| Year |
Citation |
Score |
| 2021 |
Han J, Andreu V, Langreck C, Pekarskaya EA, Grinnell SG, Allain F, Magalong V, Pintar J, Kieffer BL, Harris AZ, Javitch JA, Hen R, Nautiyal KM. Mu opioid receptors on hippocampal GABAergic interneurons are critical for the antidepressant effects of tianeptine. Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology. PMID 34593976 DOI: 10.1038/s41386-021-01192-2 |
0.796 |
|
| 2021 |
Uprety R, Che T, Zaidi SA, Grinnell SG, Varga BR, Faouzi A, Slocum ST, Allaoa A, Varadi A, Nelson M, Bernhard SM, Kulko E, LeRouzic V, Eans SO, Simons CA, et al. Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site. Elife. 10. PMID 33555255 DOI: 10.7554/eLife.56519 |
0.859 |
|
| 2020 |
Grinnell SG, Uprety R, Varadi A, Subrath J, Hunkele A, Pan YX, Pasternak GW, Majumdar S. Synthesis and Characterization of Azido Aryl Analogs of IBNtxA for Radio-Photoaffinity Labeling Opioid Receptors in Cell Lines and in Mouse Brain. Cellular and Molecular Neurobiology. PMID 32424771 DOI: 10.1007/S10571-020-00867-6 |
0.865 |
|
| 2019 |
Kruegel AC, Uprety R, Grinnell SG, Langreck C, Pekarskaya EA, Le Rouzic V, Ansonoff M, Gassaway MM, Pintar JE, Pasternak GW, Javitch JA, Majumdar S, Sames D. 7-Hydroxymitragynine Is an Active Metabolite of Mitragynine and a Key Mediator of Its Analgesic Effects. Acs Central Science. 5: 992-1001. PMID 31263758 DOI: 10.1021/Acscentsci.9B00141 |
0.788 |
|
| 2018 |
Marcott PF, Gong S, Donthamsetti P, Grinnell SG, Nelson MN, Newman AH, Birnbaumer L, Martemyanov KA, Javitch JA, Ford CP. Regional Heterogeneity of D2-Receptor Signaling in the Dorsal Striatum and Nucleus Accumbens. Neuron. PMID 29656874 DOI: 10.1016/J.Neuron.2018.03.038 |
0.534 |
|
| 2017 |
Samuels BA, Nautiyal KM, Kruegel AC, Levinstein MR, Magalong VM, Gassaway MM, Grinnell SG, Han J, Ansonoff MA, Pintar JE, Javitch JA, Sames D, Hen R. The Behavioral Effects of the Antidepressant Tianeptine Require the Mu Opioid Receptor. Neuropsychopharmacology : Official Publication of the American College of Neuropsychopharmacology. PMID 28303899 DOI: 10.1038/Npp.2017.60 |
0.751 |
|
| 2016 |
Váradi A, Marrone GF, Palmer TC, Narayan A, Szabó MR, Le Rouzic V, Grinnell SG, Subrath JJ, Warner E, Kalra S, Hunkele A, Pagirsky J, Eans SO, Medina JM, Xu J, et al. Mitragynine/corynantheidine pseudoindoxyls as opioid analgesics with mu agonism and delta antagonism which do not recruit β-arrestin-2. Journal of Medicinal Chemistry. PMID 27556704 DOI: 10.1021/Acs.Jmedchem.6B00748 |
0.86 |
|
| 2016 |
Grinnell SG, Ansonoff M, Marrone GF, Lu Z, Narayan A, Xu J, Rossi G, Majumdar S, Pan YX, Bassoni DL, Pintar J, Pasternak G. Mediation of buprenorphine analgesia by a combination of traditional and truncated mu opioid receptor splice variants. Synapse (New York, N.Y.). PMID 27223691 DOI: 10.1002/Syn.21914 |
0.805 |
|
| 2016 |
Marrone GF, Grinnell SG, Lu Z, Rossi GC, Le Rouzic V, Xu J, Majumdar S, Pan YX, Pasternak GW. Truncated mu opioid GPCR variant involvement in opioid-dependent and opioid-independent pain modulatory systems within the CNS. Proceedings of the National Academy of Sciences of the United States of America. PMID 26976581 DOI: 10.1073/Pnas.1523894113 |
0.817 |
|
| 2015 |
Pickett JE, Váradi A, Palmer TC, Grinnell SG, Schrock JM, Pasternak GW, Karimov RR, Majumdar S. Mild, Pd-catalyzed stannylation of radioiodination targets. Bioorganic & Medicinal Chemistry Letters. 25: 1761-4. PMID 25777268 DOI: 10.1016/J.Bmcl.2015.02.055 |
0.668 |
|
| 2014 |
Grinnell SG, Majumdar S, Narayan A, Le Rouzic V, Ansonoff M, Pintar JE, Pasternak GW. Pharmacologic characterization in the rat of a potent analgesic lacking respiratory depression, IBNtxA. The Journal of Pharmacology and Experimental Therapeutics. 350: 710-8. PMID 24970924 DOI: 10.1124/Jpet.114.213199 |
0.807 |
|
| 2013 |
Váradi A, Hosztafi S, Le Rouzic V, Tóth G, Urai Á, Noszál B, Pasternak GW, Grinnell SG, Majumdar S. Novel 6β-acylaminomorphinans with analgesic activity. European Journal of Medicinal Chemistry. 69: 786-9. PMID 24103580 DOI: 10.1016/J.Ejmech.2013.09.031 |
0.85 |
|
| 2013 |
Pickett JE, Nagakura K, Pasternak AR, Grinnell SG, Majumdar S, Lewis JS, Pasternak GW. Sandmeyer reaction repurposed for the site-selective, non-oxidizing radioiodination of fully-deprotected peptides: studies on the endogenous opioid peptide α-neoendorphin. Bioorganic & Medicinal Chemistry Letters. 23: 4347-50. PMID 23796454 DOI: 10.1016/J.Bmcl.2013.05.090 |
0.802 |
|
| 2012 |
Majumdar S, Subrath J, Le Rouzic V, Polikar L, Burgman M, Nagakura K, Ocampo J, Haselton N, Pasternak AR, Grinnell S, Pan YX, Pasternak GW. Synthesis and evaluation of aryl-naloxamide opiate analgesics targeting truncated exon 11-associated μ opioid receptor (MOR-1) splice variants. Journal of Medicinal Chemistry. 55: 6352-62. PMID 22734622 DOI: 10.1021/Jm300305C |
0.845 |
|
| 2011 |
Majumdar S, Grinnell S, Le Rouzic V, Burgman M, Polikar L, Ansonoff M, Pintar J, Pan YX, Pasternak GW. Truncated G protein-coupled mu opioid receptor MOR-1 splice variants are targets for highly potent opioid analgesics lacking side effects. Proceedings of the National Academy of Sciences of the United States of America. 108: 19778-83. PMID 22106286 DOI: 10.1073/Pnas.1115231108 |
0.853 |
|
| 2011 |
Majumdar S, Burgman M, Haselton N, Grinnell S, Ocampo J, Pasternak AR, Pasternak GW. Generation of novel radiolabeled opiates through site-selective iodination. Bioorganic & Medicinal Chemistry Letters. 21: 4001-4. PMID 21621410 DOI: 10.1016/J.Bmcl.2011.05.008 |
0.821 |
|
| 2011 |
Pan YX, Grinnell S, Pasternak GW. Alternative Pre-mRNA splicing of G protein-coupled receptors Neuromethods. 60: 19-34. DOI: 10.1007/978-1-61779-179-6_2 |
0.583 |
|
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