Year |
Citation |
Score |
2013 |
Ye L, Dickerson T, Kaur H, Takada YK, Fujita M, Liu R, Knapp JM, Lam KS, Schore NE, Kurth MJ, Takada Y. Identification of inhibitors against interaction between pro-inflammatory sPLA2-IIA protein and integrin αvβ3. Bioorganic & Medicinal Chemistry Letters. 23: 340-5. PMID 23164706 DOI: 10.1016/J.Bmcl.2012.10.080 |
0.496 |
|
2012 |
Knapp JM, Zhu JS, Tantillo DJ, Kurth MJ. Multicomponent assembly of highly substituted indoles by dual palladium-catalyzed coupling reactions. Angewandte Chemie (International Ed. in English). 51: 10588-91. PMID 23001913 DOI: 10.1002/Anie.201204633 |
0.513 |
|
2012 |
Knapp JM, Wood AB, Phuan PW, Lodewyk MW, Tantillo DJ, Verkman AS, Kurth MJ. Structure-activity relationships of cyanoquinolines with corrector-potentiator activity in ΔF508 cystic fibrosis transmembrane conductance regulator protein. Journal of Medicinal Chemistry. 55: 1242-51. PMID 22214395 DOI: 10.1021/Jm201372Q |
0.5 |
|
2012 |
Knapp JM, Zhu JS, Wood AB, Kurth MJ. Expedient synthesis of a 72-membered isoxazolino-β-ketoamide library by a 2·3-component reaction. Acs Combinatorial Science. 14: 85-8. PMID 22181856 DOI: 10.1021/Co200199H |
0.54 |
|
2011 |
Knapp JM, Fettinger JC, Kurth MJ. Multicomponent macrocyclization reactions (MCMRs) employing highly reactive acyl ketene and nitrile oxide intermediates. Organic Letters. 13: 4732-5. PMID 21827181 DOI: 10.1021/Ol202024A |
0.512 |
|
2011 |
Phuan PW, Yang B, Knapp JM, Wood AB, Lukacs GL, Kurth MJ, Verkman AS. Cyanoquinolines with independent corrector and potentiator activities restore ΔPhe508-cystic fibrosis transmembrane conductance regulator chloride channel function in cystic fibrosis. Molecular Pharmacology. 80: 683-93. PMID 21730204 DOI: 10.1124/Mol.111.073056 |
0.522 |
|
2010 |
Ye L, Knapp JM, Sangwung P, Fettinger JC, Verkman AS, Kurth MJ. Pyrazolylthiazole as DeltaF508-cystic fibrosis transmembrane conductance regulator correctors with improved hydrophilicity compared to bithiazoles. Journal of Medicinal Chemistry. 53: 3772-81. PMID 20373765 DOI: 10.1021/Jm100235H |
0.52 |
|
Show low-probability matches. |