| Year |
Citation |
Score |
| 2018 |
Tiwari D, Park SW, Essawy MM, Dawadi S, Mason A, Nandakumar M, Zimmerman M, Mina M, Ho HP, Engelhart CA, Ioerger T, Sacchettini JC, Rhee K, Ehrt S, Aldrich CC, et al. Targeting protein biotinylation enhances tuberculosis chemotherapy. Science Translational Medicine. 10. PMID 29695454 DOI: 10.1126/Scitranslmed.Aal1803 |
0.614 |
|
| 2018 |
Dawadi S, Boshoff HIM, Park SW, Schnappinger D, Aldrich CC. Conformationally Constrained Cinnolinone Nucleoside Analogues as Siderophore Biosynthesis Inhibitors for Tuberculosis. Acs Medicinal Chemistry Letters. 9: 386-391. PMID 29670706 DOI: 10.1021/Acsmedchemlett.8B00090 |
0.633 |
|
| 2018 |
Bockman MR, Engelhart CA, Dawadi S, Larson P, Tiwari D, Ferguson DM, Schnappinger D, Aldrich CC. Avoiding Antibiotic Inactivation in Mycobacterium tuberculosis by Rv3406 through Strategic Nucleoside Modification. Acs Infectious Diseases. PMID 29663798 DOI: 10.1021/Acsinfecdis.8B00038 |
0.601 |
|
| 2018 |
Minato Y, Dawadi S, Kordus SL, Sivanandam A, Aldrich CC, Baughn AD. Mutual potentiation drives synergy between trimethoprim and sulfamethoxazole. Nature Communications. 9: 1003. PMID 29520101 DOI: 10.1038/S41467-018-03447-X |
0.585 |
|
| 2017 |
Dawadi S, Kordus SL, Baughn AD, Aldrich CC. Synthesis and Analysis of Bacterial Folate Metabolism Intermediates and Antifolates. Organic Letters. PMID 28926267 DOI: 10.1021/Acs.Orglett.7B02487 |
0.642 |
|
| 2017 |
Okon A, Han J, Dawadi S, Demosthenous C, Aldrich CC, Gupta M, Wagner CR. Anchimerically Activated ProTides as Inhibitors of Cap-Dependent Translation and Inducers of Chemosensitization in Mantle Cell Lymphoma. Journal of Medicinal Chemistry. PMID 28858511 DOI: 10.1021/Acs.Jmedchem.7B00916 |
0.566 |
|
| 2017 |
Liu F, Dawadi S, Maize KM, Dai R, Park SW, Schnappinger D, Finzel BC, Aldrich CC. Structure-Based Optimization of Pyridoxal 5'-Phosphate (PLP)-Dependent Transaminase Enzyme (BioA) Inhibitors that Target Biotin Biosynthesis in Mycobacterium tuberculosis. Journal of Medicinal Chemistry. PMID 28594172 DOI: 10.1021/Acs.Jmedchem.7B00189 |
0.653 |
|
| 2016 |
Krajczyk A, Zeidler J, Januszczyk P, Dawadi S, Boshoff HI, Barry CE, Ostrowski T, Aldrich CC. 2-Aryl-8-aza-3-deazaadenosine analogues of 5'-O-[N-(salicyl)sulfamoyl]adenosine: Nucleoside antibiotics that block siderophore biosynthesis in Mycobacterium tuberculosis. Bioorganic & Medicinal Chemistry. PMID 27265685 DOI: 10.1016/J.Bmc.2016.05.037 |
0.621 |
|
| 2016 |
Dawadi S, Kawamura S, Rubenstein A, Remmel R, Aldrich CC. Synthesis and pharmacological evaluation of nucleoside prodrugs designed to target siderophore biosynthesis in Mycobacterium tuberculosis. Bioorganic & Medicinal Chemistry. PMID 26875934 DOI: 10.1016/J.Bmc.2016.02.002 |
0.64 |
|
| 2015 |
Bockman MR, Kalinda AS, Petrelli R, De la Mora-Rey T, Tiwari D, Liu F, Dawadi S, Nandakumar M, Rhee KY, Schnappinger D, Finzel BC, Aldrich CC. Targeting Mycobacterium tuberculosis Biotin Protein Ligase (MtBPL) with Nucleoside-Based Bisubstrate Adenylation Inhibitors. Journal of Medicinal Chemistry. 58: 7349-69. PMID 26299766 DOI: 10.1021/Acs.Jmedchem.5B00719 |
0.65 |
|
| 2015 |
Sutivisedsak N, Dawadi S, Spilling CD. Trapping Hemiacetals with Phosphono Substituted Palladium π-Allyl Complexes for the Synthesis of Substituted Cyclic Ethers. Tetrahedron Letters. 56: 3534-3537. PMID 26236053 DOI: 10.1016/J.Tetlet.2015.01.050 |
0.313 |
|
| 2015 |
Nelson KM, Viswanathan K, Dawadi S, Duckworth BP, Boshoff HI, Barry CE, Aldrich CC. Synthesis and Pharmacokinetic Evaluation of Siderophore Biosynthesis Inhibitors for Mycobacterium tuberculosis. Journal of Medicinal Chemistry. 58: 5459-75. PMID 26110337 DOI: 10.1021/Acs.Jmedchem.5B00391 |
0.678 |
|
| 2015 |
Dawadi S, Viswanathan K, Boshoff HI, Barry CE, Aldrich CC. Investigation and conformational analysis of fluorinated nucleoside antibiotics targeting siderophore biosynthesis. The Journal of Organic Chemistry. 80: 4835-50. PMID 25916415 DOI: 10.1021/Acs.Joc.5B00550 |
0.677 |
|
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