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Małgorzata Dukat - Publications

Affiliations: 
Medicinal Chemistry Virginia Commonwealth University, Richmond, VA, United States 
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Year Citation  Score
2023 Hemanth P, Nistala P, Nguyen VT, Eltit JM, Glennon RA, Dukat M. Binding and functional structure-activity similarities of 4-substituted 2,5-dimethoxyphenyl isopropylamine analogues at 5-HT and 5-HT serotonin receptors. Frontiers in Pharmacology. 14: 1101290. PMID 36762110 DOI: 10.3389/fphar.2023.1101290  0.427
2021 Alwassil OI, Abdrakhmanova GR, Dukat M. Computational analysis of non-competitive antagonist arylguanidine-α7 nAChR complexes. Journal of Molecular Graphics & Modelling. 107: 107943. PMID 34058639 DOI: 10.1016/j.jmgm.2021.107943  0.718
2021 Alwassil OI, Khatri S, Schulte MK, Aripaka SS, Mikkelsen JD, Dukat M. NH- and N-Substituted Phenylguanidines as α7 Nicotinic Acetylcholine (nACh) Receptor Antagonists: Structure-Activity Relationship Studies. Acs Chemical Neuroscience. PMID 34043311 DOI: 10.1021/acschemneuro.1c00212  0.725
2021 de la Fuente Revenga M, Shah UH, Nassehi N, Jaster AM, Hemanth P, Sierra S, Dukat M, González-Maeso J. Psychedelic-like Properties of Quipazine and Its Structural Analogues in Mice. Acs Chemical Neuroscience. 12: 831-844. PMID 33400504 DOI: 10.1021/acschemneuro.0c00291  0.303
2020 Abdelkhalek AS, Musayev FN, Iyer KA, Hemanth P, Safo MK, Dukat M. X-Ray Crystal Structure of a 2-Amino-3,4-dihydroquinazoline 5-HT Serotonin Receptor Antagonist and Related Analogs. Journal of Molecular Structure. 1202. PMID 32616964 DOI: 10.1016/j.molstruc.2019.127276  0.763
2019 Iyer KA, Alix K, Eltit JM, Solis E, Pan X, Argade MD, Khatri S, De Felice LJ, Sweet DH, Schulte MK, Dukat M. Multi-modal antidepressant-like action of 6- and 7-chloro-2-aminodihydroquinazolines in the mouse tail suspension test. Psychopharmacology. PMID 30805668 DOI: 10.1007/S00213-019-05203-5  0.618
2019 Shah UH, Gaitonde SA, Moreno JL, Glennon RA, Dukat M, González-Maeso J. A revised pharmacophore model for 5-HT2A receptor antagonists derived from the atypical antipsychotic agent risperidone. Acs Chemical Neuroscience. PMID 30609893 DOI: 10.1021/Acschemneuro.8B00637  0.463
2018 Abdelkhalek AS, Alley GS, Alwassil OI, Khatri S, Mosier PD, Nyce HL, White MM, Schulte MK, Dukat M. "Methylene Bridge" to 5-HT3 Receptor Antagonists: Conformationally-Constrained Phenylguanidines". Acs Chemical Neuroscience. PMID 30375852 DOI: 10.1021/Acschemneuro.8B00431  0.769
2018 Dukat M, Jain AD, German N, Ferrara-Pontoriero R, Huang Y, Ma Y, Schulte MK, Glennon RA. des-Formylflustrabromine (dFBr): A Structure-Activity Study on its Ability to Potentiate the Action of Acetylcholine at α4β2 Nicotinic Acetylcholine Receptors. Acs Chemical Neuroscience. PMID 30028943 DOI: 10.1021/Acschemneuro.8B00156  0.356
2017 Pan X, Iyer KA, Liu H, Sweet DH, Dukat M. A new chemotype inhibitor for the human organic cation transporter 3 (hOCT3). Bioorganic & Medicinal Chemistry Letters. PMID 28811134 DOI: 10.1016/J.Bmcl.2017.08.008  0.724
2017 Sguazzini E, Schmidt HR, Iyer KA, Kruse AC, Dukat M. Reevaluation of fenpropimorph as a σ receptor ligand: Structure-affinity relationship studies at human σ1 receptors. Bioorganic & Medicinal Chemistry Letters. 27: 2912-2919. PMID 28495085 DOI: 10.1016/j.bmcl.2017.04.088  0.742
2016 Glennon RA, Dukat M. Structure-Activity Relationships of Synthetic Cathinones. Current Topics in Behavioral Neurosciences. PMID 27830576 DOI: 10.1007/7854_2016_41  0.308
2016 Alix K, Khatri S, Mosier PD, Casterlow S, Yan D, Nyce HL, White MM, Schulte MK, Dukat M. Super-agonist, full agonist, partial agonist and antagonist actions of arylguanidines at h5-HT3A receptors. Acs Chemical Neuroscience. PMID 27533595 DOI: 10.1021/Acschemneuro.6B00196  0.459
2016 Younkin J, Gaitonde SA, Ellaithy A, Vekariya RH, Baki L, Moreno JL, Shah S, Drossopoulos P, Hideshima KS, Eltit JM, González-Maeso J, Logothetis DE, Dukat M, Glennon RA. Reformulating a Pharmacophore for 5-HT2A Serotonin Receptor Antagonists. Acs Chemical Neuroscience. PMID 27385190 DOI: 10.1021/Acschemneuro.6B00162  0.458
2014 Rao BK, Samanta D, Joshi S, Basu K, Baldwin SD, Jha A, Dukat M, Glennon RA, Jena P. Receptor-ligand interaction at 5-HT3 serotonin receptors: a cluster approach. The Journal of Physical Chemistry. A. 118: 8471-6. PMID 24878072 DOI: 10.1021/Jp5017906  0.394
2013 Dukat M, Alix K, Worsham J, Khatri S, Schulte MK. 2-Amino-6-chloro-3,4-dihydroquinazoline: A novel 5-HT3 receptor antagonist with antidepressant character. Bioorganic & Medicinal Chemistry Letters. 23: 5945-8. PMID 24035337 DOI: 10.1016/J.Bmcl.2013.08.072  0.484
2012 Rahman AA, Daoud MK, Dukat M, Herrick-Davis K, Purohit A, Teitler M, do Amaral AT, Malvezzi A, Glennon RA. Corrigendum to “Conformationally-restricted analogues and partition coefficients of the 5-HT3 serotonin receptor ligands meta-Chlorophenylbiguanide (mCPBG) and meta-Chlorophenylguanidine (mCPG)” [Bioorg. Med. Chem. Lett. 15 (2005) 3434–3438] Bioorganic & Medicinal Chemistry Letters. 22: 6526. DOI: 10.1016/J.Bmcl.2012.08.076  0.351
2011 German N, Kim JS, Jain A, Dukat M, Pandya A, Ma Y, Weltzin M, Schulte MK, Glennon RA. Deconstruction of the α4β2 nicotinic acetylcholine receptor positive allosteric modulator desformylflustrabromine Journal of Medicinal Chemistry. 54: 7259-7267. PMID 21905680 DOI: 10.1021/Jm200834X  0.361
2011 Klein MT, Dukat M, Glennon RA, Teitler M. Toward selective drug development for the human 5-hydroxytryptamine 1E receptor: a comparison of 5-hydroxytryptamine 1E and 1F receptor structure-affinity relationships. The Journal of Pharmacology and Experimental Therapeutics. 337: 860-7. PMID 21422162 DOI: 10.1124/Jpet.111.179606  0.499
2010 Glennon RA, Siripurapu U, Roth BL, Kolanos R, Bondarev ML, Sikazwe D, Lee M, Dukat M. The medicinal chemistry of 5-HT6 receptor ligands with a focus on arylsulfonyltryptamine analogs. Current Topics in Medicinal Chemistry. 10: 579-95. PMID 20166945 DOI: 10.2174/156802610791111542  0.52
2010 Glennon RA, Lee M, Rangisetty JB, Dukat M, Roth BL, Savage JE, McBride A, Rauser L, Hufeisen S, Lee DKH. ChemInform Abstract: 2-Substituted Tryptamines: Agents with Selectivity for 5-HT6 Serotonin Receptors. Cheminform. 31: no-no. DOI: 10.1002/CHIN.200023120  0.424
2010 HONG S, DUKAT M, TEITLER M, HERRICK-DAVIS K, MCCALLUM K, KAMBOJ R, GLENNON RA. ChemInform Abstract: Binding of 5-Arylalkyloxytryptamines at Human 5-HT1Dβ Serotonin Receptors. Cheminform. 27: no-no. DOI: 10.1002/CHIN.199621126  0.399
2010 DUKAT M, DAMAJ MI, GLASSCO W, DUMAS D, MAY EL, MARTIN BR, GLENNON RA. ChemInform Abstract: Epibatidine: A Very High Affinity Nicotine-Receptor Ligand. Cheminform. 26: no-no. DOI: 10.1002/chin.199513270  0.318
2008 Dukat M, Mosier PD, Kolanos R, Roth BL, Glennon RA. Binding of serotonin and N1-benzenesulfonyltryptamine-related analogs at human 5-HT6 serotonin receptors: receptor modeling studies. Journal of Medicinal Chemistry. 51: 603-11. PMID 18201064 DOI: 10.1021/Jm070910S  0.467
2007 Dukat M, Glennon RA, Young S. MD-354: What is it good for? Cns Drug Reviews. 13: 1-20. PMID 17461887 DOI: 10.1111/J.1527-3458.2007.00002.X  0.447
2006 Kolanos R, Dukat M, Roth BL, Glennon RA. Interaction of N1-unsubstituted and N1-benzenesulfonyltryptamines at h5-HT6 receptors. Bioorganic & Medicinal Chemistry Letters. 16: 5832-5. PMID 16945532 DOI: 10.1016/J.Bmcl.2006.08.068  0.433
2006 Sikazwe D, Bondarev ML, Dukat M, Rangisetty JB, Roth BL, Glennon RA. Binding of sulfonyl-containing arylalkylamines at human 5-HT6 serotonin receptors. Journal of Medicinal Chemistry. 49: 5217-25. PMID 16913710 DOI: 10.1021/Jm060469Q  0.485
2006 Ragab HM, Kim JS, Dukat M, Navarro H, Glennon RA. Aryloxyethylamines: Binding at α7 nicotinic acetylcholine receptors Bioorganic and Medicinal Chemistry Letters. 16: 4283-4286. PMID 16765047 DOI: 10.1016/J.Bmcl.2006.05.080  0.34
2006 Siripurapu U, Kolanos R, Dukat M, Roth BL, Glennon RA. Binding of methoxy-substituted N1-benzenesulfonylindole analogs at human 5-HT6 serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 16: 3793-6. PMID 16709453 DOI: 10.1016/J.Bmcl.2006.04.094  0.473
2005 Pullagurla M, Siripurapu U, Kolanos R, Bondarev ML, Dukat M, Setola V, Roth BL, Glennon RA. Binding of amine-substituted N1-benzenesulfonylindoles at human 5-HT6 serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 15: 5298-302. PMID 16183286 DOI: 10.1016/J.Bmcl.2005.08.059  0.461
2005 Abate C, Kolanos R, Dukat M, Setola V, Roth BL, Glennon RA. Interaction of chiral MS-245 analogs at h5-HT6 receptors. Bioorganic & Medicinal Chemistry Letters. 15: 3510-3. PMID 15990303 DOI: 10.1016/J.Bmcl.2005.05.092  0.394
2005 Setola V, Dukat M, Glennon RA, Roth BL. Molecular determinants for the interaction of the valvulopathic anorexigen norfenfluramine with the 5-HT2B receptor. Molecular Pharmacology. 68: 20-33. PMID 15831837 DOI: 10.1124/Mol.104.009266  0.409
2005 Kolanos R, Siripurapu U, Pullagurla M, Riaz M, Setola V, Roth BL, Dukat M, Glennon RA. Binding of isotryptamines and indenes at h5-HT6 serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 15: 1987-91. PMID 15808453 DOI: 10.1016/J.Bmcl.2005.02.070  0.369
2005 Lee M, Rangisetty JB, Pullagurla MR, Dukat M, Setola V, Roth BL, Glennon RA. 1-(1-Naphthyl)piperazine as a novel template for 5-HT6 serotonin receptor ligands. Bioorganic & Medicinal Chemistry Letters. 15: 1707-11. PMID 15745826 DOI: 10.1016/J.Bmcl.2005.01.031  0.446
2005 Pullagurla M, Dukat M, Roth BL, Setola V, Glennon RA. 5-Azatryptamine analogs as h5-HT6 serotonin receptor ligands Medicinal Chemistry Research. 14: 1-18. DOI: 10.1007/S00044-004-0121-8  0.455
2005 Lee M, Rangisetty JB, Pullagurla MR, Dukat M, Setola V, Roth BL, Glennon RA. 1-(1-Naphthyl)piperazine as a Novel Template for 5-HT6 Serotonin Receptor Ligands. Cheminform. 36. DOI: 10.1002/CHIN.200529171  0.422
2004 Prisinzano T, Dukat M, Law H, Slassi A, MacLean N, DeLannoy I, Glennon RA. 2-(Anilino)imidazolines and 2-(benzyl)imidazoline derivatives as h5-HT 1D serotonin receptor ligands Bioorganic and Medicinal Chemistry Letters. 14: 4697-4699. PMID 15324890 DOI: 10.1016/J.Bmcl.2004.06.085  0.408
2004 Shelton KL, Dukat M, Allan AM. Effect of 5-HT3 receptor over-expression on the discriminative stimulus effects of ethanol. Alcoholism, Clinical and Experimental Research. 28: 1161-71. PMID 15318114 DOI: 10.1097/01.ALC.0000138687.27452.E2  0.364
2004 Dukat M, Taroua M, Dahdouh A, Siripurapu U, Damaj MI, Martin BR, Glennon RA. (+/-)8-Amino-5,6,7,8-tetrahydroisoquinolines as novel antinociceptive agents. Bioorganic & Medicinal Chemistry Letters. 14: 3651-4. PMID 15203136 DOI: 10.1016/J.Bmcl.2004.05.020  0.318
2004 Dukat M, Smith C, Herrick-Davis K, Teitler M, Glennon RA. Binding of tryptamine analogs at h5-HT1E receptors: A structure-affinity investigation Bioorganic and Medicinal Chemistry. 12: 2545-2552. PMID 15110837 DOI: 10.1016/J.Bmc.2004.03.026  0.455
2004 Chang-Fong J, Rangisetty JB, Dukat M, Setola V, Raffay T, Roth B, Glennon RA. 1,2,3,4-Tetrahydrocarbazoles as 5-HT6 serotonin receptor ligands Bioorganic and Medicinal Chemistry Letters. 14: 1961-1964. PMID 15050637 DOI: 10.1016/J.Bmcl.2004.01.071  0.44
2004 Glennon RA, Dukat M, Liao L. Musings on alpha4beta2 nicotinic acetylcholine (nACh) receptor pharmacophore models. Current Topics in Medicinal Chemistry. 4: 631-44. PMID 14965299 DOI: 10.2174/1568026043451122  0.338
2004 Dogruer D, Lee M, Dukat M, Damaj MI, Martin BR, Glennon RA. 3-(4-Aminobutyn-1-yl)pyridines: binding at alpha 4 beta 2 nicotinic cholinergic receptors. Bioorganic & Medicinal Chemistry Letters. 14: 523-6. PMID 14698195 DOI: 10.1016/J.Bmcl.2003.10.033  0.343
2004 Dukat M. 5-HT3 Serotonin Receptor Agonists: A Pharmacophoric Journey Current Medicinal Chemistry-Central Nervous System Agents. 4: 77-94. DOI: 10.2174/1568015043356995  0.435
2004 Chang-Fong J, Rangisetty JB, Dukat M, Setola V, Raffay T, Roth B, Glennon RA. 1,2,3,4-Tetrahydrocarbazoles as 5-HT6 Serotonin Receptor Ligands. Cheminform. 35. DOI: 10.1002/CHIN.200431116  0.413
2004 Pullagurla MR, Dukat M, Setola V, Roth B, Glennon RA. N1-Benzenesulfonylgramine (I) and N1-Benzenesulfonylskatole (II): Novel 5-HT6 Receptor Ligand Templates. Cheminform. 35. DOI: 10.1002/chin.200401186  0.37
2003 Simsek R, Chang-Fong J, Lee M, Dukat M, Imad Damaj M, Martin BR, Glennon RA. Quaternary ammonium 3-(aminoethoxy)pyridines as antinociceptive agents. Bioorganic & Medicinal Chemistry Letters. 13: 2917-20. PMID 14611857 DOI: 10.1016/S0960-894X(03)00585-7  0.322
2003 Glennon RA, Daoud MK, Dukat MS, Teitler M, Herrick-Davis K, Purohit A, Syed H. Arylguanidine and arylbiguanide binding at 5-HT3 serotonin receptors: A QSAR study Bioorganic and Medicinal Chemistry. 11: 4449-4454. PMID 13129581 DOI: 10.1016/S0968-0896(03)00488-7  0.474
2003 Pullagurla MR, Dukat M, Setola V, Roth B, Glennon RA. N1-benzenesulfonylgramine and N1-benzenesulfonylskatole: novel 5-HT6 receptor ligand templates. Bioorganic & Medicinal Chemistry Letters. 13: 3355-9. PMID 12951125 DOI: 10.1016/S0960-894X(03)00612-7  0.411
2003 Khorana N, Smith C, Herrick-Davis K, Purohit A, Teitler M, Grella B, Dukat M, Glennon RA. Binding of tetrahydrocarboline derivatives at human 5-HT5A receptors. Journal of Medicinal Chemistry. 46: 3930-7. PMID 12930153 DOI: 10.1021/Jm030080S  0.423
2003 Rahman AA, Daoud MK, Dukat M, Herrick-Davis K, Purohit A, Teitler M, do Amaral AT, Malvezzi A, Glennon RA. Conformationally-restricted analogues and partition coefficients of the 5-HT3 serotonin receptor ligands meta-chlorophenylbiguanide (mCPBG) and meta-chlorophenylguanidine (mCPG). Bioorganic & Medicinal Chemistry Letters. 13: 1119-23. PMID 12643925 DOI: 10.1016/S0960-894X(03)00044-1  0.353
2002 Ferretti G, Dukat M, Giannella M, Piergentili A, Pigini M, Quaglia W, Damaj MI, Martin BR, Glennon RA. Homoazanicotine: a structure-affinity study for nicotinic acetylcholine (nACh) receptor binding. Journal of Medicinal Chemistry. 45: 4724-31. PMID 12361399 DOI: 10.1021/Jm020188S  0.371
2002 Glennon RA, Metwally K, Dukat M, Ismaiel AM, De los Angeles J, Herndon J, Teitler M, Khorana N. Ketanserin and spiperone as templates for novel serotonin 5-HT(2A) antagonists. Current Topics in Medicinal Chemistry. 2: 539-58. PMID 12052193 DOI: 10.2174/1568026023393787  0.424
2002 Chang-Fong J, Addo J, Dukat M, Smith C, Mitchell NA, Herrick-Davis K, Teitler M, Glennon RA. Evaluation of isotryptamine derivatives at 5-HT(2) serotonin receptors. Bioorganic & Medicinal Chemistry Letters. 12: 155-8. PMID 11755343 DOI: 10.1016/S0960-894X(01)00713-2  0.434
2001 Rangisetty JB, Dukat M, Dowd CS, Herrick-Davis K, DuPre A, Gadepalli S, Teitler M, Kelley CR, Sharif NA, Glennon RA. 1-[2-methoxy-5-(3-phenylpropyl)]-2-aminopropane unexpectedly shows 5-HT(2A) serotonin receptor affinity and antagonist character. Journal of Medicinal Chemistry. 44: 3283-91. PMID 11563927 DOI: 10.1021/Jm0100739  0.435
2001 Dukat M, Choi YN, Teitler M, Du Pre A, Herrick-Davis K, Smith C, Glennon RA. The binding of arylguanidines at 5-HT(3) serotonin receptors: a structure-affinity investigation. Bioorganic & Medicinal Chemistry Letters. 11: 1599-603. PMID 11412989 DOI: 10.1016/S0960-894X(01)00291-8  0.46
2001 Prisinzano T, Law H, Dukat M, Slassi A, MaClean N, Demchyshyn L, Glennon RA. Imidazoline-modified benzylimidazolines as h5-HT(1D/1B) serotonergic ligands. Bioorganic & Medicinal Chemistry. 9: 613-9. PMID 11310595 DOI: 10.1016/S0968-0896(00)00275-3  0.352
2001 Tsai Y, Dukat M, Slassi A, MacLean N, Demchyshyn L, Savage JE, Roth BL, Hufesein S, Lee M, Glennon RA. ChemInform Abstract: N1-(Benzenesulfonyl)tryptamines as Novel 5-HT6 Antagonists. Cheminform. 32: no-no. DOI: 10.1002/CHIN.200103235  0.369
2000 Tsai Y, Dukat M, Slassi A, MacLean N, Demchyshyn L, Savage JE, Roth BL, Hufesein S, Lee M, Glennon RA. N1-(Benzenesulfonyl)tryptamines as novel 5-HT6 antagonists. Bioorganic & Medicinal Chemistry Letters. 10: 2295-9. PMID 11055342 DOI: 10.1016/S0960-894X(00)00453-4  0.425
2000 Glennon RA, Dukat M, Grella B, Hong SS, Costantino L, Teitler M, Smith C, Egan C, Davis K, Mattson MV. Binding of β-carbolines and related agents at serotonin (5-HT2 and 5- HT(1A)), dopamine (D2) and benzodiazepine receptors Drug and Alcohol Dependence. 60: 121-132. PMID 10940539 DOI: 10.1016/S0376-8716(99)00148-9  0.44
2000 Dukat M, Young R, Darmani NN, Ahmed B, Glennon RA. The 5-HT3 agent N-(3-chlorophenyl)guanidine (MD-354) serves as a discriminative stimulus in rats and displays partial agonist character in a shrew emesis assay Psychopharmacology. 150: 200-207. PMID 10907673 DOI: 10.1007/S002130000410  0.401
2000 Glennon RA, Lee M, Rangisetty JB, Dukat M, Roth BL, Savage JE, McBride A, Rauser L, Hufeisen S, Lee DK. 2-Substituted tryptamines: agents with selectivity for 5-HT(6) serotonin receptors. Journal of Medicinal Chemistry. 43: 1011-8. PMID 10715164 DOI: 10.1021/Jm990550B  0.43
2000 Glennon RA, Dukat M. Central nicotinic receptor ligands and pharmacophores Pharmacochemistry Library. 31: 103-114. DOI: 10.1016/S0031-6865(99)00022-9  0.374
1999 Flammia D, Dukat M, Damaj MI, Martin B, Glennon RA. Lobeline: Structure-affinity investigation of nicotinic acetylcholinergic receptor binding Journal of Medicinal Chemistry. 42: 3726-3731. PMID 10479304 DOI: 10.1021/Jm990286M  0.309
1999 Gyermek L, Sun X, Nguyen N, Dukat M. Is there a functional response-overlap between 5-HT3 and nicotinic ion channel receptors? Annals of the New York Academy of Sciences. 861: 255-7. PMID 9928275 DOI: 10.1111/J.1749-6632.1998.TB10209.X  0.312
1999 Cheng YX, Dukat M, Dowd M, Fiedler W, Martin B, Damaj MI, Glennon RA. Synthesis and binding of 6,7,8,9-tetrahydro-5H-pyrido[3,4-d]azepine and related ring-opened analogs at central nicotinic receptors European Journal of Medicinal Chemistry. 34: 177-190. DOI: 10.1016/S0223-5234(99)80051-8  0.332
1999 Dukat M, Dowd M, Damaj MI, Martin B, El-Zahabi MA, Glennon RA. Synthesis, receptor binding and QSAR studies on 6-substituted nicotine derivatives as cholinergic ligands European Journal of Medicinal Chemistry. 34: 31-40. DOI: 10.1016/S0223-5234(99)80038-5  0.322
1998 Metwally KA, Dukat M, Egan CT, Smith C, DuPre A, Gauthier CB, Herrick-Davis K, Teitler M, Glennon RA. Spiperone: Influence of spiro ring substituents on 5-HT(2A) serotonin receptor binding Journal of Medicinal Chemistry. 41: 5084-5093. PMID 9836624 DOI: 10.1021/Jm980452A  0.48
1998 Law H, Dukat M, Teitler M, Lee DKH, Mazzocco L, Kamboj R, Rampersad V, Prisinzano T, Glennon RA. Benzylimidazolines as h5-HT(1B/1D) serotonin receptor ligands: A structure-affinity investigation Journal of Medicinal Chemistry. 41: 2243-2251. PMID 9632357 DOI: 10.1021/Jm970513P  0.409
1997 Ismaiel AM, Dukat M, Law H, Kamboj R, Fan E, Lee DKH, Mazzocco L, Buekschkens D, Teitler M, Pierson ME, Glennon RA. 2-(1-naphthyloxy)ethylamines with enhanced affinity for human 5-HT(1Dβ) (h5-HT(1B)) serotonin receptors Journal of Medicinal Chemistry. 40: 4415-4419. PMID 9435911 DOI: 10.1021/Jm970507T  0.454
1996 Dukat M, Abdel-Rahman AA, Ismaiel AM, Ingher S, Teitler M, Gyermek L, Glennon RA. Structure-activity relationships for the binding of arylpiperazines and arylbiguanides at 5-HT3 serotonin receptors Journal of Medicinal Chemistry. 39: 4017-4026. PMID 8831767 DOI: 10.1021/Jm9603936  0.448
1996 Glennon RA, Hong SS, Bondarev M, Law H, Dukat M, Rakhit S, Power P, Fan E, Kinneau D, Kamboj R, Teitler M, Herrick-Davis K, Smith C. Binding of O-alkyl derivatives of serotonin at human 5-HT1Dβ receptors Journal of Medicinal Chemistry. 39: 314-322. PMID 8568822 DOI: 10.1021/Jm950498T  0.432
1996 Imad Damaj M, Glassco W, Dukat M, May EL, Glennon RA, Martin BR. Pharmacology of novel nicotinic analogs Drug Development Research. 38: 177-187. DOI: 10.1002/(Sici)1098-2299(199607/08)38:3/4<177::Aid-Ddr6>3.0.Co;2-J  0.316
1994 Glennon RA, Hong SS, Dukat M, Teitler M, Davis K. 5-(Nonyloxy)tryptamine: A novel high-affinity 5-HTIDβ serotonin receptor agonist Journal of Medicinal Chemistry. 37: 2828-2830. PMID 8071931 DOI: 10.1021/Jm00044A001  0.443
1994 Glennon RA, Dukat M, El-Bermawy M, Law H, De Los Angeles J, Teitler M, King A, Herrick-Davis K. Influence of amine substituents on 5-HT2A versus 5-HT2C binding of phenylalkyl- and indolylalkylamines Journal of Medicinal Chemistry. 37: 1929-1935. PMID 8027974 DOI: 10.1021/Jm00039A004  0.429
1992 Glennon RA, Dukat M. Serotonin receptors and their ligands: a lack of selective agents. Pharmacology, Biochemistry, and Behavior. 40: 1009-17. PMID 1816555 DOI: 10.1016/0091-3057(91)90121-H  0.404
1992 Glennon RA, Young R, Dukat M. 5-HT3 agonist 2-methylserotonin as a training drug in discrimination studies. Pharmacology, Biochemistry, and Behavior. 41: 361-4. PMID 1574526 DOI: 10.1016/0091-3057(92)90111-R  0.323
1990 MISZTAL S, DUKAT M, MOKROSZ JL. ChemInform Abstract: Structure and Spectral Properties of β-Carbolines. Part 3. Synthesis and Stereochemistry of 1,2,3,4,6,7,9,10,15b,15c-Decahydropyrido(1′′,2′′:1′,2′)pyrazino(4′,3′:1,2)pyrido(3,4-b)indoles. Cheminform. 21. DOI: 10.1002/CHIN.199046227  0.575
1990 Mokrosz JL, Dukat M, Misztal S. Structure and Spectral Properties of β-Carbolines, I:13C-NMR and Mass Spectra of Decahydro-5H-pyrido[1′,2′;5,1]-imidazo[3,4-a]-β-carbolines Archiv Der Pharmazie. 323: 453-457. DOI: 10.1002/ARDP.19903230803  0.578
1986 MISZTAL S, DUKAT M. ChemInform Abstract: The threo and erythro Products of the Catalytic Hydrogenation of 1-(2-Pyridyl)- 1,2,3,4-tetrahydro-β-carboline. Chemischer Informationsdienst. 17. DOI: 10.1002/CHIN.198605205  0.562
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