☰

Thomas L. Mindt, Ph.D. - Publications

Affiliations: 
2003 Brown University, Providence, RI 
Area:
Natural product total synthesis
Tree Info Similar researchers PubMed Report error

34 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Rečnik LM, Kandioller W, Mindt TL. 1,4-Disubstituted 1,2,3-Triazoles as Amide Bond Surrogates for the Stabilisation of Linear Peptides with Biological Activity. Molecules (Basel, Switzerland). 25. PMID 32781656 DOI: 10.3390/Molecules25163576  0.358
2020 Vrettos EI, Valverde IE, Mascarin A, Pallier PN, Cerofolini L, Fragai M, Parigi G, Hirmiz B, Bekas N, Grob NM, Stylos EΚ, Shaye H, Del Borgo M, Aguilar MI, Magnani F, ... ... Mindt TL, et al. Single Peptide Backbone Surrogate Mutations to Regulate Angiotensin GPCR Subtype Selectivity. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 32691857 DOI: 10.1002/Chem.202000924  0.326
2020 Giammei C, Balber T, Benčurová K, Cardinale J, Berroterán-Infante N, Brandt M, Jouini N, Hacker M, Mitterhauser M, Mindt TL. Sorbitol as a Polar Pharmacological Modifier to Enhance the Hydrophilicity of Tc-Tricarbonyl-Based Radiopharmaceuticals. Molecules (Basel, Switzerland). 25. PMID 32527027 DOI: 10.3390/Molecules25112680  0.379
2020 Grob NM, Behe M, von Guggenberg E, Schibli R, Mindt TL. Corrigendum concerning "Methoxinine-An alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates". Journal of Peptide Science : An Official Publication of the European Peptide Society. 26: e3242. PMID 32026540 DOI: 10.1002/Psc.3242  0.315
2017 Briand M, Aulsebrook ML, Mindt TL, Gasser G. A solid phase-assisted approach for the facile synthesis of a highly water-soluble zirconium-89 chelator for radiopharmaceutical development. Dalton Transactions (Cambridge, England : 2003). PMID 29130082 DOI: 10.1039/C7Dt03639F  0.35
2017 Maina T, Kaloudi A, Valverde IE, Mindt TL, Nock BA. Amide-to-triazole switch vs. in vivo NEP-inhibition approaches to promote radiopeptide targeting of GRPR-positive tumors. Nuclear Medicine and Biology. 52: 57-62. PMID 28636973 DOI: 10.1016/J.Nucmedbio.2017.06.001  0.302
2017 Grob NM, Behe M, von Guggenberg E, Schibli R, Mindt TL. Methoxinine - an alternative stable amino acid substitute for oxidation-sensitive methionine in radiolabelled peptide conjugates. Journal of Peptide Science : An Official Publication of the European Peptide Society. PMID 28054429 DOI: 10.1002/Psc.2948  0.343
2016 Römhild K, Fischer CA, Mindt TL. Glycated (99m) Tc-Tricarbonyl-Labeled Peptide Conjugates for Tumor Targeting by "Click-to-Chelate". Chemmedchem. PMID 27902882 DOI: 10.1002/Cmdc.201600485  0.36
2016 Valverde IE, Vomstein S, Mindt TL. Towards the Optimization of Bombesin-Based Radiotracers for Tumor Targeting. Journal of Medicinal Chemistry. PMID 27054526 DOI: 10.1021/Acs.Jmedchem.6B00025  0.325
2016 Chiotellis A, Sladojevich F, Mu L, Müller Herde A, Valverde IE, Tolmachev V, Schibli R, Ametamey SM, Mindt TL. Novel chemoselective (18)F-radiolabeling of thiol-containing biomolecules under mild aqueous conditions. Chemical Communications (Cambridge, England). PMID 27043419 DOI: 10.1039/C6Cc01982J  0.33
2016 Mascarin A, Valverde IE, Mindt TL. Radiolabeled analogs of neurotensin (8–13) containing multiple 1,2,3-triazoles as stable amide bond mimics in the backbone Medchemcomm. 7: 1640-1646. DOI: 10.1039/C6Md00208K  0.327
2015 Mascarin A, Valverde IE, Mindt TL. Structure-Activity Relationship Studies of Amino Acid Substitutions in Radiolabeled Neurotensin Conjugates. Chemmedchem. PMID 26593062 DOI: 10.1002/Cmdc.201500468  0.367
2015 Mascarin A, Valverde IE, Vomstein S, Mindt TL. 1,2,3-Triazole Stabilized Neurotensin-Based Radiopeptidomimetics for Improved Tumor Targeting. Bioconjugate Chemistry. 26: 2143-52. PMID 26347939 DOI: 10.1021/Acs.Bioconjchem.5B00444  0.378
2015 Valverde IE, Vomstein S, Fischer CA, Mascarin A, Mindt TL. Probing the Backbone Function of Tumor Targeting Peptides by an Amide-to-Triazole Substitution Strategy. Journal of Medicinal Chemistry. 58: 7475-84. PMID 26309061 DOI: 10.1021/Acs.Jmedchem.5B00994  0.361
2015 Parker KA, Mindt TL. Regioselective 1,2-addition of organometallic reagents to unprotected juglones Tetrahedron Letters. 56: 3500-3502. DOI: 10.1016/J.Tetlet.2014.12.108  0.527
2014 Fischer CA, Vomstein S, Mindt TL. A bombesin-shepherdin radioconjugate designed for combined extra- and intracellular targeting. Pharmaceuticals (Basel, Switzerland). 7: 662-75. PMID 24871806 DOI: 10.3390/Ph7060662  0.328
2014 Valverde IE, Huxol E, Mindt TL. Radiolabeled antagonistic bombesin peptidomimetics for tumor targeting. Journal of Labelled Compounds & Radiopharmaceuticals. 57: 275-8. PMID 24327435 DOI: 10.1002/Jlcr.3162  0.354
2013 Valverde IE, Mindt TL. 1,2,3-Triazoles as amide-bond surrogates in peptidomimetics. Chimia. 67: 262-6. PMID 23967702 DOI: 10.2533/Chimia.2013.262  0.366
2013 Kluba CA, Mindt TL. Click-to-Chelate: development of technetium and rhenium-tricarbonyl labeled radiopharmaceuticals. Molecules (Basel, Switzerland). 18: 3206-26. PMID 23481882 DOI: 10.3390/Molecules18033206  0.373
2012 Kluba CA, Bauman A, Valverde IE, Vomstein S, Mindt TL. Dual-targeting conjugates designed to improve the efficacy of radiolabeled peptides. Organic & Biomolecular Chemistry. 10: 7594-602. PMID 22898743 DOI: 10.1039/C2Ob26127H  0.353
2011 Parker KA, Mindt TL. Convergent Synthesis of 2H-Chromenes - a Formal [3+3] Cycloaddition by a One-pot, Three-Step Cascade. Tetrahedron. 67: 9779-9786. PMID 22259219 DOI: 10.1016/J.Tet.2011.09.068  0.615
2011 Arrowsmith RL, Waghorn PA, Jones MW, Bauman A, Brayshaw SK, Hu Z, Kociok-Köhn G, Mindt TL, Tyrrell RM, Botchway SW, Dilworth JR, Pascu SI. Fluorescent gallium and indium bis(thiosemicarbazonates) and their radiolabelled analogues: synthesis, structures and cellular confocal fluorescence imaging investigations. Dalton Transactions (Cambridge, England : 2003). 40: 6238-52. PMID 21594287 DOI: 10.1039/C1Dt10126A  0.309
2010 Mindt TL, Struthers H, Spingler B, Brans L, Tourwé D, García-Garayoa E, Schibli R. Molecular assembly of multifunctional 99mTc radiopharmaceuticals using "clickable" amino acid derivatives Chemmedchem. 5: 2026-2038. PMID 20922747 DOI: 10.1002/Cmdc.201000342  0.393
2010 Struthers H, Mindt TL, Schibli R. Metal chelating systems synthesized using the copper(I) catalyzed azide-alkyne cycloaddition. Dalton Transactions (Cambridge, England : 2003). 39: 675-96. PMID 20066208 DOI: 10.1039/B912608B  0.321
2009 Mindt TL, Müller C, Stuker F, Salazar JF, Hohn A, Mueggler T, Rudin M, Schibli R. A "click chemistry" approach to the efficient synthesis of multiple imaging probes derived from a single precursor. Bioconjugate Chemistry. 20: 1940-9. PMID 19803478 DOI: 10.1021/Bc900276B  0.369
2009 Mindt TL, Schweinsberg C, Brans L, Hagenbach A, Abram U, Tourwé D, Garcia-Garayoa E, Schibli R. A click approach to structurally diverse conjugates containing a central di-1,2,3-triazole metal chelate. Chemmedchem. 4: 529-39. PMID 19235821 DOI: 10.1002/Cmdc.200800418  0.372
2008 Ross TL, Honer M, Lam PYH, Mindt TL, Groehn V, Schibli R, Schubiger PA, Ametamey SM. Fluorine-18 click radiosynthesis and preclinical evaluation of a new 18F-labeled folic acid derivative Bioconjugate Chemistry. 19: 2462-2470. PMID 19053298 DOI: 10.1021/Bc800356R  0.319
2008 Mindt TL, Müller C, Melis M, de Jong M, Schibli R. "Click-to-chelate": in vitro and in vivo comparison of a 99mTc(CO)3-labeled N(tau)-histidine folate derivative with its isostructural, clicked 1,2,3-triazole analogue. Bioconjugate Chemistry. 19: 1689-95. PMID 18646835 DOI: 10.1021/Bc800183R  0.371
2008 Struthers H, Spingler B, Mindt TL, Schibli R. "Click-to-chelate": design and incorporation of triazole-containing metal-chelating systems into biomolecules of diagnostic and therapeutic interest. Chemistry (Weinheim An Der Bergstrasse, Germany). 14: 6173-6183. PMID 18494020 DOI: 10.1002/Chem.200702024  0.347
2007 Mindt TL, Schibli R. Cu(I)-catalyzed intramolecular cyclization of alkynoic acids in aqueous media: a "click side reaction". The Journal of Organic Chemistry. 72: 10247-50. PMID 18044929 DOI: 10.1021/Jo702030E  0.329
2007 Mindt T, Struthers H, Garcia-Garayoa E, Desbouis D, Schibli R. Strategies for the development of novel tumor targeting technetium and rhenium radiopharmaceuticals Chimia. 61: 725-731. DOI: 10.2533/Chimia.2007.725  0.329
2006 Parker KA, Mindt TL, Koh YH. TESOTf-induced rearrangement of quinols. Efficient construction of the fully functionalized carbon skeleton of the griseusins by a divergent-reconvergent approach. Organic Letters. 8: 1759-62. PMID 16623544 DOI: 10.1021/Ol060206Q  0.524
2002 Parker KA, Mindt TL. Heterocycle annulation of enolizable vinyl quinone imides. Dihydroquinolines and quinolines from thermal 6pi-electrocyclizations and indoles from photochemical cyclizations. Organic Letters. 4: 4265-8. PMID 12443074 DOI: 10.1021/Ol026849X  0.532
2001 Parker KA, Mindt TL. Electrocyclic ring closure of the enols of vinyl quinones. A 2H-chromene synthesis. Organic Letters. 3: 3875-8. PMID 11720558 DOI: 10.1021/Ol0167199  0.541
Show low-probability matches.