Frederik Diness - Publications

Affiliations: 
2006 Chemistry Carlsberg Laboratory, Copenhagen 

37 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2022 Fischer NH, Lopes van den Broek SI, Herth MM, Diness F. Radiolabeled albumin through SAr of cysteines as a potential pretargeting theranostic agent. Rsc Advances. 12: 35032-35036. PMID 36540259 DOI: 10.1039/d2ra06406e  0.751
2022 Fischer NH, Oliveira MT, Diness F. Chemical modification of proteins - challenges and trends at the start of the 2020s. Biomaterials Science. PMID 36519403 DOI: 10.1039/d2bm01237e  0.772
2022 Yang Y, Fischer NH, Oliveira MT, Hadaf GB, Liu J, Brock-Nannestad T, Diness F, Lee JW. Carbon dioxide enhances sulphur-selective conjugate addition reactions. Organic & Biomolecular Chemistry. PMID 35605989 DOI: 10.1039/d2ob00831a  0.771
2021 Fischer NH, Fumi E, Oliveira MT, Thulstrup PW, Diness F. Tuning peptide structure and function through fluorobenzene stapling. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 34897848 DOI: 10.1002/chem.202103788  0.783
2020 Fischer NH, Nielsen DS, Palmer D, Meldal M, Diness F. C-Terminal lactamization of peptides. Chemical Communications (Cambridge, England). PMID 33367306 DOI: 10.1039/d0cc06018f  0.764
2020 Wang Y, Oliveira MT, Madsen D, Thompson A, Meldal M, Diness F. Dihydroquinazolinones via A3-Type Reactions of N-Carbamoyliminium Ions. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32790088 DOI: 10.1002/Chem.202003117  0.75
2020 Madsen D, Jørgensen FP, Palmer D, Roux M, Olsen JV, Bols M, Schoffelen S, Diness F, Meldal M. Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12. Acs Combinatorial Science. PMID 32027120 DOI: 10.1021/Acscombsci.9B00197  0.767
2019 Hoang HN, Hill TA, Ruiz-Gómez G, Diness F, Mason JM, Wu C, Abbenante G, Shepherd NE, Fairlie DP. Twists or turns: stabilising alpha beta turns in tetrapeptides. Chemical Science. 10: 10595-10600. PMID 32110345 DOI: 10.1039/C9Sc04153B  0.42
2019 Jacobsen CBB, Nielsen DS, Meldal M, Diness F. Azotides as Modular Peptide-Based Ligands for Asymmetric Lewis Acid Catalysis. The Journal of Organic Chemistry. PMID 31033291 DOI: 10.1021/Acs.Joc.9B00732  0.611
2019 Hu H, Kofoed C, Li M, Gonçalves JPL, Hansen J, Wolfram M, Hansen AK, Friis Hansen CH, Diness F, Schoffelen S, Meldal M. Computational Evolution of Threonine-Rich β-Hairpin Peptides Mimicking Specificity and Affinity of Antibodies. Acs Central Science. 5: 259-269. PMID 30834314 DOI: 10.1021/Acscentsci.8B00614  0.745
2018 Embaby AM, Lelieveldt LPWM, Diness F, Meldal M. Metallo-Organozymes with Specific Proteolytic Activity. Chemistry: a European Journal. 24: 17424-17428. PMID 30146681 DOI: 10.1002/Chem.201803666  0.669
2018 Hu H, Nikitin SV, Berthelsen AB, Diness F, Schoffelen S, Meldal M. Sustainable Flow Synthesis of Encoded Beads for Combinatorial Chemistry and Chemical Biology. Acs Combinatorial Science. PMID 29969235 DOI: 10.1021/Acscombsci.8B00052  0.745
2018 Diness F, Bjerrum NJ, Begtrup M. Synthesis and stability of strongly acidic benzamide derivatives. Beilstein Journal of Organic Chemistry. 14: 523-530. PMID 29623113 DOI: 10.3762/Bjoc.14.38  0.443
2018 Embaby AM, Schoffelen S, Kofoed C, Meldal M, Diness F. Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification Angewandte Chemie. 57: 8022-8026. PMID 29469231 DOI: 10.1002/Anie.201712589  0.771
2018 Embaby AM, Schoffelen S, Kofoed C, Meldal M, Diness F. Inside Back Cover: Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification (Angew. Chem. Int. Ed. 27/2018) Angewandte Chemie. 57: 8831-8831. DOI: 10.1002/Anie.201805102  0.76
2018 Embaby AM, Schoffelen S, Kofoed C, Meldal M, Diness F. Innenrücktitelbild: Rational Tuning of Fluorobenzene Probes for Cysteine‐Selective Protein Modification (Angew. Chem. 27/2018) Angewandte Chemie. 130: 8463-8463. DOI: 10.1002/Ange.201805102  0.761
2017 Palmer D, Gonçalves JPL, Hansen LV, Wu B, Hald H, Schoffelen S, Diness F, Le Quement ST, Nielsen TE, Meldal M. Click Chemistry-Mediated Synthesis of Selective Melanocortin Receptor-4 Agonists. Journal of Medicinal Chemistry. PMID 28972753 DOI: 10.1021/Acs.Jmedchem.7B00353  0.612
2017 Wang Y, Madsen AØ, Diness F, Meldal M. Diversity oriented syntheses by combining CuAAC and stereoselective INCIC reactions with peptides. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 28833706 DOI: 10.1002/Chem.201702900  0.654
2017 Jacobsen CB, Meldal M, Diness F. Mechanism and Scope of Base‐Controlled Catalyst‐Free N‐Arylation of Amines with Unactivated Fluorobenzenes Chemistry: a European Journal. 23: 846-851. PMID 27739610 DOI: 10.1002/Chem.201604098  0.618
2016 Nikitin S, Palmer D, Meldal M, Diness F. Comparative studies of adhesion peptides based on l- or d-amino acids Journal of Peptide Science. 22: 642-646. PMID 27580849 DOI: 10.1002/Psc.2913  0.652
2016 Hansen J, Diness F, Meldal M. C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles. Organic & Biomolecular Chemistry. 14: 3238-45. PMID 26924021 DOI: 10.1039/C6Ob00213G  0.682
2015 Diness F, Meldal M. Fmox: A Base‐Labile Aldehyde Protecting Group European Journal of Organic Chemistry. 2015: 1433-1436. DOI: 10.1002/Ejoc.201403643  0.577
2014 Hill TA, Shepherd NE, Diness F, Fairlie DP. Constraining cyclic peptides to mimic protein structure motifs. Angewandte Chemie (International Ed. in English). 53: 13020-41. PMID 25287434 DOI: 10.1002/Anie.201401058  0.559
2014 Diness F, Begtrup M. Sequential direct SNAr reactions of pentafluorobenzenes with azole or indole derivatives. Organic Letters. 16: 3130-3. PMID 24869660 DOI: 10.1021/Ol5012554  0.467
2014 de Araujo AD, Hoang HN, Kok WM, Diness F, Gupta P, Hill TA, Driver RW, Price DA, Liras S, Fairlie DP. Comparative α-helicity of cyclic pentapeptides in water. Angewandte Chemie (International Ed. in English). 53: 6965-9. PMID 24828311 DOI: 10.1002/Anie.201310245  0.423
2014 Hill TA, Shepherd NE, Diness F, Fairlie DP. Fixierung cyclischer Peptide: Mimetika von Proteinstrukturmotiven Angewandte Chemie. 126: 13234-13257. DOI: 10.1002/Ange.201401058  0.493
2012 Nielsen DS, Hoang HN, Lohman RJ, Diness F, Fairlie DP. Total synthesis, structure, and oral absorption of a thiazole cyclic peptide, sanguinamide A. Organic Letters. 14: 5720-3. PMID 23130644 DOI: 10.1021/Ol3027347  0.463
2012 Jensen JM, Simonsen FC, Mastali A, Hald H, Lillebro I, Diness F, Olsen L, Mirza O. Biophysical characterization of the proton-coupled oligopeptide transporter YjdL. Peptides. 38: 89-93. PMID 22940668 DOI: 10.1016/J.Peptides.2012.08.012  0.418
2012 Diness F, Fairlie DP. Catalyst-free N-arylation using unactivated fluorobenzenes. Angewandte Chemie (International Ed. in English). 51: 8012-6. PMID 22865561 DOI: 10.1002/Anie.201202149  0.438
2011 Diness F, Nielsen DS, Fairlie DP. Synthesis of the thiazole-thiazoline fragment of largazole analogues. The Journal of Organic Chemistry. 76: 9845-51. PMID 22032297 DOI: 10.1021/Jo201675R  0.423
2011 Meldal M, Wu B, Diness F, Michael R, Hagel G. Metabolically stable cellular adhesion to inert surfaces. Chembiochem : a European Journal of Chemical Biology. 12: 2463-70. PMID 21928441 DOI: 10.1002/Cbic.201100382  0.611
2010 Meldal M, Tornøe CW, Nielsen TE, Diness F, Le Quement ST, Christensen CA, Jensen JF, Worm-Leonhard K, Groth T, Bouakaz L, Wu B, Hagel G, Keinicke L. Ralph F. Hirschmann award address 2009: Merger of organic chemistry with peptide diversity. Biopolymers. 94: 161-82. PMID 20225304 DOI: 10.1002/Bip.21344  0.782
2010 Diness F, Meldal M. Amino acid derived 1,4-dialkyl substituted imidazolones. Biopolymers. 94: 236-241. PMID 20225297 DOI: 10.1002/Bip.21359  0.601
2009 Diness F, Meldal M. Imidazolones in Diastereoselective Cyclization Reactions and CuII‐Catalysed Cross‐Coupling Reactions Chemistry: a European Journal. 15: 7044-7047. PMID 19544506 DOI: 10.1002/Chem.200900633  0.597
2006 Diness F, Beyer J, Meldal M. Solid‐Phase Synthesis of Tetrahydro‐β‐carbolines and Tetrahydroisoquinolines by Stereoselective Intramolecular N‐Carbamyliminium Pictet–Spengler Reactions Chemistry: a European Journal. 12: 8056-8066. PMID 16881029 DOI: 10.1002/Chem.200600138  0.64
2004 Diness F, Beyer J, Meldal M. Synthesis of 3‐Boc‐(1,3)‐oxazinane‐Protected Amino Aldehydes from Amino Acids and Their Conversion into Urea Precursors. Novel Building Blocks for Combinatorial Synthesis Qsar & Combinatorial Science. 23: 130-144. DOI: 10.1002/Qsar.200320012  0.599
2003 Nielsen TE, Diness F, Meldal M. The Pictet-Spengler reaction in solid-phase combinatorial chemistry. Current Opinion in Drug Discovery & Development. 6: 801-14. PMID 14758752  0.578
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