Year |
Citation |
Score |
2021 |
Elhalem E, Bellomo A, Cooke M, Scravaglieri A, Pearce LV, Peach ML, Gandolfi Donadío L, Kazanietz MG, Comin MJ. Design, Synthesis, and Characterization of Novel -1 Heterocyclic DAG-Lactones as PKC Activators. Journal of Medicinal Chemistry. PMID 34279947 DOI: 10.1021/acs.jmedchem.1c00739 |
0.681 |
|
2017 |
Elhalem E, Donadío LG, Zhou X, Lewin NE, Garcia LC, Lai CC, Kelley JA, Peach ML, Blumberg PM, Comin MJ. Exploring the influence of indololactone structure on selectivity for binding to the C1 domains of PKCα, PKCε, and RasGRP. Bioorganic & Medicinal Chemistry. PMID 28392275 DOI: 10.1016/J.Bmc.2017.03.022 |
0.686 |
|
2014 |
Elhalem E, Recio R, Werner S, Lieder F, Calderón-Montaño JM, López-Lázaro M, Fernández I, Khiar N. Sulforaphane homologues: Enantiodivergent synthesis of both enantiomers, activation of the Nrf2 transcription factor and selective cytotoxic activity. European Journal of Medicinal Chemistry. 87: 552-63. PMID 25299679 DOI: 10.1016/j.ejmech.2014.09.052 |
0.324 |
|
2010 |
Elhalem E, Pujol CA, Damonte EB, Rodriguez JB. Synthesis and biological evaluation of N-thia-carba-thymidine as an antiherpetic agent Tetrahedron. 66: 3332-3340. DOI: 10.1016/J.TET.2010.02.092 |
0.522 |
|
2010 |
Szajnman SH, Yan W, Bailey BN, Docampo R, Elhalem E, Rodriguez JB. ChemInform Abstract: Design and Synthesis of Aryloxyethyl Thiocyanate Derivatives as Potent Inhibitors of Trypanosoma cruzi Proliferation. Cheminform. 31: no-no. DOI: 10.1002/chin.200029071 |
0.695 |
|
2006 |
Elhalem E, Comin MJ, Rodriguez JB. Synthesis of Conformationally Locked Carbocyclic Nucleosides Built on a Thiabicyclo[3.1.0]hexane System as a Pseudosugar Surrogate European Journal of Organic Chemistry. 2006: 4473-4482. DOI: 10.1002/EJOC.200600488 |
0.681 |
|
2005 |
Elhalem E, Comin MJ, Leitofuter J, García-Liñares G, Rodriguez JB. Synthetic studies toward the preparation of (4R,5R)-(−)-3-[(benzyloxy)methyl]-4,5-O-isopropylidene-cyclopenten-2-one: an important synthetic intermediate for carbanucleosides Tetrahedron: Asymmetry. 16: 425-431. DOI: 10.1016/J.TETASY.2004.11.069 |
0.636 |
|
2004 |
Gao ZG, Jeong LS, Moon HR, Kim HO, Choi WJ, Shin DH, Elhalem E, Comin MJ, Melman N, Mamedova L, Gross AS, Rodriguez JB, Jacobson KA. Structural determinants of efficacy at A3 adenosine receptors: modification of the ribose moiety. Biochemical Pharmacology. 67: 893-901. PMID 15104242 DOI: 10.1016/J.Bcp.2003.10.006 |
0.657 |
|
2004 |
Comin MJ, Elhalem E, Rodriguez JB. Cerium ammonium nitrate: a new catalyst for regioselective protection of glycols Tetrahedron. 60: 11851-11860. DOI: 10.1016/J.TET.2004.09.097 |
0.634 |
|
2002 |
Elhalem E, Bailey BN, Docampo R, Ujváry I, Szajnman SH, Rodriguez JB. Design, synthesis, and biological evaluation of aryloxyethyl thiocyanate derivatives against Trypanosoma cruzi. Journal of Medicinal Chemistry. 45: 3984-99. PMID 12190320 DOI: 10.1021/Jm0201518 |
0.688 |
|
2000 |
Szajnman SH, Yan W, Bailey BN, Docampo R, Elhalem E, Rodriguez JB. Design and synthesis of aryloxyethyl thiocyanate derivatives as potent inhibitors of Trypanosoma cruzi proliferation. Journal of Medicinal Chemistry. 43: 1826-40. PMID 10794699 DOI: 10.1021/Jm9905007 |
0.68 |
|
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