JC, Meldal M, Christensen U, Winther JR. Kinetic Analysis of the Mechanism and Specificity of Protein-disulfide Isomerase Using Fluorescence-quenched Peptides Journal of Biological Chemistry. 273: 24992-24999. PMID 9737954 DOI: 10.1074/Jbc.273.39.24992  0.439
1998 Parolis LAS, Parolis H, Kenne L, Meldal M, Bock K. The extracellular polysaccharide of Pichia (Hansenula) holstii NRRLL Y-2448: The phosphorylated side chains Carbohydrate Research. 309: 77-87. PMID 9720238 DOI: 10.1016/S0008-6215(98)00101-3  0.62
1998 Meldal M, Svendsen IB, Juliano L, Juliano MA, Nery ED, Scharfstein J. Inhibition of cruzipain visualized in a fluorescence quenched solid-phase inhibitor library assay. D-amino acid inhibitors for cruzipain, cathepsin B and cathepsin L. Journal of Peptide Science : An Official Publication of the European Peptide Society. 4: 83-91. PMID 9620612 DOI: 10.1002/(Sici)1099-1387(199804)4:2<83::Aid-Psc124>3.0.Co;2-Z  0.414
1998 Davy A, Svendsen I, Sørensen SO, Sørensen MB, Rouster J, Meldal M, Simpson DJ, Cameron-Mills V. Substrate Specificity of Barley Cysteine Endoproteases EP-A and EP-B Plant Physiology. 117: 255-261. PMID 9576795 DOI: 10.1104/Pp.117.1.255  0.318
1998 Meldal M. Preparation of Biocompatible Resins for Library Syntheses Methods of Molecular Biology. 87: 59-63. PMID 9523259 DOI: 10.1385/0-89603-392-9:59  0.32
1998 Spetzler JC, Meldal M, Felding J, Vedsø P, Begtrup M. Novel acylation catalysts in peptide synthesis: derivatives of N-hydroxytriazoles and N-hydroxytetrazoles Journal of the Chemical Society-Perkin Transactions 1. 1727-1732. DOI: 10.1039/A707313E  0.384
1998 Meinjohanns E, Meldal M, Paulsen H, Dwek RA, Bock K. Novel sequential solid-phase synthesis of N-linked glycopeptides from natural sources Journal of the Chemical Society-Perkin Transactions 1. 549-560. DOI: 10.1039/A705528E  0.663
1998 Duus J, Meldal M, Winkler JR. Fluorescence energy-transfer probes of conformation in peptides: The 2-aminobenzamide/nitrotyrosine pair Journal of Physical Chemistry B. 102: 6413-6418. DOI: 10.1021/Jp973352+  0.618
1998 Lowary T, Meldal M, Helmboldt A, Vasella A, Bock K. Novel type of rigid C-linked glycosylacetylene-phenylalanine building blocks for combinatorial synthesis of C-linked glycopeptides Journal of Organic Chemistry. 63: 9657-9668. DOI: 10.1021/Jo980517H  0.704
1998 Buchardt J, Meldal M. A chemically inert hydrophilic resin for solid phase organic synthesis Tetrahedron Letters. 39: 8695-8698. DOI: 10.1016/S0040-4039(98)01737-7  0.778
1998 Tedebark U, Meldal M, Panza L, Bock K. C-linked glycosyl azido acid in novel solid-phase C-glycopeptide synthesis Tetrahedron Letters. 39: 1815-1818. DOI: 10.1016/S0040-4039(98)00095-1  0.64
1998 Ito AS, Turchiello RDF, Hirata IY, Cezari MHS, Meldal M, Juliano L. Fluorescent properties of amino acids labeled withortho-aminobenzoic acid Biospectroscopy. 4: 395-402. DOI: 10.1002/(Sici)1520-6343(1998)4:6<395::Aid-Bspy4>3.0.Co;2-Y  0.394
1998 Renil M, Ferreras M, Delaisse JM, Foged NT, Meldal M. PEGA supports for combinatorial peptide synthesis and solid-phase enzymatic library assays. Journal of Peptide Science. 4: 195-210. DOI: 10.1002/(Sici)1099-1387(199805)4:3<195::Aid-Psc141>3.0.Co;2-R  0.452
1998 Spetzler JC, Westphal V, Winther JR, Meldal M. Preparation of fluorescence quenched libraries containing interchain disulphide bonds for studies of protein disulphide isomerases. Journal of Peptide Science. 4: 128-137. DOI: 10.1002/(Sici)1099-1387(199804)4:2<128::Aid-Psc137>3.0.Co;2-E  0.455
1997 Meldal M, Hilaire PMS. Synthetic methods of glycopeptide assembly, and biological analysis of glycopeptide products. Current Opinion in Chemical Biology. 1: 552-563. PMID 9667891 DOI: 10.1016/S1367-5931(97)80052-X  0.439
1997 Meldal M. Properties of solid supports. Methods in Enzymology. 289: 83-104. PMID 9353719 DOI: 10.1016/S0076-6879(97)89045-3  0.409
1997 Nery ED, Juliano MA, Meldal M, Svendsen I, Scharfstein J, Walmsley A, Juliano L. Characterization of the substrate specificity of the major cysteine protease (cruzipain) from Trypanosoma cruzi using a portion-mixing combinatorial library and fluorogenic peptides. The Biochemical Journal. 427-33. PMID 9163334 DOI: 10.1042/Bj3230427  0.323
1997 Klich G, Paulsen H, Meyer B, Meldal M, Bock K. Synthesis and characterisation of highly glycosylated glycopeptides with T(n)-antigenic structures corresponding to human glycophorin A(N) Carbohydrate Research. 299: 33-48. PMID 9129295 DOI: 10.1016/S0008-6215(96)00337-0  0.64
1997 Franzyk H, Christensen MK, Jørgensen RM, Meldal M, Cordes H, Mouritsen S, Bock K. Constrained glycopeptide ligands for MPRs. Limitations of unprotected phosphorylated building blocks. Bioorganic & Medicinal Chemistry. 5: 21-40. PMID 9043655 DOI: 10.1016/S0968-0896(96)00194-0  0.691
1997 Lay L, Meldal M, Nicotra F, Panza L, Russo G. Stereoselective synthesis of the C-analogue ofβ-d-glucopyranosyl serine Chemical Communications. 1469-1470. DOI: 10.1039/A703063K  0.334
1997 Mathieux N, Paulsen H, Meldal M, Bock K. Synthesis of glycopeptide sequences of repeating units of the mucins MUC 2 and MUC 3 containing oligosaccharide side-chains with core 1, core 2, core 3, core 4 and core 6 structure Journal of the Chemical Society-Perkin Transactions 1. 2359-2368. DOI: 10.1039/A701742A  0.33
1997 Mehta S, Meldal M, Ferro V, Duus J, Bock K. Internally quenched fluorogenic, α-helical dimeric peptides and glycopeptides for the evaluation of the effect of glycosylation on the conformation of peptides Journal of the Chemical Society - Perkin Transactions 1. 1365-1374. DOI: 10.1039/A607624F  0.766
1997 Meinjohanns E, Meldal M, Jensen T, Werdelin O, Galli-Stampino L, Mouritsen S, Bock K. Versatile solid-phase thiolytic reduction of azido and N-Dts groups in the synthesis of haemoglobin (67-76) O-glycopeptides and photoaffinity labelled analogues to study glycan T-cell specificity Journal of the Chemical Society - Perkin Transactions 1. 871-884. DOI: 10.1039/A606725E  0.682
1997 Paulsen H, Schleyer A, Mathieux N, Meldal M, Bock K. New solid-phase oligosaccharide synthesis on glycopeptides bound to a solid phase Journal of the Chemical Society - Perkin Transactions 1. 281-293. DOI: 10.1039/A604123J  0.664
1997 Jensen T, Hansen P, Galli-Stampino L, Mouritsen S, Frische K, Meinjohanns E, Meldal M, Werdelin O. Glycopeptide specific T cell hybridomas raised against an αGalNAc O-glycosylated self peptide are discriminating between highly related carbohydrate groups Immunology Letters. 56: 449. DOI: 10.1016/S0165-2478(97)86827-7  0.334
1997 Meldal* M, Juliano MA, Jansson AM. Azido Acids in a Novel Method of Solid-Phase Peptide Synthesis. Tetrahedron Letters. 38: 2531-2534. DOI: 10.1016/S0040-4039(97)00393-6  0.437
1997 Spetzler JC, Meldal M. Evaluation of strategies for ‘one-pot’ deprotection, cleavage and disulfide bond formation in the preparation of cystine-containing peptides Letters in Peptide Science. 3: 327-332. DOI: 10.1007/Bf00127963  0.387
1997 Schleyer A, Meldal M, Manat R, Paulsen H, Bock K. Direct Solid-Phase Glycosylations Of Peptide Templates On A Novel Peg-Based Resin Angewandte Chemie. 36: 1976-1978. DOI: 10.1002/Anie.199719761  0.405
1997 Schleyer A, Meldal M, Renil M, Paulsen H, Bock K. Direkte Festphasen-Glycosylierung von Peptiden an einem neuartigen Polyethylenglycol-Harz Angewandte Chemie. 109: 2064-2067. DOI: 10.1002/Ange.19971091814  0.553
1997 Spetzler JC, Meldal M, Meinjohanns E, Steinaa L, Mouritsen S, Bock K. Synthetic hFSH peptide constructs in the evaluation of previous studies on the hFSH receptor interaction. Journal of Peptide Science. 3: 397-414. DOI: 10.1002/(Sici)1099-1387(199711)3:6<397::Aid-Psc113>3.0.Co;2-K  0.433
1996 Frische K, Meldal M, Werdelin O, Mouritsen S, Jensen T, Galli-Stampino L, Bock K. Multiple column synthesis of a library of T-cell stimulating Tn-antigenic glycopeptide analogues for the molecular characterization of T-cell-glycan specificity Journal of Peptide Science. 2: 212-222. PMID 9231328 DOI: 10.1002/Psc.64  0.695
1996 Franzyk H, Meldal M, Paulsen H, Thiel S, Jensenius JC, Bock K. Glycopeptide mimics of mammalian Man9GlcNAc2. Ligand binding to mannan-binding proteins (MBPs) Bioorganic and Medicinal Chemistry. 4: 1881-1899. PMID 9007273 DOI: 10.1016/S0968-0896(96)00171-X  0.653
1996 Parolis LA, Duus JO, Parolis H, Meldal M, Bock K. The extracellular polysaccharide of Pichia (Hansenula) holstii NRRL Y-2448: the structure of the phosphomannan backbone. Carbohydrate Research. 293: 101-17. PMID 8916546 DOI: 10.1016/0008-6215(96)00190-5  0.703
1996 Brockhausen I, Toki D, Brockhausen J, Peters S, Bielfeldt T, Kleen A, Paulsen H, Meldal M, Hagen F, Tabak LA. Specificity of O-glycosylation by bovine colostrum UDP-GalNAc: Polypeptide α-N-acetylgalactosaminyltransferase using synthetic glycopeptide substrates Glycoconjugate Journal. 13: 849-856. PMID 8910012 DOI: 10.1007/Bf00702349  0.408
1996 Löffler A, Doucey MA, Jansson AM, Müller DR, De Beer T, Hess D, Meldal M, Richter WJ, Vliegenthart JFG, Hofsteenge J. Spectroscopic and protein chemical analyses demonstrate the presence of C-mannosylated tryptophan in intact human RNase 2 and its isoforms Biochemistry. 35: 12005-12014. PMID 8810905 DOI: 10.1021/Bi9610515  0.337
1996 Grøn H, Bech LM, Sørensen SB, Meldal M, Breddam K. Studies of Binding Sites in the Subtilisin from Bacillus Lentus by Means of Site Directed Mutagenesis and Kinetic Investigations Advances in Experimental Medicine and Biology. 379: 105-112. PMID 8796314 DOI: 10.1007/978-1-4613-0319-0_11  0.333
1996 Jensen T, Galli-Stampino L, Mouritsen S, Frische K, Peters S, Meldal M, Werdelin O. T Cell Recognition Of Tn-Glycosylated Peptide Antigens European Journal of Immunology. 26: 1342-1349. PMID 8647215 DOI: 10.1002/Eji.1830260625  0.375
1996 Jansson AM, Jensen KJ, Meldal M, Lomako J, Lomako WM, Olsen CE, Bock K. Solid-phase glycopeptide synthesis of tyrosine-glycosylated glycogenin fragments as substrates for glucosylation by glycogenin Journal of the Chemical Society - Perkin Transactions 1. 1001-1006. DOI: 10.1039/P19960001001  0.661
1996 Meinjohanns E, Meldal M, Schleyer A, Paulsen H, Bock K. Efficient syntheses of core 1, core 2, core 3 and core 4 building blocks for SPS of mucin O-glycopeptides based on the N-Dts-method Journal of the Chemical Society - Perkin Transactions 1. 985-993. DOI: 10.1039/P19960000985  0.642
1996 Renil M, Meldal M. Poepop And Poeps : Inert Polyethylene Glycol Crosslinked Polymeric Supports For Solid Synthesis Tetrahedron Letters. 37: 6185-6188. DOI: 10.1016/0040-4039(96)01319-6  0.446
1995 Auzanneau FI, Meldal M, Bock K. Synthesis, characterization and biocompatibility of PEGA resins Journal of Peptide Science : An Official Publication of the European Peptide Society. 1: 31-44. PMID 9222982 DOI: 10.1002/Psc.310010106  0.673
1995 Paulsen H, Peters S, Bielfeldt T, Meldal M, Bock K. Synthesis of the glycosyl amino acids Nα-Fmoc-Ser[Ac4-β-d-Gal p-(1 → 3)-Ac2-α-d-GalN3 p]-OPfp and Nα-Fmoc-Thr[Ac4-β-d-Gal p-(1 → 3)-Ac2-α-d-GalN3 p]-OPfp and the application in the solid-phase peptide synthesis of multiply glycosylated mucin peptides with T.. Carbohydrate Research. 268: 17-34. PMID 7736464 DOI: 10.1016/0008-6215(94)00292-N  0.671
1995 Peters S, Lowary TL, Hindsgaul O, Meldal M, Bock K. Solid-phase synthesis of a fucosylated glycopeptide of human factor IX with a fucose-α-(1→O)-serine linkage Journal of the Chemical Society, Perkin Transactions 1. 3017-3022. DOI: 10.1039/P19950003017  0.785
1995 Franzyk H, Meldal M, Paulsen H, Bock K. Synthesis of aliphatic O-dimannosyl amino acid building blocks for solid-phase assembly of glycopeptide libraries Journal of the Chemical Society-Perkin Transactions 1. 2883-2898. DOI: 10.1039/P19950002883  0.406
1995 Meinjohanns E, Vargas-Berenguel A, Meldal M, Paulsen H, Bock K. Comparison of N-Dts and N-Aloc in the solid-phase syntheses of O-GlcNAc glycopeptide fragments of RNA-polymerase II and mammalian neurofilaments Journal of the Chemical Society, Perkin Transactions 1. 2165-2175. DOI: 10.1039/P19950002165  0.663
1995 Meldal M, Svendsen I. Direct visualization of enzyme inhibitors using a portion mixing inhibitor library containing a quenched fluorogenic peptide substrate. Part 1. Inhibitors for subtilisin Carlsberg Journal of the Chemical Society-Perkin Transactions 1. 1591-1596. DOI: 10.1039/P19950001591  0.396
1995 Rio-Anneheim S, Paulsen H, Meldal M, Bock K. Synthesis of the building blocks Nα-Fmoc-O-[α-D-Ac3,GalN3,p-(1→3)-α-D-ac2,gain3,p]-Thr-Opfp and nα -fmoc-o-[α-D-ac3,GalN3,p-(1→6)=α-D-ac2,GalN3,p] -Thr-Opfp and their application in the solid phase glycopeptide synthesis of core 5 and core 7 mucin o-glycopeptides Journal of the Chemical Society, Perkin Transactions 1. 1071-1080. DOI: 10.1039/P19950001071  0.663
1995 Meinjohanns E, Meldal M, Paulsen H, Bock K. Dithiasuccinoyl (Dts) amino-protecting group used in syntheses of 1,2-trans-amino sugar glycosides Journal of the Chemical Society, Perkin Transactions 1. 405-415. DOI: 10.1039/P19950000405  0.658
1995 Meinjohanns E, Meldal M, Bock K. Efficient synthesis of O-(2-acetamido-2-deoxy-β-d-glucopyranosyl)-ser/thr building blocks for spps of o-glcnac glycopeptides Tetrahedron Letters. 36: 9205-9208. DOI: 10.1016/0040-4039(95)01941-A  0.646
1995 Renil M, Meldal M. Synthesis And Application Of A Pega Polymeric Support For High Capacity Continuous Flow Solid-Phase Peptide Synthesis Tetrahedron Letters. 36: 4647-4650. DOI: 10.1016/0040-4039(95)00808-P  0.445
1994 Mouritsen S, Meldal M, Christiansen-Brams I, Elsner H, Werdelin O. Attachment of oligosaccharides to peptide antigen profoundly affects binding to major histocompatibility complex class II molecules and peptide immunogenicity European Journal of Immunology. 24: 1066-1072. PMID 8181518 DOI: 10.1002/Eji.1830240509  0.383
1994 Granovsky M, Bielfeldt T, Peters S, Paulsen H, Meldal M, Brockhausen J, Brockhausen I. UDPgalactose:glycoprotein–N‐acetyl‐d‐galactosamine 3‐β‐d‐galactosyltransferase activity synthesizing O‐glycan core 1 is controlled by the amino acid sequence and glycosylation of glycopeptide substrates Febs Journal. 221: 1039-1046. PMID 8181460 DOI: 10.1111/J.1432-1033.1994.Tb18822.X  0.424
1994 Meldal M, Svendsen I, Breddam K, Auzanneau F. Portion-mixing peptide libraries of quenched fluorogenic substrates for complete subsite mapping of endoprotease specificity. Proceedings of the National Academy of Sciences of the United States of America. 91: 3314-3318. PMID 8159745 DOI: 10.1073/Pnas.91.8.3314  0.415
1994 Rønnow TECL, Meldal M, Bock K. Gram-scale synthesis of α,α-trehalose 6-monophosphate and α,α-trehalose 6,6′-diphosphate Carbohydrate Research. 260: 323-328. PMID 8069876 DOI: 10.1016/0008-6215(94)84050-4  0.591
1994 Meldal M, Bielfeldt T, Peters S, Jensen KJ, Paulsen H, Bock K. Susceptibility of glycans to β-elimination in Fmoc-based O-glycopeptide synthesis International Journal of Peptide and Protein Research. 43: 529-536. PMID 7928083 DOI: 10.1111/J.1399-3011.1994.Tb00554.X  0.639
1994 Meldal M, Bock K. A general approach to the synthesis of O- and N-linked glycopeptides Glycoconjugate Journal. 11: 59-63. PMID 7804007 DOI: 10.1007/Bf00731144  0.616
1994 Christiansen-Brams I, Jansson AM, Meldal M, Breddam K, Bock K. Silyl protection in the solid-phase synthesis of N-linked glycopeptides. Preparation of glycosylated fluorogenic substrates for subtilisins Bioorganic and Medicinal Chemistry. 2: 1153-1167. PMID 7757413 DOI: 10.1016/S0968-0896(00)82067-2  0.664
1994 Bundle DR, Eichler E, Gidney MA, Meldal M, Ragauskas A, Sigurskjold BW, Sinnott B, Watson DC, Yaguchi M, Young NM. Molecular recognition of a Salmonella trisaccharide epitope by monoclonal antibody Se155-4. Biochemistry. 33: 5172-82. PMID 7513555 DOI: 10.1021/Bi00183A022  0.522
1994 Vargas-Berenguel A, Meldal M, Paulsen H, Jensen KJ, Bock K. Synthesis of glycosyltyrosine building blocks for solid-phase glycopeptide assembly: Use of aryl tert-butyl ethers as glycosyl acceptors in aromatic glycosylations Journal of the Chemical Society, Perkin Transactions 1. 3287-3294. DOI: 10.1039/P19940003287  0.648
1994 Vargas-Berenguel A, Meldal M, Paulsen H, Bock K. Convenient synthesis of O-(2-acetamido-2-deoxy-β-D-glucopyranosyl)- serine and -threonine building blocks for solid-phase glycopeptide assembly Journal of the Chemical Society, Perkin Transactions 1. 2615-2619. DOI: 10.1039/P19940002615  0.661
1994 Ferro V, Meldal M, Bock K. Synthesis of 2′- and 2″-O-acylated maltotriosides as potential fluorescence-quenched substrates for α-amylase Journal of the Chemical Society, Perkin Transactions 1. 2169-2176. DOI: 10.1039/P19940002169  0.64
1994 Christensen MK, Meldal M, Bock K, Cordes H, Mouritsen S, Elsner H. Synthesis of glycosylated peptide templates containing 6′-O-phosphorylated mannose disaccharides and their binding to the cation-independent mannose 6-phosphate receptor Journal of the Chemical Society, Perkin Transactions 1. 1299-1310. DOI: 10.1039/P19940001299  0.657
1994 Meldal M, Auzanneau FI, Hindsgaul O, Palcic MM. A PEGA resin for use in the solid-phase chemical-enzymatic synthesis of glycopeptides Journal of the Chemical Society, Chemical Communications. 1849-1850. DOI: 10.1039/C39940001849  0.567
1994 Meldal M. Recent developments in glycopeptide and oligosaccharide synthesis Current Opinion in Structural Biology. 4: 710-718. DOI: 10.1016/S0959-440X(94)90169-4  0.402
1994 Ronnow TECL, Meldal M, Bock K. The use of O-glycosyl trichloroacetimidates in the synthesis of unsymmetrical trehalose analogues Tetrahedron: Asymmetry. 5: 2109-2122. DOI: 10.1016/S0957-4166(00)86287-4  0.659
1994 Meldal M. Multiple Column Synthesis of Quenched Solid-Phase Bound Fluorogenic Substrates for Characterization of Endoprotease Specificity Methods. 6: 417-424. DOI: 10.1006/Meth.1994.1044  0.43
1994 Paulsen H, Bielfeldt T, Peters S, Meldal M, Bock K. Eine neue Strategie zur Festphasensynthese vonO-Glycopeptiden über 2-Azidoglycopeptide Liebigs Annalen Der Chemie. 1994: 369-379. DOI: 10.1002/Jlac.199419940410  0.676
1993 Sorensen SB, Bech LM, Meldal M, Breddam K. Mutational replacements of the amino acid residues forming the hydrophobic S4 binding pocket of subtilisin 309 from Bacillus lentus. Biochemistry. 32: 8994-8999. PMID 8369272 DOI: 10.1021/Bi00086A003  0.339
1993 Jensen KJ, Meldal M, Bock K. Glycosylation of phenols: preparation of 1,2-cis and 1,2-trans glycosylated tyrosine derivatives to be used in solid-phase glycopeptide synthesis Journal of the Chemical Society-Perkin Transactions 1. 2119-2129. DOI: 10.1039/P19930002119  0.363
1993 Christiansen-Brams I, Meldal M, Bock K. Protected-mode synthesis of N-linked glycopeptides: single-step preparation of building blocks as peracetyl glycosylated NαFmoc asparagine OPfp esters Journal of the Chemical Society-Perkin Transactions 1. 1461-1471. DOI: 10.1039/P19930001461  0.367
1993 Christensen MK, Meldal M, Bock K. Synthesis of mannose 6-phosphate-containing disaccharide threonine building blocks and their use in solid-phase glycopeptide synthesis Journal of the Chemical Society-Perkin Transactions 1. 1453-1460. DOI: 10.1039/P19930001453  0.377
1993 Reimer KB, Meldal M, Kusumoto S, Fukaseb K, Bocka K. Small-scale solid-phase O-glycopeptide synthesis of linear and cyclized hexapeptides from blood-clotting factor IX containing O-(α-D-Xyl-1→3-α-D-Xyl-1→3-β-D-Glc)-L-ser Journal of the Chemical Society-Perkin Transactions 1. 925-932. DOI: 10.1039/P19930000925  0.392
1993 Christiansen-Brams I, Meldal M, Bock K. Silyl protection in the solid-phase synthesis of N-linked neoglycopeptides. One-step deprotection of fully protected neoglycopeptides Tetrahedron Letters. 34: 3315-3318. DOI: 10.1016/S0040-4039(00)73692-6  0.705
1993 Christiansen-Brams I, Meldal M, Bock K. S17.2 Solid phase synthesis of di- N -Glycosylated RGD-Analogues Glycoconjugate Journal. 10: 324-324. DOI: 10.1007/Bf01210125  0.338
1992 Breddam K, Meldal M. Substrate preferences of glutamic-acid-specific endopeptidases assessed by synthetic peptide substrates based on intramolecular fluorescence quenching. Febs Journal. 206: 103-107. PMID 1587264 DOI: 10.1111/J.1432-1033.1992.Tb16906.X  0.369
1992 Szwajcer-Dey E, Rasmussen J, Meldal M, Breddam K. Proline-specific endopeptidases from microbial sources: isolation of an enzyme from a Xanthomonas sp. Journal of Bacteriology. 174: 2454-2459. PMID 1556065 DOI: 10.1128/Jb.174.8.2454-2459.1992  0.382
1992 Ida CB, Meldal M, Bock K. Synthesis of the 1-amino-alditols derived from cellobiose, lactose and maltose Journal of Carbohydrate Chemistry. 11: 813-835. DOI: 10.1080/07328309208018272  0.652
1992 Jansson AM, Meldal M, Bock K. Solid-phase synthesis and characterization of O-dimannosylated heptadecapeptide analogues of human insulin-like growth factor 1 (IGF-1) Journal of the Chemical Society, Perkin Transactions 1. 1699-1708. DOI: 10.1039/P19920001699  0.654
1992 Meldal M. Pega: a flow stable polyethylene glycol dimethyl acrylamide copolymer for solid phase synthesis. Tetrahedron Letters. 33: 3077-3080. DOI: 10.1016/S0040-4039(00)79604-3  0.422
1992 Peters S, Bielfeldt T, Meldal M, Bock K, Paulsen H. Solid phase peptide synthesis of mucin glycopeptides Tetrahedron Letters. 33: 6445-6448. DOI: 10.1016/S0040-4039(00)79011-3  0.701
1992 Meldal M, Christensen MK, Bock K. Large-scale synthesis of d-mannose 6-phosphate and other hexose 6-phosphates Carbohydrate Research. 235: 115-127. DOI: 10.1016/0008-6215(92)80082-C  0.625
1992 Bielfeldt T, Peters S, Meldal M, Bock K, Paulsen H. Eine neue Strategie zur Festphasensynthese vonO-Glycopeptiden Angewandte Chemie. 104: 881-883. DOI: 10.1002/Ange.19921040719  0.572
1991 Meldal M, Breddam K. Anthranilamide and nitrotyrosine as a donor-acceptor pair in internally quenched fluorescent substrates for endopeptidases: multicolumn peptide synthesis of enzyme substrates for subtilisin Carlsberg and pepsin. Analytical Biochemistry. 195: 141-147. PMID 1888010 DOI: 10.1016/0003-2697(91)90309-H  0.442
1991 Bock K, Meldal M, Refn S. Controlled reduction of acarbose: conformational analysis of acarbose and the resulting saturated products Carbohydrate Research. 221: 1-16. PMID 1816915 DOI: 10.1016/0008-6215(91)80045-O  0.616
1991 Peters S, Bielfeldt T, Meldal M, Bock K, Paulsena H. Multiple column solid phase glycopeptide synthesis Tetrahedron Letters. 32: 5067-5070. DOI: 10.1016/S0040-4039(00)93429-4  0.667
1990 Jakobsen MH, Buchardt O, Holm A, Meldal M. A facile one-pot synthesis of 3,4-dihydro-3-hydroxy-4-oxo-1,2,3-benzotriazine and derivatives Synthesis. 1990: 1008-1010. DOI: 10.1055/S-1990-27078  0.391
1990 Meldal M, Jensen KJ. Pentafluorophenyl esters for the temporary protection of the α-carboxy group in solid phase glycopeptide synthesis Journal of the Chemical Society, Chemical Communications. 483-485. DOI: 10.1039/C39900000483  0.369
1990 Jansson AM, Meldal M, Back K. The active ester N-fmoc-3-O-[Ac4-α-D-Manp-(1→2)-Ac3-α-D-Manp-1-]=thre-O-Pfp as a building block in solid-phase synthesis of an o-linked dimannosyl glycopeptide. Tetrahedron Letters. 31: 6991-6994. DOI: 10.1016/S0040-4039(00)97224-1  0.353
1990 Meldal M, Book K. Pentafluorophenyl esters for temporary carboxyl group protection in solid phase synthesis of N-linked glycopeptides Tetrahedron Letters. 31: 6987-6990. DOI: 10.1016/S0040-4039(00)97223-X  0.375
1989 Mouritsen S, Meldal M, Rubin B, Holm A, Werdelin O. The T-lymphocyte proliferative response to synthetic peptide antigens of defined secondary structure. Scandinavian Journal of Immunology. 30: 723-730. PMID 2481338 DOI: 10.1111/J.1365-3083.1989.Tb02482.X  0.385
1988 Cameron LR, Holder JL, Meldal M, Sheppard RC. Peptide synthesis. Part 13. Feedback control in solid phase synthesis. Use of fluorenylmethoxycarbonyl amino acid 3,4-dihydro-4-oxo-1,2,3-benzotriazin-3-yl esters in a fully automated system Journal of the Chemical Society-Perkin Transactions 1. 2895-2901. DOI: 10.1039/P19880002895  0.461
1988 Atherton E, Holder JL, Meldal M, Sheppard RC, Valerio RM. Peptide synthesis. Part 12. 3,4-Dihydro-4-oxo-1,2,3-benzotriazin-3-yl esters of fluorenylmethoxycarbonyl amino acids as self-indicating reagents for solid phase peptide synthesis Journal of the Chemical Society-Perkin Transactions 1. 2887-2894. DOI: 10.1039/P19880002887  0.467
1987 Krogfelt KA, Meldal M, Klemm P. K88 fimbrial antigens: identification of antigenic determinants by the use of synthetic peptides Microbial Pathogenesis. 2: 465-472. PMID 2467165 DOI: 10.1016/0882-4010(87)90053-2  0.354
1987 Cameron L, Meldal M, Sheppard RC. Feedback control in organic synthesis. A system for solid phase peptide synthesis with true automation Journal of the Chemical Society, Chemical Communications. 270-272. DOI: 10.1039/C39870000270  0.422
1986 Meldal M. Synthesis of a putative subtype specific antigenic heptapeptide from Escherichia coli K88 ad protein fimbriae. Acta Chemica Scandinavica. 40: 242-249. PMID 2873700 DOI: 10.3891/Acta.Chem.Scand.40B-0242  0.41
1986 Atherton E, Cameron L, Meldal M, Sheppard RC. Self-indicating activated esters for use in solid phase peptide synthesis. Fluorenylmethoxycarbonylamino acid derivatives of 3-hydroxy-4-oxodihydrobenzotriazine Journal of the Chemical Society, Chemical Communications. 1763-1765. DOI: 10.1039/C39860001763  0.438
1985 Norberg T, Svenson SB, Bock K, Meldal M. Immunochemistry of SalmonellaO-antigens: Studies of Salmonella BO antigen epitopes by enzyme-linked immunosorbent inhibition assays Fems Microbiology Letters. 28: 171-176. DOI: 10.1111/J.1574-6968.1985.Tb00786.X  0.614
1984 Bock K, Meldal M, Bundle DR, Iversen T, Pinto BM, Garegg PJ, Kvanström I, Norberg T, Lindberg AA, Svenson SB. The conformation of Salmonella O-antigenic oligosaccharides of serogroups A, B, and D1 inferred from 1H- and 13C-nuclear magnetic resonance spectroscopy. Carbohydrate Research. 130: 35-53. PMID 6478461 DOI: 10.1016/0008-6215(84)85268-4  0.689
1984 Bock K, Meldal M, Bundle DR, Iversen T, Garegg PJ, Norberg T, Lindberg AA, Svenson SB. The conformation of Salmonella O-antigenic polysaccharide chains of serogroups A, B, and D1 predicted by semi-empirical, Hard-Sphere (HSEA) calculations. Carbohydrate Research. 130: 23-34. PMID 6478459 DOI: 10.1016/0008-6215(84)85267-2  0.693
1984 Bock K, Meldal M. Synthesis of tetrasaccharides related to the O-specific determinants of Salmonella serogroups A, B and D1 Acta Chemica Scandinavica. 15: 255-266. DOI: 10.3891/Acta.Chem.Scand.38B-0255  0.618
1984 Bock K, Meldal M. Synthesis of the branchpoint tetrasaccharide of the O-specific determinant of Salmonella serogroup B Cheminform. 15: 71-77. DOI: 10.1002/Chin.198433296  0.606
1983 Bock K, Meldal M, Meyer B, Wiebe L. Isomerization of D-glucose with glucose-isomerase. A mechanistic study. Acta Chemica Scandinavica. Series B: Organic Chemistry and Biochemistry. 37: 101-8. PMID 6880523 DOI: 10.3891/Acta.Chem.Scand.37B-0101  0.567
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