Year |
Citation |
Score |
2023 |
Stazi G, Taglieri L, Nicolai A, Romanelli A, Fioravanti R, Morrone S, Sabatino M, Ragno R, Taurone S, Nebbioso M, Carletti R, Artico M, Valente S, Scarpa S, Mai A. Retraction Note: Dissecting the role of novel EZH2 inhibitors in primary glioblastoma cell cultures: effects on proliferation, epithelialmesenchymal transition, migration, and on the pro-inflammatory phenotype. Clinical Epigenetics. 15: 179. PMID 37936214 DOI: 10.1186/s13148-023-01595-6 |
0.528 |
|
2023 |
Schiavone V, Romasco T, Di Pietrantonio N, Garzoli S, Palmerini C, Di Tomo P, Pipino C, Mandatori D, Fioravanti R, Butturini E, Sabatino M, Baldassarre MPA, Ragno R, Pandolfi A, Di Pietro N. Essential Oils from Mediterranean Plants Inhibit In Vitro Monocyte Adhesion to Endothelial Cells from Umbilical Cords of Females with Gestational Diabetes Mellitus. International Journal of Molecular Sciences. 24. PMID 37108387 DOI: 10.3390/ijms24087225 |
0.542 |
|
2022 |
Proia E, Ragno A, Antonini L, Sabatino M, Mladenovič M, Capobianco R, Ragno R. Ligand-based and structure-based studies to develop predictive models for SARS-CoV-2 main protease inhibitors through the 3d-qsar.com portal. Journal of Computer-Aided Molecular Design. PMID 35716228 DOI: 10.1007/s10822-022-00460-7 |
0.608 |
|
2022 |
Artini M, Papa R, Sapienza F, Božović M, Vrenna G, Tuccio Guarna Assanti V, Sabatino M, Garzoli S, Fiscarelli EV, Ragno R, Selan L. Essential Oils Biofilm Modulation Activity and Machine Learning Analysis on Isolates from Cystic Fibrosis Patients. Microorganisms. 10. PMID 35630332 DOI: 10.3390/microorganisms10050887 |
0.555 |
|
2022 |
Kurtanović N, Tomašević N, Matić S, Proia E, Sabatino M, Antonini L, Mladenović M, Ragno R. Human Estrogen Receptor Alpha Antagonists, Part 3: 3-D Pharmacophore and 3-D QSAR Guided Brefeldin A Hit-to-Lead Optimization toward New Breast Cancer Suppressants. Molecules (Basel, Switzerland). 27. PMID 35566172 DOI: 10.3390/molecules27092823 |
0.578 |
|
2022 |
Taglienti A, Donati L, Ferretti L, Tomassoli L, Sapienza F, Sabatino M, Di Massimo G, Fiorentino S, Vecchiarelli V, Nota P, Ragno R. Antiphytoviral Activity of Essential Oils and Hydrosols From , , and to Control Zucchini Yellow Mosaic Virus and Tomato Leaf Curl New Delhi Virus in L. Frontiers in Microbiology. 13: 840893. PMID 35547120 DOI: 10.3389/fmicb.2022.840893 |
0.538 |
|
2022 |
Valentini E, D'Aguanno S, Di Martile M, Montesano C, Ferraresi V, Patsilinakos A, Sabatino M, Antonini L, Chiacchiarini M, Valente S, Mai A, Colotti G, Ragno R, Trisciuoglio D, Del Bufalo D. Targeting the anti-apoptotic Bcl-2 family proteins: machine learning virtual screening and biological evaluation of new small molecules. Theranostics. 12: 2427-2444. PMID 35265218 DOI: 10.7150/thno.64233 |
0.753 |
|
2021 |
Nowak RP, Tumber A, Hendrix E, Ansari MSZ, Sabatino M, Antonini L, Andrijes R, Salah E, Mautone N, Pellegrini FR, Simelis K, Kawamura A, Johansson C, Passeri D, Pellicciari R, et al. First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53. Journal of Medicinal Chemistry. 64: 17031-17050. PMID 34843649 DOI: 10.1021/acs.jmedchem.1c00605 |
0.601 |
|
2021 |
Paglia G, Antonini L, Cervoni L, Ragno R, Sabatino M, Minacori M, Rubini E, Altieri F. A Comparative Analysis of Punicalagin Interaction with PDIA1 and PDIA3 by Biochemical and Computational Approaches. Biomedicines. 9. PMID 34829762 DOI: 10.3390/biomedicines9111533 |
0.538 |
|
2021 |
Kurtanović N, Tomašević N, Matić S, Mitrović MM, Kostić DA, Sabatino M, Antonini L, Ragno R, Mladenović M. Human estrogen receptor α antagonists, part 2: Synthesis driven by rational design, in vitro antiproliferative, and in vivo anticancer evaluation of innovative coumarin-related antiestrogens as breast cancer suppressants. European Journal of Medicinal Chemistry. 227: 113869. PMID 34710747 DOI: 10.1016/j.ejmech.2021.113869 |
0.549 |
|
2021 |
Mihović N, Tomašević N, Matić S, Mitrović MM, Kostić DA, Sabatino M, Antonini L, Ragno R, Mladenović M. Human Estrogen Receptor α Antagonists. Part 1: 3-D QSAR-Driven Rational Design of Innovative Coumarin-Related Antiestrogens as Breast Cancer Suppressants through Structure-Based and Ligand-Based Studies. Journal of Chemical Information and Modeling. 61: 5028-5053. PMID 34648283 DOI: 10.1021/acs.jcim.1c00530 |
0.559 |
|
2021 |
Di Martile M, Garzoli S, Sabatino M, Valentini E, D'Aguanno S, Ragno R, Del Bufalo D. Antitumor effect of Melaleuca alternifolia essential oil and its main component terpinen-4-ol in combination with target therapy in melanoma models. Cell Death Discovery. 7: 127. PMID 34059622 DOI: 10.1038/s41420-021-00510-3 |
0.587 |
|
2020 |
Papa R, Garzoli S, Vrenna G, Sabatino M, Sapienza F, Relucenti M, Donfrancesco O, Fiscarelli EV, Artini M, Selan L, Ragno R. Essential Oils Biofilm Modulation Activity, Chemical and Machine Learning Analysis. Application on Isolates from Cystic Fibrosis Patients. International Journal of Molecular Sciences. 21. PMID 33291608 DOI: 10.3390/ijms21239258 |
0.583 |
|
2020 |
Rinaldi F, Oliva A, Sabatino M, Imbriano A, Hanieh PN, Garzoli S, Mastroianni CM, De Angelis M, Miele MC, Arnaut M, Di Timoteo F, Marianecci C, Ragno R, Carafa M. Antimicrobial Essential Oil Formulation: Chitosan Coated Nanoemulsions for Nose to Brain Delivery. Pharmaceutics. 12. PMID 32709076 DOI: 10.3390/Pharmaceutics12070678 |
0.565 |
|
2020 |
Sabatino M, Fabiani M, Božović M, Garzoli S, Antonini L, Marcocci ME, Palamara AT, De Chiara G, Ragno R. Experimental Data Based Machine Learning Classification Models with Predictive Ability to Select in Vitro Active Antiviral and Non-Toxic Essential Oils. Molecules (Basel, Switzerland). 25. PMID 32466318 DOI: 10.3390/Molecules25102452 |
0.616 |
|
2020 |
Matutino Bastos T, Botelho Pereira Soares M, Haddad Franco C, Alcântara L, Antonini L, Sabatino M, Mautone N, Holanda Freitas-Junior L, Moraes CB, Ragno R, Rotili D, Schenkman S, Mai A, Silvio Moretti N. Identification of Inhibitors to Sirtuins Based on Compounds Developed to Human Enzymes. International Journal of Molecular Sciences. 21. PMID 32455951 DOI: 10.3390/Ijms21103659 |
0.638 |
|
2020 |
Di Vito M, Bellardi MG, Sanguinetti M, Mondello F, Girolamo A, Barbanti L, Garzoli S, Sabatino M, Ragno R, Vitali A, Palucci I, Posteraro B, Gasbarrini A, Prati GM, Aragona G, et al. Potent Activity of Essential Oil and Hydrolate Against Gut Yeast Isolates from Irritable Bowel Syndrome Patients-The Right Mix for Potential Therapeutic Use. Nutrients. 12. PMID 32392768 DOI: 10.3390/Nu12051329 |
0.59 |
|
2020 |
Caroselli S, Zwergel C, Pirolli A, Sabatino M, Xu Z, Kirsch G, Mai A, Colotti G, Altieri F, Canipari R, Valente S, Ragno R. Discovery of the First Human Arylsulfatase A Reversible Inhibitor Impairing Mouse Oocyte Fertilization. Acs Chemical Biology. PMID 32239919 DOI: 10.1021/Acschembio.9B00999 |
0.744 |
|
2019 |
Stazi G, Taglieri L, Nicolai A, Romanelli A, Fioravanti R, Morrone S, Sabatino M, Ragno R, Taurone S, Nebbioso M, Carletti R, Artico M, Valente S, Scarpa S, Mai A. Dissecting the role of novel EZH2 inhibitors in primary glioblastoma cell cultures: effects on proliferation, epithelial-mesenchymal transition, migration, and on the pro-inflammatory phenotype. Clinical Epigenetics. 11: 173. PMID 31791385 DOI: 10.1186/S13148-019-0763-5 |
0.589 |
|
2019 |
Patsilinakos A, Artini M, Papa R, Sabatino M, Božović M, Garzoli S, Vrenna G, Buzzi R, Manfredini S, Selan L, Ragno R. Machine Learning Analyses on Data including Essential Oil Chemical Composition and In Vitro Experimental Antibiofilm Activities against Species. Molecules (Basel, Switzerland). 24. PMID 30832446 DOI: 10.3390/Molecules24050890 |
0.75 |
|
2019 |
Oliva A, Garzoli S, Sabatino M, Tadić V, Costantini S, Ragno R, Božović M. Chemical composition and antimicrobial activity of essential oil of Helichrysum italicum (Roth) G. Don fil. (Asteraceae) from Montenegro. Natural Product Research. 1-4. PMID 30602287 DOI: 10.1080/14786419.2018.1538218 |
0.572 |
|
2019 |
Valentini E, Martile MD, Desideri M, Carcasole S, Patsilinakos A, Sabatino M, Mai A, Colotti G, Ragno R, Trisciuoglio D, Bufalo DD. Abstract 2502: Targeting anti-apoptotic Bcl-2 family for cancer therapy Cancer Research. DOI: 10.1158/1538-7445.Sabcs18-2502 |
0.721 |
|
2018 |
Artini M, Patsilinakos A, Papa R, Božović M, Sabatino M, Garzoli S, Vrenna G, Tilotta M, Pepi F, Ragno R, Selan L. Antimicrobial and Antibiofilm Activity and Machine Learning Classification Analysis of Essential Oils from Different Mediterranean Plants against Pseudomonas aeruginosa. Molecules (Basel, Switzerland). 23. PMID 29473844 DOI: 10.3390/Molecules23020482 |
0.757 |
|
2018 |
Sabatino M, Rotili D, Patsilinakos A, Forgione M, Tomaselli D, Alby F, Arimondo PB, Mai A, Ragno R. Disruptor of telomeric silencing 1-like (DOT1L): disclosing a new class of non-nucleoside inhibitors by means of ligand-based and structure-based approaches. Journal of Computer-Aided Molecular Design. PMID 29335872 DOI: 10.1007/S10822-018-0096-Z |
0.769 |
|
2018 |
Garzoli S, Božović M, Baldisserotto A, Sabatino M, Cesa S, Pepi F, Vicentini CB, Manfredini S, Ragno R. Essential oil extraction, chemical analysis and anti-Candida activity of Foeniculum vulgare Miller - new approaches. Natural Product Research. 32: 1254-1259. PMID 28617136 DOI: 10.1080/14786419.2017.1340291 |
0.577 |
|
2017 |
Carradori S, Bizzarri B, D'Ascenzio M, De Monte C, Grande R, Rivanera D, Zicari A, Mari E, Sabatino M, Patsilinakos A, Ragno R, Secci D. Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity. European Journal of Medicinal Chemistry. 140: 274-292. PMID 28963991 DOI: 10.1016/J.Ejmech.2017.09.026 |
0.773 |
|
2017 |
Mladenović M, Patsilinakos A, Pirolli A, Sabatino M, Ragno R. Understanding the Molecular Determinant of Reversible Human Monoamine Oxidase B Inhibitors Containing 2H-Chromen-2-One Core: Structure-Based and Ligand-Based Derived Three-Dimensional Quantitative Structure-Activity Relationships Predictive Models. Journal of Chemical Information and Modeling. 57: 787-814. PMID 28291352 DOI: 10.1021/Acs.Jcim.6B00608 |
0.734 |
|
2017 |
Božović M, Garzoli S, Sabatino M, Pepi F, Baldisserotto A, Andreotti E, Romagnoli C, Mai A, Manfredini S, Ragno R. Essential Oil Extraction, Chemical Analysis and Anti-Candida Activity of Calamintha nepeta (L.) Savi subsp. glandulosa (Req.) Ball-New Approaches. Molecules (Basel, Switzerland). 22. PMID 28134788 DOI: 10.3390/Molecules22020203 |
0.574 |
|
2017 |
Venditti A, Frezza C, Salutari G, di Cecco M, Ciaschetti G, Oliva A, De Angelis M, Vullo V, Sabatino M, Garzoli S, Pepi F, Ragno R, Serafini M, Bianco A. Composition of the Essential Oil of Coristospermum cuneifolium and Antimicrobial Activity Evaluation Planta Medica International Open. 4: e74-e81. DOI: 10.1055/S-0043-118131 |
0.553 |
|
2016 |
Coluccia A, Passacantilli S, Famiglini V, Sabatino M, Patsilinakos A, Ragno R, Mazzoccoli C, Sisinni L, Okuno A, Takikawa O, Silvestri R, La Regina G. New Inhibitors of Indoleamine 2,3-Dioxygenase 1: Molecular Modeling Studies, Synthesis, and Biological Evaluation. Journal of Medicinal Chemistry. 59: 9760-9773. PMID 27690429 DOI: 10.1021/Acs.Jmedchem.6B00718 |
0.779 |
|
2016 |
Consalvi S, Poce G, Ragno R, Sabatino M, La Motta C, Sartini S, Calderone V, Martelli A, Ghelardini C, Di Cesare Mannelli L, Biava M. A Series of COX-2 Inhibitors Endowed with NO-Releasing Properties: Synthesis, Biological Evaluation, and Docking Analysis. Chemmedchem. 11: 1804-11. PMID 27229194 DOI: 10.1002/Cmdc.201600086 |
0.635 |
|
2015 |
Consalvi S, Alfonso S, Di Capua A, Poce G, Pirolli A, Sabatino M, Ragno R, Anzini M, Sartini S, La Motta C, Di Cesare Mannelli L, Ghelardini C, Biava M. Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors. Bioorganic & Medicinal Chemistry. 23: 810-20. PMID 25596758 DOI: 10.1016/J.Bmc.2014.12.041 |
0.764 |
|
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