Year |
Citation |
Score |
2021 |
Biswas S, Van Steijvoort BF, Waeterschoot M, Bheemireddy NR, Evano G, Maes BU. Expedient synthesis of bridged bicyclic nitrogen scaffolds via orthogonal tandem catalysis. Angewandte Chemie (International Ed. in English). PMID 34143924 DOI: 10.1002/anie.202106716 |
0.34 |
|
2019 |
Bomon J, Van Den Broeck E, Bal M, Liao Y, Sergeyev S, Van Speybroeck V, Sels BF, Maes BU. Brønsted Acid Catalyzed Tandem Defunctionalization of Biorenewable Ferulic acid and Derivates into Bio-catechol. Angewandte Chemie (International Ed. in English). PMID 31765514 DOI: 10.1002/Anie.201913023 |
0.34 |
|
2019 |
Dobi Z, Reddy NB, Renders E, Van Raemdonck L, Mensch C, De Smet G, Chen C, Bheeter C, Sergeyev S, Herrebout WA, Maes BU. Carbamate Synthesis Via a Shelf Stable and Renewable C1 Reactant. Chemsuschem. PMID 30921504 DOI: 10.1002/Cssc.201900406 |
0.32 |
|
2018 |
Ronson TO, Renders E, Van Steijvoort BF, Wang X, Wybon CCD, Prokopcová H, Meerpoel L, Maes BU. Ruthenium-Catalyzed Reductive Arylation of N-(2-Pyridinyl)amides with Isopropanol and Arylboronate Esters. Angewandte Chemie (International Ed. in English). PMID 30380163 DOI: 10.1002/Anie.201810947 |
0.435 |
|
2016 |
Morel B, Franck P, Bidange J, Sergeyev S, Smith D, Moseley J, Maes BU. Concise Xanthine Synthesis via a Double Amidination Reaction of a 6-Chlorouracil with Amidines using Base Metal Catalysis. Chemsuschem. PMID 27899009 DOI: 10.1002/Cssc.201601483 |
0.461 |
|
2016 |
Zhu YP, Sergeyev S, Franck P, Orru RV, Maes BU. Amine Activation: Synthesis of N-(Hetero)arylamides from Isothioureas and Carboxylic Acids. Organic Letters. PMID 27570902 DOI: 10.1021/Acs.Orglett.6B02247 |
0.403 |
|
2016 |
Mampuys P, Zhu Y, Sergeyev S, Ruijter E, Orru RV, Van Doorslaer S, Maes BU. Iodide-Catalyzed Synthesis of Secondary Thiocarbamates from Isocyanides and Thiosulfonates. Organic Letters. PMID 27276236 DOI: 10.1021/Acs.Orglett.6B01023 |
0.446 |
|
2016 |
Wu XF, Zhu F, Li Y, Wang Z, Orru RV, Maes BU. Palladium-Catalyzed Construction of Amidines from Arylboronic acids under Oxidative Conditions. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 27061735 DOI: 10.1002/Chem.201601262 |
0.444 |
|
2016 |
Sterckx H, De Houwer J, Mensch C, Herrebout W, Tehrani KA, Maes BU. Base metal-catalyzed benzylic oxidation of (aryl)(heteroaryl)methanes with molecular oxygen. Beilstein Journal of Organic Chemistry. 12: 144-53. PMID 26877817 DOI: 10.3762/Bjoc.12.16 |
0.679 |
|
2016 |
Sergeyev S, Yadav AK, Franck P, Michiels J, Lewi P, Heeres J, Vanham G, Ariën KK, Vande Velde CM, De Winter H, Maes BU. 2,6-Di(arylamino)-3-fluoropyridine Derivatives as HIV Non-Nucleoside Reverse Transcriptase Inhibitors. Journal of Medicinal Chemistry. 59: 1854-68. PMID 26785139 DOI: 10.1021/Acs.Jmedchem.5B01336 |
0.329 |
|
2015 |
Hervé M, Lefèvre G, Mitchell EA, Maes BU, Jutand A. On the Triple Role of Fluoride Ions in Palladium-Catalyzed Stille Reactions. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26548772 DOI: 10.1002/Chem.201503309 |
0.513 |
|
2015 |
Maes BU, Verbeeck S, Verhelst T, Ekomié A, von Wolff N, Lefèvre G, Mitchell EA, Jutand A. Oxidative Addition of Haloheteroarenes to Palladium(0): Concerted versus SN Ar-Type Mechanism. Chemistry (Weinheim An Der Bergstrasse, Germany). 21: 7858-65. PMID 25858175 DOI: 10.1002/Chem.201406210 |
0.537 |
|
2014 |
Mampuys P, Zhu Y, Vlaar T, Ruijter E, Orru RV, Maes BU. Sustainable three-component synthesis of isothioureas from isocyanides, thiosulfonates, and amines. Angewandte Chemie (International Ed. in English). 53: 12849-54. PMID 25223494 DOI: 10.1002/Anie.201406717 |
0.405 |
|
2014 |
Verbeeck S, Yadav AK, Maes BU, Augustyns K, Van Der Veken P, Cos P, Maes L, Pieters L. Antiprotozoal activity of synthetic amino substituted 1-methyl-1 H-alpha-carbolines. Die Pharmazie. 69: 83-5. PMID 24640594 DOI: 10.1691/Ph.2014.3748 |
0.321 |
|
2013 |
Vlaar T, Orru RV, Maes BU, Ruijter E. Palladium-catalyzed synthesis of 2-aminobenzoxazinones by aerobic oxidative coupling of anthranilic acids and isocyanides. The Journal of Organic Chemistry. 78: 10469-75. PMID 24063265 DOI: 10.1021/Jo401924H |
0.446 |
|
2013 |
Smout V, Peschiulli A, Verbeeck S, Mitchell EA, Herrebout W, Bultinck P, Vande Velde CM, Berthelot D, Meerpoel L, Maes BU. Removal of the pyridine directing group from α-substituted N-(pyridin-2-yl)piperidines obtained via directed Ru-catalyzed sp3 C-H functionalization. The Journal of Organic Chemistry. 78: 9803-14. PMID 24007399 DOI: 10.1021/Jo401521Y |
0.424 |
|
2013 |
Peschiulli A, Smout V, Storr TE, Mitchell EA, Eliáš Z, Herrebout W, Berthelot D, Meerpoel L, Maes BU. Ruthenium-catalyzed α-(hetero)arylation of saturated cyclic amines: reaction scope and mechanism. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 10378-87. PMID 23780756 DOI: 10.1002/Chem.201204438 |
0.426 |
|
2013 |
Vlaar T, Mampuys P, Helliwell M, Maes BU, Orru RV, Ruijter E. Multicomponent synthesis of 4-aminophthalazin-1(2H)-ones by palladium-catalyzed isocyanide insertion. The Journal of Organic Chemistry. 78: 6735-45. PMID 23768066 DOI: 10.1021/Jo401131P |
0.436 |
|
2013 |
Vlaar T, Ruijter E, Maes BU, Orru RV. Palladium-catalyzed migratory insertion of isocyanides: an emerging platform in cross-coupling chemistry. Angewandte Chemie (International Ed. in English). 52: 7084-97. PMID 23754476 DOI: 10.1002/Anie.201300942 |
0.433 |
|
2013 |
Maes J, Rauws TR, Maes BU. Synthesis of C8-N9 annulated purines by iron-catalyzed C-H amination. Chemistry (Weinheim An Der Bergstrasse, Germany). 19: 9137-41. PMID 23733404 DOI: 10.1002/Chem.201301248 |
0.356 |
|
2013 |
Yadav AK, Verbeeck S, Hostyn S, Franck P, Sergeyev S, Maes BU. "Base effect" in the auto-tandem palladium-catalyzed synthesis of amino-substituted 1-methyl-1H-α-carbolines. Organic Letters. 15: 1060-3. PMID 23410177 DOI: 10.1021/Ol400064R |
0.477 |
|
2012 |
Vlaar T, Cioc RC, Mampuys P, Maes BU, Orru RV, Ruijter E. Sustainable synthesis of diverse privileged heterocycles by palladium-catalyzed aerobic oxidative isocyanide insertion. Angewandte Chemie (International Ed. in English). 51: 13058-61. PMID 23161862 DOI: 10.1002/Anie.201207410 |
0.405 |
|
2012 |
Mitchell EA, Peschiulli A, Lefevre N, Meerpoel L, Maes BU. Direct α-functionalization of saturated cyclic amines. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 10092-142. PMID 22829434 DOI: 10.1002/Chem.201201539 |
0.323 |
|
2012 |
Bergman SD, Storr TE, Prokopcová H, Aelvoet K, Diels G, Meerpoel L, Maes BU. The role of the alcohol and carboxylic acid in directed ruthenium-catalyzed C(sp3)-H α-alkylation of cyclic amines. Chemistry (Weinheim An Der Bergstrasse, Germany). 18: 10393-8. PMID 22786664 DOI: 10.1002/Chem.201201072 |
0.429 |
|
2012 |
De Houwer J, Abbaspour Tehrani K, Maes BU. Synthesis of aryl(di)azinyl ketones through copper- and iron-catalyzed oxidation of the methylene group of aryl(di)azinylmethanes. Angewandte Chemie (International Ed. in English). 51: 2745-8. PMID 22290611 DOI: 10.1002/Anie.201108540 |
0.428 |
|
2012 |
Rauws TR, Maes BU. Transition metal-catalyzed N-arylations of amidines and guanidines. Chemical Society Reviews. 41: 2463-97. PMID 22222274 DOI: 10.1039/C1Cs15236J |
0.331 |
|
2012 |
Smeulders G, Meynen V, Houthoofd K, Mullens S, Martens JA, Maes BU, Cool P. Is their potential for post-synthetic brominating reactions on benzene bridged PMOs? Microporous and Mesoporous Materials. 164: 49-55. DOI: 10.1016/J.Micromeso.2012.06.033 |
0.378 |
|
2011 |
Van Baelen G, Kuijer S, Rý?ek L, Sergeyev S, Janssen E, de Kanter FJ, Maes BU, Ruijter E, Orru RV. Synthesis of 4-aminoquinazolines by palladium-catalyzed intramolecular imidoylation of N-(2-bromoaryl)amidines. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 15039-44. PMID 22125085 DOI: 10.1002/Chem.201102468 |
0.444 |
|
2011 |
Vlaar T, Ruijter E, Znabet A, Janssen E, de Kanter FJ, Maes BU, Orru RV. Palladium-catalyzed synthesis of 4-aminophthalazin-1(2H)-ones by isocyanide insertion. Organic Letters. 13: 6496-9. PMID 22085248 DOI: 10.1021/Ol202784D |
0.429 |
|
2011 |
Verhelst T, Liu Z, Maes J, Maes BU. Synthesis of (hetero)arylated pyridazin-3(2H)-ones via Negishi reaction involving zincated pyridazin-3(2H)-ones. The Journal of Organic Chemistry. 76: 9648-59. PMID 22017314 DOI: 10.1021/Jo201587J |
0.402 |
|
2011 |
Verhelst T, Maes J, Liu Z, Sergeyev S, Maes BU. Synthesis of functionalized pyridazin-3(2H)-ones via selective bromine-magnesium exchange and lactam directed ortho C-H magnesiation. The Journal of Organic Chemistry. 76: 6670-7. PMID 21732644 DOI: 10.1021/Jo201009M |
0.358 |
|
2011 |
Masters KS, Rauws TR, Yadav AK, Herrebout WA, Van der Veken B, Maes BU. On the importance of an acid additive in the synthesis of pyrido[1,2-a]benzimidazoles by direct copper-catalyzed amination. Chemistry (Weinheim An Der Bergstrasse, Germany). 17: 6315-20. PMID 21509841 DOI: 10.1002/Chem.201100574 |
0.435 |
|
2011 |
Verhelst T, Verbeeck S, Ryabtsova O, Depraetere S, Maes BU. Synthesis of functionalized pyridazin-3(2H)-ones via nucleophilic substitution of hydrogen (SNH). Organic Letters. 13: 272-5. PMID 21138319 DOI: 10.1021/Ol102703W |
0.424 |
|
2010 |
Prokopcová H, Bergman SD, Aelvoet K, Smout V, Herrebout W, Van der Veken B, Meerpoel L, Maes BU. C-2 arylation of piperidines through directed transition-metal-catalyzed sp3 C-H activation. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 13063-7. PMID 20981669 DOI: 10.1002/Chem.201001887 |
0.338 |
|
2010 |
Verbeeck S, Meyers C, Franck P, Jutand A, Maes BU. Dual effect of halides in the Stille reaction: in situ halide metathesis and catalyst stabilization. Chemistry (Weinheim An Der Bergstrasse, Germany). 16: 12831-7. PMID 20967805 DOI: 10.1002/Chem.201002267 |
0.587 |
|
2010 |
Verbeeck S, Herrebout WA, Gulevskaya AV, van der Veken BJ, Maes BU. ONSH: optimization of oxidative alkylamination reactions through study of the reaction mechanism. The Journal of Organic Chemistry. 75: 5126-33. PMID 20617847 DOI: 10.1021/Jo100858N |
0.449 |
|
2009 |
Ryabtsova O, Verhelst T, Baeten M, Vande Velde CM, Maes BU. Synthesis of functionalized pyridazin-3(2H)-ones via bromine-magnesium exchange on bromopyridazin-3(2H)-ones. The Journal of Organic Chemistry. 74: 9440-5. PMID 19928756 DOI: 10.1021/Jo9020985 |
0.433 |
|
2009 |
El Sayed I, Van der Veken P, Steert K, Dhooghe L, Hostyn S, Van Baelen G, Lemière G, Maes BU, Cos P, Maes L, Joossens J, Haemers A, Pieters L, Augustyns K. Synthesis and antiplasmodial activity of aminoalkylamino-substituted neocryptolepine derivatives. Journal of Medicinal Chemistry. 52: 2979-88. PMID 19364118 DOI: 10.1021/Jm801490Z |
0.35 |
|
2008 |
Meyers C, Yáñez M, Elmaatougi A, Verhelst T, Coelho A, Fraiz N, Lemière GL, García-Mera X, Laguna R, Cano E, Maes BU, Sotelo E. 2-Substituted 4-, 5-, and 6-[(1E)-3-oxo-3-phenylprop-1-en-1-yl]pyridazin-3(2H)-ones and 2-substituted 4,5-bis[(1E)-3-oxo-3-phenylprop-1-en-1-yl]pyridazin-3(2H)-ones as potent platelet aggregation inhibitors: design, synthesis, and SAR studies. Bioorganic & Medicinal Chemistry Letters. 18: 793-7. PMID 18053717 DOI: 10.1016/J.Bmcl.2007.11.034 |
0.35 |
|
2008 |
Franck P, Hostyn S, Dajka-Halász B, Polonka-Bálint Á, Monsieurs K, Mátyus P, Maes BU. Pd-catalyzed intramolecular direct arylations at high temperature Tetrahedron. 64: 6030-6037. DOI: 10.1016/J.Tet.2008.01.060 |
0.417 |
|
2007 |
Loones KT, Maes BU, Herrebout WA, Dommisse RA, Lemière GL, Van der Veken BJ. Examination of the mechanism of the intramolecular amination of N-(3-bromopyridin-2-yl)azaheteroarylamines and N-(2-chloropyridin-3-yl)azaheteroarylamines: a Pd-catalyzed amination and/or a base-assisted nucleophilic aromatic substitution? Tetrahedron. 63: 3818-3825. DOI: 10.1016/J.Tet.2007.02.041 |
0.403 |
|
2006 |
Loones KT, Maes BU, Meyers C, Deruytter J. Orthogonal and auto-tandem catalysis: synthesis of dipyrido[1,2-a:2',3'-d]imidazole and its benzo and aza analogues via inter- and intramolecular C-N bond formation. The Journal of Organic Chemistry. 71: 260-4. PMID 16388645 DOI: 10.1021/Jo052091U |
0.421 |
|
2006 |
Crespo A, Meyers C, Coelho A, Yáñez M, Fraiz N, Sotelo E, Maes BU, Laguna R, Cano E, Lemière GL, Raviña E. Pyridazines part 41: synthesis, antiplatelet activity and SAR of 2,4,6-substituted 5-(3-oxo-3-phenylprop-1-en-1-yl)- or 5-(3-phenylprop-2-enoyl)pyridazin-3(2H)-ones. Bioorganic & Medicinal Chemistry Letters. 16: 1080-3. PMID 16290144 DOI: 10.1016/J.Bmcl.2005.10.073 |
0.356 |
|
2006 |
Riedl Z, Monsieurs K, Krajsovszky G, Dunkel P, Maes BU, Tapolcsányi P, Egyed O, Boros S, Mátyus P, Pieters L, Lemière GL, Hajós G. Synthesis of novel 1-methyl-1H-pyridazino[3,4-b]indoles Tetrahedron. 62: 121-129. DOI: 10.1016/J.Tet.2005.09.136 |
0.415 |
|
2004 |
Loones KT, Maes BU, Dommisse RA, Lemière GL. The first tandem double palladium-catalyzed aminations: synthesis of dipyrido[1,2-a:3',2'-d]imidazole and its benzo- and aza-analogues. Chemical Communications (Cambridge, England). 2466-7. PMID 15514818 DOI: 10.1002/CHIN.200514036 |
0.412 |
|
2004 |
Meyers C, Maes BU, Loones KT, Bal G, Lemière GL, Dommisse RA. Study of a new rate increasing "base effect" in the palladium-catalyzed amination of aryl iodides. The Journal of Organic Chemistry. 69: 6010-7. PMID 15373485 DOI: 10.1021/Jo049774E |
0.369 |
|
2004 |
Dajka-Halász B, Monsieurs K, Éliás O, Károlyházy L, Tapolcsányi P, Maes BU, Riedl Z, Hajós G, Dommisse RA, Lemière GL, Košmrlj J, Mátyus P. Synthesis of 5H-pyridazino[4,5-b]indoles and their benzofurane analogues utilizing an intramolecular Heck-type reaction Tetrahedron. 60: 2283-2291. DOI: 10.1016/J.Tet.2004.01.024 |
0.433 |
|
2003 |
Hajós G, Riedl Z, Timári G, Mátyus P, Maes B, Lemière G. Synthesis of New Polyfused Heterocycles of Biological Importance by Means of Pd(0) Catalysis Molecules. 8: 480-487. DOI: 10.3390/80600480 |
0.381 |
|
2002 |
Tapolcsányi P, Krajsovszky G, Andó R, Lipcsey P, Horváth G, Mátyus P, Riedl Z, Hajós G, Maes BU, Lemière GL. Synthesis of some diazino-fused tricyclic systems via Suzuki cross-coupling and regioselective nitrene insertion reactions Tetrahedron. 58: 10137-10143. DOI: 10.1016/S0040-4020(02)01400-X |
0.424 |
|
2002 |
Maes BU, Monsieurs K, Loones KT, Lemière GL, Dommisse R, Mátyus P, Riedl Z, Hajós G. Synthesis of 4-aryl-5-hydroxy- and 5-aryl-4-hydroxypyridazin-3(2H)-ones and their use in the preparation of 4,5-diarylpyridazin-3(2H)-ones and hitherto unknown isochromeno[3,4-d]pyridazinediones Tetrahedron. 58: 9713-9721. DOI: 10.1016/S0040-4020(02)01285-1 |
0.4 |
|
2002 |
Riedl Z, Maes BU, Monsieurs K, Lemière GL, Mátyus P, Hajós G. Synthesis of new pyridazino[4,5-c]isoquinolinones by Suzuki cross-coupling reaction Tetrahedron. 58: 5645-5650. DOI: 10.1016/S0040-4020(02)00531-8 |
0.451 |
|
1976 |
Heeres J, Mostmans JH, Maes B, Backx LJ. Synthesis And Antiprotozoal Activity Of Nitroimidazoles- Carbamates And Thiocarbamates Cheminform. 7. DOI: 10.1002/Chin.197642259 |
0.335 |
|
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