| Year |
Citation |
Score |
| 2023 |
Choi JY, Noguchi Y, Alburger JM, Bayle S, Chung E, Grant W, Chaikuad A, Knapp S, Duckett DR, Roush WR. Structure-Based Development of Isoform-Selective Inhibitors of Casein Kinase 1ε vs Casein Kinase 1δ. Journal of Medicinal Chemistry. PMID 37204207 DOI: 10.1021/acs.jmedchem.2c01180 |
0.44 |
|
| 2022 |
Shahoei R, Pangeni S, Sanders MA, Zhang H, Mladenovic-Lucas L, Roush WR, Halvorsen G, Kelly CV, Granneman JG, Huang YM. Molecular Modeling of ABHD5 Structure and Ligand Recognition. Frontiers in Molecular Biosciences. 9: 935375. PMID 35836935 DOI: 10.3389/fmolb.2022.935375 |
0.764 |
|
| 2020 |
Jílková A, Rubešová P, Fanfrlík J, Fajtová P, Řezáčová P, Brynda J, Lepšík M, Mertlíková-Kaiserová H, Emal CD, Renslo AR, Roush WR, Horn M, Caffrey CR, Mareš M. Druggable Hot Spots in the Schistosomiasis Cathepsin B1 Target Identified by Functional and Binding Mode Analysis of Potent Vinyl Sulfone Inhibitors. Acs Infectious Diseases. PMID 33175511 DOI: 10.1021/acsinfecdis.0c00501 |
0.773 |
|
| 2019 |
Doebelin C, He Y, Campbell S, Nuhant P, Kumar N, Koenig M, Garcia-Ordonez R, Chang MR, Roush WR, Lin L, Kahn S, Cameron MD, Griffin PR, Solt LA, Kamenecka TM. Discovery and optimization of a series of sulfonamide inverse agonists for the retinoic acid receptor-related receptor-α. Medicinal Chemistry (Shariqah (United Arab Emirates)). PMID 30799793 DOI: 10.2174/1573406415666190222124745 |
0.69 |
|
| 2019 |
Mahmud I, Tian G, Wang J, Stowe R, Huo Z, Zhang Y, Purayil HT, Helm E, Drashansky T, Avram D, Daaka Y, Roush WR, Liao D. Abstract 4718: SR-4370, a potent and selective inhibitor of class I HDACs, suppresses AR signaling and in vivo prostate tumor growth Cancer Research. DOI: 10.1158/1538-7445.Sabcs18-4718 |
0.681 |
|
| 2018 |
Zyserman I, Mondal D, Sarabia F, McKerrow JH, Roush WR, Debnath A. Identification of cysteine protease inhibitors as new drug leads against Naegleria fowleri. Experimental Parasitology. PMID 29551628 DOI: 10.1016/J.Exppara.2018.03.010 |
0.506 |
|
| 2018 |
Tian G, Mahmud I, Stowe R, Zhang Y, Purayil HT, Roush W, Daaka Y, Liao D. Abstract B004: A combination of two chemically distinct inhibitors of class I HDACs is highly effective to suppress AR signaling and in vivo growth of prostate cancer xenograft Cancer Research. 78. DOI: 10.1158/1538-7445.Prca2017-B004 |
0.685 |
|
| 2018 |
Mahmud I, Garrett TJ, Stowe R, Roush WR, Liao D. Abstract LB-248: Chemically distinct class I HDAC inhibitors synergize to inhibit global lipid metabolism in cancer Cancer Research. 78. DOI: 10.1158/1538-7445.Am2018-Lb-248 |
0.696 |
|
| 2017 |
Monastyrskyi A, Nilchan N, Quereda V, Noguchi Y, Ruiz C, Grant W, Cameron M, Duckett D, Roush W. Development of dual casein kinase 1δ/1ε (CK1δ/ε) inhibitors for treatment of breast cancer. Bioorganic & Medicinal Chemistry. PMID 29289448 DOI: 10.1016/J.Bmc.2017.12.020 |
0.487 |
|
| 2017 |
Rondini EA, Mladenovic-Lucas L, Roush WR, Halvorsen G, Green AE, Granneman JG. Novel pharmacological probes reveal ABHD5 as a locus of lipolysis control in white and brown adipocytes. The Journal of Pharmacology and Experimental Therapeutics. PMID 28928121 DOI: 10.1124/Jpet.117.243253 |
0.768 |
|
| 2017 |
Allais C, Roush WR. Enantio- and Diastereoselective Synthesis of 1,5-syn-(Z)-Amino Alcohols via Imine Double Allylboration: Synthesis of trans-1,2,3,6-Tetrahydropyridines and Total Synthesis of Andrachcine. Organic Letters. PMID 28471668 DOI: 10.1021/Acs.Orglett.7B00995 |
0.767 |
|
| 2017 |
Ho T, Fieser M, Danheiser R, Roush W, Fieser L. Tetrakis(triphenylphosphine)nickel(0) Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos09647 |
0.383 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Rhodium(II) carboxylates Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos08768.Pub6 |
0.436 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Phosphorus(V) sulfide Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos08273.Pub3 |
0.407 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Phenyliodine(III) dichloride Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos07987 |
0.311 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Palladium(II) chloride Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos07690.Pub6 |
0.411 |
|
| 2017 |
Ho T, Fieser M, Danheiser R, Roush W, Fieser L. Palladium(II) acetate Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos07552.Pub6 |
0.448 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Manganese(II) Chloride Fieser and Fieser's Reagents For Organic Synthesis. 368-368. DOI: 10.1002/9780471264194.Fos06703.Pub2 |
0.345 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Magnesium Bromide Etherate Fieser and Fieser's Reagents For Organic Synthesis. 364-364. DOI: 10.1002/9780471264194.Fos06647.Pub2 |
0.395 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Lithium 2,2,6,6‐Tetramethylpiperidide, LiTMP Fieser and Fieser's Reagents For Organic Synthesis. 361-362. DOI: 10.1002/9780471264194.Fos06576.Pub4 |
0.502 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Lithium diisopropylamide (LDA) Fieser and Fieser's Reagents For Organic Synthesis. 358-359. DOI: 10.1002/9780471264194.Fos06433.Pub6 |
0.4 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Lithium aluminum hydride Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos06257.Pub3 |
0.361 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Dihydridotetrakis(triphenylphosphine)ruthenium(II) Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos04013.Pub2 |
0.382 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Copper(I) Iodide Fieser and Fieser's Reagents For Organic Synthesis. 194-198. DOI: 10.1002/9780471264194.Fos02911.Pub6 |
0.471 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Copper(I) cyanide Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos02897.Pub5 |
0.448 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Copper(II) Chloride Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos02878.Pub6 |
0.412 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Copper(I) t-Butoxide Fieser and Fieser's Reagents For Organic Synthesis. 225-225. DOI: 10.1002/9780471264194.Fos02868.Pub4 |
0.408 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Boron trifluoride etherate Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos01542.Pub6 |
0.5 |
|
| 2017 |
Ho T, Fieser M, Danheiser R, Roush W, Fieser L. Bis(dibenzylideneacetone)palladium(0) Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos01118.Pub3 |
0.442 |
|
| 2017 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Copper(I) Chloride Fieser and Fieser's Reagents For Organic Synthesis. 1-4. DOI: 10.1002/047084289X.Rc215.Pub2 |
0.424 |
|
| 2016 |
Getun IV, Wu Z, Fallahi M, Ouizem S, Liu Q, Li W, Costi R, Roush WR, Cleveland JL, Bois PR. Functional Roles of Acetylated Histone Marks at Mouse Meiotic Recombination Hotspots. Molecular and Cellular Biology. PMID 27821479 DOI: 10.1128/Mcb.00942-15 |
0.745 |
|
| 2016 |
Nair RN, Mishra JK, Li F, Tortosa M, Yang C, Doherty JR, Cameron M, Cleveland JL, Roush WR, Bannister TD. Exploiting the co-reliance of tumours upon transport of amino acids and lactate: Gln and Tyr conjugates of MCT1 inhibitors. Medchemcomm. 7: 900-905. PMID 27347360 DOI: 10.1039/C5Md00579E |
0.764 |
|
| 2016 |
Jones BD, Tochowicz A, Tang Y, Cameron MD, McCall LI, Hirata K, Siqueira-Neto JL, Reed SL, McKerrow JH, Roush WR. Synthesis and Evaluation of Oxyguanidine Analogues of the Cysteine Protease Inhibitor WRR-483 against Cruzain. Acs Medicinal Chemistry Letters. 7: 77-82. PMID 26819670 DOI: 10.1021/Acsmedchemlett.5B00336 |
0.308 |
|
| 2015 |
Rosenberg LH, Lafitte M, Quereda V, Grant W, Chen W, Bibian M, Noguchi Y, Fallahi M, Yang C, Chang JC, Roush WR, Cleveland JL, Duckett DR. Therapeutic targeting of casein kinase 1δ in breast cancer. Science Translational Medicine. 7: 318ra202. PMID 26676609 DOI: 10.1126/scitranslmed.aac8773 |
0.425 |
|
| 2015 |
Sanders MA, Madoux F, Mladenovic L, Zhang H, Ye X, Angrish M, Mottillo EP, Caruso JA, Halvorsen G, Roush WR, Chase P, Hodder P, Granneman JG. Endogenous and Synthetic ABHD5 Ligands Regulate ABHD5-Perilipin Interactions and Lipolysis in Fat and Muscle. Cell Metabolism. PMID 26411340 DOI: 10.1016/J.Cmet.2015.08.023 |
0.765 |
|
| 2015 |
Schreiber SL, Kotz JD, Li M, Aubé J, Austin CP, Reed JC, Rosen H, White EL, Sklar LA, Lindsley CW, Alexander BR, Bittker JA, Clemons PA, de Souza A, Foley MA, ... ... Roush WR, et al. Advancing Biological Understanding and Therapeutics Discovery with Small-Molecule Probes. Cell. 161: 1252-1265. PMID 26046436 DOI: 10.1016/J.Cell.2015.05.023 |
0.388 |
|
| 2015 |
Ghalei H, Schaub FX, Doherty JR, Noguchi Y, Roush WR, Cleveland JL, Stroupe ME, Karbstein K. Hrr25/CK1δ-directed release of Ltv1 from pre-40S ribosomes is necessary for ribosome assembly and cell growth. The Journal of Cell Biology. 208: 745-59. PMID 25778921 DOI: 10.1083/Jcb.201409056 |
0.503 |
|
| 2015 |
Wang Y, Stowe RL, Pinello CE, Tian G, Madoux F, Li D, Zhao LY, Li JL, Wang Y, Wang Y, Ma H, Hodder P, Roush WR, Liao D. Identification of histone deacetylase inhibitors with benzoylhydrazide scaffold that selectively inhibit class I histone deacetylases. Chemistry & Biology. 22: 273-84. PMID 25699604 DOI: 10.1016/J.Chembiol.2014.12.015 |
0.695 |
|
| 2015 |
Corzo CA, Mari Y, Chang MR, Khan T, Kuruvilla D, Nuhant P, Kumar N, West GM, Duckett DR, Roush WR, Griffin PR. Antiproliferation activity of a small molecule repressor of liver receptor homolog 1. Molecular Pharmacology. 87: 296-304. PMID 25473120 DOI: 10.1124/Mol.114.095554 |
0.698 |
|
| 2015 |
El Hilali X, Roush WR. ChemInform Abstract: Enantio- and Diastereoselective Synthesis of syn-β-Hydroxy-α-alkenyl Carboxamides via Reductive Aldol Reactions of Morpholine 4-Methyl-2,3-pentadienoic Carboxamide with Diisopinocampheylborane. Cheminform. 46: no-no. DOI: 10.1002/chin.201540027 |
0.33 |
|
| 2015 |
Abbott JR, Allais C, Roush WR. Enantioselective Reductive Syn-Aldol Reactions of 4-Acryloylmorpholine: Preparation of (2R, 3S)-3-Hydroxy-2-methyl-1-morpholino-5-phenylpentan-1-one Organic Syntheses. 92: 38-57. DOI: 10.1002/0471264229.Os092.04 |
0.727 |
|
| 2014 |
Wang H, Yang C, Doherty JR, Roush WR, Cleveland JL, Bannister TD. Synthesis and structure-activity relationships of pteridine dione and trione monocarboxylate transporter 1 inhibitors. Journal of Medicinal Chemistry. 57: 7317-24. PMID 25068893 DOI: 10.1021/Jm500640X |
0.637 |
|
| 2014 |
Doherty JR, Yang C, Scott KE, Cameron MD, Fallahi M, Li W, Hall MA, Amelio AL, Mishra JK, Li F, Tortosa M, Genau HM, Rounbehler RJ, Lu Y, Dang CV, ... ... Roush WR, et al. Blocking lactate export by inhibiting the Myc target MCT1 Disables glycolysis and glutathione synthesis. Cancer Research. 74: 908-20. PMID 24285728 DOI: 10.1158/0008-5472.Can-13-2034 |
0.763 |
|
| 2014 |
Wang Y, Stowe R, Pinello CE, Zhao LY, Tian G, Hodder P, Roush WR, Liao D. Abstract 2525: Identification and characterization of class I HDAC-specific small-molecule inhibitors with a novel pharmacophore Cancer Research. 74: 2525-2525. DOI: 10.1158/1538-7445.Am2014-2525 |
0.694 |
|
| 2014 |
Knochel P, Haas D, Allais C, Tsai AS, Nuhant P, Roush WR. 1,4-Reductive Aldol Reactions of Substituted α,β-Unsaturated Amides Synfacts. 10: 188-188. DOI: 10.1055/S-0033-1340576 |
0.383 |
|
| 2014 |
El Hilali X, Roush WR. Enantio- and diastereoselective synthesis of syn-β-hydroxy-α-alkenyl carboxamides via reductive aldol reactions of morpholine 4-methyl-2,3-pentadienoic carboxamide with diisopinocampheylborane Tetrahedron Letters. DOI: 10.1016/J.Tetlet.2015.01.018 |
0.449 |
|
| 2014 |
Allais C, Tsai AS, Nuhant P, Roush WR. ChemInform Abstract: Generation of Stereochemically Defined Tetrasubstituted Enolborinates by 1,4-Hydroboration of α,β-Unsaturated Morpholine Carboxamides with (Diisopinocampheyl)borane. Cheminform. 45: no-no. DOI: 10.1002/chin.201419048 |
0.709 |
|
| 2013 |
Allais C, Tsai AS, Nuhant P, Roush WR. Generation of stereochemically defined tetrasubstituted enolborinates by 1,4-hydroboration of α,β-unsaturated morpholine carboxamides with (diisopinocampheyl)borane. Angewandte Chemie (International Ed. in English). 52: 12888-91. PMID 24281884 DOI: 10.1002/Anie.201307302 |
0.825 |
|
| 2013 |
Kister J, Ess DH, Roush WR. Enantio- and diastereoselective synthesis of syn-β-hydroxy-α-vinyl carboxylic esters via reductive aldol reactions of ethyl allenecarboxylate with 10-TMS-9-Borabicyclo[3.3.2]decane and DFT analysis of the hydroboration pathway. Organic Letters. 15: 5436-9. PMID 24138187 DOI: 10.1021/Ol4025277 |
0.656 |
|
| 2013 |
Chen M, Roush WR. Enantiodivergent hydroboration reactions of a racemic allenylsilane with diisopinocampheylborane and Curtin-Hammett controlled double asymmetric crotylboration reactions of (S)-E-αphenyldimethylsilyl( (d) diisopinocampheyl)-crotylborane. Tetrahedron. 69: 7551-7558. PMID 24068848 DOI: 10.1016/j.tet.2013.06.053 |
0.396 |
|
| 2013 |
Chen M, Roush WR. Enantiodivergent Hydroboration Reactions of a Racemic Allenylsilane with Diisopinocampheylborane and Curtin-Hammett Controlled Double Asymmetric Crotylboration Reactions of (S)-E-α-phenyldimethylsilyl( (d) diisopinocampheyl)-crotylborane. Tetrahedron. 69: 5468-5475. PMID 24039304 DOI: 10.1016/J.Tet.2013.04.098 |
0.484 |
|
| 2013 |
Allais C, Nuhant P, Roush WR. (Diisopinocampheyl)borane-mediated reductive aldol reactions of acrylate esters: enantioselective synthesis of anti-aldols. Organic Letters. 15: 3922-5. PMID 23885946 DOI: 10.1021/Ol401679G |
0.833 |
|
| 2013 |
Nuhant P, Allais C, Roush WR. Diisopinocampheylborane-mediated reductive aldol reactions: highly enantio- and diastereoselective synthesis of syn aldols from N-acryloylmorpholine. Angewandte Chemie (International Ed. in English). 52: 8703-7. PMID 23818095 DOI: 10.1002/Anie.201302535 |
0.846 |
|
| 2013 |
Bibian M, Rahaim RJ, Choi JY, Noguchi Y, Schürer S, Chen W, Nakanishi S, Licht K, Rosenberg LH, Li L, Feng Y, Cameron MD, Duckett DR, Cleveland JL, Roush WR. Development of highly selective casein kinase 1δ/1ε (CK1δ/ε) inhibitors with potent antiproliferative properties. Bioorganic & Medicinal Chemistry Letters. 23: 4374-80. PMID 23787102 DOI: 10.1016/J.Bmcl.2013.05.075 |
0.507 |
|
| 2013 |
Chen M, Roush WR. Enantioselective synthesis of (Z)- and (E)-2-methyl-1,5-anti-pentenediols via an allene hydroboration-double-allylboration reaction sequence. Journal of the American Chemical Society. 135: 9512-7. PMID 23758559 DOI: 10.1021/Ja4033633 |
0.488 |
|
| 2013 |
Tsai AS, Chen M, Roush WR. Chiral Brønsted Acid Catalyzed Enantioselective Synthesis of anti-Homopropargyl Alcohols via Kinetic Resolution-Aldehyde Allenylboration Using Racemic Allenylboronates. Organic Letters. 15: 2325. PMID 23578147 DOI: 10.1021/Ol400932E |
0.601 |
|
| 2013 |
Chen M, Roush WR. Enantioselective synthesis of (E)-δ-silyl-anti-homoallylic alcohols via an enantiodivergent hydroboration-crotylboration reaction of a racemic allenylsilane. Organic Letters. 15: 1662-5. PMID 23534391 DOI: 10.1021/Ol4004405 |
0.45 |
|
| 2013 |
Nuhant P, Roush WR. Enantio- and diastereoselective synthesis of N-acetyl dihydrotetrafibricin methyl ester. Journal of the American Chemical Society. 135: 5340-3. PMID 23530855 DOI: 10.1021/Ja401918R |
0.792 |
|
| 2013 |
Tsai AS, Chen M, Roush WR. Chiral Brønsted acid catalyzed enantioselective synthesis of anti-homopropargyl alcohols via kinetic resolution-aldehyde allenylboration using racemic allenylboronates. Organic Letters. 15: 1568-71. PMID 23484801 DOI: 10.1021/Ol4003459 |
0.625 |
|
| 2013 |
Geist JG, Barth R, Roush WR. Enantioselective synthesis of the C1-C11 fragment of tedanolide C. Organic Letters. 15: 58-61. PMID 23249423 DOI: 10.1021/Ol303089W |
0.745 |
|
| 2013 |
Abbott JR, Roush WR. Stereoselective synthesis of the disaccharide unit of incednine. Organic Letters. 15: 62-4. PMID 23249392 DOI: 10.1021/Ol303093Z |
0.439 |
|
| 2013 |
Chen M, Roush WR. Crotylboron-based synthesis of the polypropionate units of chaxamycins A/D, salinisporamycin, and rifamycin S. The Journal of Organic Chemistry. 78: 3-8. PMID 22703288 DOI: 10.1021/Jo3008226 |
0.461 |
|
| 2013 |
Chen YT, Brinen LS, Kerr ID, Hansell E, Doyle PS, McKerrow JH, Roush WR. Structure of WRR-483 bound to cruzain Plos Neglected Tropical Diseases. DOI: 10.1371/Journal.Pntd.0000825.G003 |
0.441 |
|
| 2013 |
Nuhant P, Allais C, Roush WR. ChemInform Abstract: Diisopinocampheylborane-Mediated Reductive Aldol Reactions: Highly Enantio- and Diastereoselective Synthesis of syn Aldols from N-Acryloylmorpholine. Cheminform. 45: no-no. DOI: 10.1002/chin.201402025 |
0.737 |
|
| 2013 |
Allais C, Nuhant P, Roush WR. ChemInform Abstract: (Diisopinocampheyl)borane-Mediated Reductive Aldol Reactions of Acrylate Esters: Enantioselective Synthesis of anti-Aldols. Cheminform. 44: no-no. DOI: 10.1002/chin.201350057 |
0.749 |
|
| 2013 |
Chen M, Roush WR. ChemInform Abstract: Enantioselective Synthesis of (Z)- and (E)-2-Methyl-1,5-anti-pentenediols via an Allene Hydroboration-Double-Allylboration Reaction Sequence. Cheminform. 44: no-no. DOI: 10.1002/chin.201349045 |
0.344 |
|
| 2013 |
Chen M, Roush WR. ChemInform Abstract: Enantiodivergent Hydroboration Reactions of a Racemic Allenylsilane with Diisopinocampheylborane and Curtin-Hammett Controlled Double Asymmetric Crotylboration Reactions of (S)-E-α-Phenyldimethylsilyl (ddiisopinocampheyl)-crotylborane Cheminform. 44: no-no. DOI: 10.1002/chin.201345023 |
0.403 |
|
| 2013 |
Chen M, Roush WR. ChemInform Abstract: Enantioselective Synthesis of (E)-δ-Silyl-anti-homoallylic Alcohols via an Enantiodivergent Hydroboration-Crotylboration Reaction of a Racemic Allenylsilane. Cheminform. 44: no-no. DOI: 10.1002/chin.201333198 |
0.302 |
|
| 2013 |
Tsai AS, Chen M, Roush WR. ChemInform Abstract: Chiral Broensted Acid Catalyzed Enantioselective Synthesis of anti-Homopropargyl Alcohols via Kinetic Resolution-Aldehyde Allenylboration Using Racemic Allenylboronates. Cheminform. 44: no-no. DOI: 10.1002/chin.201333039 |
0.541 |
|
| 2013 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. 4‐Dimethylaminopyridine (DMAP) Fieser and Fieser's Reagents For Organic Synthesis. 254-255. DOI: 10.1002/9780471264194.Fos04311.Pub5 |
0.396 |
|
| 2013 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Diisobutylaluminum Hydride, (DIBAL‐H) Fieser and Fieser's Reagents For Organic Synthesis. 253-253. DOI: 10.1002/9780471264194.Fos04085.Pub5 |
0.394 |
|
| 2013 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. 2,3-Dichloro-5,6-Dicyano-1,4-Benzoquinone (DDQ) Fieser and Fieser's Reagents For Organic Synthesis. 207-209. DOI: 10.1002/9780471264194.Fos03620.Pub5 |
0.306 |
|
| 2013 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. t‐Butyl Hydroperoxide Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos01966.Pub5 |
0.321 |
|
| 2012 |
Dossey AT, Whitaker JM, Dancel MC, Vander Meer RK, Bernier UR, Gottardo M, Roush WR. Defensive spiroketals from Asceles glaber (Phasmatodea): absolute configuration and effects on ants and mosquitoes. Journal of Chemical Ecology. 38: 1105-15. PMID 22976590 DOI: 10.1007/S10886-012-0183-X |
0.542 |
|
| 2012 |
Chen M, Roush WR. Enantioselective synthesis of anti- and syn-homopropargyl alcohols via chiral Brønsted acid catalyzed asymmetric allenylboration reactions. Journal of the American Chemical Society. 134: 10947-52. PMID 22731887 DOI: 10.1021/Ja3031467 |
0.53 |
|
| 2012 |
Han JL, Chen M, Roush WR. Diastereo- and enantioselective synthesis of (E)-2-Methyl-1,2-syn- and (E)-2-Methyl-1,2-anti-3-pentenediols via allenylboronate kinetic resolution with ((d)Ipc)2BH and aldehyde allylboration. Organic Letters. 14: 3028-31. PMID 22646839 DOI: 10.1021/Ol3010968 |
0.438 |
|
| 2012 |
Chen M, Roush WR. Enantioselective synthesis of (+)-crocacin C. An example of a highly challenging mismatched double asymmetric δ-stannylcrotylboration reaction. Organic Letters. 14: 1880-3. PMID 22409510 DOI: 10.1021/Ol300476F |
0.579 |
|
| 2012 |
Chen M, Roush WR. Enantioselective synthesis of (-)-basiliskamide A. Organic Letters. 14: 1556-9. PMID 22372693 DOI: 10.1021/Ol300282E |
0.555 |
|
| 2012 |
Chen M, Roush WR. Highly stereoselective synthesis of anti,anti-dipropionate stereotriads: a solution to the long-standing problem of challenging mismatched double asymmetric crotylboration reactions. Journal of the American Chemical Society. 134: 3925-31. PMID 22332989 DOI: 10.1021/Ja300472A |
0.537 |
|
| 2012 |
Chen M, Roush WR. Total synthesis of (-)-tirandamycin C. Organic Letters. 14: 426-8. PMID 22148850 DOI: 10.1021/Ol203161U |
0.523 |
|
| 2012 |
Nuhant P, Kister J, Lira R, Sorg A, Roush WR. Development of a double allylboration reagent targeting 1,5-syn-(E)-diols: application to the synthesis of the C(23)–C(40) fragment of tetrafibricin [Tetrahedron 67 (35) (2011) 6497–6512] Tetrahedron. 68: 774. DOI: 10.1016/J.Tet.2011.10.077 |
0.814 |
|
| 2012 |
Chen M, Roush WR. ChemInform Abstract: Enantioselective Synthesis of anti- and syn-Homopropargyl Alcohols via Chiral Broensted Acid Catalyzed Asymmetric Allenylboration Reactions. Cheminform. 43: no-no. DOI: 10.1002/chin.201251026 |
0.329 |
|
| 2012 |
Sun H, Roush WR, Candito DA, Blanchot M, Lautens M. Synthesis of (S,S)‐Diisopropyl Tartrate (E)‐Crotylboronate and Its Reaction with Aldehydes: (2R,3R,4R)‐1,2‐Dideoxy‐2‐Ethenyl‐4,5‐O‐(1‐Methylethylidene)‐Xylitol Organic Syntheses. 88: 181-196. DOI: 10.1002/0471264229.Os088.17 |
0.79 |
|
| 2011 |
Sun H, Roush WR, Hughes D. SYNTHESIS OF (+)-B-ALLYLDIISOPINOCAMPHEYLBORANE AND ITS REACTION WITH ALDEHYDES. Organic Syntheses; An Annual Publication of Satisfactory Methods For the Preparation of Organic Chemicals. 88: 87-102. PMID 22962503 DOI: 10.1002/0471264229.Os088.09 |
0.778 |
|
| 2011 |
Ying M, Roush WR. Studies on the Synthesis of Reidispongiolide A: Stereoselective Synthesis of the C(22)-C(36) Fragment. Tetrahedron. 67: 10274-10280. PMID 22711935 DOI: 10.1016/J.Tet.2011.10.029 |
0.519 |
|
| 2011 |
Roth J, Minond D, Darout E, Liu Q, Lauer J, Hodder P, Fields GB, Roush WR. Identification of novel, exosite-binding matrix metalloproteinase-13 inhibitor scaffolds. Bioorganic & Medicinal Chemistry Letters. 21: 7180-4. PMID 22018790 DOI: 10.1016/J.Bmcl.2011.09.077 |
0.751 |
|
| 2011 |
Nuhant P, Kister J, Lira R, Sorg A, Roush WR. Development of a Double Allylboration Reagent Targeting 1,5-syn-(E)-Diols: Application to the Synthesis of the C(23)-C(40) Fragment of Tetrafibricin. Tetrahedron. 67: 6497-6512. PMID 21857752 DOI: 10.1016/J.Tet.2011.06.008 |
0.819 |
|
| 2011 |
Zhou Y, Agudelo J, Lu K, Goetz DH, Hansell E, Chen YT, Roush WR, McKerrow J, Craik CS, Amberg SM, Simmons G. Inhibitors of SARS-CoV entry--identification using an internally-controlled dual envelope pseudovirion assay. Antiviral Research. 92: 187-94. PMID 21820471 DOI: 10.1016/J.Antiviral.2011.07.016 |
0.48 |
|
| 2011 |
Sun H, Roush WR, Candito DA, Blanchot M, Lautens M. SYNTHESIS OF (S,S)-DIISOPROPYL TARTRATE (E)-CROTYLBORONATE AND ITS REACTION WITH ALDEHYDES: (2R,3R,4R)-1,2-DIDEOXY-2-ETHENYL-4,5-O-(1-METHYLETHYLIDENE)-XYLITOL. Organic Syntheses; An Annual Publication of Satisfactory Methods For the Preparation of Organic Chemicals. 88: 181-196. PMID 21666877 |
0.784 |
|
| 2011 |
Sun H, Abbott JR, Roush WR. Stereoselective synthesis of a model C(18)-C(35) spiroketal fragment of integramycin. Organic Letters. 13: 2734-7. PMID 21510632 DOI: 10.1021/Ol200834P |
0.827 |
|
| 2011 |
Halvorsen GT, Roush WR. Stereoselective Synthesis of the Decahydrofluorene Core of the Hirsutellones. Tetrahedron Letters. 52: 2072-2075. PMID 21503271 DOI: 10.1016/J.Tetlet.2010.10.111 |
0.838 |
|
| 2011 |
Solt LA, Kumar N, Nuhant P, Wang Y, Lauer JL, Liu J, Istrate MA, Kamenecka TM, Roush WR, Vidovi? D, Schürer SC, Xu J, Wagoner G, Drew PD, Griffin PR, et al. Suppression of TH17 differentiation and autoimmunity by a synthetic ROR ligand. Nature. 472: 491-4. PMID 21499262 DOI: 10.1038/Nature10075 |
0.691 |
|
| 2011 |
Chen M, Roush WR. Enantioconvergent hydroboration of a racemic allene: enantioselective synthesis of (E)-δ-stannyl-anti-homoallylic alcohols via aldehyde crotylboration. Journal of the American Chemical Society. 133: 5744-7. PMID 21449594 DOI: 10.1021/Ja2010187 |
0.42 |
|
| 2011 |
Chen M, Roush WR. Enantioselective syntheses of syn- and anti-β-hydroxyallylsilanes via allene hydroboration-aldehyde allylboration reactions. Organic Letters. 13: 1992-5. PMID 21410173 DOI: 10.1021/Ol200392U |
0.459 |
|
| 2011 |
Kister J, Nuhant P, Lira R, Sorg A, Roush WR. Enantio- and diastereoselective synthesis of (E)-1,5-syn-diols: application to the synthesis of the C(23)-C(40) fragment of tetrafibricin. Organic Letters. 13: 1868-71. PMID 21375316 DOI: 10.1021/Ol2003836 |
0.833 |
|
| 2011 |
Stewart PS, Chen M, Roush WR, Ess DH. Thermodynamic control of 1,3-boratropic shifts of α- and γ-stannyl-substituted allylboranes: hyperconjugation outweighs steric effects. Organic Letters. 13: 1478-81. PMID 21323387 DOI: 10.1021/Ol2001599 |
0.415 |
|
| 2011 |
Kumar N, Kojetin DJ, Solt LA, Kumar KG, Nuhant P, Duckett DR, Cameron MD, Butler AA, Roush WR, Griffin PR, Burris TP. Identification of SR3335 (ML-176): a synthetic RORα selective inverse agonist. Acs Chemical Biology. 6: 218-22. PMID 21090593 DOI: 10.1021/Cb1002762 |
0.693 |
|
| 2011 |
Chen M, Roush WR. ChemInform Abstract: Enantioselective Syntheses of syn- and anti-β-Hydroxyallylsilanes via Allene Hydroboration-Aldehyde Allylboration Reactions. Cheminform. 42: no-no. DOI: 10.1002/chin.201130185 |
0.309 |
|
| 2011 |
Kister J, Nuhant P, Lira R, Sorg A, Roush WR. ChemInform Abstract: Enantio- and Diastereoselective Synthesis of (E)-1,5-syn-Diols: Application to the Synthesis of the C(23)-C(40) Fragment of Tetrafibricin. Cheminform. 42: no-no. DOI: 10.1002/chin.201127068 |
0.813 |
|
| 2011 |
Ho T, Fieser M, Danheiser R, Roush W, Smith J, Fieser L. Phase‐transfer catalysts Fieser and Fieser's Reagents For Organic Synthesis. 452-452. DOI: 10.1002/9780471264194.Fos07867.Pub4 |
0.469 |
|
| 2011 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Mercury(II) Trifluoroacetate Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos06777.Pub3 |
0.391 |
|
| 2011 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Mercury(II) Acetate Fieser and Fieser's Reagents For Organic Synthesis. 369-369. DOI: 10.1002/9780471264194.Fos06741.Pub2 |
0.409 |
|
| 2011 |
Ho T, Fieser M, Danheiser R, Roush W, Fieser L. Lithium Naphthalenide, LN Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos06537.Pub3 |
0.449 |
|
| 2011 |
Ho T, Fieser M, Danheiser R, Roush W, Fieser L. Cerium(III) Chloride Fieser and Fieser's Reagents For Organic Synthesis. 119-120. DOI: 10.1002/9780471264194.Fos02299.Pub3 |
0.463 |
|
| 2011 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. 9-Borabicyclo[3.3.1]nonane Fieser and Fieser's Reagents For Organic Synthesis. 98-98. DOI: 10.1002/9780471264194.Fos01498.Pub3 |
0.485 |
|
| 2010 |
Chen YT, Brinen LS, Kerr ID, Hansell E, Doyle PS, McKerrow JH, Roush WR. In vitro and in vivo studies of the trypanocidal properties of WRR-483 against Trypanosoma cruzi. Plos Neglected Tropical Diseases. 4. PMID 20856868 DOI: 10.1371/Journal.Pntd.0000825 |
0.478 |
|
| 2010 |
Winbush SM, Roush WR. Enantioselective synthesis of (Z)-1,2-anti-2,5-anti-triol monosilyl ethers using a cross-metathesis allylboration sequence. Organic Letters. 12: 4344-7. PMID 20806914 DOI: 10.1021/Ol101789G |
0.382 |
|
| 2010 |
Wang Y, Kumar N, Nuhant P, Cameron MD, Istrate MA, Roush WR, Griffin PR, Burris TP. Identification of SR1078, a synthetic agonist for the orphan nuclear receptors RORα and RORγ. Acs Chemical Biology. 5: 1029-34. PMID 20735016 DOI: 10.1021/Cb100223D |
0.686 |
|
| 2010 |
Gianni D, Taulet N, Zhang H, DerMardirossian C, Kister J, Martinez L, Roush WR, Brown SJ, Bokoch GM, Rosen H. A novel and specific NADPH oxidase-1 (Nox1) small-molecule inhibitor blocks the formation of functional invadopodia in human colon cancer cells. Acs Chemical Biology. 5: 981-93. PMID 20715845 DOI: 10.1021/Cb100219N |
0.53 |
|
| 2010 |
Chen M, Ess DH, Roush WR. Enantioselective synthesis of (E)-delta-stannyl homoallylic alcohols via aldehyde allylboration using alpha-stannylallylboranes generated by allene hydroboration followed by a highly diastereoselective 1,3-boratropic shift. Journal of the American Chemical Society. 132: 7881-3. PMID 20496899 DOI: 10.1021/Ja103041U |
0.481 |
|
| 2010 |
Chen M, Roush WR. Highly (E)-selective BF(3).Et(2)O-promoted allylboration of chiral nonracemic alpha-substituted allylboronates and analysis of the origin of stereocontrol. Organic Letters. 12: 2706-9. PMID 20476769 DOI: 10.1021/Ol1007444 |
0.403 |
|
| 2010 |
Barth R, Roush WR. Enantioselective synthesis of alpha-methylene-beta-hydroxy carboxylic acid derivatives via a diastereoselective aldol/beta-elimination sequence: application to the C(15)-C(21) fragment of tedanolide C. Organic Letters. 12: 2342-5. PMID 20405855 DOI: 10.1021/Ol1006955 |
0.636 |
|
| 2010 |
He C, Nora GP, Schneider EL, Kerr ID, Hansell E, Hirata K, Gonzalez D, Sajid M, Boyd SE, Hruz P, Cobo ER, Le C, Liu WT, Eckmann L, Dorrestein PC, ... ... Roush WR, et al. A novel Entamoeba histolytica cysteine proteinase, EhCP4, is key for invasive amebiasis and a therapeutic target. The Journal of Biological Chemistry. 285: 18516-27. PMID 20378535 DOI: 10.1074/Jbc.M109.086181 |
0.731 |
|
| 2010 |
Barth R, Roush WR. ChemInform Abstract: Enantioselective Synthesis of α-Methylene-β-hydroxy Carboxylic Acid Derivatives via a Diastereoselective Aldol/β-Elimination Sequence: Application to the C(15)-C(21) Fragment of Tedanolide C. Cheminform. 41: no-no. DOI: 10.1002/chin.201038213 |
0.588 |
|
| 2010 |
Chen M, Handa M, Roush WR. ChemInform Abstract: Enantioselective Synthesis of 2-Methyl-1,2-syn- and 2-Methyl-1,2-anti-3-butenediols via Allene Hydroboration-Aldehyde Allylboration Reaction Sequences. Cheminform. 41. DOI: 10.1002/chin.201008052 |
0.585 |
|
| 2010 |
Kister J, DeBaillie AC, Lira R, Roush WR. ChemInform Abstract: Stereoselective Synthesis of γ-Substituted (Z)-Allylic Boranes via Kinetically Controlled Hydroboration of Allenes with 10-TMS-9-Borabicyclo[3.3.2]decane. Cheminform. 41. DOI: 10.1002/chin.201008040 |
0.614 |
|
| 2010 |
Frank SA, Roush WR. ChemInform Abstract: Studies on the Synthesis of (-)-Spinosyn A: Application of the Steric Directing Group Strategy to Transannular Diels-Alder Reactions. Cheminform. 33: no-no. DOI: 10.1002/chin.200247200 |
0.622 |
|
| 2010 |
Frank SA, Mergott DJ, Roush WR. ChemInform Abstract: The Vinylogous Intramolecular Morita-Baylis-Hillman Reaction: Synthesis of Functionalized Cyclopentenes and Cyclohexenes with Trialkylphosphines as Nucleophilic Catalysts. Cheminform. 33: no-no. DOI: 10.1002/chin.200232041 |
0.825 |
|
| 2010 |
Roush WR, Madar DJ, Coffey DS. ChemInform Abstract: Synthesis of Highly Functionalized Naphthoate Precursors to Damavaricin D - Observation of Kinetically Stable Benzocyclohexadienones in the Bromination Reactions of Highly Functionalized β-Naphthol Derivatives. Cheminform. 33: no-no. DOI: 10.1002/chin.200226213 |
0.314 |
|
| 2010 |
Micalizio GC, Roush WR. ChemInform Abstract: Studies on the Synthesis of Pectenotoxin II: Synthesis of a C(11)-C(26) Fragment Precursor (VI) via [3 + 2]-Annulation Reactions of Chiral Allylsilanes. Cheminform. 32: no-no. DOI: 10.1002/chin.200150222 |
0.69 |
|
| 2010 |
Roush WR, Dilley GJ. ChemInform Abstract: Studies on the Synthesis of 2,6-Disubstituted Dihydropyrans: Intervention of Oxonia-Cope Rearrangements in the Lewis Acid Mediated Cyclodehydrative Reactions of Aldehydes and β-Hydroxyallylsilanes. Cheminform. 32: no-no. DOI: 10.1002/chin.200141159 |
0.772 |
|
| 2010 |
Yakelis NA, Roush WR. ChemInform Abstract: Lewis Acid Catalyzed Intramolecular Diels-Alder Reactions of Acyclic (Z)-Substituted 1,3-Dienes. Cheminform. 32: no-no. DOI: 10.1002/chin.200130041 |
0.809 |
|
| 2010 |
Powell NA, Roush WR. ChemInform Abstract: Studies on the Total Synthesis of Formamicin: Synthesis of the C(1)-C(11) Fragment. Cheminform. 32: no-no. DOI: 10.1002/chin.200121194 |
0.329 |
|
| 2010 |
Frank SA, Chen H, Kunz RK, Schnaderbeck MJ, Roush WR. ChemInform Abstract: Use of Thallium(I) Ethoxide in Suzuki Cross-Coupling Reactions. Cheminform. 31: no-no. DOI: 10.1002/chin.200046042 |
0.548 |
|
| 2010 |
Roush WR, Pfeifer LA. ChemInform Abstract: Total Synthesis of Mycalamide A (IX) and 7-epi-Mycalamide A (V). Cheminform. 31: no-no. DOI: 10.1002/chin.200027232 |
0.762 |
|
| 2010 |
Micalizio GC, Roush WR. ChemInform Abstract: A Three-Component Coupling Strategy for Tetrahydrofuran Synthesis: Application of the Diisopropyl Tartrate, Modified (E)-γ-(Dimethylphenylsilyl)allylboronate as an α,γ-Allyl Dianion Equivalent. Cheminform. 31: no-no. DOI: 10.1002/chin.200021109 |
0.615 |
|
| 2010 |
Roush WR, Narayan S, Bennett CE, Briner K. ChemInform Abstract: Iodoacetoxylation of Glycals Using Cerium(IV) Ammonium Nitrate, Sodium Iodide, and Acetic Acid: Stereoselective Synthesis of 2-Deoxy-2-iodo-α-mannopyranosyl Acetates. Cheminform. 30: no-no. DOI: 10.1002/chin.199948214 |
0.716 |
|
| 2010 |
Roush WR, Narayan S. ChemInform Abstract: 2-Deoxy-2-iodo-α-mannopyranosyl and -talopyranosyl Acetates: Highly Stereoselective Glycosyl Donors for the Synthesis of 2-Deoxy-α-glycosides. Cheminform. 30: no-no. DOI: 10.1002/chin.199947218 |
0.544 |
|
| 2010 |
Roush WR, Gung BW, Bennett CE. ChemInform Abstract: 2-Deoxy-2-iodo- and 2-Deoxy-2-bromo-α-glucopyranosyl Trichloroacetimidates: Highly Reactive and Stereoselective Donors for the Synthesis of 2-Deoxy-β-glycosides. Cheminform. 30: no-no. DOI: 10.1002/chin.199947217 |
0.591 |
|
| 2010 |
Roush WR, Lane GC. ChemInform Abstract: Synthesis of Tedanolide: Synthesis of the C5-C21 Segment via a Highly Stereoselective Fragment Assembly Aldol Reaction of a Chiral β,γ-Unsaturated Methyl Ketone. Cheminform. 30: no-no. DOI: 10.1002/chin.199941265 |
0.81 |
|
| 2010 |
Roush WR, Dilley GJ. ChemInform Abstract: Studies of Fragment Assembly Aldol Reactions of Chiral Aldehydes and Chiral Methyl Ketones: Stereoselective Synthesis of the C(13)-C(25) Segment of Scytophycin C. Cheminform. 30: no-no. DOI: 10.1002/chin.199935262 |
0.792 |
|
| 2010 |
Scheidt KA, Tasaka A, Bannister TD, Wendt MD, Roush WR. ChemInform Abstract: Total Synthesis of (-)-Bafilomycin A1 (I): Application of Diastereoselective Crotylboration and Methyl Ketone Aldol Reactions. Cheminform. 30: no-no. DOI: 10.1002/chin.199934259 |
0.592 |
|
| 2010 |
Roush WR, Bennett CE. ChemInform Abstract: A Highly Stereoselective Synthesis of 2-Deoxy-β-glycosides Using 2-Deoxy-2-iodo-glucopyranosyl Acetate Donors. Cheminform. 30: no-no. DOI: 10.1002/chin.199934229 |
0.604 |
|
| 2010 |
Chemler SR, Roush WR. ChemInform Abstract: Stereochemically Divergent Pathways for the Allylation and Crotylation Reactions of anti- and syn-β-Hydroxy-α-methyl Aldehydes with Allyl- and Crotyltrifluorosilanes. Cheminform. 30: no-no. DOI: 10.1002/chin.199934040 |
0.646 |
|
| 2010 |
Roush WR, Hartz RA, Gustin DJ. ChemInform Abstract: Total Synthesis of Olivomycin A. Cheminform. 30: no-no. DOI: 10.1002/chin.199925222 |
0.334 |
|
| 2010 |
Chemler SR, Coffey DS, Roush WR. ChemInform Abstract: An Improved Synthesis of the (E,Z)-Dienoate Precursor of (+)-Damavaricin D via a Vinylogous Horner-Wadsworth-Emmons Reaction. Cheminform. 30: no-no. DOI: 10.1002/chin.199919259 |
0.669 |
|
| 2010 |
ROUSH WR, GWALTNEY SLI, CHENG J, SCHEIDT KA, MCKERROW JH, HANSELL E. ChemInform Abstract: Vinyl Sulfonate Esters and Vinyl Sulfonamides: Potent, Irreversible Inhibitors of Cysteine Proteases. Cheminform. 30: no-no. DOI: 10.1002/chin.199909224 |
0.515 |
|
| 2010 |
SCHEIDT KA, CHEN H, FOLLOWS BC, CHEMLER SR, COFFEY DS, ROUSH WR. ChemInform Abstract: Tris(dimethylamino)sulfonium Difluorotrimethylsilicate, a Mild Reagent for the Removal of Silicon Protecting Groups. Cheminform. 30: no-no. DOI: 10.1002/chin.199907076 |
0.674 |
|
| 2010 |
ROUSH WR, SCIOTTI RJ. ChemInform Abstract: Enantioselective Total Synthesis of (-)-Chlorothricolide via the Tandem Inter- and Intramolecular Diels-Alder Reaction of a Hexaenoate Intermediate. Cheminform. 29: no-no. DOI: 10.1002/chin.199849291 |
0.416 |
|
| 2010 |
CHEMLER SR, ROUSH WR. ChemInform Abstract: Concerning the Syntheses of the Elusive anti,anti-Dipropionate Stereotriad via the Crotylation of β-Hydroxy α-Methyl Aldehydes with (Z)-Crotyltrifluorosilane. Application to the Synthesis of the C7-C16 Segment of Zincophorin. Cheminform. 29: no-no. DOI: 10.1002/chin.199845046 |
0.646 |
|
| 2010 |
ROUSH WR, PFEIFER LA. ChemInform Abstract: Stereoselective N-Acylation Reactions of α-Alkoxy Carbamates. Cheminform. 29: no-no. DOI: 10.1002/chin.199832087 |
0.77 |
|
| 2010 |
ROUSH WR, PFEIFER LA, MARRON TG. ChemInform Abstract: Studies on the Synthesis of the Mycalamides: Stereocontrolled Synthesis of a Model N-Glycosylpederamide (VIII) via a Stereoselective Aldol Reaction. Cheminform. 29: no-no. DOI: 10.1002/chin.199831268 |
0.805 |
|
| 2010 |
ROUSH WR, REILLY ML, KOYAMA K, BROWN BB. ChemInform Abstract: A Formal Total Synthesis of (+)-Tetronolide, the Aglycon of the Tetrocarcins: Enantio- and Diastereoselective Syntheses of the Octahydronaphthalene (Bottom-Half) and Spirotetronate (Top-Half) Fragments. Cheminform. 29: no-no. DOI: 10.1002/chin.199819249 |
0.338 |
|
| 2010 |
ROUSH WR, BARDA DA. ChemInform Abstract: Highly Selective Lewis Acid Catalyzed Diels-Alder Reactions of Acyclic (Z)-1,3-Dienes. Cheminform. 28: no-no. DOI: 10.1002/chin.199748038 |
0.326 |
|
| 2010 |
ROUSH WR, SEBESTA DP, BENNETT CE. ChemInform Abstract: Stereoselective Synthesis of 2-Deoxy-β-glycosides from Glycal Precursors. Part 1. Stereochemistry of the Reactions of D-Glucal Derivatives with Phenylsulfenyl Chloride and Phenylselenenyl Chloride. Cheminform. 28: no-no. DOI: 10.1002/chin.199744233 |
0.65 |
|
| 2010 |
ROUSH WR, SEBESTA DP, JAMES RA. ChemInform Abstract: Stereoselective Synthesis of 2-Deoxy-β-glycosides from Glycal Precursors. Part 2. Stereochemistry of Glycosidation Reactions of 2- Thiophenyl- and 2-Selenophenyl-α-D-gluco-pyranosyl Donors. Cheminform. 28: no-no. DOI: 10.1002/chin.199743240 |
0.301 |
|
| 2010 |
HUNT JA, ROUSH WR. ChemInform Abstract: 4,5-Diisopropyl-B-((E)-((3′-menthofuryl)dimethylsilyl)allyl)-1,3,2- dioxaborolane, an Improved Chiral Reagent for the anti-α- Hydroxyallylation of Aldehydes: Application to the Enantioselective Synthesis of (-)-Swainsonine. Cheminform. 28: no-no. DOI: 10.1002/chin.199727035 |
0.307 |
|
| 2010 |
ROUSH WR, MARRON TG, PFEIFER LA. ChemInform Abstract: Highly Diastereoselective Synthesis of Pederic Acid Derivatives. Cheminform. 28: no-no. DOI: 10.1002/chin.199723273 |
0.781 |
|
| 2010 |
ROUSH WR, KOYAMA K, CURTIN ML, MORIARTY KJ. ChemInform Abstract: Studies on the Synthesis of Nargenicin A1: Highly Stereoselective Synthesis of the Complete Carbon Framework via the Transannular Diels- Alder Reaction of an 18-Membered Macrolide. Cheminform. 27: no-no. DOI: 10.1002/chin.199651203 |
0.351 |
|
| 2010 |
GUSTIN DJ, VANNIEUWENHZE MS, ROUSH WR. ChemInform Abstract: Diastereoselective Aldol Reactions of Chiral Aldehydes and Chiral Methyl Ketones: Dependence of Stereoselectivity on the Metal Enolate, the Aldehyde 2,3-Stereochemistry, and the Aldehyde β-Alkoxy Protecting Group. Cheminform. 26: no-no. DOI: 10.1002/chin.199536035 |
0.325 |
|
| 2010 |
ROUSH WR, LIN X. ChemInform Abstract: Synthesis of Aureolic Acid Antibiotics: Highly Stereoselective Synthesis of Aryl 2-Deoxy-β-glycosides via the Mitsunobu Reaction and Synthesis of the Olivomycin A-B Disaccharide. Cheminform. 26: no-no. DOI: 10.1002/chin.199529313 |
0.4 |
|
| 2010 |
ROUSH WR, SCIOTTI RJ. ChemInform Abstract: Enantioselective Total Synthesis of (-)-Chlorothricolide (XIV). Cheminform. 25: no-no. DOI: 10.1002/chin.199451288 |
0.36 |
|
| 2010 |
ROUSH WR, FOLLOWS BC. ChemInform Abstract: Asymmetric Synthesis of the Hydroxylamino Sugar of Calicheamicin. Cheminform. 25: no-no. DOI: 10.1002/chin.199447045 |
0.359 |
|
| 2010 |
ROUSH WR, BANNISTER TD, WENDT MD. ChemInform Abstract: Concerning the Diastereofacial Selectivity of Aldol Reactions of Chiral Methyl Ketone Enolates: Evidence for Remote Chelation in the Bafilomycin Aldol Reaction. Cheminform. 25: no-no. DOI: 10.1002/chin.199416043 |
0.343 |
|
| 2010 |
ROUSH WR, MARRON TG. ChemInform Abstract: Toward the Synthesis of Mycalamides A, B, and Onnamide A: A Highly Stereoselective Synthesis of the Trioxadecalin Ring System. Cheminform. 25: no-no. DOI: 10.1002/chin.199407078 |
0.325 |
|
| 2010 |
ROUSH WR, BROWN BB. ChemInform Abstract: A Highly Diastereo- and Enantioselective Synthesis of the Top Half of Kijanolide. Cheminform. 24: no-no. DOI: 10.1002/chin.199334291 |
0.375 |
|
| 2010 |
ROUSH WR, BROWN BB. ChemInform Abstract: Studies on the Synthesis of Kijanolide: Synthesis of the 2-Acyl Spiro Tetronate and Investigations Concerning the Coupling of the Tope and Bottom Half Fragments. Cheminform. 24: no-no. DOI: 10.1002/chin.199334290 |
0.325 |
|
| 2010 |
ROUSH WR, MURPHY M. ChemInform Abstract: An Improved Synthesis of Naphthoate Precursors to Olivin. Cheminform. 24: no-no. DOI: 10.1002/chin.199314149 |
0.303 |
|
| 2010 |
ROUSH WR, BROWN BB. ChemInform Abstract: Enantioselective Synthesis of 2-Alkyl-5-methylene-1,3-dioxolan-4-ones and Exo-Selective Diels-Alder Reactions with Cyclopentadiene. Cheminform. 23: no-no. DOI: 10.1002/chin.199245177 |
0.413 |
|
| 2010 |
ROUSH WR, PARK JC. ChemInform Abstract: Asymmetric Allylborations of 3-Decynaldicobalt Hexacarbonyl: Cobalt- Induced Reversal of Enantioselectivity and Applications to Highly Diastereoselective Intramolecular Pauson-Khand Reactions. Cheminform. 23: no-no. DOI: 10.1002/chin.199226059 |
0.336 |
|
| 2010 |
ROUSH WR, LIN X. ChemInform Abstract: A Highly Stereoselective Synthesis of Aryl 2-Deoxy-β-glycosides via the Mitsunobu Reaction. Cheminform. 23: no-no. DOI: 10.1002/chin.199208299 |
0.368 |
|
| 2010 |
ROUSH WR, MORIARTY KJ, BROWN BB. ChemInform Abstract: Stereoselective Synthesis of Z,E-2-Bromodienes via the Palladium(0)- Catalyzed Cross Coupling Reactions of 1,1-Dibromoolefins and Vinylboronic Acids. Cheminform. 23: no-no. DOI: 10.1002/chin.199207102 |
0.347 |
|
| 2010 |
ROUSH WR, STRAUB JA, VANNIEUWENHZE MS. ChemInform Abstract: A Stereochemically General Synthesis of 2-Deoxyhexoses via the Asymmetric Allylboration of 2,3-Epoxy Aldehydes. Cheminform. 22: no-no. DOI: 10.1002/chin.199128093 |
0.357 |
|
| 2010 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Silver(I) trifluoromethanesulfonate (triflate) Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos08967.Pub3 |
0.436 |
|
| 2010 |
Ho T, Fieser M, Danheiser R, Roush W, Fieser L. 4-Phenyl-1,2,4-triazoline-3,5-dione (PTAD) Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos08190 |
0.467 |
|
| 2009 |
Ess DH, Kister J, Chen M, Roush WR. Origin of thermodynamic versus kinetic control of allene hydroboration with 9-borabicyclo[3.3.1]nonane and 10(R)-trimethylsilyl-9-borabicyclo[3.3.2]decane. Organic Letters. 11: 5538-41. PMID 19899749 DOI: 10.1021/Ol902364D |
0.623 |
|
| 2009 |
Ess DH, Kister J, Chen M, Roush WR. Quantum-mechanical study of 10-R-9-borabicyclo[3.3.2]decane alkene hydroboration. The Journal of Organic Chemistry. 74: 8626-37. PMID 19824624 DOI: 10.1021/Jo901737D |
0.575 |
|
| 2009 |
Chen M, Handa M, Roush WR. Enantioselective synthesis of 2-methyl-1,2-syn- and 2-methyl-1,2-anti-3-butenediols via allene hydroboration-aldehyde allylboration reaction sequences. Journal of the American Chemical Society. 131: 14602-3. PMID 19778012 DOI: 10.1021/Ja904599H |
0.661 |
|
| 2009 |
Kister J, DeBaillie AC, Lira R, Roush WR. Stereoselective synthesis of gamma-substituted (Z)-allylic boranes via kinetically controlled hydroboration of allenes with 10-TMS-9-borabicyclo[3.3.2]decane. Journal of the American Chemical Society. 131: 14174-5. PMID 19775159 DOI: 10.1021/Ja905494C |
0.637 |
|
| 2009 |
Dossey AT, Gottardo M, Whitaker JM, Roush WR, Edison AS. Alkyldimethylpyrazines in the defensive spray of Phyllium westwoodii: a first for order Phasmatodea. Journal of Chemical Ecology. 35: 861-70. PMID 19685263 DOI: 10.1007/S10886-009-9666-9 |
0.521 |
|
| 2009 |
Li F, Roush WR. Stereoselective synthesis of syn,syn- and syn,anti-1,3,5-triols via intramolecular hydrosilylation of substituted pent-3-en-1,5-diols. Organic Letters. 11: 2932-5. PMID 19507846 DOI: 10.1021/Ol9009877 |
0.583 |
|
| 2009 |
Li F, Roush WR. ChemInform Abstract: Stereoselective Synthesis of syn,syn- and syn,anti-1,3,5-Triols via Intramolecular Hydrosilylation of Substituted Pent-3-ene-1,5-diols. Cheminform. 40. DOI: 10.1002/chin.200946047 |
0.558 |
|
| 2009 |
Tortosa M, Yakelis NA, Roush WR. ChemInform Abstract: Total Synthesis of (+)-Superstolide A. Cheminform. 40. DOI: 10.1002/chin.200915209 |
0.805 |
|
| 2009 |
Halvorsen GT, Roush WR. ChemInform Abstract: Siloxacyclopentenes as Dienophile-Linked Directing Groups in Intramolecular Diels-Alder Reactions. Cheminform. 40. DOI: 10.1002/chin.200915035 |
0.814 |
|
| 2009 |
Bates RH, Chen M, Roush WR. ChemInform Abstract: Applications of Chiral Allylmetallating Agents Toward the Synthesis of Oxygen Heterocycles Cheminform. 40. DOI: 10.1002/chin.200911272 |
0.34 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Tetrabutylammonium Fluoride, TBAF Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos09497.Pub2 |
0.457 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Sodium bis(2‐methoxyethoxy)aluminum hydride (SMEAH, Red‐AlÒ) Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos09016.Pub2 |
0.333 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Potassium t‐amyloxide Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos08377.Pub2 |
0.373 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Phosphoryl chloride (Phosphorus oxychloride) Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos08277.Pub2 |
0.342 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Hydrogen chloride, anhydrous Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos05591.Pub2 |
0.359 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Ethylenebis(triphenylphosphine)platinum(0) Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos05108 |
0.346 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Diisobutylaluminum Hydride (DIBAH, DIBAL) Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos04085.Pub2 |
0.387 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W. Chlorotris(triphenylphosphine)rhodium(I) (Wilkinson's catalyst) Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos02718.Pub2 |
0.441 |
|
| 2009 |
Ho T, Fieser M, Fieser L, Danheiser R, Roush W, Smith J. Chloromethyl methyl ether Fieser and Fieser's Reagents For Organic Synthesis. DOI: 10.1002/9780471264194.Fos02563.Pub2 |
0.323 |
|
| 2009 |
Ho T, Fieser M, Danheiser R, Roush W, Smith J, Fieser L. N,N′‐Carbonyldiimidazole Fieser and Fieser's Reagents For Organic Synthesis. 0-0. DOI: 10.1002/9780471264194.Fos02244.Pub2 |
0.459 |
|
| 2008 |
Dunetz JR, Julian LD, Newcom JS, Roush WR. Total syntheses of (+)-tedanolide and (+)-13-deoxytedanolide. Journal of the American Chemical Society. 130: 16407-16. PMID 18980317 DOI: 10.1021/Ja8063205 |
0.82 |
|
| 2008 |
Tortosa M, Yakelis NA, Roush WR. Total synthesis of (+)-superstolide A. The Journal of Organic Chemistry. 73: 9657-67. PMID 18956845 DOI: 10.1021/Jo801794S |
0.845 |
|
| 2008 |
Halvorsen GT, Roush WR. Siloxacyclopentenes as dienophile-linked directing groups in intramolecular Diels-Alder reactions. Organic Letters. 10: 5313-6. PMID 18954061 DOI: 10.1021/Ol802266S |
0.834 |
|
| 2008 |
Bates RH, Chen M, Roush WR. Applications of chiral allylmetallating agents toward the synthesis of oxygen heterocyles. Current Opinion in Drug Discovery & Development. 11: 778-92. PMID 18946843 |
0.667 |
|
| 2008 |
Pragani R, Roush WR. Studies on the synthesis of durhamycin A: stereoselective synthesis of a model aglycone. Organic Letters. 10: 4613-6. PMID 18808128 DOI: 10.1021/Ol8018727 |
0.395 |
|
| 2008 |
Bates RH, Shotwell JB, Roush WR. Stereoselective syntheses of the C(1)-C(9) fragment of amphidinolide C. Organic Letters. 10: 4343-6. PMID 18783230 DOI: 10.1021/Ol801852J |
0.675 |
|
| 2008 |
Huh CW, Roush WR. Highly stereoselective and modular syntheses of 10-hydroxytrilobacin and three diastereomers via stereodivergent [3 + 2]-annulation reactions. Organic Letters. 10: 3371-4. PMID 18588305 DOI: 10.1021/Ol801242D |
0.448 |
|
| 2008 |
Chen YT, Lira R, Hansell E, McKerrow JH, Roush WR. Synthesis of macrocyclic trypanosomal cysteine protease inhibitors. Bioorganic & Medicinal Chemistry Letters. 18: 5860-3. PMID 18585034 DOI: 10.1016/J.Bmcl.2008.06.012 |
0.533 |
|
| 2008 |
Roush WR. Total synthesis of biologically active natural products. Journal of the American Chemical Society. 130: 6654-6. PMID 18491856 DOI: 10.1021/Ja8028813 |
0.343 |
|
| 2008 |
Dunetz JR, Roush WR. Concerning the synthesis of the tedanolide C(13)-C(23) fragment via anti-aldol reaction. Organic Letters. 10: 2059-62. PMID 18422319 DOI: 10.1021/Ol800546G |
0.817 |
|
| 2008 |
Tortosa M, Yakelis NA, Roush WR. Total synthesis of +-superstolide A. Journal of the American Chemical Society. 130: 2722-3. PMID 18254629 DOI: 10.1021/Ja710238H |
0.85 |
|
| 2008 |
Winbush SM, Mergott DJ, Roush WR. Total synthesis of (-)-spinosyn A: examination of structural features that govern the stereoselectivity of the key transannular Diels-Alder reaction. The Journal of Organic Chemistry. 73: 1818-29. PMID 18215065 DOI: 10.1021/Jo7024515 |
0.806 |
|
| 2008 |
Hicks JD, Roush WR. Synthesis of the C(26)-C(42) and C(43)-C(67) pyran-containing fragments of amphidinol 3 via a common pyran intermediate. Organic Letters. 10: 681-4. PMID 18205377 DOI: 10.1021/Ol703042Q |
0.597 |
|
| 2008 |
Handa M, Smith WJ, Roush WR. Studies on the synthesis of apoptolidin A. 2. Synthesis of the disaccharide unit. The Journal of Organic Chemistry. 73: 1036-9. PMID 18163646 DOI: 10.1021/Jo7022526 |
0.702 |
|
| 2008 |
Handa M, Scheidt KA, Bossart M, Zheng N, Roush WR. Studies on the synthesis of apoptolidin A. 1. Synthesis of the C(1)-C(11) fragment. The Journal of Organic Chemistry. 73: 1031-5. PMID 18163645 DOI: 10.1021/Jo702250Z |
0.771 |
|
| 2008 |
Tortosa M, Yakelis NA, Roush WR. Synthesis of (+)-Superstolide A Synfacts. 2008: 786-786. DOI: 10.1055/S-2008-1078534 |
0.829 |
|
| 2008 |
Winbush SM, Mergott DJ, Roush WR. Synthesis of (-)-Spinosyn A Synfacts. 2008: 785-785. DOI: 10.1055/S-2008-1078533 |
0.453 |
|
| 2008 |
Winbush SM, Mergott DJ, Roush WR. ChemInform Abstract: Total Synthesis of (-)-Spinosyn A (Ib): Examination of Structural Features that Govern the Stereoselectivity of the Key Transannular Diels-Alder Reaction. Cheminform. 39. DOI: 10.1002/chin.200829202 |
0.797 |
|
| 2008 |
Hicks JD, Huh CW, Legg AD, Roush WR. ChemInform Abstract: Concerning the Selective Protection of (Z)-1,5-syn-Ene-diols and (E)-1,5-anti-Ene-diols as Allylic Triethylsilyl Ethers. Cheminform. 39. DOI: 10.1002/chin.200823067 |
0.548 |
|
| 2008 |
Handa M, Scheidt KA, Bossart M, Zheng N, Roush WR. ChemInform Abstract: Studies on the Synthesis of Apoptolidin A (I). Part 1. Synthesis of the C(1)-C(11) Fragment. Cheminform. 39. DOI: 10.1002/chin.200822211 |
0.705 |
|
| 2008 |
Handa M, Smith WJI, Roush WR. ChemInform Abstract: Studies on the Synthesis of Apoptolidin A. Part 2. Synthesis of the Disaccaride Unit. Cheminform. 39. DOI: 10.1002/chin.200819223 |
0.597 |
|
| 2007 |
Va P, Roush WR. Total Synthesis of Amphidinolide E and Amphidinolide E Stereoisomers. Tetrahedron. 63: 5768-5796. PMID 18575572 DOI: 10.1016/J.Tet.2007.02.058 |
0.406 |
|
| 2007 |
Hicks JD, Huh CW, Legg AD, Roush WR. Concerning the selective protection of (Z)-1,5-syn-ene-diols and (E)-1,5-anti-ene-diols as allylic triethylsilyl ethers. Organic Letters. 9: 5621-4. PMID 18027963 DOI: 10.1021/Ol702588H |
0.585 |
|
| 2007 |
Lira R, Roush WR. Enantio- and diastereoselective synthesis of syn-beta-hydroxyallylsilanes via a chiral (Z)-gamma-silylallylboronate. Organic Letters. 9: 4315-8. PMID 17867698 DOI: 10.1021/Ol7018746 |
0.389 |
|
| 2007 |
Goetz DH, Choe Y, Hansell E, Chen YT, McDowell M, Jonsson CB, Roush WR, McKerrow J, Craik CS. Substrate specificity profiling and identification of a new class of inhibitor for the major protease of the SARS coronavirus. Biochemistry. 46: 8744-52. PMID 17605471 DOI: 10.1021/Bi0621415 |
0.494 |
|
| 2007 |
Halvorsen GT, Roush WR. Intramolecular diels-alder reactions of siloxacyclopentene constrained trienes Organic Letters. 9: 2243-2246. PMID 17480094 DOI: 10.1021/Ol070858U |
0.829 |
|
| 2007 |
Lira R, Roush WR. Stereoselective synthesis of the C(1)-C(19) fragment of tetrafibricin Organic Letters. 9: 533-536. PMID 17249805 DOI: 10.1021/Ol0629869 |
0.457 |
|
| 2007 |
Va P, Roush WR. Synthesis of 2-epi-amphidinolide E: An unexpected and highly selective C(2) inversion during an esterification reaction Organic Letters. 9: 307-310. PMID 17217291 DOI: 10.1021/Ol0628098 |
0.468 |
|
| 2006 |
Va P, Roush WR. Total synthesis of amphidinolide E. Journal of the American Chemical Society. 128: 15960-1. PMID 17165709 DOI: 10.1021/ja066663j |
0.394 |
|
| 2006 |
Trullinger TK, Qi J, Roush WR. Studies on the synthesis of quartromicins a(3) and d(3): synthesis of the vertical and horizontal bis-spirotetronate fragments. The Journal of Organic Chemistry. 71: 6915-22. PMID 16930045 DOI: 10.1021/Jo061059C |
0.558 |
|
| 2006 |
Qi J, Roush WR. Synthesis of precursors of the agalacto (exo) fragment of the quartromicins via an auxiliary-controlled exo-selective Diels-Alder reaction. Organic Letters. 8: 2795-8. PMID 16774259 DOI: 10.1021/Ol0609208 |
0.609 |
|
| 2005 |
Flamme EM, Roush WR. Synthesis of 2,6-trans-disubstituted 5,6-dihydropyrans from (Z)-1,5-syn-endiols. Beilstein Journal of Organic Chemistry. 1: 7. PMID 16542020 DOI: 10.1186/1860-5397-1-7 |
0.813 |
|
| 2005 |
Dias LC, Aguilar AM, Salles AG, Steil LJ, Roush WR. Concerning the application of the1H NMR ABX analysis for assignment of stereochemistry to aldols deriving from aldehydes lacking β-branches Journal of Organic Chemistry. 70: 10461-10465. PMID 16323858 DOI: 10.1021/Jo051773E |
0.362 |
|
| 2005 |
Thalji RK, Roush WR. Remarkable phosphine-effect on the intramolecular aldol reactions of unsaturated 1,5-diketones: highly regioselective synthesis of cross-conjugated dienones. Journal of the American Chemical Society. 127: 16778-9. PMID 16316211 DOI: 10.1021/Ja054085L |
0.806 |
|
| 2005 |
Hicks JD, Flamme EM, Roush WR. Synthesis of the C(43)-C(67) fragment of amphidinol 3. Organic Letters. 7: 5509-12. PMID 16288543 DOI: 10.1021/Ol052322J |
0.838 |
|
| 2005 |
Lambert WT, Roush WR. Synthesis of the A-B subunit of angelmicin B. Organic Letters. 7: 5501-4. PMID 16288541 DOI: 10.1021/Ol052321R |
0.685 |
|
| 2005 |
Mertz E, Tinsley JM, Roush WR. [3 + 2]-annulation reactions of chiral allylsilanes and chiral aldehydes. studies on the synthesis of bis-tetrahydrofuran substructures of annonaceous acetogenins. The Journal of Organic Chemistry. 70: 8035-46. PMID 16277325 DOI: 10.1021/Jo0511290 |
0.738 |
|
| 2005 |
Tinsley JM, Mertz E, Chong PY, Rarig RA, Roush WR. Synthesis of (+)-bullatacin via the highly diastereoselective [3+2] annulation reaction of a racemic aldehyde and a nonracemic allylsilane. Organic Letters. 7: 4245-8. PMID 16146398 DOI: 10.1021/Ol051719K |
0.758 |
|
| 2005 |
Owen RM, Roush WR. Stereoselective synthesis of the C(1)-C(11) fragment of peloruside A. Organic Letters. 7: 3941-4. PMID 16119937 DOI: 10.1021/Ol0514303 |
0.423 |
|
| 2005 |
Tinsley JM, Roush WR. Total synthesis of asimicin via highly stereoselective [3 + 2] annulation reactions of substituted allylsilanes. Journal of the American Chemical Society. 127: 10818-9. PMID 16076173 DOI: 10.1021/Ja051986L |
0.757 |
|
| 2005 |
Heitzman CL, Lambert WT, Mertz E, Shotwell JB, Tinsley JM, Va P, Roush WR. Efficient protiodesilylation of unactivated C(sp3)-SiMe2Ph bonds using tetrabutylammonium fluoride. Organic Letters. 7: 2405-8. PMID 15932209 DOI: 10.1021/Ol0506821 |
0.787 |
|
| 2005 |
Julian LD, Newcom JS, Roush WR. Total synthesis of (+)-13-deoxytedanolide. Journal of the American Chemical Society. 127: 6186-7. PMID 15853320 DOI: 10.1021/Ja050729D |
0.838 |
|
| 2005 |
Liu CM, Smith WJ, Gustin DJ, Roush WR. Experimental evidence for chair-like transition states in aldol reactions of methyl ketone lithium enolates: stereoselective synthesis and utilization of a deuterium-labeled enolate as a probe of reaction stereochemistry. Journal of the American Chemical Society. 127: 5770-1. PMID 15839658 DOI: 10.1021/Ja050730C |
0.697 |
|
| 2005 |
Flamme EM, Roush WR. Synthesis of the C(1)-C(25) fragment of amphidinol 3: application of the double-allylboration reaction for synthesis of 1,5-diols. Organic Letters. 7: 1411-4. PMID 15787519 DOI: 10.1021/Ol050250Q |
0.837 |
|
| 2005 |
Dineen TA, Roush WR. Stereoselective synthesis of the octahydronaphthalene unit of integramycin via an intramolecular Diels-Alder reaction. Organic Letters. 7: 1355-8. PMID 15787505 DOI: 10.1021/Ol050191G |
0.807 |
|
| 2005 |
Narayan S, Roush WR. Studies Toward the Total Synthesis of Angelmicin B (Hibarimicin B) (II): Synthesis of a Model CD?D? Arylnaphthoquinone (I). Cheminform. 36. DOI: 10.1002/chin.200507215 |
0.513 |
|
| 2004 |
Shotwell JB, Roush WR. Synthesis of the C11-C29 fragment of amphidinolide F. Organic Letters. 6: 3865-8. PMID 15469369 DOI: 10.1021/ol048381z |
0.346 |
|
| 2004 |
Narayan S, Roush WR. Studies toward the total synthesis of angelmicin B (hibarimicin B): synthesis of a model CD-D' arylnaphthoquinone. Organic Letters. 6: 3789-92. PMID 15469350 DOI: 10.1021/Ol048436X |
0.569 |
|
| 2004 |
Durham TB, Blanchard N, Savall BM, Powell NA, Roush WR. Total synthesis of formamicin. Journal of the American Chemical Society. 126: 9307-17. PMID 15281821 DOI: 10.1021/Ja048493L |
0.838 |
|
| 2004 |
Roush WR, Neitz RJ. Studies on the synthesis of landomycin A. Synthesis of the originally assigned structure of the aglycone, landomycinone, and revision of structure. The Journal of Organic Chemistry. 69: 4906-12. PMID 15255715 DOI: 10.1021/Jo049426C |
0.778 |
|
| 2004 |
Dineen TA, Roush WR. Total synthesis of cochleamycin A. Organic Letters. 6: 2043-6. PMID 15176814 DOI: 10.1021/Ol049331X |
0.82 |
|
| 2004 |
Mergott DJ, Frank SA, Roush WR. Total synthesis of (-)-spinosyn A. Proceedings of the National Academy of Sciences of the United States of America. 101: 11955-9. PMID 15173590 DOI: 10.1073/Pnas.0401247101 |
0.845 |
|
| 2004 |
Methot JL, Roush WR. Nucleophilic phosphine organocatalysis Advanced Synthesis and Catalysis. 346: 1035-1050. DOI: 10.1002/Adsc.200404087 |
0.442 |
|
| 2004 |
Roush WR. Recent studies in carbonyl allylation reactions: Application to the synthesis of oxygen heterocycles Actualite Chimique. 21-22. |
0.32 |
|
| 2003 |
Dineen TA, Roush WR. Probing the Lewis acid-catalyzed intramolecular Diels-Alder cyclizations of allylic alkoxy-substituted (Z)-1,3-dienes. Organic Letters. 5: 4725-8. PMID 14627425 DOI: 10.1021/Ol035900+ |
0.79 |
|
| 2003 |
Methot JL, Roush WR. Synthetic studies toward FR182877. Remarkable solvent effect in the vinylogous morita-baylis-hillman cyclization. Organic Letters. 5: 4223-6. PMID 14572290 DOI: 10.1021/Ol0357550 |
0.414 |
|
| 2003 |
Boitano A, Emal CD, Leonetti F, Blatt NB, Dineen TA, Ellman JA, Roush WR, Opipari AW, Glick GD. Structure activity studies of a novel cytotoxic benzodiazepine. Bioorganic & Medicinal Chemistry Letters. 13: 3327-30. PMID 12951119 DOI: 10.1016/S0960-894X(03)00683-8 |
0.763 |
|
| 2003 |
Reddick JJ, Cheng J, Roush WR. Relative rates of Michael reactions of 2'-(phenethyl)thiol with vinyl sulfones, vinyl sulfonate esters, and vinyl sulfonamides relevant to vinyl sulfonyl cysteine protease inhibitors. Organic Letters. 5: 1967-70. PMID 12762698 DOI: 10.1021/Ol034555L |
0.395 |
|
| 2003 |
Durham TB, Roush WR. Stereoselective synthesis of functionalized precursors of the CDEF and CDE 2,6-dideoxy-tetra- and trisaccharide units of durhamycins A and B. Organic Letters. 5: 1875-8. PMID 12762675 DOI: 10.1021/Ol034395D |
0.721 |
|
| 2003 |
Durham TB, Roush WR. Stereoselective synthesis of 2-deoxy-beta-galactosides via 2-deoxy-2-bromo- and 2-deoxy-2-iodo-galactopyranosyl donors. Organic Letters. 5: 1871-4. PMID 12762674 DOI: 10.1021/Ol034393T |
0.735 |
|
| 2003 |
Yakelis NA, Roush WR. Synthesis of the C(21)-C(26) fragment of superstolide A: concerning the stereochemistry of (E)-crotylboration reactions of alaninal derivatives. The Journal of Organic Chemistry. 68: 3838-43. PMID 12737561 DOI: 10.1021/Jo0341012 |
0.817 |
|
| 2003 |
Heo JN, Holson EB, Roush WR. Common-intermediate strategy for synthesis of conduritols and inositols via beta-hydroxy cyclohexenylsilanes. Organic Letters. 5: 1697-700. PMID 12735755 DOI: 10.1021/Ol034349D |
0.738 |
|
| 2003 |
Heo JN, Micalizio GC, Roush WR. Enantio- and diastereoselective synthesis of cyclic beta-hydroxy allylsilanes via sequential aldehyde gamma-silylallylboration and ring-closing metathesis reactions. Organic Letters. 5: 1693-6. PMID 12735754 DOI: 10.1021/Ol034347T |
0.681 |
|
| 2003 |
Chemler SR, Roush WR. Stereochemistry of the allylation and crotylation reactions of alpha-methyl-beta-hydroxy aldehydes with allyl- and crotyltrifluorosilanes. Synthesis of anti,anti-dipropionate stereotriads and stereodivergent pathways for the reactions with 2,3-anti- and 2,3-syn-alpha-methyl-beta-hydroxy aldehydes. The Journal of Organic Chemistry. 68: 1319-33. PMID 12585871 DOI: 10.1021/Jo0267908 |
0.665 |
|
| 2003 |
Savall BM, Blanchard N, Roush WR. Total synthesis of the formamicin aglycon, formamicinone. Organic Letters. 5: 377-9. PMID 12556196 DOI: 10.1021/Ol027569K |
0.825 |
|
| 2003 |
Blanchard N, Roush WR. 2-Deoxy-2-iodo-beta-glucopyranosyl fluorides: mild and highly stereoselective glycosyl donors for the synthesis of 2-deoxy-beta-glycosides from beta-hydroxy ketones. Organic Letters. 5: 81-4. PMID 12509896 DOI: 10.1021/Ol027257H |
0.546 |
|
| 2003 |
Shenai BR, Lee BJ, Alvarez-Hernandez A, Chong PY, Emal CD, Neitz RJ, Roush WR, Rosenthal PJ. Structure-activity relationships for inhibition of cysteine protease activity and development of Plasmodium falciparum by peptidyl vinyl sulfones. Antimicrobial Agents and Chemotherapy. 47: 154-60. PMID 12499184 DOI: 10.1128/Aac.47.1.154-160.2003 |
0.779 |
|
| 2003 |
Gung BW, Xue X, Roush WR. The Origin of Diastereofacial Control in Allylboration Reactions Using Tartrate Ester Derived Allylboronates: Attractive Interactions between the Lewis Acids Coordinated Aldehyde Carbonyl Group and an Ester Carbonyl Oxygen [J. Am. Chem. Soc.2002,124, 10692−10697]. Journal of the American Chemical Society. 125: 3668-3668. DOI: 10.1021/Ja025125D |
0.372 |
|
| 2002 |
Roush WR, Newcom JS. Studies on the synthesis of tedanolide. 2. Stereoselective synthesis of a protected C(1)-C(12) fragment. Organic Letters. 4: 4739-42. PMID 12489975 DOI: 10.1021/Ol0272343 |
0.827 |
|
| 2002 |
Chong PY, Roush WR. Concerning the origin of the high beta-selectivity of glycosidation reactions of 2-deoxy-2-iodo-glucopyranosyl trichloroacetimidates. Organic Letters. 4: 4523-6. PMID 12465928 DOI: 10.1021/Ol027066E |
0.376 |
|
| 2002 |
Flamme EM, Roush WR. Enantioselective synthesis of 1,5-anti- and 1,5-syn-diols using a highly diastereoselective one-pot double allylboration reaction sequence. Journal of the American Chemical Society. 124: 13644-5. PMID 12431072 DOI: 10.1021/Ja028055J |
0.836 |
|
| 2002 |
Holson EB, Roush WR. Synthesis of the C(2)-C(13) fragment (the A-B spiroketal unit) of spongistatin 1 (altohyrtin A): use of a common intermediate for the synthesis of both spongistatin spiroketals. Organic Letters. 4: 3723-5. PMID 12375928 DOI: 10.1021/Ol026688X |
0.758 |
|
| 2002 |
Holson EB, Roush WR. Diastereoselective synthesis of the C(17)-C(28) fragment (the C-D spiroketal unit) of spongistatin 1 (altohyrtin A) via a kinetically controlled iodo-spiroketalization reaction. Organic Letters. 4: 3719-22. PMID 12375927 DOI: 10.1021/Ol0266875 |
0.747 |
|
| 2002 |
Gung BW, Xue X, Roush WR. The origin of diastereofacial control in allylboration reactions using tartrate ester derived allylboronates: attractive interactions between the Lewis acid coordinated aldehyde carbonyl group and an ester carbonyl oxygen. Journal of the American Chemical Society. 124: 10692-7. PMID 12207523 DOI: 10.1021/Ja026373C |
0.306 |
|
| 2002 |
Mergott DJ, Frank SA, Roush WR. Application of the intramolecular vinylogous Morita-Baylis-Hillman reaction toward the synthesis of the spinosyn A tricyclic nucleus. Organic Letters. 4: 3157-60. PMID 12201741 DOI: 10.1021/Ol026540D |
0.837 |
|
| 2002 |
Hernandez AA, Roush WR. Recent advances in the synthesis, design and selection of cysteine protease inhibitors. Current Opinion in Chemical Biology. 6: 459-65. PMID 12133721 DOI: 10.1016/S1367-5931(02)00345-9 |
0.322 |
|
| 2002 |
Scheidt KA, Bannister TD, Tasaka A, Wendt MD, Savall BM, Fegley GJ, Roush WR. Total synthesis of (-)-bafilomycin A(1). Journal of the American Chemical Society. 124: 6981-90. PMID 12059221 DOI: 10.1021/Ja017885E |
0.849 |
|
| 2002 |
Frank SA, Roush WR. Studies on the synthesis of (-)-spinosyn a: application of the steric directing group strategy to transannular Diels-Alder reactions. The Journal of Organic Chemistry. 67: 4316-24. PMID 12054969 DOI: 10.1021/Jo025580S |
0.676 |
|
| 2002 |
Roush WR, Bannister TD, Wendt MD, VanNieuwenhze MS, Gustin DJ, Dilley GJ, Lane GC, Scheidt KA, Smith WJ. An NMR method for assigning relative stereochemistry to beta-hydroxy ketones deriving from aldol reactions of methyl ketones. The Journal of Organic Chemistry. 67: 4284-9. PMID 12054964 DOI: 10.1021/Jo0164148 |
0.798 |
|
| 2002 |
Roush WR, Bannister TD, Wendt MD, Jablonowski JA, Scheidt KA. Studies on the synthesis of bafilomycin A(1): stereochemical aspects of the fragment assembly aldol reaction for construction of the C(13)-C25) segment. The Journal of Organic Chemistry. 67: 4275-83. PMID 12054963 DOI: 10.1021/Jo016413F |
0.789 |
|
| 2002 |
Roush WR, Limberakis C, Kunz RK, Barda DA. Diastereoselective synthesis of the endo- and exo-spirotetronate subunits of the quartromicins. The first enantioselective Diels-Alder reaction of an acyclic (Z)-1,3-diene. Organic Letters. 4: 1543-6. PMID 11975624 DOI: 10.1021/Ol025772+ |
0.808 |
|
| 2002 |
Frank SA, Mergott DJ, Roush WR. The vinylogous intramolecular Morita-Baylis-Hillman reaction: synthesis of functionalized cyclopentenes and cyclohexenes with trialkylphosphines as nucleophilic catalysts. Journal of the American Chemical Society. 124: 2404-5. PMID 11890766 DOI: 10.1021/Ja017123J |
0.839 |
|
| 2002 |
Roush WR, Chen H, Reilly ML. Studies on the synthesis of kijanolide: Synthesis of an advanced seco-acid intermediate Heterocycles. 58: 259-282. DOI: 10.3987/Com-02-S(M)17 |
0.492 |
|
| 2002 |
Roush WR, James RA. Towards the synthesis of aureolic acid analogue conjugates: Synthesis and glycosidation reactions of 3-o-acetyl-4-azido-2,4,6-trideoxy-L-glucopyranose derivatives Australian Journal of Chemistry. 55: 141-146. DOI: 10.1071/Ch01199 |
0.462 |
|
| 2002 |
Roush WR, Powell NA, James RA. Synthesis of structurally simplified aureolic acid aglycone-C-D-E trisaccharide analogues Australian Journal of Chemistry. 55: 113-121. DOI: 10.1071/Ch01198 |
0.438 |
|
| 2002 |
Holson EB, Roush WR. Diastereoselective synthesis of the C(17)-C(28) fragment (the C-D spiroketal unit) of spongistatin 1 (altohyrtin A) via a kinetically controlled lodo-spiroketalization reaction Organic Letters. 4: 3719-3722. DOI: 10.1021/ol0266875 |
0.698 |
|
| 2002 |
Roush WR, Limberakis C, Kunz RK, Barda DA. Diastereoselective Synthesis of the endo- and exo-Spirotetronate Subunits of the Quartromicins. The First Enantioselective Diels - Alder Reaction of an Acyclic (Z)-1,3-Diene Organic Letters. 4: 1543-1546. DOI: 10.1021/ol025772+ |
0.794 |
|
| 2002 |
Roush WR, Blizzard TA. Synthesis of verrucarin B Cheminform. 14. DOI: 10.1021/Jo00197A002 |
0.347 |
|
| 2002 |
Roush WR, Hertel L, Schnaderbeck MJ, Yakelis NA. Synthesis of the C(18)-C(26) segment of superstolide A Tetrahedron Letters. 43: 4885-4887. DOI: 10.1016/S0040-4039(02)00903-6 |
0.806 |
|
| 2002 |
Roush WR, Barda DA, Limberakis C, Kunz RK. Studies on the synthesis of the quartromicins: Partial stereochemical assignment of quartromicins A3 and D3 and diastereoselective synthesis of the endo- and exo-spirotetronate subunits Tetrahedron. 58: 6433-6454. DOI: 10.1016/S0040-4020(02)00656-7 |
0.786 |
|
| 2002 |
Johns BA, Grant CM, Marshall JA, Holson EB, Roush WR. Synthesis and utilization of indium (i) iodide for in situ formation of enantioenriched allenylindium reagents and their addition to aldehydes: (2r,3s,4s)-1-(tertbutyldiphenylsilyloxy)-2,4-dimethyl-5-hexyn-3-ol Organic Syntheses. 79: 59-70. DOI: 10.1002/0471264180.Os079.08 |
0.673 |
|
| 2002 |
Abiko A, Flamme EM, Roush WR. Anti-selective boron-mediated asymmetric aldol reaction of carboxylic esters: Synthesis of (2S, 3R)-2,4-dimethyl-1,3-pentanediol Organic Syntheses. 79: 116-123. |
0.821 |
|
| 2002 |
Abiko A, Flamme EM, Roush WR. Dicyclohexylboron trifluoromethanesulfonate Organic Syntheses. 79: 103-107. |
0.782 |
|
| 2001 |
Caffrey CR, Hansell E, Lucas KD, Brinen LS, Alvarez Hernandez A, Cheng J, Gwaltney SL, Roush WR, Stierhof YD, Bogyo M, Steverding D, McKerrow JH. Active site mapping, biochemical properties and subcellular localization of rhodesain, the major cysteine protease of Trypanosoma brucei rhodesiense. Molecular and Biochemical Parasitology. 118: 61-73. PMID 11704274 DOI: 10.1016/S0166-6851(01)00368-1 |
0.763 |
|
| 2001 |
Roush WR, Cheng J, Knapp-Reed B, Alvarez-Hernandez A, McKerrow JH, Hansell E, Engel JC. Potent second generation vinyl sulfonamide inhibitors of the trypanosomal cysteine protease cruzain. Bioorganic & Medicinal Chemistry Letters. 11: 2759-62. PMID 11591518 DOI: 10.1016/S0960-894X(01)00566-2 |
0.77 |
|
| 2001 |
Roush WR, Bennett CE, Roberts SE. Studies on the synthesis of landomycin A: synthesis and glycosidation reactions of L-rhodinosyl acetate derivatives. The Journal of Organic Chemistry. 66: 6389-93. PMID 11559191 DOI: 10.1021/Jo015756A |
0.691 |
|
| 2001 |
Savall BM, Powell NA, Roush WR. Highly diastereoselective synthesis of propargylic 1,2-anti-diol derivatives using alpha-alkoxypropargylstannanes. Organic Letters. 3: 3057-60. PMID 11554842 DOI: 10.1021/Ol016536M |
0.768 |
|
| 2001 |
Powell NA, Roush WR. Studies on the total synthesis of formamicin: synthesis of the C(1)-C(11) fragment. Organic Letters. 3: 453-6. PMID 11428037 DOI: 10.1021/Ol0069610 |
0.437 |
|
| 2001 |
Micalizio GC, Roush WR. Studies on the synthesis of pectenotoxin II: synthesis of a C(11)-C(26) fragment precursor via [3 + 2]-annulation reactions of chiral allylsilanes. Organic Letters. 3: 1949-52. PMID 11405752 DOI: 10.1021/Ol0160250 |
0.729 |
|
| 2001 |
Yakelis NA, Roush WR. Lewis acid catalyzed intramolecular Diels-Alder reactions of acyclic (Z)-substituted 1,3-dienes. Organic Letters. 3: 957-60. PMID 11263925 DOI: 10.1021/Ol015667K |
0.783 |
|
| 2001 |
Roush WR, Madar DJ, Coffey DS. Synthesis of highly functionalized naphthoate precursors to damavaricin D - Observation of kinetically stable benzocyclohexadienones in the bromination reactions of highly functionalized β-naphthol derivatives Canadian Journal of Chemistry. 79: 1711-1726. DOI: 10.1139/V01-135 |
0.513 |
|
| 2001 |
Roush WR, Dilley GJ. Studies on the synthesis of 2,6-disubstituted dihydropyrans: Intervention of oxonia-cope rearrangements in the lewis acid mediated cyclodehydrative reactions of aldehydes and β-hydroxyallylsilanes Synlett. 955-959. DOI: 10.1055/S-2001-14632 |
0.782 |
|
| 2001 |
Micalizio GC, Pinchuk AN, Roush WR. ChemInform Abstract: Synthesis of the C(29)-C(45) Bis-pyran Subunit (E-F) of Spongistatin 1 (Altohyrtin A). Cheminform. 32: no-no. DOI: 10.1002/chin.200115240 |
0.613 |
|
| 2001 |
Roush WR, Pinchuk AN, Micalizio GC. ChemInform Abstract: [(E)-γ-(Dimethylphenylsilyl)allyl]diisopinocampheylborane: A Highly Enantioselective Reagent for the Synthesis of anti-β-Hydroxyallylsilanes. Cheminform. 32: no-no. DOI: 10.1002/chin.200110042 |
0.636 |
|
| 2000 |
Micalizio GC, Pinchuk AN, Roush WR. Synthesis of the C(29)-C(45) bis-pyran subunit (E-F) of spongistatin 1 (Altohyrtin A). The Journal of Organic Chemistry. 65: 8730-6. PMID 11112596 DOI: 10.1021/Jo001236O |
0.706 |
|
| 2000 |
Frank SA, Chen H, Kunz RK, Schnaderbeck MJ, Roush WR. Use of thallium(I) ethoxide in Suzuki cross coupling reactions. Organic Letters. 2: 2691-4. PMID 10990429 DOI: 10.1021/Ol0062446 |
0.804 |
|
| 2000 |
Micalizio GC, Roush WR. A three-component coupling strategy for tetrahydrofuran synthesis: application of the diisopropyl tartrate modified (E)-gamma-(dimethylphenylsilyl)allylboronate as an alpha,gamma-allyl dianion equivalent. Organic Letters. 2: 461-4. PMID 10814351 DOI: 10.1021/Ol9913082 |
0.671 |
|
| 2000 |
Roush WR, Pfeifer LA. Total synthesis of mycalamide A and 7-epi-mycalamide A. Organic Letters. 2: 859-62. PMID 10754688 DOI: 10.1021/ol005629l |
0.773 |
|
| 2000 |
Frank SA, Works AB, Roush WR. Studies on the synthesis of the decahydro-as-indacene ring system of (-)-spinosyn A via transannular Diels-Alder reactions of substituted (E,E,E)-cyclododeca-1,6,8-trienes Canadian Journal of Chemistry. 78: 757-771. DOI: 10.1139/V00-045 |
0.658 |
|
| 2000 |
Roush WR, Bennett CE. A highly stereoselective synthesis of the landomycin a hexasaccharide unit [10] Journal of the American Chemical Society. 122: 6124-6125. DOI: 10.1021/Ja000743K |
0.631 |
|
| 2000 |
Roush WR, Pinchuk AN, Micalizio GC. [(E)-γ-(Dimethylphenylsilyl)allyl]diisopinocampheylborane: A highly enantioselective reagent for the synthesis of anti-β-hydroxyallylsilanes Tetrahedron Letters. 41: 9413-9417. DOI: 10.1016/S0040-4039(00)01526-4 |
0.657 |
|
| 2000 |
Roush WR, Hernandez AA, McKerrow JH, Selzer PM, Hansell E, Engel JC. Design, synthesis and evaluation of D-Homophenylalanyl epoxysuccinate inhibitors of the trypanosomal cysteine protease cruzain Tetrahedron. 56: 9747-9762. DOI: 10.1016/S0040-4020(00)00882-6 |
0.32 |
|
| 2000 |
Micalizio GC, Roush WR. A three-component coupling strategy for tetrahydrofuran synthesis: Application of the diisopropyl tartrate modified (E)-γ-(dimethylphenylsilyl)allylboronate as an α,γ-allyl dianion equivalent Organic Letters. 2: 461-464. |
0.611 |
|
| 1999 |
Scheidt KA, Tasaka A, Bannister TD, Wendt MD, Roush WR. Total Synthesis of (-)-Bafilomycin A : Application of Diastereoselective Crotylboration and Methyl Ketone Aldol Reactions. Angewandte Chemie (International Ed. in English). 38: 1652-1655. PMID 29710989 DOI: 10.1002/(Sici)1521-3773(19990601)38:11<1652::Aid-Anie1652>3.0.Co;2-K |
0.792 |
|
| 1999 |
Roush WR, Narayan S. 2-Deoxy-2-iodo-alpha-mannopyranosyl and -talopyranosyl acetates: highly stereoselective glycosyl donors for the synthesis of 2-deoxy-alpha-glycosides. Organic Letters. 1: 899-902. PMID 10823220 DOI: 10.1021/Ol9908068 |
0.557 |
|
| 1999 |
Roush WR, Narayan S, Bennett CE, Briner K. Iodoacetoxylation of glycals using cerium(IV) ammonium nitrate, sodium iodide, and acetic acid: stereoselective synthesis of 2-deoxy-2-iodo-alpha-mannopyranosyl acetates. Organic Letters. 1: 895-7. PMID 10823219 DOI: 10.1021/Ol990815G |
0.737 |
|
| 1999 |
Roush WR, Gung BW, Bennett CE. 2-Deoxy-2-iodo- and 2-deoxy-2-bromo-alpha-glucopyranosyl trichloroacetimidates: highly reactive and stereoselective donors for the synthesis of 2-deoxy-beta-glycosides. Organic Letters. 1: 891-3. PMID 10823218 DOI: 10.1021/Ol9908070 |
0.63 |
|
| 1999 |
Roush WR, Lane GC. Studies on the synthesis of tedanolide: synthesis of the C(5)-C(21) segment via a highly stereoselective fragment assembly aldol reaction of a chiral beta,gamma-unsaturated methyl ketone. Organic Letters. 1: 95-8. PMID 10822542 DOI: 10.1021/Ol990572S |
0.814 |
|
| 1999 |
Roush WR, Hernandez AA, Zepeda G. A new synthesis of peptidyl epoxysuccinates for probing cysteine protease-inhibitor P3/S3 binding interactions Synthesis. 1500-1504. DOI: 10.1055/S-1999-3648 |
0.387 |
|
| 1999 |
Roush WR, Hartz RA, Gustin DJ. Total Synthesis of Olivomycin AJ. Am. Chem. Soc.1999,121, 1990−1991 Journal of the American Chemical Society. 121: 4092-4092. DOI: 10.1021/Ja9955060 |
0.36 |
|
| 1999 |
Roush WR, Bennett CE. A highly stereoselective synthesis of 2-deoxy-β-glycosides using 2- deoxy-2-iodo-glucopyranosyl acetate donors [7] Journal of the American Chemical Society. 121: 3541-3542. DOI: 10.1021/Ja984365J |
0.635 |
|
| 1999 |
Roush WR, Hartz RA, Gustin DJ. Total synthesis of olivomycin A [19] Journal of the American Chemical Society. 121: 1990-1991. DOI: 10.1021/Ja984229E |
0.438 |
|
| 1999 |
Roush WR, Dilley GJ. Studies of fragment assembly aldol reactions of chiral aldehydes and chiral methyl ketones: Stereoselective synthesis of the C(13)-C(25) segment of scytophycin C Tetrahedron Letters. 40: 4955-4959. DOI: 10.1016/S0040-4039(99)00868-0 |
0.81 |
|
| 1999 |
Chemler SR, Roush WR. Stereochemically divergent pathways for the allylation and crotylation reactions of anti- and syn-β-hydroxy-α-methyl aldehydes with allyl- and crotyltrifluorosilanes Tetrahedron Letters. 40: 4643-4647. DOI: 10.1016/S0040-4039(99)00730-3 |
0.677 |
|
| 1999 |
Micalizio GC, Roush WR. Towards the synthesis of spongistatin 1: Diastereoselective synthesis of the C(36)-C(45) subunit Tetrahedron Letters. 40: 3351-3354. DOI: 10.1016/S0040-4039(99)00464-5 |
0.724 |
|
| 1999 |
Chemler SR, Coffey DS, Roush WR. An improved synthesis of the (E,Z)-dienoate precursor of (+)-damavaricin D via a vinylogous Horner-Wadsworth-Emmons reaction Tetrahedron Letters. 40: 1269-1272. DOI: 10.1016/S0040-4039(98)02638-0 |
0.71 |
|
| 1999 |
Scheldt KA, Tasaka A, Bannister TD, Wendt MD, Roush WR. Total synthesis of (-)-bafilomycin A1: Application of diastereoselective crotylboration and methyl ketone aldol reactions Angewandte Chemie - International Edition. 38: 1652-1655. DOI: 10.1002/(SICI)1521-3773(19990601)38:11<1652::AID-ANIE1652>3.0.CO;2-K |
0.325 |
|
| 1999 |
Scheidt KA, Tasaka A, Bannister TD, Wendt MD, Roush WR. Totalsynthese von (−)-Bafilomycin A1: Anwendung von diastereoselektiver Crotylborierung und Methylketon-Aldolreaktionen Angewandte Chemie. 111: 1760-1762. DOI: 10.1002/(Sici)1521-3757(19990601)111:11<1760::Aid-Ange1760>3.0.Co;2-A |
0.491 |
|
| 1998 |
Scheidt KA, Roush WR, McKerrow JH, Selzer PM, Hansell E, Rosenthal PJ. Structure-based design, synthesis and evaluation of conformationally constrained cysteine protease inhibitors. Bioorganic & Medicinal Chemistry. 6: 2477-94. PMID 9925304 DOI: 10.1016/S0968-0896(98)80022-9 |
0.546 |
|
| 1998 |
Roush WR, González FV, McKerrow JH, Hansell E. Design and synthesis of dipeptidyl alpha',beta'-epoxy ketones, potent irreversible inhibitors of the cysteine protease cruzain. Bioorganic & Medicinal Chemistry Letters. 8: 2809-12. PMID 9873627 DOI: 10.1016/S0960-894X(98)00494-6 |
0.321 |
|
| 1998 |
Ley SV, Osborn HMI, Priepke HWM, Warriner SL, Scheidt KA, Roush WR. (1'S, 2'S)-Methyl-30,40-(1', 2' -Dimethoxycyclohexane-1', 2'-Diyl)-Alpha -D-Mannopyranoside : (Alpha -D-Mannopyranoside, Methyl 3,4-O-(1,2-Dimethoxy-1 ,2 -Cyclohexanediyl)-, 3S(S)-) Organic Syntheses. 75: 170-176. DOI: 10.15227/Orgsyn.075.0170 |
0.506 |
|
| 1998 |
Scheidt KA, Chen H, Follows BC, Chemler SR, Coffey DS, Roush WR. Tris(dimethylamino)sulfonium Difluorotrimethylsilicate, a Mild Reagent for the Removal of Silicon Protecting Groups The Journal of Organic Chemistry. 63: 6436-6437. DOI: 10.1021/Jo981215I |
0.715 |
|
| 1998 |
Chemler SR, Roush WR. Concerning the Synthesis of the Elusiveanti,anti-Dipropionate Stereotriad via the Crotylation of β-Hydroxy α-Methyl Aldehydes with (Z)-Crotyltrifluorosilane. Application to the Synthesis of the C(7)−C(16) Segment of Zincophorin The Journal of Organic Chemistry. 63: 3800-3801. DOI: 10.1021/Jo980387C |
0.687 |
|
| 1998 |
Roush WR, Sciotti RJ. Studies on the Synthesis of Chlorothricolide: Diastereo- and Enantioselective Syntheses of Model Top-Half Spirotetronate Units The Journal of Organic Chemistry. 63: 5473-5482. DOI: 10.1021/Jo980379W |
0.428 |
|
| 1998 |
Roush WR, Pfeifer LA, Marron TG. Studies on the synthesis of the mycalamides: Stereocontrolled synthesis of a model N-glycosylpederamide via a stereoselective aldol reaction Journal of Organic Chemistry. 63: 2064-2065. DOI: 10.1021/Jo980023K |
0.813 |
|
| 1998 |
Roush WR, Gwaltney SL, Cheng J, Scheidt KA, McKerrow JH, Hansell E. Vinyl sulfonate esters and vinyl sulfonamides: Potent, irreversible inhibitors of cysteine proteases [10] Journal of the American Chemical Society. 120: 10994-10995. DOI: 10.1021/Ja981792O |
0.554 |
|
| 1998 |
Roush WR, Sciotti RJ. Enantioselective Total Synthesis of (−)-Chlorothricolide via the Tandem Inter- and Intramolecular Diels−Alder Reaction of a Hexaenoate Intermediate Journal of the American Chemical Society. 120: 7411-7419. DOI: 10.1021/Ja980611F |
0.515 |
|
| 1997 |
Roush WR, Marron TG, Pfeifer LA. Highly Diastereoselective Synthesis of Pederic Acid Derivatives. The Journal of Organic Chemistry. 62: 474-478. PMID 11671436 DOI: 10.1021/Jo961841K |
0.823 |
|
| 1997 |
Roush WR, Reilly ML, Koyama K, Brown BB. A Formal Total Synthesis of (+)-Tetronolide, the Aglycon of the Tetrocarcins: Enantio- and Diastereoselective Syntheses of the Octahydronaphthalene (Bottom-Half) and Spirotetronate (Top-Half) Fragments The Journal of Organic Chemistry. 62: 8708-8721. DOI: 10.1021/Jo970960C |
0.523 |
|
| 1997 |
Hunt JA, Roush WR. 4,5-Diisopropyl-B-[(E)-[(3‘-menthofuryl)dimethylsilyl]allyl]-1,3,2- dioxaborolane, an Improved Chiral Reagent for the Anti α-Hydroxyallylation of Aldehydes: Application to the Enantioselective Synthesis of (−)-Swainsonine The Journal of Organic Chemistry. 62: 1112-1124. DOI: 10.1021/Jo961840S |
0.463 |
|
| 1997 |
Roush WR, Coffey DS, Madar DJ. Total synthesis of (+)-damavaricin D Journal of the American Chemical Society. 119: 11331-11332. DOI: 10.1021/Ja971828X |
0.338 |
|
| 1997 |
Roush WR, Barda DA. Highly Selective Lewis Acid Catalyzed Diels−Alder Reactions of Acyclic (Z)-1,3-Dienes Journal of the American Chemical Society. 119: 7402-7403. DOI: 10.1021/Ja971070H |
0.417 |
|
| 1997 |
Roush WR, Barda DA. Second generation synthesis of the quartromicin spirotetronic acid subunits via a Claisen rearrangement-intramolecular aldol sequence Tetrahedron Letters. 38: 8785-8788. DOI: 10.1016/S0040-4039(97)10416-6 |
0.461 |
|
| 1997 |
Roush WR, Barda DA. An intramolecular Diels-Alder approach to the spirotetronic acid subunits of the quartromicins Tetrahedron Letters. 38: 8781-8784. DOI: 10.1016/S0040-4039(97)10415-4 |
0.426 |
|
| 1997 |
Roush WR, Sebesta DP, James RA. Stereoselective synthesis of 2-deoxy-β-glycosides from glycal precursors. 2. Stereochemistry of glycosidation reactions of 2-thiophenyl- and 2-selenophenyl-α-d-gluco-pyranosyl donors Tetrahedron. 53: 8837-8852. DOI: 10.1016/S0040-4020(97)90395-1 |
0.415 |
|
| 1997 |
Roush WR, Sebesta DP, Bennett CE. Stereoselective synthesis of 2-deoxy-β-glycosides from glycal precursors. 1. Stereochemistry of the reactions of d-glucal derivatives with phenylsulfenyl chloride and phenylselenenyl chloride Tetrahedron. 53: 8825-8836. DOI: 10.1016/S0040-4020(97)90394-X |
0.674 |
|
| 1996 |
Roush WR, Briner K, Kesler BS, Murphy M, Gustin DJ. Studies on the Synthesis of Aureolic Acid Antibiotics: Acyloin Glycosidation Studies. The Journal of Organic Chemistry. 61: 6098-6099. PMID 11667440 DOI: 10.1021/Jo960932E |
0.764 |
|
| 1996 |
Hunt JA, Roush WR. Solid-Phase Synthesis of 6-Deoxyoligosaccharides Journal of the American Chemical Society. 118: 9998-9999. DOI: 10.1021/Ja962128F |
0.307 |
|
| 1996 |
Roush WR, Koyama K, Curtin ML, Moriarty KJ. Studies on the synthesis of nargenicin A1: Highly stereoselective synthesis of the complete carbon framework via the transannular Diels-Alder reaction of an 18-membered macrolide Journal of the American Chemical Society. 118: 7502-7512. DOI: 10.1021/Ja9607796 |
0.517 |
|
| 1996 |
Roush WR, Champoux JA, Peterson BC. Diastereoselective synthesis of the cis-octahydronaphthalene nucleus of superstolides A and B Tetrahedron Letters. 37: 8989-8992. DOI: 10.1016/S0040-4039(96)02110-7 |
0.478 |
|
| 1996 |
Roush WR, Works AB. Diastereoselective synthesis of the trans-anti-cis-decahydro-as-indacene ring system via the transannular Diels-Alder reaction of a functionalized (E,E,E)-cyclododeca-1,6,8-triene Tetrahedron Letters. 37: 8065-8068. DOI: 10.1016/0040-4039(96)01840-0 |
0.411 |
|
| 1995 |
Roush WR, Coffey DS. Synthesis of the Naphthoquinone Nucleus of Awamycin The Journal of Organic Chemistry. 60: 4412-4418. DOI: 10.1021/Jo00119A018 |
0.374 |
|
| 1995 |
Roush WR, Lin X. Studies on the Synthesis of Aureolic Acid Antibiotics: Highly Stereoselective Synthesis of Aryl 2-Deoxy-.beta.-glycosides via the Mitsunobu Reaction and Synthesis of the Olivomycin A-B Disaccharide Journal of the American Chemical Society. 117: 2236-2250. DOI: 10.1021/Ja00113A013 |
0.482 |
|
| 1995 |
Gustin DJ, VanNieuwenhze MS, Roush WR. Synthesis of the C(3)C(15) segment of rutamycin B via a C(8)C(9) fragment assembly aldol reaction: Metal dependence of the aldehyde and enolate diastereofacial selectivities Tetrahedron Letters. 36: 3447-3450. DOI: 10.1016/0040-4039(95)00628-P |
0.682 |
|
| 1995 |
Gustin DJ, VanNieuwenhze MS, Roush WR. Diastereoselective aldol reactions of chiral aldehydes and chiral methyl ketones: Dependence of stereoselectivity on the metal enolate, the aldehyde 2,3-stereochemistry, and the aldehyde β-alkoxy protecting group Tetrahedron Letters. 36: 3443-3446. DOI: 10.1016/0040-4039(95)00626-N |
0.684 |
|
| 1995 |
Marron TG, Roush WR. Diastereoselective synthesis of N-benzoyl mycalamine, the fully elaborated trioxadecalin nucleus of mycalamide. A. Control of the key N-acyl aminal stereocenter via carbamate acylation Tetrahedron Letters. 36: 1581-1584. DOI: 10.1016/0040-4039(95)00093-R |
0.423 |
|
| 1995 |
Hunt J, Roush WR. Diisopropyl tartrate-modified (E)-γ-[(menthofuryl)dimethylsilyl]-allyl boronate, an improved chiral reagent for the anti α-hydroxyallylation of aldehydes. Application to the enantioselective synthesis of (−)-swainsonine Tetrahedron Letters. 36: 501-504. DOI: 10.1016/0040-4039(94)02295-M |
0.474 |
|
| 1994 |
Roush WR, VanNieuwenhze MS. [(Z)-.gamma.-[(Diisopropylidene-.alpha.-D-mannopyranosyl)oxy]allyl]tributylstannane: A New Chiral Reagent for the Asymmetric .alpha.-Hydroxyallylation of Aldehydes Journal of the American Chemical Society. 116: 8536-8543. DOI: 10.1021/Ja00098A014 |
0.602 |
|
| 1994 |
Roush WR, Sciotti RJ. Enantioselective Total Synthesis of (-)-Chlorothricolide Journal of the American Chemical Society. 116: 6457-6458. DOI: 10.1021/Ja00093A065 |
0.463 |
|
| 1994 |
Roush WR, Wada CK. Application of .eta.4-Diene Iron Tricarbonyl Complexes in Acyclic Stereocontrol: Asymmetric Synthesis of the as-Indacene Unit of Ikarugamycin (A Formal Total Synthesis) Journal of the American Chemical Society. 116: 2151-2152. DOI: 10.1021/Ja00084A068 |
0.366 |
|
| 1994 |
Roush WR, Follows BC. Asymmetric synthesis of the hydroxylamino sugar of calicheamicin Tetrahedron Letters. 35: 4935-4938. DOI: 10.1016/S0040-4039(00)73286-2 |
0.396 |
|
| 1994 |
Roush WR, Gustin D. A stereochemically general synthesis of methyl 2,4,6-trideoxy-4-methylthio-α-D-ribo-pyranoside, the thio sugar of esperamicin A1 Tetrahedron Letters. 35: 4931-4934. DOI: 10.1016/S0040-4039(00)73285-0 |
0.436 |
|
| 1994 |
Wada CK, Roush WR. Highly stereoselective 1,4-addition reactions of alkylidene malonate substituted η4-(1,3-butadienyl)iron(tricarbonyl) complexes Tetrahedron Letters. 35: 7351-7354. DOI: 10.1016/0040-4039(94)85311-8 |
0.384 |
|
| 1994 |
Roush WR, Wada CK. Highly stereoselective substitution reactions of functionalized η4-[3(E),5(E)-heptadien-2-ol]iron tricarbonyl complexes Tetrahedron Letters. 35: 7347-7350. DOI: 10.1016/0040-4039(94)85310-X |
0.408 |
|
| 1993 |
Roush WR, Briner K, Sebesta DP. Highly Stereoselective Synthesis of α-L-Olivomycosides via Trimethylsilyl Triflate Mediated Glycosidations of 1-O-Acetyl-4-O-isobutyryl-2,6-dideoxy-2-iodo-3-C-methyl-α-L-mannopyranose Synlett. 1993: 264-266. DOI: 10.1055/S-1993-22425 |
0.32 |
|
| 1993 |
Roush WR, Brown BB. Studies on the synthesis of kijanolide: synthesis of the 2-acyl spirotetronate and investigations concerning the coupling of the top and bottom half fragments The Journal of Organic Chemistry. 58: 2162-2172. DOI: 10.1021/Jo00060A036 |
0.476 |
|
| 1993 |
Roush WR, Brown BB. A highly diastereo- and enantioselective synthesis of the top half of kijanolide The Journal of Organic Chemistry. 58: 2151-2161. DOI: 10.1021/Jo00060A035 |
0.465 |
|
| 1993 |
Roush WR, Brown BB. Application of the steric directing group strategy to the stereoselective synthesis of the octahydronaphthalene substructure of kijanolide and tetronolide Journal of the American Chemical Society. 115: 2268-2278. DOI: 10.1021/Ja00059A024 |
0.483 |
|
| 1993 |
Roush WR, Lin X. Synthesis of naphthyl A–B disaccharides corresponding to olivomycin A and mithramycin Tetrahedron Letters. 34: 6829-6832. DOI: 10.1016/S0040-4039(00)91806-9 |
0.454 |
|
| 1993 |
Roush WR, Marron TG. Toward the synthesis of mycalamides A, B and onnamide A: a highly stereoselective synthesis of the trioxadecalin ring system Tetrahedron Letters. 34: 5421-5424. DOI: 10.1016/S0040-4039(00)73924-4 |
0.42 |
|
| 1993 |
Roush WR, Bannister TD, Wendt MD. Concerning the diastereofacial selectivity of aldol reactions of chiral methyl ketone enolates: Evidence for remote chelation in the bafilomycin aldol reaction Tetrahedron Letters. 34: 8387-8390. DOI: 10.1016/S0040-4039(00)61340-0 |
0.72 |
|
| 1993 |
Roush WR, Warmus JS, Works AB. Synthesis and transannular diels-alder reactions of (E,E,E)-cyclotetradeca-2,8,10-trienones Tetrahedron Letters. 34: 4427-4430. DOI: 10.1016/0040-4039(93)88050-S |
0.388 |
|
| 1993 |
Roush WR, Madar DJ. Towards the synthesis of streptovaricin D: Synthesis of fully elaborated aromatic precursors and coupling with ansa chain fragments Tetrahedron Letters. 34: 1553-1556. DOI: 10.1016/0040-4039(93)85004-G |
0.401 |
|
| 1992 |
Roush WR, Murphy M. An improved synthesis of naphthoate precursors to olivin The Journal of Organic Chemistry. 57: 6622-6629. DOI: 10.1021/Jo00050A047 |
0.458 |
|
| 1992 |
Sebesta DP, Roush WR. Synthesis of C-D-E trisaccharide precursors of olivomycin A. The Journal of Organic Chemistry. 57: 4799-4802. DOI: 10.1021/Jo00044A010 |
0.359 |
|
| 1992 |
Roush WR, Brown BB. Enantioselective synthesis of 2-alkyl-5-methylene-1,3-dioxolan-4-ones and exo-selective Diels-Alder reactions with cyclopentadiene The Journal of Organic Chemistry. 57: 3380-3387. DOI: 10.1021/Jo00038A028 |
0.363 |
|
| 1992 |
Roush WR, Ratz AM, Jablonowski JA. Solid-state and solution conformational analysis of tartrate-derived 1,3-dioxolanes and 1,3,2-dioxaborolanes The Journal of Organic Chemistry. 57: 2047-2052. DOI: 10.1021/Jo00033A027 |
0.304 |
|
| 1992 |
Roush WR, Bannister TD. Stereoselective synthesis of the C(13)–C(25) segment of bafilomycin A1 Tetrahedron Letters. 33: 3587-3590. DOI: 10.1016/S0040-4039(00)92509-7 |
0.716 |
|
| 1992 |
Roush WR, Sciotti RJ. Enantioselective synthesis of the top half of chlorothricolide Tetrahedron Letters. 33: 4691-4694. DOI: 10.1016/S0040-4039(00)61260-1 |
0.472 |
|
| 1992 |
Roush WR, Koyama K. Enantioselective synthesis of the top half of tetronolide Tetrahedron Letters. 33: 6227-6230. DOI: 10.1016/S0040-4039(00)60939-5 |
0.461 |
|
| 1992 |
Roush WR, Grover PT. Diisopropyl tartrate modified (E)-γ-[(cyclohexyloxy)dimethylsilyl]- and (E)-γ-(dimethylphenylsilyl)allylboronates: Chiral Reagents for the Enantio- and Diastereoselective synthesis of anti 1,2-diols and 2-butene-1,4-diols via the formal α- and γ-hydroxyallylation of aldehydes Tetrahedron. 48: 1981-1998. DOI: 10.1016/S0040-4020(01)88869-4 |
0.446 |
|
| 1991 |
Roush WR, Lin XF. A highly stereoselective synthesis of aryl 2-deoxy-.beta.-glycosides via the Mitsunobu reaction The Journal of Organic Chemistry. 56: 5740-5742. DOI: 10.1021/Jo00020A003 |
0.44 |
|
| 1991 |
Roush WR. Concerning the diastereofacial selectivity of the aldol reactions of .alpha.-methyl chiral aldehydes and lithium and boron propionate enolates The Journal of Organic Chemistry. 56: 4151-4157. DOI: 10.1021/Jo00013A015 |
0.455 |
|
| 1991 |
Roush WR, Lin X, Straub JA. A highly stereoselective synthesis of the AB disaccharide unit of olivomycin A The Journal of Organic Chemistry. 56: 1649-1655. DOI: 10.1021/Jo00004A054 |
0.474 |
|
| 1991 |
Roush WR, Straub JA, VanNieuwenhze MS. A stereochemically general synthesis of 2-deoxyhexoses via the asymmetric allylboration of 2,3-epoxy aldehydes The Journal of Organic Chemistry. 56: 1636-1648. DOI: 10.1021/Jo00004A053 |
0.66 |
|
| 1991 |
Roush WR, Kageyama M, Riva R, Brown BB, Warmus JS, Moriarty KJ. Enantioselective synthesis of the bottom half of chlorothricolide. 3. Studies of the steric directing group strategy for stereocontrol in intramolecular Diels-Alder reactions The Journal of Organic Chemistry. 56: 1192-1210. DOI: 10.1021/Jo00003A049 |
0.5 |
|
| 1991 |
Roush WR, Park JC. Asymmetric allylborations of 3-decynal dicobalt hexacarbonyl: cobalt induced reversal of enantioselectivity and applications to highly diastereoselective intramolecular pauson-khand reactions Tetrahedron Letters. 32: 6285-6288. DOI: 10.1016/0040-4039(91)80148-Y |
0.426 |
|
| 1990 |
Roush WR, Hoong LK, Palmer MAJ, Straub JA, Palkowitz AD. Asymmetric synthesis using tartrate ester modified allylboronates. 2. Single and double asymmetric reactions with alkoxy-substituted aldehydes The Journal of Organic Chemistry. 55: 4117-4126. DOI: 10.1021/Jo00300A032 |
0.404 |
|
| 1990 |
Roush WR, Hoong LK, Palmer MAJ, Park JC. Asymmetric synthesis using tartrate ester modified allylboronates. 1. Factors influencing stereoselectivity The Journal of Organic Chemistry. 55: 4109-4117. DOI: 10.1021/Jo00300A031 |
0.322 |
|
| 1990 |
Roush WR, Park JC. Use of metal carbonyl complexes to achieve high enantioselectivity in the asymmetric allylboration of unsaturated aldehydes The Journal of Organic Chemistry. 55: 1143-1144. DOI: 10.1021/Jo00291A009 |
0.308 |
|
| 1990 |
Roush WR, Palkowitz AD, Ando K. Acyclic diastereoselective synthesis using tartrate ester-modified crotylboronates. Double asymmetric reactions with .alpha.-methyl chiral aldehydes and synthesis of the C(19)-C(29) segment of rifamycin S Journal of the American Chemical Society. 112: 6348-6359. DOI: 10.1021/Ja00173A024 |
0.477 |
|
| 1990 |
Roush WR, Ando K, Powers DB, Palkowitz AD, Halterman RL. Asymmetric synthesis using diisopropyl tartrate modified (E)- and (Z)-crotylboronates: preparation of the chiral crotylboronates and reactions with achiral aldehydes Journal of the American Chemical Society. 112: 6339-6348. DOI: 10.1021/Ja00173A023 |
0.492 |
|
| 1990 |
Roush WR, Grover PT. Diisopropyl tartrate (E)-γ-(dimethylphenylsilyl)allylboronate, a chiral allylic alcohol β-carbanion equivalent for the enantioselective synthesis of 2-butene-1,4-diols from aldehydes Tetrahedron Letters. 31: 7567-7570. DOI: 10.1016/S0040-4039(00)97300-3 |
0.49 |
|
| 1990 |
Roush WR, Gover PT, Lin X. Diisopropyl tartrate modified (E)-γ-[(cyclohexyloxy)dimethylsilyl-allylboronate, a chiral reagent for the stereoselective synthesis of anti 1,2-diols via the formal α-hydroxyallylation of aldehydes Tetrahedron Letters. 31: 7563-7566. DOI: 10.1016/S0040-4039(00)97299-X |
0.493 |
|
| 1990 |
Roush WR, Moriarty KJ, Brown BB. Stereoselective synthesis of (Z,E)-2-bromo-1,3-dienes via the palladium (O) catalyzed cross coupling reactions of 1,1-dibromoolefins and vinylboronic acids Tetrahedron Letters. 31: 6509-6512. DOI: 10.1016/S0040-4039(00)97103-X |
0.438 |
|
| 1990 |
ROUSH WR, PALKOWITZ AD, ANDO K. ChemInform Abstract: Acyclic Diastereoselective Synthesis Using Tartrate Ester Modified Crotylboronates. Double Asymmetric Reactions with α-Methyl Chiral Aldehydes and Synthesis of the C(19)-C(29) Segment of Rifamycin S. Cheminform. 21. DOI: 10.1002/chin.199049076 |
0.419 |
|
| 1990 |
ROUSH WR, ANDO K, POWERS DB, PALKOWITZ AD, HALTERMAN RL. ChemInform Abstract: Asymmetric Synthesis Using Diisopropyl Tartrate Modified (E)- and (Z)-Crotylboronates: Preparation of the Chiral Crotylboronates and Reactions with Achiral Aldehydes. Cheminform. 21. DOI: 10.1002/chin.199049075 |
0.391 |
|
| 1990 |
ROUSH WR, HOONG LK, PALMER MAJ, PARK JC. ChemInform Abstract: Asymmetric Synthesis Using Tartrate Ester Modified Allylboronates. Part 1. Factors Influencing Stereoselectivity. Cheminform. 21. DOI: 10.1002/chin.199045065 |
0.304 |
|
| 1990 |
ROUSH WR, HOONG LK, PALMER MAJ, STRAUB JA, PALKOWITZ AD. ChemInform Abstract: Asymmetric Synthesis Using Tartrate Ester-Modified Allylboronates. Part 2. Single and Double Asymmetric Reactions with Alkoxy-Substituted Aldehydes. Cheminform. 21. DOI: 10.1002/chin.199045064 |
0.426 |
|
| 1990 |
ROUSH WR. ChemInform Abstract: Stereochemical and Synthetic Studies of the Intramolecular Diels-Alder Reaction Cheminform. 21. DOI: 10.1002/chin.199044337 |
0.34 |
|
| 1990 |
ROUSH WR, BROWN BB. ChemInform Abstract: Diastereoselective Synthesis of the Top Half of Kijanolide. Cheminform. 21. DOI: 10.1002/chin.199033305 |
0.359 |
|
| 1990 |
ROUSH WR, ESSENFELD AP, WARMUS JS, BROWN BB. ChemInform Abstract: Synthesis and Diels-Alder Reactions of 2-Alkyl-5-methylene-1,3-dioxolan-4-ones (Va), (Vb) and 2-Alkyl-3-acyl-5-methylene-1,3-oxazolidin-4-ones (Vc): Highly Exo and Diastereoface Selective Chiral Ketene Equivalents. Cheminform. 21. DOI: 10.1002/chin.199032059 |
0.417 |
|
| 1990 |
ROUSH WR. ChemInform Abstract: Evolution of a Strategy for the Synthesis of Olivomycin A: Development of Methodology for the Diastereo- and Enantioselective Synthesis of Carbohydrates from Acyclic Precursors Cheminform. 21. DOI: 10.1002/chin.199016344 |
0.353 |
|
| 1989 |
Roush WR, Palkowitz AD. Synthesis of the C(1)-C(15) segment of streptovaricin D The Journal of Organic Chemistry. 54: 3009-3011. DOI: 10.1021/Jo00274A008 |
0.35 |
|
| 1989 |
Coe JW, Roush WR. Studies of an intramolecular Diels-Alder approach to the nargenicins: involvement of boatlike transition states in the cyclizations of substituted 1,7,9-decatrien-3-ones The Journal of Organic Chemistry. 54: 915-930. DOI: 10.1021/Jo00265A036 |
0.316 |
|
| 1989 |
Roush WR, Michaelides MR, Tai DF, Lesur BM, Chong WKM, Harris DJ. A highly stereoselective synthesis of (+)-olivin, the aglycon of olivomycin A Journal of the American Chemical Society. 111: 2984-2995. DOI: 10.1021/Ja00190A036 |
0.773 |
|
| 1989 |
Roush WR, Banfi L, Park JC, Hoong LK. The asymmetric allylboration reaction: Dependence of rate and enantioselectivity on the chiral auxiliary Tetrahedron Letters. 30: 6457-6460. DOI: 10.1016/S0040-4039(01)88993-0 |
0.804 |
|
| 1989 |
Roush WR, Brown BB. Diastereoselective synthesis of the top half of kijanolide Tetrahedron Letters. 30: 7309-7312. DOI: 10.1016/S0040-4039(00)70684-8 |
0.515 |
|
| 1989 |
Roush WR, Essenfeld AP, Warmus JS, Brown BB. Synthesis and Diels-Alder reactions of 2-alkyl-5-methylene-1,3-dioxolan-4-ones and 2-alkyl-3-acyl-5-methylene-1,3-oxazolidin-4-ones: Highly exo and diastereoface selective chiral ketene equivalents Tetrahedron Letters. 30: 7305-7308. DOI: 10.1016/S0040-4039(00)70683-6 |
0.481 |
|
| 1989 |
Roush WR. Evolution of a Strategy for the Synthesis of Olivomycin a: Development of Methodology for the Diastereo- and Enantioselective Synthesis of Carbohydrates from Acyclic Precursors Strategies and Tactics in Organic Synthesis. 2: 323-367. DOI: 10.1016/B978-0-08-092429-8.50015-5 |
0.453 |
|
| 1989 |
ROUSH WR, MICHAELIDES MR, TAI DF, LESUR BM, CHONG WKM, HARRIS DJ. ChemInform Abstract: A Highly Stereoselective Synthesis of (+)-Olivin, the Aglycon of Olivomycin A. Cheminform. 20. DOI: 10.1002/chin.198932317 |
0.755 |
|
| 1989 |
ROUSH WR, ANDO K, POWERS DB, HALTERMAN RL, PALKOWITZ AD. ChemInform Abstract: Enantioselective Synthesis Using Diisopropyl Tartrate Modified E- (I) and Z-Crotylboronates (II): Reactions with Achiral Aldehydes (III). Cheminform. 20. DOI: 10.1002/chin.198918154 |
0.313 |
|
| 1988 |
Roush WR, Riva R. Enantioselective synthesis of the bottom half of chlorothricolide. 2. A comparative study of substituent effects on the stereoselectivity of the key intramolecular Diels-Alder reaction The Journal of Organic Chemistry. 53: 710-712. DOI: 10.1021/Jo00238A049 |
0.477 |
|
| 1988 |
Roush WR, Ando K, Powers DB, Halterman RL, Palkowitz AD. Enantioselective synthesis using diisopropyl tartrate modified (E)- and (Z)-crotylboronates: Reactions with achiral aldehydes Tetrahedron Letters. 29: 5579-5582. DOI: 10.1016/S0040-4039(00)80816-3 |
0.418 |
|
| 1988 |
Roush WR, Brown BB, Drozda SE. A highly stereoselective synthesis of the octahydronaphthalene subunit of kijanolide and tetronolide Tetrahedron Letters. 29: 3541-3544. DOI: 10.1016/0040-4039(88)85287-0 |
0.491 |
|
| 1988 |
ROUSH WR, BROWN BB, DROZDA SE. ChemInform Abstract: A Highly Stereoselective Synthesis of the Octahydronaphthalene Subunit of Kijanolide and Tetronolide. Cheminform. 19. DOI: 10.1002/chin.198852125 |
0.328 |
|
| 1988 |
ROUSH WR, RIVA R. ChemInform Abstract: Enantioselective Synthesis of the Bottom Half of Chlorothricolide. Part 2. A Comparative Study of Substituent Effects on the Stereoselectivity of the Key Intramolecular Diels-Alder Reaction. Cheminform. 19. DOI: 10.1002/chin.198825163 |
0.421 |
|
| 1988 |
ROUSH WR, STRAUB JA, BROWN RJ. ChemInform Abstract: Stereochemistry of the Epoxidations of Acyclic Allylic Amides. Applications toward the Synthesis of 2,3,6-Trideoxy-3-aminohexoses. Cheminform. 19. DOI: 10.1002/chin.198817158 |
0.36 |
|
| 1988 |
ROUSH WR, MICHAELIDES MR, TAI DF, CHONG WKM. ChemInform Abstract: A Highly Stereoselective Total Synthesis of the Natural Enantiomer of Olivin (XIIb). Cheminform. 19. DOI: 10.1002/chin.198812347 |
0.358 |
|
| 1987 |
Halterman RL, Roush WR, Hoong LK. Analytical resolution of secondary methyl ethers by chiral complexation gas chromatography The Journal of Organic Chemistry. 52: 1152-1155. DOI: 10.1021/Jo00382A036 |
0.312 |
|
| 1987 |
Roush WR, Russo-Rodriguez S. Trichothecene degradation studies. 3. Synthesis of 12,13-deoxy-12,13-methanoanguidine and 12-epianguidine, two optically active analogs of the epoxytrichothecene mycotoxin anguidine The Journal of Organic Chemistry. 52: 603-606. DOI: 10.1021/Jo00380A022 |
0.754 |
|
| 1987 |
Roush WR, Russo-Rodriguez S. Trichothecene degradation studies. 2. Synthesis of [13-14C]anguidine The Journal of Organic Chemistry. 52: 598-603. DOI: 10.1021/Jo00380A021 |
0.791 |
|
| 1987 |
Roush WR, Palkowitz AD, Palmer MJ. Reactions of diisopropyl tartrate modified allyl- and (E)- and (Z)-crotylboronates with .beta.-alkoxy-.alpha.-methylpropionaldehydes: a reagent-based solution to the acyclic dipropionate problem The Journal of Organic Chemistry. 52: 316-318. DOI: 10.1021/Jo00378A041 |
0.393 |
|
| 1987 |
Roush WR, Straub JA, Brown RJ. Total synthesis of carbohydrates. 5. Stereochemistry of the epoxidations of acyclic allylic amides. Applications towards the synthesis of 2,3,6-trideoxy-3-aminohexoses The Journal of Organic Chemistry. 52: 5127-5136. DOI: 10.1021/Jo00232A014 |
0.468 |
|
| 1987 |
Roush WR, Michaelides MR, Tai DF, Chong WKM. A highly stereoselective total synthesis of the natural enantiomer of olivin Journal of the American Chemical Society. 109: 7575-7577. DOI: 10.1021/Ja00258A077 |
0.46 |
|
| 1987 |
Roush WR, Palkowitz AD. Application of tartrate ester modified allylic boronates in organic synthesis: an efficient, highly stereoselective synthesis of the carbon(19)-carbon(29) segment of rifamycin S Journal of the American Chemical Society. 109: 953-955. DOI: 10.1021/Ja00237A082 |
0.354 |
|
| 1987 |
Roush WR, Coe JW. Studies on the synthesis of nargenicin A1. An example of anintramolecular diels-alder reaction that proceeds with a boat-likeconformation of the connecting chain Tetrahedron Letters. 28: 931-934. DOI: 10.1016/S0040-4039(00)95877-5 |
0.444 |
|
| 1987 |
Roush WR, Essenfeld AP, Warmus JS. Effect of dienophile activating group on the stereoselectivity of the intramolecular diels-alder reaction Tetrahedron Letters. 28: 2447-2450. DOI: 10.1016/S0040-4039(00)95437-6 |
0.388 |
|
| 1987 |
ROUSH WR, RUSSO-RODRIGUEZ S. ChemInform Abstract: Trichothecene Degradation Studies. Part 3. Synthesis of 12,13-Deoxy- 12,13-methanoanguidine (I) and 12-Epianguidine (II), Two Optically Active Analogues of the Epoxytrichothecene Mycotoxin Anguidine. Cheminform. 18. DOI: 10.1002/chin.198733365 |
0.738 |
|
| 1987 |
ROUSH WR, RUSSO-RODRIGUEZ S. ChemInform Abstract: Trichothecene Degradation Studies. Part 2. Synthesis of (13-14C)Anguidine (I). Cheminform. 18. DOI: 10.1002/chin.198733364 |
0.784 |
|
| 1987 |
ROUSH WR, COE JW. ChemInform Abstract: Studies on the Synthesis of Nargenicin A1. An Example of an Intramolecular Diels-Alder Reaction that Proceeds with a Boat-Like Conformation of the Connecting Chain. Cheminform. 18. DOI: 10.1002/chin.198733087 |
0.306 |
|
| 1987 |
ROUSH WR, PALKOWITZ AD. ChemInform Abstract: Applications of Tartrate Ester Modified Allylic Boronates in Organic Synthesis: An Efficient, Highly Stereoselective Synthesis of the C(19)-C(29) Segment (X) of Rifamycin S. Cheminform. 18. DOI: 10.1002/chin.198724334 |
0.322 |
|
| 1986 |
Roush WR, Adam MA, Walts AE, Harris DJ. Stereochemistry of the reactions of substituted allylboronates with chiral aldehydes. Factors influencing aldehyde diastereofacial selectivity Journal of the American Chemical Society. 108: 3422-3434. DOI: 10.1021/Ja00272A043 |
0.427 |
|
| 1986 |
Roush WR, Halterman RL. Diisopropyl tartrate modified (E)-crotylboronates: highly enantioselective propionate (E)-enolate equivalents Journal of the American Chemical Society. 108: 294-296. DOI: 10.1021/Ja00262A018 |
0.323 |
|
| 1986 |
Roush WR, Michaelides MR. Studies on the total synthesis of sesbanimide: A highly diastereoselective synthesis of the ab ring system Tetrahedron Letters. 27: 3353-3356. DOI: 10.1016/S0040-4039(00)84794-2 |
0.441 |
|
| 1986 |
Roush WR, Straub JA. Total synthesis of the AB disaccharide unit of olivomycin A Tetrahedron Letters. 27: 3349-3352. DOI: 10.1016/S0040-4039(00)84793-0 |
0.428 |
|
| 1986 |
ROUSH WR, ADAM MA, WALTS AE, HARRIS DJ. ChemInform Abstract: Stereochemistry of the Reactions of Substituted Allylboronates with Chiral Aldehydes. Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198641265 |
0.471 |
|
| 1986 |
ROUSH WR, RUSSO-RODRIGUEZ S. ChemInform Abstract: Trichothecene Degradation Studies: Synthesis of 12,13-Deoxyanguidine (I) and 12,13-Deoxyverrucarol (II). Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198625329 |
0.76 |
|
| 1986 |
ROUSH WR, WALTS AE, HOONG LK. ChemInform Abstract: Diastereo- and Enantioselective Aldehyde Addition Reactions of 2-Allyl-1,3,2-dioxaborolane-4,5-dicarboxylic Esters, a Useful Class of Tartrate Ester Modified Allylboronates. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198616250 |
0.353 |
|
| 1986 |
ROUSH WR, RUSSO-RODRIGUEZ S. ChemInform Abstract: Synthesis of 4β-Acetoxyscirpene-3α,15-diol. Chemischer Informationsdienst. 17. DOI: 10.1002/Chin.198607225 |
0.76 |
|
| 1986 |
ROUSH WR, KAGEYAMA M. ChemInform Abstract: Enantioselective Synthesis of the Bottom-Half of Chlorothricolide. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198606134 |
0.366 |
|
| 1985 |
Roush WR, Hagadorn SM. Synthesis of mycarose and epi-axenose from non-carbohydrate precursors. Carbohydrate Research. 136: 187-93. PMID 4005889 DOI: 10.1016/0008-6215(85)85195-8 |
0.484 |
|
| 1985 |
Roush WR, Russo-Rodriguez S. Trichothecene degradation studies: synthesis of 12,13-deoxyanguidine and 12,13-deoxyverrucarol The Journal of Organic Chemistry. 50: 5465-5468. DOI: 10.1021/Jo00350A004 |
0.724 |
|
| 1985 |
Roush WR, Adam MA. Directed openings of 2,3-epoxy alcohols via reactions with isocyanates: synthesis of (+)-erythro-dihydrosphingosine The Journal of Organic Chemistry. 50: 3752-3757. DOI: 10.1021/Jo00220A015 |
0.385 |
|
| 1985 |
Roush WR, Russo-Rodriguez S. Synthesis of 4.beta.-acetoxyscirpene-3.alpha.,15-diol The Journal of Organic Chemistry. 50: 3224-3226. DOI: 10.1021/Jo00217A046 |
0.745 |
|
| 1985 |
Roush WR, Walts AE, Hoong LK. Diastereo- and enantioselective aldehyde addition reactions of 2-allyl-1,3,2-dioxaborolane-4,5-dicarboxylic esters, a useful class of tartrate ester modified allylboronates Journal of the American Chemical Society. 107: 8186-8190. DOI: 10.1021/Ja00312A062 |
0.452 |
|
| 1985 |
Roush WR, Marletta MA, Russo-Rodriguez S, Recchia J. Trichothecene metabolism studies: isolation and structure determination of 15-acetyl-3.alpha.-(1'.beta.-D-glucopyranosiduronyl)scirpen-3,4.beta.,15-triol Journal of the American Chemical Society. 107: 3354-3355. DOI: 10.1021/Ja00297A055 |
0.721 |
|
| 1985 |
Roush WR, Kageyama M. Enantioselective synthesis of the bottom-half of chlorothricolide Tetrahedron Letters. 26: 4327-4330. DOI: 10.1016/S0040-4039(00)98725-2 |
0.517 |
|
| 1985 |
Roush WR, Walts AE. Stereochemistry of the reactions of pinacol allylboronate with two α,β-dialkoxyaldehydes Tetrahedron Letters. 26: 3427-3430. DOI: 10.1016/S0040-4039(00)98655-6 |
0.387 |
|
| 1985 |
Roush WR, Marletta MA, Russo-Rodriguez S, Recchia J. Trichothecene metabolism studies. 2. Structure of 3α-(1″gb-D-glucopyranosiduronyl)-8α-isovaleryloxy-scirpen-3,4β, 15-triol 15-acetate produced from T-2 toxin IN VITRO Tetrahedron Letters. 26: 5231-5234. DOI: 10.1016/S0040-4039(00)95002-0 |
0.736 |
|
| 1985 |
Walts AE, Roush WR. A stereorational total synthesis of (−)-ptilocaulin Tetrahedron. 41: 3463-3478. DOI: 10.1016/S0040-4020(01)96701-8 |
0.428 |
|
| 1985 |
WALTS AE, ROUSH WR. ChemInform Abstract: A STEREORATIONAL TOTAL SYNTHESIS OF (-)-PTILOCAULIN Chemischer Informationsdienst. 16. DOI: 10.1002/chin.198551324 |
0.334 |
|
| 1985 |
ROUSH WR, MARLETTA MA, RUSSO-RODRIGUEZ S, RECCHIA J. ChemInform Abstract: TRICHOTHECENE METABOLISM STUDIES: ISOLATION AND STRUCTURE DETERMINATION OF 15-ACETYL-3α-(1′β-D-GLUCOPYRANOSIDURONYL)SCIRPEN-3,4β,15-TRIOL Chemischer Informationsdienst. 16. DOI: 10.1002/Chin.198538346 |
0.734 |
|
| 1985 |
ROUSH WR, HAGADORN SM. ChemInform Abstract: TOTAL SYNTHESIS OF CARBOHYDRATES, PART 4. SYNTHESIS OF MYCAROSE AND EPI-AXENOSE FROM NON-CARBOHYDRATE PRECURSORS Chemischer Informationsdienst. 16. DOI: 10.1002/chin.198534354 |
0.335 |
|
| 1985 |
ROUSH WR, GILLIS HR, ESSENFELD AP. ChemInform Abstract: HYDROFLUORIC ACID CATALYZED INTRAMOLECULAR DIELS-ALDER REACTIONS Chemischer Informationsdienst. 16. DOI: 10.1002/chin.198522143 |
0.321 |
|
| 1984 |
Roush WR, Blizzard TA. Synthesis of epoxytrichothecenes: verrucarin J and verrucarin J isomers The Journal of Organic Chemistry. 49: 1772-1783. DOI: 10.1021/Jo00184A021 |
0.384 |
|
| 1984 |
Blanchette MA, Choy W, Davis JT, Essenfeld AP, Masamune S, Roush WR, Sakai T. Horner-wadsworth-emmons reaction: Use of lithium chloride and an amine for base-sensitive compounds Tetrahedron Letters. 25: 2183-2186. DOI: 10.1016/S0040-4039(01)80205-7 |
0.39 |
|
| 1984 |
Roush WR, Gillis HR, Essenfeld AP. Hydrofluoric acid catalyzed intramolecular Diels-Alder reactions The Journal of Organic Chemistry. 49: 4674-4682. DOI: 10.1002/Chin.198522143 |
0.42 |
|
| 1984 |
ROUSH WR, BROWN RJ. ChemInform Abstract: TOTAL SYNTHESIS OF CARBOHYDRATES. 3. EFFICIENT ENANTIOSELECTIVE SYNTHESES OF 2,6-DIDEOXYHEXOSES Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198428336 |
0.332 |
|
| 1984 |
ROUSH WR, WALTS AE. ChemInform Abstract: TOTAL SYNTHESIS OF (-)-PTILOCAULIN Chemischer Informationsdienst. 15. DOI: 10.1002/chin.198419339 |
0.334 |
|
| 1984 |
Roush WR, Walts AE. Total synthesis of (-)-ptilocaulin Journal of the American Chemical Society. 106: 721-723. DOI: 10.1002/Chin.198419339 |
0.438 |
|
| 1983 |
Roush WR, Blizzard TA. Synthesis of verrucarin J The Journal of Organic Chemistry. 48: 758-759. DOI: 10.1021/Jo00153A035 |
0.422 |
|
| 1983 |
Roush WR, D'Ambra TE. Total synthesis of (.+-.)-verrucarol Journal of the American Chemical Society. 105: 1058-1060. DOI: 10.1021/Ja00342A071 |
0.438 |
|
| 1983 |
Roush WR, Spada AP. Synthesis of trichoverrol B Tetrahedron Letters. 24: 3693-3696. DOI: 10.1016/S0040-4039(00)94511-8 |
0.406 |
|
| 1983 |
Roush WR, Lesur BM. Stereochemistry of Vinyl Cuprate Additions to Carbohydrate-Derived Enones and α,β-Unsaturated Esters Tetrahedron Letters. 24: 2231-2234. DOI: 10.1016/S0040-4039(00)81891-2 |
0.71 |
|
| 1983 |
Roush WR, Harris DJ, Lesur BM. Studies on the Synthesis of Olivin: Diastereoselective Synthesis of a Functionalized D-Fucose Derivative Tetrahedron Letters. 24: 2227-2230. DOI: 10.1016/S0040-4039(00)81890-0 |
0.752 |
|
| 1983 |
Roush WR, Adam MA, Peseckis SM. Regioselectivity of the reactions of trialkylaluminum reagents with 2,3-epoxyalcohols: Application to the synthesis of α-chiral aldehydes Tetrahedron Letters. 24: 1377-1380. DOI: 10.1016/S0040-4039(00)81660-3 |
0.462 |
|
| 1983 |
Roush WR, Brown RJ. Total synthesis of carbohydrates. 3. Efficient enantioselective syntheses of 2,6-dideoxyhexoses The Journal of Organic Chemistry. 48: 5093-5101. DOI: 10.1002/Chin.198428336 |
0.431 |
|
| 1983 |
Roush WR, Brown RJ, DiMare M. Total synthesis of carbohydrates. 2. Regiochemical control of nucleophilic ring opening of acylated 2,3-epoxy alcohols The Journal of Organic Chemistry. 48: 5083-5093. DOI: 10.1002/Chin.198428086 |
0.339 |
|
| 1983 |
ROUSH WR, HARRIS DJ, LESUR BM. ChemInform Abstract: STUDIES ON THE SYNTHESIS OF OLIVIN: DIASTEREOSELECTIVE SYNTHESIS OF A FUNCTIONALIZED D-FUCOSE DERIVATIVE Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198339356 |
0.727 |
|
| 1983 |
ROUSH WR, LESUR BM. ChemInform Abstract: STEREOCHEMISTRY OF VINYL CUPRATE ADDITIONS TO CARBOHYDRATE-DERIVED ENONES AND α,β-UNSATURATED ESTERS Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198339111 |
0.683 |
|
| 1983 |
ROUSH WR, BLIZZARD TA. ChemInform Abstract: SYNTHESIS OF VERRUCARIN J Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198331263 |
0.313 |
|
| 1983 |
ROUSH WR, ADAM MA, PESECKIS SM. ChemInform Abstract: REGIOSELECTIVITY OF THE REACTIONS OF TRIALKYLALUMINUM REAGENTS WITH 2,3-EPOXY ALCOHOLS: APPLICATION TO THE SYNTHESIS OF α-CHIRAL ALDEHYDES Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198329230 |
0.32 |
|
| 1983 |
ROUSH WR, D'AMBRA TE. ChemInform Abstract: TOTAL SYNTHESIS OF (.+-.)-VERRUCAROL Chemischer Informationsdienst. 14. DOI: 10.1002/Chin.198322355 |
0.444 |
|
| 1982 |
Roush WR, Brown RJ. Total synthesis of carbohydrates: stereoselective syntheses of 2,6-dideoxy-D-arabino-hexose and 2,6-dideoxy-D-ribo-hexose The Journal of Organic Chemistry. 47: 1371-1373. DOI: 10.1021/Jo00346A050 |
0.321 |
|
| 1982 |
Roush WR, Gillis HR. Further stereochemical aspects of intramolecular Diels-Alder reactions in the undeca-2,8,10-trienoate ester series The Journal of Organic Chemistry. 47: 4825-4829. DOI: 10.1021/Jo00146A001 |
0.456 |
|
| 1982 |
Hall SE, Roush WR. Synthesis of the bottom half of chlorothricolide The Journal of Organic Chemistry. 47: 4611-4621. DOI: 10.1021/Jo00145A002 |
0.447 |
|
| 1982 |
Roush WR, Gillis HR, Ko AI. Stereochemical aspects of the intramolecular Diels-Alder reactions of deca-2,7,9-trienoate esters. 3. Thermal, Lewis acid catalyzed, and asymmetric cyclizations Journal of the American Chemical Society. 104: 2269-2283. DOI: 10.1021/Ja00372A027 |
0.431 |
|
| 1982 |
Roush WR, Spada AP. Enantio- and stereoselective syntheses of the dihydroxyoctadienoic acid framents of the roridins and trichoverrins Tetrahedron Letters. 23: 3773-3776. DOI: 10.1016/S0040-4039(00)87703-5 |
0.348 |
|
| 1982 |
Roush WR, Blizzard TA, Basha FZ. Methodology for the synthesis of the acyclic portions of verrucarins A and J Tetrahedron Letters. 23: 2331-2334. DOI: 10.1016/S0040-4039(00)87334-7 |
0.677 |
|
| 1982 |
ROUSH WR, BLIZZARD TA, BASHA FZ. ChemInform Abstract: METHODOLOGY FOR THE SYNTHESIS OF THE ACYCLIC PORTIONS OF VERRUCARINS A AND J Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198243273 |
0.673 |
|
| 1982 |
ROUSH WR, GILLIS HR, KO AI. ChemInform Abstract: STEREOCHEMICAL ASPECTS OF THE INTRAMOLECULAR DIELS-ALDER REACTIONS OF DECA-2,7,9-TRIENOATE ESTERS. 3. THERMAL, LEWIS ACID CATALYZED, AND ASYMMETRIC C CYCLIZATIONS Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198233092 |
0.36 |
|
| 1982 |
ROUSH WR, PESECKIS SM. ChemInform Abstract: INTRAMOLECULAR DIELS-ALDER REACTIONS: THE ANGULARLY METHYLATED TRANS-PERHYDROINDAN RING SYSTEM Chemischer Informationsdienst. 13. DOI: 10.1002/chin.198207163 |
0.302 |
|
| 1981 |
Roush WR, D'Ambra TE. Synthesis of a bicyclic precursor to verrucarol: application of a trimethylsilyl-controlled Diels-Alder reaction and Wagner-Meerwein rearrangement sequence The Journal of Organic Chemistry. 46: 5045-5047. DOI: 10.1021/Jo00337A059 |
0.429 |
|
| 1981 |
Roush WR, Myers AG. Antibiotic X-14547A: total synthesis of the right-hand half The Journal of Organic Chemistry. 46: 1509-1511. DOI: 10.1021/Jo00320A060 |
0.512 |
|
| 1981 |
Roush WR, Peseckis SM. Intramolecular Diels-Alder reactions: the angularly methylated trans-perhydroindan ring system Journal of the American Chemical Society. 103: 6696-6704. DOI: 10.1021/Ja00412A027 |
0.408 |
|
| 1981 |
Roush WR, Hall SE. Studies on the total synthesis of chlorothricolide: stereochemical aspects of the intramolecular Diels-Alder reactions of methyl undeca-2,8,10-trienoates Journal of the American Chemical Society. 103: 5200-5211. DOI: 10.1021/Ja00407A042 |
0.48 |
|
| 1981 |
ROUSH WR, HALL SE. ChemInform Abstract: STUDIES ON THE TOTAL SYNTHESIS OF CHLOROTHRICOLIDE: STEREOCHEMICAL ASPECTS OF THE INTRAMOLECULAR DIELS-ALDER REACTIONS OF METHYL UNDECA-2,8,10-TRIENOATES Chemischer Informationsdienst. 12. DOI: 10.1002/chin.198149169 |
0.383 |
|
| 1981 |
ROUSH WR, MYERS AG. ChemInform Abstract: ANTIBIOTIC X-14547A: TOTAL SYNTHESIS OF THE RIGHT-HAND HALF Chemischer Informationsdienst. 12. DOI: 10.1002/chin.198133345 |
0.463 |
|
| 1980 |
Roush WR, Gillis HR. Improved synthesis of the perhydroindenone precursor of dendrobine The Journal of Organic Chemistry. 45: 4283-4287. DOI: 10.1021/Jo01310A006 |
0.405 |
|
| 1980 |
Roush WR, Gillis HR. Stereochemical aspects of the intramolecular Diels-Alder reactions of methyl deca-2,7,9-trienoates. 2. Lewis acid catalysis The Journal of Organic Chemistry. 45: 4267-4268. DOI: 10.1021/Jo01309A055 |
0.417 |
|
| 1980 |
Roush WR, Ko AI, Gillis HR. Stereochemical aspects of the intramolecular Diels-Alder reactions of methyl deca-2,7,9-trienoates. 1. Thermal cyclizations The Journal of Organic Chemistry. 45: 4264-4267. DOI: 10.1021/Jo01309A054 |
0.392 |
|
| 1980 |
Roush WR, D'Ambra TE. Total synthesis of verrucarol: a stereoselective synthesis of 13,14-dinor-15-hydroxytrichothec-9-ene The Journal of Organic Chemistry. 45: 3927-3929. DOI: 10.1021/Jo01307A045 |
0.469 |
|
| 1980 |
Roush WR. Total synthesis of (.+-.)-dendrobine Journal of the American Chemical Society. 102: 1390-1404. DOI: 10.1021/ja00524a027 |
0.326 |
|
| 1979 |
Roush WR. Stereochemical aspects of the intramolecular Diels-Alder reactions of methyl (E,E,E)- and (Z,E,E)-6-alkoxy-11-methyldodeca-2,7,9-trienoate The Journal of Organic Chemistry. 44: 4008-4010. DOI: 10.1021/Jo01336A067 |
0.302 |
|
| 1978 |
Roush WR. Total synthesis of (.+-.)-dendrobine Journal of the American Chemical Society. 100: 3599-3601. DOI: 10.1021/Ja00479A053 |
0.438 |
|
| 1978 |
ROUSH WR. ChemInform Abstract: TOTAL SYNTHESIS OF (.+-.)-DENDROBINE Chemischer Informationsdienst. 9. DOI: 10.1002/chin.197836323 |
0.334 |
|
| Show low-probability matches. |
