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Andrew D. Abell - Publications

Affiliations: 
University of Adelaide, Adelaide, South Australia, Australia 
Area:
design, synthesis and biological testing of inhibitors of enzymes of mechanistic and therapeutic importance
Website:
http://www.adelaide.edu.au/directory/andrew.abell

117 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2020 Yeoh YQ, Horsley J, Yu J, Polyak SW, Jovcevski B, Abell AD. Short Photoswitchable Antibacterial Peptides. Chemmedchem. PMID 32558320 DOI: 10.1002/Cmdc.202000280  0.3
2020 Yeoh YQ, Horsley JR, Polyak SW, Abell AD. A hypoxia-activated antibacterial prodrug. Bioorganic & Medicinal Chemistry Letters. 127140. PMID 32247730 DOI: 10.1016/J.Bmcl.2020.127140  0.3
2019 Lee KJ, Tieu W, Blanco-Rodriguez B, Paparella AS, Yu J, Hayes A, Feng J, Marshall AC, Noll B, Milne R, Cini D, Wilce MCJ, Booker GW, Bruning JB, Polyak SW, ... Abell AD, et al. Sulfonamide-based inhibitors of biotin protein ligase as new antibiotic leads. Acs Chemical Biology. PMID 31407891 DOI: 10.1021/Acschembio.9B00463  0.339
2018 Pehere AD, Nguyen S, Garlick SK, Wilson DW, Hudson I, Sykes MJ, Morton JD, Abell AD. Tripeptide analogues of MG132 as protease inhibitors. Bioorganic & Medicinal Chemistry. PMID 30581047 DOI: 10.1016/J.Bmc.2018.12.022  0.314
2018 Schumann NC, Bruning J, Marshall AC, Abell AD. The role of N-terminal heterocycles in hydrogen bonding to α-chymotrypsin. Bioorganic & Medicinal Chemistry Letters. PMID 30579793 DOI: 10.1016/J.Bmcl.2018.12.032  0.302
2018 Abell AD, Yu J, Polyak S, Horsley J, Yeoh YQ. Photopharmacological Control of Cyclic Antimicrobial Peptides. Chembiochem : a European Journal of Chemical Biology. PMID 30324702 DOI: 10.1002/Cbic.201800618  0.302
2018 Hochscherf J, Pietsch M, Tieu W, Kuan K, Abell AD, Gütschow M, Niefind K. Crystal structure of highly glycosylated human leukocyte elastase in complex with an S2' site binding inhibitor. Acta Crystallographica. Section F, Structural Biology Communications. 74: 480-489. PMID 30084397 DOI: 10.1107/S2053230X1800537X  0.311
2018 Wegener KL, McGrath AE, Dixon NE, Oakley AJ, Scanlon DB, Abell AD, Bruning J. Rational design of a 310-helical PIP-box mimetic targeting PCNA - the human sliding clamp. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 29917264 DOI: 10.1002/Chem.201801734  0.309
2017 Paparella AS, Lee KJ, Hayes A, Feng J, Feng Z, Cini D, Deshmukh S, Booker GW, Wilce MCJ, Polyak SW, Abell AD. Halogenation of biotin protein ligase inhibitors improves whole cell activity against Staphylococcus aureus. Acs Infectious Diseases. PMID 29131575 DOI: 10.1021/Acsinfecdis.7B00134  0.302
2017 Blanco B, Palasis KA, Adwal A, Callen DF, Abell AD. Azobenzene-containing photoswitchable proteasome inhibitors with selective activity and cellular toxicity. Bioorganic & Medicinal Chemistry. PMID 28642029 DOI: 10.1016/J.Bmc.2017.06.011  0.312
2017 Frkic RL, Rodriguez BB, Chang MR, Kuruvilla D, Ciesla A, Abell AD, Kamenecka TM, Griffin PR, Bruning JB. Structure-Activity Relationship of 2,4-dichloro-N-(3,5-dichloro-4-(quinolin-3-yloxy)phenyl)benzenesulfonamide (INT131) Analogs for PPARγ-Targeted Antidiabetics. Journal of Medicinal Chemistry. PMID 28485590 DOI: 10.1021/Acs.Jmedchem.6B01727  0.305
2017 Pehere AD, Zhang X, Abell AD. Macrocyclic Peptidomimetics Prepared by Ring-Closing Metathesis and Azide–Alkyne Cycloaddition Australian Journal of Chemistry. 70: 138. DOI: 10.1071/Ch16532  0.336
2016 Feng J, Paparella AS, Tieu W, Heim D, Clark S, Hayes A, Booker GW, Polyak SW, Abell AD. New Series of BPL Inhibitors To Probe the Ribose-Binding Pocket of Staphylococcus aureus Biotin Protein Ligase. Acs Medicinal Chemistry Letters. 7: 1068-1072. PMID 27994739 DOI: 10.1021/Acsmedchemlett.6B00248  0.337
2016 Feng J, Paparella AS, Booker GW, Polyak SW, Abell AD. Biotin Protein Ligase Is a Target for New Antibacterials. Antibiotics (Basel, Switzerland). 5. PMID 27463729 DOI: 10.3390/Antibiotics5030026  0.305
2016 Zhang X, Bruning JB, George JH, Abell AD. A mechanistic study on the inhibition of α-chymotrypsin by a macrocyclic peptidomimetic aldehyde. Organic & Biomolecular Chemistry. PMID 27349772 DOI: 10.1039/C6Ob01159D  0.314
2015 Zhang X, Heng S, Abell AD. Photoregulation of α-Chymotrypsin Activity by Spiropyran-Based Inhibitors in Solution and Attached to an Optical Fiber. Chemistry (Weinheim An Der Bergstrasse, Germany). PMID 26100654 DOI: 10.1002/Chem.201501488  0.313
2015 Tieu W, Polyak SW, Paparella AS, Yap MY, Soares da Costa TP, Ng B, Wang G, Lumb R, Bell JM, Turnidge JD, Wilce MC, Booker GW, Abell AD. Improved Synthesis of Biotinol-5'-AMP: Implications for Antibacterial Discovery. Acs Medicinal Chemistry Letters. 6: 216-20. PMID 25699152 DOI: 10.1021/Ml500475N  0.315
2014 Tieu W, Jarrad AM, Paparella AS, Keeling KA, Soares da Costa TP, Wallace JC, Booker GW, Polyak SW, Abell AD. Heterocyclic acyl-phosphate bioisostere-based inhibitors of Staphylococcus aureus biotin protein ligase. Bioorganic & Medicinal Chemistry Letters. 24: 4689-93. PMID 25193234 DOI: 10.1016/J.Bmcl.2014.08.030  0.311
2014 Chua KC, Pietsch M, Zhang X, Hautmann S, Chan HY, Bruning JB, Gütschow M, Abell AD. Macrocyclic protease inhibitors with reduced peptide character. Angewandte Chemie (International Ed. in English). 53: 7828-31. PMID 24903745 DOI: 10.1002/Anie.201404301  0.341
2014 Paparella AS, Soares da Costa TP, Yap MY, Tieu W, Wilce MCJ, Booker GW, Abell AD, Polyak SW. Structure guided design of Biotin protein ligase inhibitors for antibiotic discovery Current Topics in Medicinal Chemistry. 14: 4-20. PMID 24236729 DOI: 10.2174/1568026613666131111103149  0.328
2014 Jones SA, Duncan J, Aitken SG, Coxon JM, Abell AD. The preparation of macrocyclic calpain inhibitors by ring closing metathesis and cross metathesis Australian Journal of Chemistry. 67: 1257-1263. DOI: 10.1071/Ch14121  0.334
2013 Pehere AD, Pietsch M, Gütschow M, Neilsen PM, Pedersen DS, Nguyen S, Zvarec O, Sykes MJ, Callen DF, Abell AD. Synthesis and extended activity of triazole-containing macrocyclic protease inhibitors Chemistry - a European Journal. 19: 7975-7981. PMID 23606616 DOI: 10.1002/Chem.201204260  0.363
2013 Neilsen PM, Pehere AD, Pishas KI, Callen DF, Abell AD. New 26S proteasome inhibitors with high selectivity for chymotrypsin-like activity and p53-dependent cytotoxicity Acs Chemical Biology. 8: 353-359. PMID 23190346 DOI: 10.1021/Cb300549D  0.311
2012 Soares da Costa TP, Tieu W, Yap MY, Zvarec O, Bell JM, Turnidge JD, Wallace JC, Booker GW, Wilce MC, Abell AD, Polyak SW. Biotin analogues with antibacterial activity are potent inhibitors of biotin protein ligase. Acs Medicinal Chemistry Letters. 3: 509-14. PMID 24900501 DOI: 10.1021/Ml300106P  0.31
2012 Chen H, Jiao W, Jones MA, Coxon JM, Morton JD, Bickerstaffe R, Pehere AD, Zvarec O, Abell AD. New tripeptide-based macrocyclic calpain inhibitors formed by N-alkylation of histidine. Chemistry & Biodiversity. 9: 2473-84. PMID 23161629 DOI: 10.1002/Cbdv.201200320  0.319
2012 Peddie V, Butcher RJ, Robinson WT, Wilce MCJ, Traore DAK, Abell AD. Synthesis and conformation of fluorinated β-peptidic compounds Chemistry - a European Journal. 18: 6655-6662. PMID 22517667 DOI: 10.1002/Chem.201200313  0.322
2012 Zvarec O, Polyak SW, Tieu W, Kuan K, Dai H, Pedersen DS, Morona R, Zhang L, Booker GW, Abell AD. 5-Benzylidenerhodanine and 5-benzylidene-2-4-thiazolidinedione based antibacterials Bioorganic and Medicinal Chemistry Letters. 22: 2720-2722. PMID 22444680 DOI: 10.1016/J.Bmcl.2012.02.100  0.307
2012 Soares Da Costa TP, Tieu W, Yap MY, Pendini NR, Polyak SW, Pedersen DS, Morona R, Turnidge JD, Wallace JC, Wilce MCJ, Booker GW, Abell AD. Selective inhibition of biotin protein ligase from Staphylococcus aureus Journal of Biological Chemistry. 287: 17823-17832. PMID 22437830 DOI: 10.1074/Jbc.M112.356576  0.301
2012 Pehere AD, Abell AD. New β-strand templates constrained by Huisgen cycloaddition Organic Letters. 14: 1330-1333. PMID 22339212 DOI: 10.1021/Ol3002199  0.317
2012 Polyak SW, Abell AD, Wilce MCJ, Zhang L, Booker GW. Structure, function and selective inhibition of bacterial acetyl-coa carboxylase Applied Microbiology and Biotechnology. 93: 983-992. PMID 22183085 DOI: 10.1007/S00253-011-3796-Z  0.317
2012 Peddie V, Abell AD. A study on the diastereoselective synthesis of α-fluorinated β3-amino acids by α-fluorination Helvetica Chimica Acta. 95: 2460-2473. DOI: 10.1002/Hlca.201200520  0.322
2011 Pedersen DS, Abell A. 1,2,3-Triazoles in peptidomimetic chemistry European Journal of Organic Chemistry. 2399-2411. DOI: 10.1002/Ejoc.201100157  0.333
2010 Pietsch M, Chua KCH, Abell AD. Calpains: Attractive targets for the development of synthetic inhibitors Current Topics in Medicinal Chemistry. 10: 270-293. PMID 20166953 DOI: 10.2174/156802610790725489  0.349
2009 Jones SA, Jones MA, McNabb SB, Aitken SG, Coxon JM, Abell AD. N-heterocyclic dipeptide aldehyde calpain inhibitors. Protein and Peptide Letters. 16: 1466-72. PMID 20001909 DOI: 10.2174/092986609789839296  0.344
2009 Abell AD, Alexander NA, Aitken SG, Chen H, Coxon JM, Jones MA, McNabb SB, Muscroft-Taylor A. Synthesis of macrocyclic beta-strand templates by ring closing metathesis. The Journal of Organic Chemistry. 74: 4354-6. PMID 19397301 DOI: 10.1021/Jo802723W  0.326
2009 Abell AD, Jones MA, Coxon JM, Morton JD, Aitken SG, McNabb SB, Lee HY, Mehrtens JM, Alexander NA, Stuart BG, Neffe AT, Bickerstaffe R. Molecular modeling, synthesis, and biological evaluation of macrocyclic calpain inhibitors. Angewandte Chemie (International Ed. in English). 48: 1455-8. PMID 19145612 DOI: 10.1002/Anie.200805014  0.649
2009 Jones MA, Coxon JM, McNabb SB, Mehrtens JM, Alexander NA, Jones S, Chen H, Buisan C, Abell AD. Efficient large-scale synthesis of CAT811, a potent calpain inhibitor of interest in the treatment of cataracts Australian Journal of Chemistry. 62: 671-675. DOI: 10.1071/Ch09101  0.331
2008 Jones MA, Morton JD, Coxon JM, McNabb SB, Lee HY, Aitken SG, Mehrtens JM, Robertson LJ, Neffe AT, Miyamoto S, Bickerstaffe R, Gately K, Wood JM, Abell AD. Synthesis, biological evaluation and molecular modelling of N-heterocyclic dipeptide aldehydes as selective calpain inhibitors. Bioorganic & Medicinal Chemistry. 16: 6911-23. PMID 18571418 DOI: 10.1016/J.Bmc.2008.05.048  0.622
2008 Edmonds MK, Graichen FHM, Gardiner J, Abell AD. Enantioselective synthesis of α-fluorinated β2-amino acids Organic Letters. 10: 885-887. PMID 18232705 DOI: 10.1021/Ol703045Z  0.322
2008 Pearson D, Abell AD. D-Leu-L-Phe-containing dipeptide inhibitors of α-chymotrypsin - The role of the N- and C-termini in enzyme affinity Arkivoc. 2008: 85-94. DOI: 10.3998/Ark.5550190.0009.C10  0.303
2008 Vernall AJ, Ballet S, Abell AD. Cross-metathesis and ring-closing metathesis reactions of amino acid-based substrates Tetrahedron. 64: 3980-3997. DOI: 10.1016/J.Tet.2008.02.043  0.33
2007 Abell AD, Jones MA, Neffe AT, Aitken SG, Cain TP, Payne RJ, McNabb SB, Coxon JM, Stuart BG, Pearson D, Lee HY, Morton JD. Investigation into the P3 binding domain of m-calpain using photoswitchable diazo- and triazene-dipeptide aldehydes: new anticataract agents. Journal of Medicinal Chemistry. 50: 2916-20. PMID 17497840 DOI: 10.1021/Jm061455N  0.624
2007 McCarthy AR, Hartmann RW, Abell AD. Evaluation of 4′-substituted bicyclic pyridones as non-steroidal inhibitors of steroid 5α-reductase Bioorganic and Medicinal Chemistry Letters. 17: 3603-3607. PMID 17490876 DOI: 10.1016/J.Bmcl.2007.04.049  0.365
2007 Payne RJ, Riboldi-Tunnicliffe A, Kerbarh O, Abell AD, Lapthorn AJ, Abell C. Design, synthesis, and structural studies on potent biaryl inhibitors of type II dehydroquinases. Chemmedchem. 2: 1010-3. PMID 17487901 DOI: 10.1002/Cmdc.200700062  0.31
2007 Payne RJ, Peyrot F, Kerbarh O, Abell AD, Abell C. Rational design, synthesis, and evaluation of nanomolar type II dehydroquinase inhibitors. Chemmedchem. 2: 1015-29. PMID 17487900 DOI: 10.1002/Cmdc.200700032  0.347
2007 Zaman S, Kitamura M, Abell AD. Synthesis of 5-phenyl 2-functionalized pyrroles by amino Heck and Tandem amino Heck carbonylation reactions Australian Journal of Chemistry. 60: 624-626. DOI: 10.1071/Ch07132  0.343
2006 Zaman S, Campaner P, Abell AD. Synthesis of amino acid derived seven-membered lactams by RCM and their evaluation against HIV protease Bioorganic and Medicinal Chemistry. 14: 8323-8331. PMID 17010620 DOI: 10.1016/J.Bmc.2006.09.009  0.341
2006 Pearson D, Abell AD. Photoswitch inhibitors of α-chymotrypsin - Increased substitution and peptidic character in peptidomimetic boronate esters Organic and Biomolecular Chemistry. 4: 3618-3625. PMID 16990937 DOI: 10.1039/B609320P  0.351
2006 Gardiner J, Aitken SG, McNabb SB, Zaman S, Abell AD. Ring closing metathesis of α- and β-amino acid derived dienes Journal of Organometallic Chemistry. 691: 5487-5496. DOI: 10.1016/J.Jorganchem.2006.09.061  0.313
2005 Neffe AT, Abell AD. Developments in the design and synthesis of calpain inhibitors Current Opinion in Drug Discovery and Development. 8: 684-700. PMID 16312145  0.607
2005 Payne RJ, Toscano MD, Bulloch EM, Abell AD, Abell C. Design and synthesis of aromatic inhibitors of anthranilate synthase. Organic & Biomolecular Chemistry. 3: 2271-81. PMID 16010361 DOI: 10.1039/B503802B  0.343
2005 Zaman S, Mitsuru K, Abell AD. Synthesis of trisubstituted imidazoles by palladium-catalyzed cyclization of O-pentafluorobenzoylamidoximes: Application to amino acid mimetics with a C-terminal imidazole Organic Letters. 7: 609-611. PMID 15704906 DOI: 10.1021/Ol047628P  0.314
2005 Abell AD, Brown KM, Coxon JM, Jones MA, Miyamoto S, Neffe AT, Nikkel JM, Stuart BG. Synthesis and evaluation of eight-membered cyclic pseudo-dipeptides Peptides. 26: 251-258. PMID 15629536 DOI: 10.1016/J.Peptides.2004.09.006  0.665
2005 Abell AD, Harvey AJ. Synthesis of a [1,4]dioxane-2,5-dione based-peptidomimetic scaffold Arkivoc. 2006: 72-76. DOI: 10.3998/Ark.5550190.0007.307  0.306
2004 Payne RJ, Daines AM, Clark BM, Abell AD. Synthesis and protein conjugation studies of vitamin K analogues Bioorganic and Medicinal Chemistry. 12: 5785-5791. PMID 15498655 DOI: 10.1016/J.Bmc.2004.08.037  0.301
2004 Daines AM, Abell AD. The preparation of side chain functionalized analogues of coenzyme Q for protein conjugation studies. Organic & Biomolecular Chemistry. 2: 2371-5. PMID 15305221 DOI: 10.1039/B407659A  0.328
2004 Gardiner J, Abell AD. Synthesis and solid state conformation of phenylalanine mimetics constrained in a proline-like conformation. Organic & Biomolecular Chemistry. 2: 2365-70. PMID 15305220 DOI: 10.1039/B406450J  0.344
2004 Gardiner J, Anderson KH, Downard A, Abell AD. Synthesis of cyclic beta-amino acid esters from methionine, allylglycine, and serine. The Journal of Organic Chemistry. 69: 3375-82. PMID 15132545 DOI: 10.1021/Jo049794G  0.32
2004 Abell AD. Chemistry at the Interface Australian Journal of Chemistry. 57: 819. DOI: 10.1071/Ch04180  0.316
2004 Payne RJ, Brown KM, Coxon JM, Morton JD, Lee HYY, Abell AD. Peptidic aldehydes based on α- and β-amino acids: Synthesis, inhibition of m-Calpain, and anti-cataract properties Australian Journal of Chemistry. 57: 877-884. DOI: 10.1071/Ch04080  0.356
2004 Le Sann C, Abell AD. Synthesis and properties of a mesylated ArgoGel resin Australian Journal of Chemistry. 57: 355-358. DOI: 10.1071/Ch03247  0.305
2003 Martyn DC, Vernall AJ, Clark BM, Abell AD. Ring-deactivated hydroxyalkylpyrrole-based inhibitors of alpha-chymotrypsin: synthesis and mechanism of action. Organic & Biomolecular Chemistry. 1: 2103-10. PMID 12945901 DOI: 10.1039/B302411C  0.301
2003 Humphries ME, Murphy J, Phillips AJ, Abell AD. Synthesis of functionalized piperidinones. The Journal of Organic Chemistry. 68: 2432-6. PMID 12636413 DOI: 10.1021/Jo0267091  0.508
2003 Le Sann C, Abell C, Abell AD. A convenient method for the synthesis of dehydroquinic acid Synthetic Communications. 33: 527-533. DOI: 10.1081/Scc-120015805  0.318
2003 Gardiner J, Abell AD. A diastereoselective synthesis of the tetrahydropyridazinone core of 2-oxo-1,6-diazobicyclo[4.3.0]nonane-9-carboxylate-based peptidomimetics starting from (S)-phenylalanine Tetrahedron Letters. 44: 4227-4230. DOI: 10.1016/S0040-4039(03)00882-7  0.33
2002 Abell AD, Gardiner J. Synthesis of substituted cyclohexenyl-based beta-amino acids by ring-closing metathesis. Organic Letters. 4: 3663-6. PMID 12375913 DOI: 10.1021/Ol0266121  0.324
2002 Le Sann C, Abell C, Abell AD. A simple method for the preparation of 3-hydroxyiminodehydroquinate, a potent inhibitor of type II dehydroquinase Journal of the Chemical Society. Perkin Transactions 1. 2065-2068. DOI: 10.1039/B206066C  0.331
2002 May BCH, Abell AD. α-methylene tetrazole-based peptidomimetics: Synthesis and inhibition of hiv protease Journal of the Chemical Society. Perkin Transactions 1. 2: 172-178. DOI: 10.1039/B109128J  0.315
2002 Abell AD. Heterocyclic-based peptidomimetics Letters in Peptide Science. 8: 267-272. DOI: 10.1023/A:1016216828677  0.333
2001 May BC, Abell AD. The synthesis and solid state structure of (8S)-8-benzyl-8,9-dihydro-7H-tetrazolo[1,5-d][1,4]diazepin-6-one. Chemical Communications (Cambridge, England). 2080-1. PMID 12240172 DOI: 10.1039/B106175P  0.315
2001 Harvey AJ, Abell AD. Alpha-ketoester-based photobiological switches: synthesis, peptide chain extension and assay against alpha-chymotrypsin. Bioorganic & Medicinal Chemistry Letters. 11: 2441-4. PMID 11549442 DOI: 10.1016/S0960-894X(01)00464-4  0.314
2001 Edmonds MK, Abell AD. Design and synthesis of a conformationally restricted trans peptide isostere based on the bioactive conformations of saquinavir and nelfinavir. The Journal of Organic Chemistry. 66: 3747-52. PMID 11374993 DOI: 10.1021/Jo0016834  0.332
2001 Martyn DC, Hoult DA, Abell AD. Stereocontrol of the Horner-Wadsworth-Emmons Reaction: Application to the Synthesis of HIV-1 Protease Inhibitors Australian Journal of Chemistry. 54: 391-396. DOI: 10.1071/Ch01093  0.339
2001 Zubarev VY, Trifonov RE, Filichev VV, Ostrovskii VA, Abell AD, Edmonds MK. Synthesis, X-ray and conformational studies of novel tetrazole-containing macrocycles: 4,13-dioxa-1,7,8,9,17,18,19,20-octaazatricyclo[14.2.1.17,10]icosa-8,10(20),16(19),17-tetraene and 4,14-dioxa-1,7,8,9,10,18,19,20-octaazatricyclo[15.2.1.07,10]icosa-8,10,17(20),18-tetraene Journal of the Chemical Society-Perkin Transactions 1. 417-421. DOI: 10.1039/B006217K  0.307
2001 May BCH, Abell AD. The synthesis and crystal structure of alpha-keto tetrazole-based dipeptide mimics Tetrahedron Letters. 42: 5641-5644. DOI: 10.1016/S0040-4039(01)01101-7  0.343
2000 Abell AD, Prince MJ, McNulty AM, Neubauer BL. Simple bi- and tricyclic inhibitors of human steroid 5alpha-reductase. Bioorganic & Medicinal Chemistry Letters. 10: 1909-11. PMID 10987415 DOI: 10.1016/S0960-894X(00)00368-1  0.325
2000 Gerrard JA, Prince MJ, Abell AD. Kinetic characterisation of ene-diol-based inhibitors of alpha-amylase. Bioorganic & Medicinal Chemistry Letters. 10: 1575-6. PMID 10915054 DOI: 10.1016/S0960-894X(00)00288-2  0.3
2000 Phillips AJ, Morris JC, Abell AD. Progress towards an intramolecular Diels-Alder ring-expansion approach to taxinine: The interplay of Lewis acids and high pressure Tetrahedron Letters. 41: 2723-2727. DOI: 10.1016/S0040-4039(00)00248-3  0.506
1999 Nabbs BK, Abell AD. The synthesis and P388 cytotoxicity of mycalazol 11 and related 5-acyl-2-hydroxymethylpyrroles. Bioorganic & Medicinal Chemistry Letters. 9: 505-8. PMID 10091711 DOI: 10.1016/S0960-894X(99)00021-9  0.321
1999 Abell AD, Oldham MD. Leucine-phenylalanine dipeptide-based N-mesyloxysuccinimides: synthesis of all four stereoisomers and their assay against serine proteases. Bioorganic & Medicinal Chemistry Letters. 9: 497-500. PMID 10091709 DOI: 10.1016/S0960-894X(99)00017-7  0.321
1999 May BCH, Abell AD. A convenient preparation of (2SR,3S)-3-amino-2-hydroxy-4-phenylbutanoic acid; an important peptide bond isostere Synthetic Communications. 29: 2515-2525. DOI: 10.1080/00397919908086259  0.345
1999 Abell AD, Oldham MD, Moore MM, Robinson WT. The synthesis and X-ray crystal structure of phenylalanine-based N-benzyloxysuccinimides Australian Journal of Chemistry. 52: 977-981. DOI: 10.1071/Ch99055  0.305
1999 Abell AD, Nabbs BK, Battersby AR, Thompson A, Dolphin D. Synthesis and properties of ring-deactivated Deuterated (hydroxymethyl)pyrroles Chemtracts. 12: 534-538. DOI: 10.1021/Ja973656+  0.531
1999 Abell AD, Nabbs BK, Battersby AR, Thompson A, Dolphin D. Synthesis and properties of ring-deactivated Deuterated (hydroxymethyl)pyrroles Chemtracts. 12: 534-538. DOI: 10.1021/ja973656+  0.453
1998 Abell AD, Phillips AJ, Budhia S, McNulty AM, Neubauer BL. The preparation and biological activity of lactam-based, non-steroidal, inhibitors of human type-1 steroid 5α-reductase Australian Journal of Chemistry. 51: 389-396. DOI: 10.1071/C97130  0.498
1998 Abell AD, Nabbs BK, Battersby AR. The reaction of N-magnesium derivatives of pyrroles with N- mesylchloromethylpyrroles: A synthesis of dipyrrylmethanes Journal of Organic Chemistry. 63: 8163-8169. DOI: 10.1021/Jo980573I  0.527
1998 Abell AD, Gardiner J, Phillips AJ, Robinson WT. Synthesis and X-ray structure of a 1,2,3,6-tetrahydropyridine-based phenylalanine mimetic Tetrahedron Letters. 39: 9563-9566. DOI: 10.1016/S0040-4039(98)02125-X  0.51
1997 Carr AC, Winterbourn CC, Blunt JW, Phillips AJ, Abell AD. Nuclear magnetic resonance characterization of 6 alpha-chloro-5 beta-cholestane-3 beta,5-diol formed from the reaction of hypochlorous acid with cholesterol. Lipids. 32: 363-7. PMID 9113623 DOI: 10.1007/S11745-997-0046-8  0.441
1997 Abell AD, Brandt M, Levy MA, Holt DA. Preparation and biological activity of tricyclic non-steroidal inhibitors of human steroid 5α-reductase Journal of the Chemical Society - Perkin Transactions 1. 1663-1667. DOI: 10.1039/A608169J  0.337
1997 Abell AD, Blunt JW, Foulds GJ, Munro MHG. Chemistry of the mycalamides: Antiviral and antitumour compounds from a New Zealand marine sponge. Part 6. The synthesis and testing of analogues of the C(7)-C(10) fragment Journal of the Chemical Society - Perkin Transactions 1. 1647-1654. DOI: 10.1039/A608168A  0.314
1997 Abell AD, Edwards RA, Oldham MD. Chemistry and X-ray crystallographic structure of N-protected (5-oxo-1,3-oxazolidin-4-yl)acetic acids: Versatile intermediates in the synthesis of peptidomimetics Journal of the Chemical Society - Perkin Transactions 1. 1655-1662. DOI: 10.1039/A608165G  0.347
1996 Abell AD, Taylor JM, Oldham MD. Self-addition products from the alkylation of amino acid-derived oxazolidinones: X-ray molecular structures of (2R,4S,1′S)-3-benzoyl-4-[benzoylamino(phenyl)methyl]-4-benzyl-2-phenyl-1, 3-oxazolidin-5-one, (2R,4S,1′S)- and (2R,4S,1′R)-3-benzoyl-4-[benzoylamino(phenyl)methyl]-4-isopropyl-2-phenyl- 1,3-oxazolidin-5-one Journal of the Chemical Society - Perkin Transactions 1. 1299-1304. DOI: 10.1039/P19960001299  0.301
1996 Abell AD, Brandt M, Levy MA, Holt DA. A comparison of steroidal and non-steroidal inhibitors of human steroid 5α-reductase: New tricyclic aryl acid inhibitors of the type-1 isozyme Bioorganic and Medicinal Chemistry Letters. 6: 481-484. DOI: 10.1016/0960-894X(96)00054-6  0.335
1995 Abell AD, Oldham MD, Taylor JM. Synthesis of phenylalanine-based cyclic acylated enamino ester dipeptide analogues: Inhibitors of α-chymotrypsin. X-ray molecular structure of (2′S,4′R)-4′-benzyl-3′-benzyloxycarbonyl-5′-oxo- 2′-phenyloxazolidin-4′-ylacetic acid Journal of the Chemical Society, Perkin Transactions 1. 953-961. DOI: 10.1039/P19950000953  0.371
1995 Abell AD, Oldham MD, Taylor JM. Synthesis of cyclic acylated enamino esters from enol lactones, 4-keto amides, and 5-hydroxy lactams Journal of Organic Chemistry. 60: 1214-1220. DOI: 10.1021/Jo00110A026  0.376
1994 Abell AD, Brandt M, Levy MA, Holt DA. A non-steroidal diene acid inhibitor of human type 2 stereoid 5α-reductase Bioorganic and Medicinal Chemistry Letters. 4: 2327-2330. DOI: 10.1016/0960-894X(94)85034-8  0.328
1993 Abell A, Litten J. Synthesis and Amino Acid Chain Extension of 1-Acylated Hydroxymethylpyrroles Australian Journal of Chemistry. 46: 1473. DOI: 10.1071/Ch9931473  0.31
1993 Abell AD, Hoult DA, Morris KM, Taylor JM, Trent JO. Halogenation of keto acid phosphoranes: Synthesis of halo enol lactones and haloallenes Journal of Organic Chemistry. 58: 1531-1537. DOI: 10.1021/Jo00058A039  0.322
1993 Abell AD, Taylor JM. Synthesis of cyclic acylated enamino ester dipeptide analogues via the bromolactonization of a keto acid phosphorane Journal of Organic Chemistry. 58: 14-15. DOI: 10.1021/Jo00053A006  0.331
1992 Abell AD, Litten JC. Synthesis and hydrolysis of dipeptide isosteres containing a proline analogue with latent reactivity Tetrahedron Letters. 33: 3005-3008. DOI: 10.1016/S0040-4039(00)79584-0  0.356
1992 Abell AD, Hoult DA, Jamieson EJ. Synthesis of 1,2-disubstituted pyrroles: A cis peptide bond surrogate Tetrahedron Letters. 33: 5831-5832. DOI: 10.1016/0040-4039(92)89043-C  0.322
1991 Abell A, Hartshorn M, Maclennan M, Robinson W, Wright G. Reactions of 1,4-Dimethyl-4-nitro-cyclohexa-2,5-dien-1-yl Acetates With Nitrogen Dioxide; the Formation of Polynitro Cyclohexenyl Esters Australian Journal of Chemistry. 44: 43. DOI: 10.1071/Ch9910043  0.341
1990 Abell AD, Morris KB, Litten JC. Synthesis and deprotection of [1-(ethoxycarbonyl)-4-[(diphenylmethoxy)carbonyl]-1-methyl-2-oxobutyl]- triphenylphosphonium chloride: A key intermediate in the Wittig reaction between a cyclic anhydride and a stabilized ylide Journal of Organic Chemistry. 55: 5217-5221. DOI: 10.1021/Jo00305A013  0.301
1989 Abell A, Hartshorn M, Robinson W, Waller A, Wright G. Reactions of 4-Methyl-1-(1′-methylethyl)-4-nitrocyclohexa-2,5-dien-1-yl Acetates With Nitrogen Dioxide; Towards a Mechanism for the Formation of Polynitro Cyclohexenyl Esters on Reaction of p-Cymene With Nitrogen Dioxide in Acetic Anhydride Australian Journal of Chemistry. 42: 2225. DOI: 10.1071/Ch9892225  0.32
1989 Abell AD, Trent JO. A novel bromo lactonization of acylated phosphoranes. A new route to bromo enol lactones Journal of the Chemical Society, Chemical Communications. 409-410. DOI: 10.1039/C39890000409  0.322
1988 Abell A, Clark B, Robinson W. A Mechanistic Study of the Wittig Reaction Between a Cyclic Anhydride and a Stabilized Phosphorane Australian Journal of Chemistry. 41: 1243. DOI: 10.1071/Ch9881243  0.314
1987 Schauder JR, Jendrezejewski S, Abell A, Hart GJ, Battersby AR. Stereochemistry of formation of the hydroxymethyl group of hydroxymethylbilane, the precursor of uro'gen-III Journal of the Chemical Society, Chemical Communications. 436-438. DOI: 10.1039/C39870000436  0.49
1986 ABELL AD, HEINICKE GW, MASSY-WESTROPP RA. ChemInform Abstract: Synthesis of Dialkyl Hex-2-yne-1,6-dioates and Hept-2-yne-1,7-dioates. Chemischer Informationsdienst. 17. DOI: 10.1002/chin.198603132  0.593
1985 Abell A, Massy-Westropp R, Reynolds G. Rearrangement of Freelingyne with Base Australian Journal of Chemistry. 38: 1129. DOI: 10.1071/Ch9851129  0.6
1985 Abell A, Massy-Westropp R. Mechanism of Acetal Cleavage with Methylmagnesium Iodide Australian Journal of Chemistry. 38: 1031. DOI: 10.1071/Ch9851031  0.612
1985 Abell AD, Heinicke GW, Massy-Westropp RA. Synthesis of Dialkyl Hex-2-yne-1,6-dioates and Hept-2-yne-1,7-dioates Synthesis. 1985: 764-766. DOI: 10.1055/S-1985-31339  0.595
1985 Abell AD, Massy-Westropp RA. Regioselective bond cleavage and coordination effects in the reduction of some acetals with lithium in ammonia Tetrahedron. 41: 2451-2464. DOI: 10.1016/S0040-4020(01)96640-2  0.62
1984 Abell A, Dimitriadis E, Massy-Westropp R. Stereospecific formation of tetrahydrofurans from substituted 2,8-Dioxabicyclo[3.2.1]oct-3-ylmethanols Australian Journal of Chemistry. 37: 395. DOI: 10.1071/Ch9840395  0.634
1984 ABELL AD, DIMITRIADIS E, MASSY-WESTROPP RA. ChemInform Abstract: STEREOSPECIFIC FORMATION OF TETRAHYDROFURANS FROM SUBSTITUTED 2,8-DIOXABICYCLO(3.2.1)OCT-3-YLMETHANOLS Chemischer Informationsdienst. 15. DOI: 10.1002/Chin.198438170  0.583
1983 ABELL AD, DOYLE IR, MASSY-WESTROPP RA. ChemInform Abstract: THE WITTIG REACTION WITH GLUTARIC AND SUCCINIC ANHYDRIDES Chemischer Informationsdienst. 14. DOI: 10.1002/chin.198314128  0.565
1982 Abell A, Doyle I, Massy-Westropp R. The Wittig reaction with glutaric and succinic anhydrides Australian Journal of Chemistry. 35: 2277. DOI: 10.1071/Ch9822277  0.634
1982 Abell A, Massy-Westropp R. Aspects of the mechanism of the Wittig reaction between cyclic anhydrides and stabilized phosphoranes Australian Journal of Chemistry. 35: 2077. DOI: 10.1071/Ch9822077  0.626
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