Year |
Citation |
Score |
2020 |
Yeoh YQ, Horsley J, Yu J, Polyak SW, Jovcevski B, Abell AD. Short Photoswitchable Antibacterial Peptides. Chemmedchem. PMID 32558320 DOI: 10.1002/Cmdc.202000280 |
0.3 |
|
2020 |
Yeoh YQ, Horsley JR, Polyak SW, Abell AD. A hypoxia-activated antibacterial prodrug. Bioorganic & Medicinal Chemistry Letters. 127140. PMID 32247730 DOI: 10.1016/J.Bmcl.2020.127140 |
0.3 |
|
2019 |
Lee KJ, Tieu W, Blanco-Rodriguez B, Paparella AS, Yu J, Hayes A, Feng J, Marshall AC, Noll B, Milne R, Cini D, Wilce MCJ, Booker GW, Bruning JB, Polyak SW, ... Abell AD, et al. Sulfonamide-based inhibitors of biotin protein ligase as new antibiotic leads. Acs Chemical Biology. PMID 31407891 DOI: 10.1021/Acschembio.9B00463 |
0.339 |
|
2018 |
Pehere AD, Nguyen S, Garlick SK, Wilson DW, Hudson I, Sykes MJ, Morton JD, Abell AD. Tripeptide analogues of MG132 as protease inhibitors. Bioorganic & Medicinal Chemistry. PMID 30581047 DOI: 10.1016/J.Bmc.2018.12.022 |
0.314 |
|
2018 |
Schumann NC, Bruning J, Marshall AC, Abell AD. The role of N-terminal heterocycles in hydrogen bonding to α-chymotrypsin. Bioorganic & Medicinal Chemistry Letters. PMID 30579793 DOI: 10.1016/J.Bmcl.2018.12.032 |
0.302 |
|
2018 |
Abell AD, Yu J, Polyak S, Horsley J, Yeoh YQ. Photopharmacological Control of Cyclic Antimicrobial Peptides. Chembiochem : a European Journal of Chemical Biology. PMID 30324702 DOI: 10.1002/Cbic.201800618 |
0.302 |
|
2018 |
Hochscherf J, Pietsch M, Tieu W, Kuan K, Abell AD, Gütschow M, Niefind K. Crystal structure of highly glycosylated human leukocyte elastase in complex with an S2' site binding inhibitor. Acta Crystallographica. Section F, Structural Biology Communications. 74: 480-489. PMID 30084397 DOI: 10.1107/S2053230X1800537X |
0.311 |
|
2018 |
Wegener KL, McGrath AE, Dixon NE, Oakley AJ, Scanlon DB, Abell AD, Bruning J. Rational design of a 310-helical PIP-box mimetic targeting PCNA - the human sliding clamp. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29917264 DOI: 10.1002/Chem.201801734 |
0.309 |
|
2017 |
Paparella AS, Lee KJ, Hayes A, Feng J, Feng Z, Cini D, Deshmukh S, Booker GW, Wilce MCJ, Polyak SW, Abell AD. Halogenation of biotin protein ligase inhibitors improves whole cell activity against Staphylococcus aureus. Acs Infectious Diseases. PMID 29131575 DOI: 10.1021/Acsinfecdis.7B00134 |
0.302 |
|
2017 |
Blanco B, Palasis KA, Adwal A, Callen DF, Abell AD. Azobenzene-containing photoswitchable proteasome inhibitors with selective activity and cellular toxicity. Bioorganic & Medicinal Chemistry. PMID 28642029 DOI: 10.1016/J.Bmc.2017.06.011 |
0.312 |
|
2017 |
Frkic RL, Rodriguez BB, Chang MR, Kuruvilla D, Ciesla A, Abell AD, Kamenecka TM, Griffin PR, Bruning JB. Structure-Activity Relationship of 2,4-dichloro-N-(3,5-dichloro-4-(quinolin-3-yloxy)phenyl)benzenesulfonamide (INT131) Analogs for PPARγ-Targeted Antidiabetics. Journal of Medicinal Chemistry. PMID 28485590 DOI: 10.1021/Acs.Jmedchem.6B01727 |
0.305 |
|
2017 |
Pehere AD, Zhang X, Abell AD. Macrocyclic Peptidomimetics Prepared by Ring-Closing Metathesis and Azide–Alkyne Cycloaddition Australian Journal of Chemistry. 70: 138. DOI: 10.1071/Ch16532 |
0.336 |
|
2016 |
Feng J, Paparella AS, Tieu W, Heim D, Clark S, Hayes A, Booker GW, Polyak SW, Abell AD. New Series of BPL Inhibitors To Probe the Ribose-Binding Pocket of Staphylococcus aureus Biotin Protein Ligase. Acs Medicinal Chemistry Letters. 7: 1068-1072. PMID 27994739 DOI: 10.1021/Acsmedchemlett.6B00248 |
0.337 |
|
2016 |
Feng J, Paparella AS, Booker GW, Polyak SW, Abell AD. Biotin Protein Ligase Is a Target for New Antibacterials. Antibiotics (Basel, Switzerland). 5. PMID 27463729 DOI: 10.3390/Antibiotics5030026 |
0.305 |
|
2016 |
Zhang X, Bruning JB, George JH, Abell AD. A mechanistic study on the inhibition of α-chymotrypsin by a macrocyclic peptidomimetic aldehyde. Organic & Biomolecular Chemistry. PMID 27349772 DOI: 10.1039/C6Ob01159D |
0.314 |
|
2015 |
Zhang X, Heng S, Abell AD. Photoregulation of α-Chymotrypsin Activity by Spiropyran-Based Inhibitors in Solution and Attached to an Optical Fiber. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26100654 DOI: 10.1002/Chem.201501488 |
0.313 |
|
2015 |
Tieu W, Polyak SW, Paparella AS, Yap MY, Soares da Costa TP, Ng B, Wang G, Lumb R, Bell JM, Turnidge JD, Wilce MC, Booker GW, Abell AD. Improved Synthesis of Biotinol-5'-AMP: Implications for Antibacterial Discovery. Acs Medicinal Chemistry Letters. 6: 216-20. PMID 25699152 DOI: 10.1021/Ml500475N |
0.315 |
|
2014 |
Tieu W, Jarrad AM, Paparella AS, Keeling KA, Soares da Costa TP, Wallace JC, Booker GW, Polyak SW, Abell AD. Heterocyclic acyl-phosphate bioisostere-based inhibitors of Staphylococcus aureus biotin protein ligase. Bioorganic & Medicinal Chemistry Letters. 24: 4689-93. PMID 25193234 DOI: 10.1016/J.Bmcl.2014.08.030 |
0.311 |
|
2014 |
Chua KC, Pietsch M, Zhang X, Hautmann S, Chan HY, Bruning JB, Gütschow M, Abell AD. Macrocyclic protease inhibitors with reduced peptide character. Angewandte Chemie (International Ed. in English). 53: 7828-31. PMID 24903745 DOI: 10.1002/Anie.201404301 |
0.341 |
|
2014 |
Paparella AS, Soares da Costa TP, Yap MY, Tieu W, Wilce MCJ, Booker GW, Abell AD, Polyak SW. Structure guided design of Biotin protein ligase inhibitors for antibiotic discovery Current Topics in Medicinal Chemistry. 14: 4-20. PMID 24236729 DOI: 10.2174/1568026613666131111103149 |
0.328 |
|
2014 |
Jones SA, Duncan J, Aitken SG, Coxon JM, Abell AD. The preparation of macrocyclic calpain inhibitors by ring closing metathesis and cross metathesis Australian Journal of Chemistry. 67: 1257-1263. DOI: 10.1071/Ch14121 |
0.334 |
|
2013 |
Pehere AD, Pietsch M, Gütschow M, Neilsen PM, Pedersen DS, Nguyen S, Zvarec O, Sykes MJ, Callen DF, Abell AD. Synthesis and extended activity of triazole-containing macrocyclic protease inhibitors Chemistry - a European Journal. 19: 7975-7981. PMID 23606616 DOI: 10.1002/Chem.201204260 |
0.363 |
|
2013 |
Neilsen PM, Pehere AD, Pishas KI, Callen DF, Abell AD. New 26S proteasome inhibitors with high selectivity for chymotrypsin-like activity and p53-dependent cytotoxicity Acs Chemical Biology. 8: 353-359. PMID 23190346 DOI: 10.1021/Cb300549D |
0.311 |
|
2012 |
Soares da Costa TP, Tieu W, Yap MY, Zvarec O, Bell JM, Turnidge JD, Wallace JC, Booker GW, Wilce MC, Abell AD, Polyak SW. Biotin analogues with antibacterial activity are potent inhibitors of biotin protein ligase. Acs Medicinal Chemistry Letters. 3: 509-14. PMID 24900501 DOI: 10.1021/Ml300106P |
0.31 |
|
2012 |
Chen H, Jiao W, Jones MA, Coxon JM, Morton JD, Bickerstaffe R, Pehere AD, Zvarec O, Abell AD. New tripeptide-based macrocyclic calpain inhibitors formed by N-alkylation of histidine. Chemistry & Biodiversity. 9: 2473-84. PMID 23161629 DOI: 10.1002/Cbdv.201200320 |
0.319 |
|
2012 |
Peddie V, Butcher RJ, Robinson WT, Wilce MCJ, Traore DAK, Abell AD. Synthesis and conformation of fluorinated β-peptidic compounds Chemistry - a European Journal. 18: 6655-6662. PMID 22517667 DOI: 10.1002/Chem.201200313 |
0.322 |
|
2012 |
Zvarec O, Polyak SW, Tieu W, Kuan K, Dai H, Pedersen DS, Morona R, Zhang L, Booker GW, Abell AD. 5-Benzylidenerhodanine and 5-benzylidene-2-4-thiazolidinedione based antibacterials Bioorganic and Medicinal Chemistry Letters. 22: 2720-2722. PMID 22444680 DOI: 10.1016/J.Bmcl.2012.02.100 |
0.307 |
|
2012 |
Soares Da Costa TP, Tieu W, Yap MY, Pendini NR, Polyak SW, Pedersen DS, Morona R, Turnidge JD, Wallace JC, Wilce MCJ, Booker GW, Abell AD. Selective inhibition of biotin protein ligase from Staphylococcus aureus Journal of Biological Chemistry. 287: 17823-17832. PMID 22437830 DOI: 10.1074/Jbc.M112.356576 |
0.301 |
|
2012 |
Pehere AD, Abell AD. New β-strand templates constrained by Huisgen cycloaddition Organic Letters. 14: 1330-1333. PMID 22339212 DOI: 10.1021/Ol3002199 |
0.317 |
|
2012 |
Polyak SW, Abell AD, Wilce MCJ, Zhang L, Booker GW. Structure, function and selective inhibition of bacterial acetyl-coa carboxylase Applied Microbiology and Biotechnology. 93: 983-992. PMID 22183085 DOI: 10.1007/S00253-011-3796-Z |
0.317 |
|
2012 |
Peddie V, Abell AD. A study on the diastereoselective synthesis of α-fluorinated β3-amino acids by α-fluorination Helvetica Chimica Acta. 95: 2460-2473. DOI: 10.1002/Hlca.201200520 |
0.322 |
|
2011 |
Pedersen DS, Abell A. 1,2,3-Triazoles in peptidomimetic chemistry European Journal of Organic Chemistry. 2399-2411. DOI: 10.1002/Ejoc.201100157 |
0.333 |
|
2010 |
Pietsch M, Chua KCH, Abell AD. Calpains: Attractive targets for the development of synthetic inhibitors Current Topics in Medicinal Chemistry. 10: 270-293. PMID 20166953 DOI: 10.2174/156802610790725489 |
0.349 |
|
2009 |
Jones SA, Jones MA, McNabb SB, Aitken SG, Coxon JM, Abell AD. N-heterocyclic dipeptide aldehyde calpain inhibitors. Protein and Peptide Letters. 16: 1466-72. PMID 20001909 DOI: 10.2174/092986609789839296 |
0.344 |
|
2009 |
Abell AD, Alexander NA, Aitken SG, Chen H, Coxon JM, Jones MA, McNabb SB, Muscroft-Taylor A. Synthesis of macrocyclic beta-strand templates by ring closing metathesis. The Journal of Organic Chemistry. 74: 4354-6. PMID 19397301 DOI: 10.1021/Jo802723W |
0.326 |
|
2009 |
Abell AD, Jones MA, Coxon JM, Morton JD, Aitken SG, McNabb SB, Lee HY, Mehrtens JM, Alexander NA, Stuart BG, Neffe AT, Bickerstaffe R. Molecular modeling, synthesis, and biological evaluation of macrocyclic calpain inhibitors. Angewandte Chemie (International Ed. in English). 48: 1455-8. PMID 19145612 DOI: 10.1002/Anie.200805014 |
0.649 |
|
2009 |
Jones MA, Coxon JM, McNabb SB, Mehrtens JM, Alexander NA, Jones S, Chen H, Buisan C, Abell AD. Efficient large-scale synthesis of CAT811, a potent calpain inhibitor of interest in the treatment of cataracts Australian Journal of Chemistry. 62: 671-675. DOI: 10.1071/Ch09101 |
0.331 |
|
2008 |
Jones MA, Morton JD, Coxon JM, McNabb SB, Lee HY, Aitken SG, Mehrtens JM, Robertson LJ, Neffe AT, Miyamoto S, Bickerstaffe R, Gately K, Wood JM, Abell AD. Synthesis, biological evaluation and molecular modelling of N-heterocyclic dipeptide aldehydes as selective calpain inhibitors. Bioorganic & Medicinal Chemistry. 16: 6911-23. PMID 18571418 DOI: 10.1016/J.Bmc.2008.05.048 |
0.622 |
|
2008 |
Edmonds MK, Graichen FHM, Gardiner J, Abell AD. Enantioselective synthesis of α-fluorinated β2-amino acids Organic Letters. 10: 885-887. PMID 18232705 DOI: 10.1021/Ol703045Z |
0.322 |
|
2008 |
Pearson D, Abell AD. D-Leu-L-Phe-containing dipeptide inhibitors of α-chymotrypsin - The role of the N- and C-termini in enzyme affinity Arkivoc. 2008: 85-94. DOI: 10.3998/Ark.5550190.0009.C10 |
0.303 |
|
2008 |
Vernall AJ, Ballet S, Abell AD. Cross-metathesis and ring-closing metathesis reactions of amino acid-based substrates Tetrahedron. 64: 3980-3997. DOI: 10.1016/J.Tet.2008.02.043 |
0.33 |
|
2007 |
Abell AD, Jones MA, Neffe AT, Aitken SG, Cain TP, Payne RJ, McNabb SB, Coxon JM, Stuart BG, Pearson D, Lee HY, Morton JD. Investigation into the P3 binding domain of m-calpain using photoswitchable diazo- and triazene-dipeptide aldehydes: new anticataract agents. Journal of Medicinal Chemistry. 50: 2916-20. PMID 17497840 DOI: 10.1021/Jm061455N |
0.624 |
|
2007 |
McCarthy AR, Hartmann RW, Abell AD. Evaluation of 4′-substituted bicyclic pyridones as non-steroidal inhibitors of steroid 5α-reductase Bioorganic and Medicinal Chemistry Letters. 17: 3603-3607. PMID 17490876 DOI: 10.1016/J.Bmcl.2007.04.049 |
0.365 |
|
2007 |
Payne RJ, Riboldi-Tunnicliffe A, Kerbarh O, Abell AD, Lapthorn AJ, Abell C. Design, synthesis, and structural studies on potent biaryl inhibitors of type II dehydroquinases. Chemmedchem. 2: 1010-3. PMID 17487901 DOI: 10.1002/Cmdc.200700062 |
0.31 |
|
2007 |
Payne RJ, Peyrot F, Kerbarh O, Abell AD, Abell C. Rational design, synthesis, and evaluation of nanomolar type II dehydroquinase inhibitors. Chemmedchem. 2: 1015-29. PMID 17487900 DOI: 10.1002/Cmdc.200700032 |
0.347 |
|
2007 |
Zaman S, Kitamura M, Abell AD. Synthesis of 5-phenyl 2-functionalized pyrroles by amino Heck and Tandem amino Heck carbonylation reactions Australian Journal of Chemistry. 60: 624-626. DOI: 10.1071/Ch07132 |
0.343 |
|
2006 |
Zaman S, Campaner P, Abell AD. Synthesis of amino acid derived seven-membered lactams by RCM and their evaluation against HIV protease Bioorganic and Medicinal Chemistry. 14: 8323-8331. PMID 17010620 DOI: 10.1016/J.Bmc.2006.09.009 |
0.341 |
|
2006 |
Pearson D, Abell AD. Photoswitch inhibitors of α-chymotrypsin - Increased substitution and peptidic character in peptidomimetic boronate esters Organic and Biomolecular Chemistry. 4: 3618-3625. PMID 16990937 DOI: 10.1039/B609320P |
0.351 |
|
2006 |
Gardiner J, Aitken SG, McNabb SB, Zaman S, Abell AD. Ring closing metathesis of α- and β-amino acid derived dienes Journal of Organometallic Chemistry. 691: 5487-5496. DOI: 10.1016/J.Jorganchem.2006.09.061 |
0.313 |
|
2005 |
Neffe AT, Abell AD. Developments in the design and synthesis of calpain inhibitors Current Opinion in Drug Discovery and Development. 8: 684-700. PMID 16312145 |
0.607 |
|
2005 |
Payne RJ, Toscano MD, Bulloch EM, Abell AD, Abell C. Design and synthesis of aromatic inhibitors of anthranilate synthase. Organic & Biomolecular Chemistry. 3: 2271-81. PMID 16010361 DOI: 10.1039/B503802B |
0.343 |
|
2005 |
Zaman S, Mitsuru K, Abell AD. Synthesis of trisubstituted imidazoles by palladium-catalyzed cyclization of O-pentafluorobenzoylamidoximes: Application to amino acid mimetics with a C-terminal imidazole Organic Letters. 7: 609-611. PMID 15704906 DOI: 10.1021/Ol047628P |
0.314 |
|
2005 |
Abell AD, Brown KM, Coxon JM, Jones MA, Miyamoto S, Neffe AT, Nikkel JM, Stuart BG. Synthesis and evaluation of eight-membered cyclic pseudo-dipeptides Peptides. 26: 251-258. PMID 15629536 DOI: 10.1016/J.Peptides.2004.09.006 |
0.665 |
|
2005 |
Abell AD, Harvey AJ. Synthesis of a [1,4]dioxane-2,5-dione based-peptidomimetic scaffold Arkivoc. 2006: 72-76. DOI: 10.3998/Ark.5550190.0007.307 |
0.306 |
|
2004 |
Payne RJ, Daines AM, Clark BM, Abell AD. Synthesis and protein conjugation studies of vitamin K analogues Bioorganic and Medicinal Chemistry. 12: 5785-5791. PMID 15498655 DOI: 10.1016/J.Bmc.2004.08.037 |
0.301 |
|
2004 |
Daines AM, Abell AD. The preparation of side chain functionalized analogues of coenzyme Q for protein conjugation studies. Organic & Biomolecular Chemistry. 2: 2371-5. PMID 15305221 DOI: 10.1039/B407659A |
0.328 |
|
2004 |
Gardiner J, Abell AD. Synthesis and solid state conformation of phenylalanine mimetics constrained in a proline-like conformation. Organic & Biomolecular Chemistry. 2: 2365-70. PMID 15305220 DOI: 10.1039/B406450J |
0.344 |
|
2004 |
Gardiner J, Anderson KH, Downard A, Abell AD. Synthesis of cyclic beta-amino acid esters from methionine, allylglycine, and serine. The Journal of Organic Chemistry. 69: 3375-82. PMID 15132545 DOI: 10.1021/Jo049794G |
0.32 |
|
2004 |
Abell AD. Chemistry at the Interface Australian Journal of Chemistry. 57: 819. DOI: 10.1071/Ch04180 |
0.316 |
|
2004 |
Payne RJ, Brown KM, Coxon JM, Morton JD, Lee HYY, Abell AD. Peptidic aldehydes based on α- and β-amino acids: Synthesis, inhibition of m-Calpain, and anti-cataract properties Australian Journal of Chemistry. 57: 877-884. DOI: 10.1071/Ch04080 |
0.356 |
|
2004 |
Le Sann C, Abell AD. Synthesis and properties of a mesylated ArgoGel resin Australian Journal of Chemistry. 57: 355-358. DOI: 10.1071/Ch03247 |
0.305 |
|
2003 |
Martyn DC, Vernall AJ, Clark BM, Abell AD. Ring-deactivated hydroxyalkylpyrrole-based inhibitors of alpha-chymotrypsin: synthesis and mechanism of action. Organic & Biomolecular Chemistry. 1: 2103-10. PMID 12945901 DOI: 10.1039/B302411C |
0.301 |
|
2003 |
Humphries ME, Murphy J, Phillips AJ, Abell AD. Synthesis of functionalized piperidinones. The Journal of Organic Chemistry. 68: 2432-6. PMID 12636413 DOI: 10.1021/Jo0267091 |
0.508 |
|
2003 |
Le Sann C, Abell C, Abell AD. A convenient method for the synthesis of dehydroquinic acid Synthetic Communications. 33: 527-533. DOI: 10.1081/Scc-120015805 |
0.318 |
|
2003 |
Gardiner J, Abell AD. A diastereoselective synthesis of the tetrahydropyridazinone core of 2-oxo-1,6-diazobicyclo[4.3.0]nonane-9-carboxylate-based peptidomimetics starting from (S)-phenylalanine Tetrahedron Letters. 44: 4227-4230. DOI: 10.1016/S0040-4039(03)00882-7 |
0.33 |
|
2002 |
Abell AD, Gardiner J. Synthesis of substituted cyclohexenyl-based beta-amino acids by ring-closing metathesis. Organic Letters. 4: 3663-6. PMID 12375913 DOI: 10.1021/Ol0266121 |
0.324 |
|
2002 |
Le Sann C, Abell C, Abell AD. A simple method for the preparation of 3-hydroxyiminodehydroquinate, a potent inhibitor of type II dehydroquinase Journal of the Chemical Society. Perkin Transactions 1. 2065-2068. DOI: 10.1039/B206066C |
0.331 |
|
2002 |
May BCH, Abell AD. α-methylene tetrazole-based peptidomimetics: Synthesis and inhibition of hiv protease Journal of the Chemical Society. Perkin Transactions 1. 2: 172-178. DOI: 10.1039/B109128J |
0.315 |
|
2002 |
Abell AD. Heterocyclic-based peptidomimetics Letters in Peptide Science. 8: 267-272. DOI: 10.1023/A:1016216828677 |
0.333 |
|
2001 |
May BC, Abell AD. The synthesis and solid state structure of (8S)-8-benzyl-8,9-dihydro-7H-tetrazolo[1,5-d][1,4]diazepin-6-one. Chemical Communications (Cambridge, England). 2080-1. PMID 12240172 DOI: 10.1039/B106175P |
0.315 |
|
2001 |
Harvey AJ, Abell AD. Alpha-ketoester-based photobiological switches: synthesis, peptide chain extension and assay against alpha-chymotrypsin. Bioorganic & Medicinal Chemistry Letters. 11: 2441-4. PMID 11549442 DOI: 10.1016/S0960-894X(01)00464-4 |
0.314 |
|
2001 |
Edmonds MK, Abell AD. Design and synthesis of a conformationally restricted trans peptide isostere based on the bioactive conformations of saquinavir and nelfinavir. The Journal of Organic Chemistry. 66: 3747-52. PMID 11374993 DOI: 10.1021/Jo0016834 |
0.332 |
|
2001 |
Martyn DC, Hoult DA, Abell AD. Stereocontrol of the Horner-Wadsworth-Emmons Reaction: Application to the Synthesis of HIV-1 Protease Inhibitors Australian Journal of Chemistry. 54: 391-396. DOI: 10.1071/Ch01093 |
0.339 |
|
2001 |
Zubarev VY, Trifonov RE, Filichev VV, Ostrovskii VA, Abell AD, Edmonds MK. Synthesis, X-ray and conformational studies of novel tetrazole-containing macrocycles: 4,13-dioxa-1,7,8,9,17,18,19,20-octaazatricyclo[14.2.1.17,10]icosa-8,10(20),16(19),17-tetraene and 4,14-dioxa-1,7,8,9,10,18,19,20-octaazatricyclo[15.2.1.07,10]icosa-8,10,17(20),18-tetraene Journal of the Chemical Society-Perkin Transactions 1. 417-421. DOI: 10.1039/B006217K |
0.307 |
|
2001 |
May BCH, Abell AD. The synthesis and crystal structure of alpha-keto tetrazole-based dipeptide mimics Tetrahedron Letters. 42: 5641-5644. DOI: 10.1016/S0040-4039(01)01101-7 |
0.343 |
|
2000 |
Abell AD, Prince MJ, McNulty AM, Neubauer BL. Simple bi- and tricyclic inhibitors of human steroid 5alpha-reductase. Bioorganic & Medicinal Chemistry Letters. 10: 1909-11. PMID 10987415 DOI: 10.1016/S0960-894X(00)00368-1 |
0.325 |
|
2000 |
Gerrard JA, Prince MJ, Abell AD. Kinetic characterisation of ene-diol-based inhibitors of alpha-amylase. Bioorganic & Medicinal Chemistry Letters. 10: 1575-6. PMID 10915054 DOI: 10.1016/S0960-894X(00)00288-2 |
0.3 |
|
2000 |
Phillips AJ, Morris JC, Abell AD. Progress towards an intramolecular Diels-Alder ring-expansion approach to taxinine: The interplay of Lewis acids and high pressure Tetrahedron Letters. 41: 2723-2727. DOI: 10.1016/S0040-4039(00)00248-3 |
0.506 |
|
1999 |
Nabbs BK, Abell AD. The synthesis and P388 cytotoxicity of mycalazol 11 and related 5-acyl-2-hydroxymethylpyrroles. Bioorganic & Medicinal Chemistry Letters. 9: 505-8. PMID 10091711 DOI: 10.1016/S0960-894X(99)00021-9 |
0.321 |
|
1999 |
Abell AD, Oldham MD. Leucine-phenylalanine dipeptide-based N-mesyloxysuccinimides: synthesis of all four stereoisomers and their assay against serine proteases. Bioorganic & Medicinal Chemistry Letters. 9: 497-500. PMID 10091709 DOI: 10.1016/S0960-894X(99)00017-7 |
0.321 |
|
1999 |
May BCH, Abell AD. A convenient preparation of (2SR,3S)-3-amino-2-hydroxy-4-phenylbutanoic acid; an important peptide bond isostere Synthetic Communications. 29: 2515-2525. DOI: 10.1080/00397919908086259 |
0.345 |
|
1999 |
Abell AD, Oldham MD, Moore MM, Robinson WT. The synthesis and X-ray crystal structure of phenylalanine-based N-benzyloxysuccinimides Australian Journal of Chemistry. 52: 977-981. DOI: 10.1071/Ch99055 |
0.305 |
|
1999 |
Abell AD, Nabbs BK, Battersby AR, Thompson A, Dolphin D. Synthesis and properties of ring-deactivated Deuterated (hydroxymethyl)pyrroles Chemtracts. 12: 534-538. DOI: 10.1021/Ja973656+ |
0.531 |
|
1999 |
Abell AD, Nabbs BK, Battersby AR, Thompson A, Dolphin D. Synthesis and properties of ring-deactivated Deuterated (hydroxymethyl)pyrroles Chemtracts. 12: 534-538. DOI: 10.1021/ja973656+ |
0.453 |
|
1998 |
Abell AD, Phillips AJ, Budhia S, McNulty AM, Neubauer BL. The preparation and biological activity of lactam-based, non-steroidal, inhibitors of human type-1 steroid 5α-reductase Australian Journal of Chemistry. 51: 389-396. DOI: 10.1071/C97130 |
0.498 |
|
1998 |
Abell AD, Nabbs BK, Battersby AR. The reaction of N-magnesium derivatives of pyrroles with N- mesylchloromethylpyrroles: A synthesis of dipyrrylmethanes Journal of Organic Chemistry. 63: 8163-8169. DOI: 10.1021/Jo980573I |
0.527 |
|
1998 |
Abell AD, Gardiner J, Phillips AJ, Robinson WT. Synthesis and X-ray structure of a 1,2,3,6-tetrahydropyridine-based phenylalanine mimetic Tetrahedron Letters. 39: 9563-9566. DOI: 10.1016/S0040-4039(98)02125-X |
0.51 |
|
1997 |
Carr AC, Winterbourn CC, Blunt JW, Phillips AJ, Abell AD. Nuclear magnetic resonance characterization of 6 alpha-chloro-5 beta-cholestane-3 beta,5-diol formed from the reaction of hypochlorous acid with cholesterol. Lipids. 32: 363-7. PMID 9113623 DOI: 10.1007/S11745-997-0046-8 |
0.441 |
|
1997 |
Abell AD, Brandt M, Levy MA, Holt DA. Preparation and biological activity of tricyclic non-steroidal inhibitors of human steroid 5α-reductase Journal of the Chemical Society - Perkin Transactions 1. 1663-1667. DOI: 10.1039/A608169J |
0.337 |
|
1997 |
Abell AD, Blunt JW, Foulds GJ, Munro MHG. Chemistry of the mycalamides: Antiviral and antitumour compounds from a New Zealand marine sponge. Part 6. The synthesis and testing of analogues of the C(7)-C(10) fragment Journal of the Chemical Society - Perkin Transactions 1. 1647-1654. DOI: 10.1039/A608168A |
0.314 |
|
1997 |
Abell AD, Edwards RA, Oldham MD. Chemistry and X-ray crystallographic structure of N-protected (5-oxo-1,3-oxazolidin-4-yl)acetic acids: Versatile intermediates in the synthesis of peptidomimetics Journal of the Chemical Society - Perkin Transactions 1. 1655-1662. DOI: 10.1039/A608165G |
0.347 |
|
1996 |
Abell AD, Taylor JM, Oldham MD. Self-addition products from the alkylation of amino acid-derived oxazolidinones: X-ray molecular structures of (2R,4S,1′S)-3-benzoyl-4-[benzoylamino(phenyl)methyl]-4-benzyl-2-phenyl-1, 3-oxazolidin-5-one, (2R,4S,1′S)- and (2R,4S,1′R)-3-benzoyl-4-[benzoylamino(phenyl)methyl]-4-isopropyl-2-phenyl- 1,3-oxazolidin-5-one Journal of the Chemical Society - Perkin Transactions 1. 1299-1304. DOI: 10.1039/P19960001299 |
0.301 |
|
1996 |
Abell AD, Brandt M, Levy MA, Holt DA. A comparison of steroidal and non-steroidal inhibitors of human steroid 5α-reductase: New tricyclic aryl acid inhibitors of the type-1 isozyme Bioorganic and Medicinal Chemistry Letters. 6: 481-484. DOI: 10.1016/0960-894X(96)00054-6 |
0.335 |
|
1995 |
Abell AD, Oldham MD, Taylor JM. Synthesis of phenylalanine-based cyclic acylated enamino ester dipeptide analogues: Inhibitors of α-chymotrypsin. X-ray molecular structure of (2′S,4′R)-4′-benzyl-3′-benzyloxycarbonyl-5′-oxo- 2′-phenyloxazolidin-4′-ylacetic acid Journal of the Chemical Society, Perkin Transactions 1. 953-961. DOI: 10.1039/P19950000953 |
0.371 |
|
1995 |
Abell AD, Oldham MD, Taylor JM. Synthesis of cyclic acylated enamino esters from enol lactones, 4-keto amides, and 5-hydroxy lactams Journal of Organic Chemistry. 60: 1214-1220. DOI: 10.1021/Jo00110A026 |
0.376 |
|
1994 |
Abell AD, Brandt M, Levy MA, Holt DA. A non-steroidal diene acid inhibitor of human type 2 stereoid 5α-reductase Bioorganic and Medicinal Chemistry Letters. 4: 2327-2330. DOI: 10.1016/0960-894X(94)85034-8 |
0.328 |
|
1993 |
Abell A, Litten J. Synthesis and Amino Acid Chain Extension of 1-Acylated Hydroxymethylpyrroles Australian Journal of Chemistry. 46: 1473. DOI: 10.1071/Ch9931473 |
0.31 |
|
1993 |
Abell AD, Hoult DA, Morris KM, Taylor JM, Trent JO. Halogenation of keto acid phosphoranes: Synthesis of halo enol lactones and haloallenes Journal of Organic Chemistry. 58: 1531-1537. DOI: 10.1021/Jo00058A039 |
0.322 |
|
1993 |
Abell AD, Taylor JM. Synthesis of cyclic acylated enamino ester dipeptide analogues via the bromolactonization of a keto acid phosphorane Journal of Organic Chemistry. 58: 14-15. DOI: 10.1021/Jo00053A006 |
0.331 |
|
1992 |
Abell AD, Litten JC. Synthesis and hydrolysis of dipeptide isosteres containing a proline analogue with latent reactivity Tetrahedron Letters. 33: 3005-3008. DOI: 10.1016/S0040-4039(00)79584-0 |
0.356 |
|
1992 |
Abell AD, Hoult DA, Jamieson EJ. Synthesis of 1,2-disubstituted pyrroles: A cis peptide bond surrogate Tetrahedron Letters. 33: 5831-5832. DOI: 10.1016/0040-4039(92)89043-C |
0.322 |
|
1991 |
Abell A, Hartshorn M, Maclennan M, Robinson W, Wright G. Reactions of 1,4-Dimethyl-4-nitro-cyclohexa-2,5-dien-1-yl Acetates With Nitrogen Dioxide; the Formation of Polynitro Cyclohexenyl Esters Australian Journal of Chemistry. 44: 43. DOI: 10.1071/Ch9910043 |
0.341 |
|
1990 |
Abell AD, Morris KB, Litten JC. Synthesis and deprotection of [1-(ethoxycarbonyl)-4-[(diphenylmethoxy)carbonyl]-1-methyl-2-oxobutyl]- triphenylphosphonium chloride: A key intermediate in the Wittig reaction between a cyclic anhydride and a stabilized ylide Journal of Organic Chemistry. 55: 5217-5221. DOI: 10.1021/Jo00305A013 |
0.301 |
|
1989 |
Abell A, Hartshorn M, Robinson W, Waller A, Wright G. Reactions of 4-Methyl-1-(1′-methylethyl)-4-nitrocyclohexa-2,5-dien-1-yl Acetates With Nitrogen Dioxide; Towards a Mechanism for the Formation of Polynitro Cyclohexenyl Esters on Reaction of p-Cymene With Nitrogen Dioxide in Acetic Anhydride Australian Journal of Chemistry. 42: 2225. DOI: 10.1071/Ch9892225 |
0.32 |
|
1989 |
Abell AD, Trent JO. A novel bromo lactonization of acylated phosphoranes. A new route to bromo enol lactones Journal of the Chemical Society, Chemical Communications. 409-410. DOI: 10.1039/C39890000409 |
0.322 |
|
1988 |
Abell A, Clark B, Robinson W. A Mechanistic Study of the Wittig Reaction Between a Cyclic Anhydride and a Stabilized Phosphorane Australian Journal of Chemistry. 41: 1243. DOI: 10.1071/Ch9881243 |
0.314 |
|
1987 |
Schauder JR, Jendrezejewski S, Abell A, Hart GJ, Battersby AR. Stereochemistry of formation of the hydroxymethyl group of hydroxymethylbilane, the precursor of uro'gen-III Journal of the Chemical Society, Chemical Communications. 436-438. DOI: 10.1039/C39870000436 |
0.49 |
|
1986 |
ABELL AD, HEINICKE GW, MASSY-WESTROPP RA. ChemInform Abstract: Synthesis of Dialkyl Hex-2-yne-1,6-dioates and Hept-2-yne-1,7-dioates. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198603132 |
0.593 |
|
1985 |
Abell A, Massy-Westropp R, Reynolds G. Rearrangement of Freelingyne with Base Australian Journal of Chemistry. 38: 1129. DOI: 10.1071/Ch9851129 |
0.6 |
|
1985 |
Abell A, Massy-Westropp R. Mechanism of Acetal Cleavage with Methylmagnesium Iodide Australian Journal of Chemistry. 38: 1031. DOI: 10.1071/Ch9851031 |
0.612 |
|
1985 |
Abell AD, Heinicke GW, Massy-Westropp RA. Synthesis of Dialkyl Hex-2-yne-1,6-dioates and Hept-2-yne-1,7-dioates Synthesis. 1985: 764-766. DOI: 10.1055/S-1985-31339 |
0.595 |
|
1985 |
Abell AD, Massy-Westropp RA. Regioselective bond cleavage and coordination effects in the reduction of some acetals with lithium in ammonia Tetrahedron. 41: 2451-2464. DOI: 10.1016/S0040-4020(01)96640-2 |
0.62 |
|
1984 |
Abell A, Dimitriadis E, Massy-Westropp R. Stereospecific formation of tetrahydrofurans from substituted 2,8-Dioxabicyclo[3.2.1]oct-3-ylmethanols Australian Journal of Chemistry. 37: 395. DOI: 10.1071/Ch9840395 |
0.634 |
|
1984 |
ABELL AD, DIMITRIADIS E, MASSY-WESTROPP RA. ChemInform Abstract: STEREOSPECIFIC FORMATION OF TETRAHYDROFURANS FROM SUBSTITUTED 2,8-DIOXABICYCLO(3.2.1)OCT-3-YLMETHANOLS Chemischer Informationsdienst. 15. DOI: 10.1002/Chin.198438170 |
0.583 |
|
1983 |
ABELL AD, DOYLE IR, MASSY-WESTROPP RA. ChemInform Abstract: THE WITTIG REACTION WITH GLUTARIC AND SUCCINIC ANHYDRIDES Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198314128 |
0.565 |
|
1982 |
Abell A, Doyle I, Massy-Westropp R. The Wittig reaction with glutaric and succinic anhydrides Australian Journal of Chemistry. 35: 2277. DOI: 10.1071/Ch9822277 |
0.634 |
|
1982 |
Abell A, Massy-Westropp R. Aspects of the mechanism of the Wittig reaction between cyclic anhydrides and stabilized phosphoranes Australian Journal of Chemistry. 35: 2077. DOI: 10.1071/Ch9822077 |
0.626 |
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