Year |
Citation |
Score |
2022 |
Picconi P, Hind CK, Sutton JM, Rahman KM. Covalent DNA Binding Is Essential for Gram-Negative Antibacterial Activity of Broad Spectrum Pyrrolobenzodiazepines. Antibiotics (Basel, Switzerland). 11. PMID 36551427 DOI: 10.3390/antibiotics11121770 |
0.731 |
|
2020 |
Picconi P, Hind C, Nahar KS, Jamshidi S, Di Maggio L, Saeed N, Evans B, Solomons J, Wand ME, Sutton JM, Rahman KM. New broad-spectrum antibiotics containing a pyrrolobenzodiazepine ring with activity against multidrug resistant Gram-negative bacteria. Journal of Medicinal Chemistry. PMID 32515951 DOI: 10.1021/acs.jmedchem.0c00328 |
0.81 |
|
2020 |
Vandera KA, Picconi P, Valero M, González-Gaitano G, Woods A, Clifton LA, Skoda MWA, Rahman KM, Harvey RD, Dreiss CA. Antibiotic-in-cyclodextrin-in-liposomes: formulation development and interactions with model bacterial membranes. Molecular Pharmaceutics. PMID 32352791 DOI: 10.1021/acs.molpharmaceut.0c00096 |
0.637 |
|
2019 |
Picconi P, Jeeves R, Moon CW, Jamshidi S, Nahar KS, Laws M, Bacon J, Rahman KM. Noncytotoxic Pyrrolobenzodiazepine-Ciprofloxacin Conjugate with Activity against . Acs Omega. 4: 20873-20881. PMID 31867477 DOI: 10.1021/acsomega.9b00834 |
0.773 |
|
2018 |
Thurston D, Corcoran D, Picconi P, Chui C, Procopiou G, Pysz I, Rahman K. Formation of a Novel C11-Acetone Adduct of a Pyrrolobenzodiazepine (PBD) with Loss of Cytotoxicity Synlett. 29: 1112-1116. DOI: 10.1055/S-0036-1591552 |
0.592 |
|
2017 |
Andriollo P, Hind C, Picconi P, Nahar KS, Jamshidi S, Varsha A, Clifford M, Sutton JM, Rahman KM. C8-linked pyrrolobenzodiazepine monomers with inverted building blocks show selective activity against MDR Gram-positive bacteria. Acs Infectious Diseases. PMID 29260545 DOI: 10.1021/acsinfecdis.7b00130 |
0.744 |
|
2017 |
Picconi P, Hind C, Jamshidi S, Nahar K, Clifford M, Wand ME, Sutton JM, Rahman KM. Triaryl benzimidazoles as a new class of antibacterial agents against resistant pathogenic microorganisms. Journal of Medicinal Chemistry. PMID 28650661 DOI: 10.1021/acs.jmedchem.7b00108 |
0.837 |
|
2017 |
Picconi P, Prabaharan P, Auer JL, Sandiford S, Cascio F, Chowdhury M, Hind C, Wand ME, Sutton JM, Rahman KM. Novel pyridyl nitrofuranyl isoxazolines show antibacterial activity against multiple drug resistant Staphylococcus species. Bioorganic & Medicinal Chemistry. PMID 28600080 DOI: 10.1016/j.bmc.2017.05.037 |
0.737 |
|
2015 |
Rossi D, Talman V, Gennäs GBA, Marra A, Picconi P, Nasti R, Serra M, Ann J, Amadio M, Pascale A, Tuominen RK, Yli-Kauhaluoma J, Lee J, Collina S. Beyond the affinity for protein kinase C: exploring 2-phenyl-3-hydroxypropyl pivalate analogues as C1 domain-targeting ligands Medchemcomm. 6: 547-554. DOI: 10.1039/C4Md00564C |
0.351 |
|
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