| Year |
Citation |
Score |
| 2023 |
El-Mowafi SA, Konshina AG, Mohammed EHM, Krylov NA, Efremov RG, Parang K. Structural Analysis and Activity Correlation of Amphiphilic Cyclic Antimicrobial Peptides Derived from the [WR] Scaffold. Molecules (Basel, Switzerland). 28. PMID 38138539 DOI: 10.3390/molecules28248049 |
0.328 |
|
| 2023 |
Helmy NM, Parang K. Cyclic Peptides with Antifungal Properties Derived from Bacteria, Fungi, Plants, and Synthetic Sources. Pharmaceuticals (Basel, Switzerland). 16. PMID 37375840 DOI: 10.3390/ph16060892 |
0.334 |
|
| 2023 |
Gupta S, Park SE, Mozaffari S, El-Aarag B, Parang K, Tiwari RK. Design, Synthesis, and Antiproliferative Activity of Benzopyran-4-One-Isoxazole Hybrid Compounds. Molecules (Basel, Switzerland). 28. PMID 37241960 DOI: 10.3390/molecules28104220 |
0.793 |
|
| 2023 |
Moreno J, Zoghebi K, Salehi D, Kim L, Shoushtari SK, Tiwari RK, Parang K. Amphiphilic Cell-Penetrating Peptides Containing Arginine and Hydrophobic Residues as Protein Delivery Agents. Pharmaceuticals (Basel, Switzerland). 16. PMID 36986567 DOI: 10.3390/ph16030469 |
0.649 |
|
| 2023 |
Mandal D, Lohan S, Sajid MI, Alhazza A, Tiwari RK, Parang K, Montazeri Aliabadi H. Modified Linear Peptides Effectively Silence STAT-3 in Breast Cancer and Ovarian Cancer Cell Lines. Pharmaceutics. 15. PMID 36839988 DOI: 10.3390/pharmaceutics15020666 |
0.644 |
|
| 2022 |
Lohan S, Konshina AG, Efremov RG, Maslennikov I, Parang K. Structure-Based Rational Design of Small α-Helical Peptides with Broad-Spectrum Activity against Multidrug-Resistant Pathogens. Journal of Medicinal Chemistry. PMID 36574364 DOI: 10.1021/acs.jmedchem.2c01708 |
0.365 |
|
| 2022 |
Kim L, Lohan S, Moreno J, Zoghebi K, Tiwari RK, Parang K. Cyclic and Linear Peptides Containing Alternate WW and RR Residues as Molecular Cargo Delivery Tools. Molecular Pharmaceutics. PMID 36445335 DOI: 10.1021/acs.molpharmaceut.2c00664 |
0.639 |
|
| 2022 |
Mohammed EHM, Lohan S, Ghaffari T, Gupta S, Tiwari RK, Parang K. Membrane-Active Cyclic Amphiphilic Peptides: Broad-Spectrum Antibacterial Activity Alone and in Combination with Antibiotics. Journal of Medicinal Chemistry. 65: 15819-15839. PMID 36442155 DOI: 10.1021/acs.jmedchem.2c01469 |
0.634 |
|
| 2022 |
Agarwal HK, Chhikara BS, Ye G, Bhavaraju S, Dixit A, Kumar A, Doncel GF, Parang K. Synthesis and Biological Evaluation of 5'--Fatty Acyl Ester Derivatives of 3'-Fluoro-2',3'-dideoxythymidine as Potential Anti-HIV Microbicides. Molecules (Basel, Switzerland). 27. PMID 35630829 DOI: 10.3390/molecules27103352 |
0.741 |
|
| 2022 |
Salehi D, Mozaffari S, Zoghebi K, Lohan S, Mandal D, Tiwari RK, Parang K. Amphiphilic Cell-Penetrating Peptides Containing Natural and Unnatural Amino Acids as Drug Delivery Agents. Cells. 11. PMID 35406720 DOI: 10.3390/cells11071156 |
0.639 |
|
| 2022 |
Mandal D, Mohammed EHM, Lohan S, Mandipoor P, Baradaran D, Tiwari RK, Parang K, Aliabadi HM. Redox-Responsive Disulfide Cyclic Peptides: A New Strategy for siRNA Delivery. Molecular Pharmaceutics. PMID 35347995 DOI: 10.1021/acs.molpharmaceut.1c00879 |
0.632 |
|
| 2022 |
Mohammed EHM, Lohan S, Tiwari RK, Parang K. Amphiphilic cyclic peptide [WKR]-Antibiotics combinations as broad-spectrum antimicrobial agents. European Journal of Medicinal Chemistry. 235: 114278. PMID 35339840 DOI: 10.1016/j.ejmech.2022.114278 |
0.57 |
|
| 2022 |
Querfurth H, Marshall J, Parang K, Rioult-Pedotti MS, Tiwari R, Kwon B, Reisinger S, Lee HK. A PDK-1 allosteric agonist neutralizes insulin signaling derangements and beta-amyloid toxicity in neuronal cells and in vitro. Plos One. 17: e0261696. PMID 35061720 DOI: 10.1371/journal.pone.0261696 |
0.532 |
|
| 2022 |
Zoghebi K, Aliabadi HM, Tiwari RK, Parang K. [(WR)WKβA]-Doxorubicin Conjugate: A Delivery System to Overcome Multi-Drug Resistance against Doxorubicin. Cells. 11. PMID 35053417 DOI: 10.3390/cells11020301 |
0.658 |
|
| 2022 |
Lohan S, Mandal D, Choi W, Konshina AG, Tiwari RK, Efremov RG, Maslennikov I, Parang K. Small Amphiphilic Peptides: Activity Against a Broad Range of Drug-Resistant Bacteria and Structural Insight into Membranolytic Properties. Journal of Medicinal Chemistry. PMID 34978443 DOI: 10.1021/acs.jmedchem.1c01782 |
0.652 |
|
| 2021 |
Nasrolahi Shirazi A, Sajid MI, Mandal D, Stickley D, Nagasawa S, Long J, Lohan S, Parang K, Tiwari RK. Cyclic Peptide-Gadolinium Nanocomplexes as siRNA Delivery Tools. Pharmaceuticals (Basel, Switzerland). 14. PMID 34832846 DOI: 10.3390/ph14111064 |
0.819 |
|
| 2021 |
El-Sayed NS, Sajid MI, Parang K, Tiwari RK. Synthesis, characterization, and cytotoxicity evaluation of dextran-myristoyl-ECGKRK peptide conjugate. International Journal of Biological Macromolecules. PMID 34597704 DOI: 10.1016/j.ijbiomac.2021.09.160 |
0.646 |
|
| 2021 |
El-Sayed NS, Jureka AS, Edwards MR, Lohan S, Williams CG, Keiser PT, Davey RA, Totonchy J, Tiwari RK, Basler CF, Parang K. Synthesis and antiviral activity of fatty acyl conjugates of remdesivir against severe acute respiratory syndrome coronavirus 2 and Ebola virus. European Journal of Medicinal Chemistry. 226: 113862. PMID 34583312 DOI: 10.1016/j.ejmech.2021.113862 |
0.542 |
|
| 2021 |
Mozaffari S, Salehi D, Mahdipoor P, Beuttler R, Tiwari R, Aliabadi HM, Parang K. Design and application of hybrid cyclic-linear peptide-doxorubicin conjugates as a strategy to overcome doxorubicin resistance and toxicity. European Journal of Medicinal Chemistry. 226: 113836. PMID 34537446 DOI: 10.1016/j.ejmech.2021.113836 |
0.613 |
|
| 2021 |
Khayyatnejad Shoushtari S, Zoghebi K, Sajid MI, Tiwari RK, Parang K. Hybrid Cyclic-Linear Cell-Penetrating Peptides Containing Alternative Positively Charged and Hydrophobic Residues as Molecular Transporters. Molecular Pharmaceutics. 18: 3909-3919. PMID 34491768 DOI: 10.1021/acs.molpharmaceut.1c00594 |
0.662 |
|
| 2021 |
Sanner MF, Zoghebi K, Hanna S, Mozaffari S, Rahighi S, Tiwari RK, Parang K. Cyclic Peptides as Protein Kinase Inhibitors: Structure-Activity Relationship and Molecular Modeling. Journal of Chemical Information and Modeling. PMID 34000187 DOI: 10.1021/acs.jcim.1c00320 |
0.64 |
|
| 2021 |
Hall R, Alasmari A, Mozaffari S, Mahdipoor P, Parang K, Montazeri Aliabadi H. Peptide/Lipid-Associated Nucleic Acids (PLANAs) as a Multicomponent siRNA Delivery System. Molecular Pharmaceutics. PMID 33496597 DOI: 10.1021/acs.molpharmaceut.0c00969 |
0.336 |
|
| 2020 |
Kumar S, Mandal D, El-Mowafi SA, Mozaffari S, Tiwari RK, Parang K. Click-Free Synthesis of a Multivalent Tricyclic Peptide as a Molecular Transporter. Pharmaceutics. 12. PMID 32899170 DOI: 10.3390/Pharmaceutics12090842 |
0.698 |
|
| 2020 |
Shirazi AN, Park SE, Rad S, Baloyan L, Mandal D, Sajid MI, Hall R, Lohan S, Zoghebi K, Parang K, Tiwari RK. Cyclic Peptide-Gadolinium Nanoparticles for Enhanced Intracellular Delivery. Pharmaceutics. 12. PMID 32825689 DOI: 10.3390/Pharmaceutics12090792 |
0.821 |
|
| 2020 |
Mohammed EHM, Mandal D, Mozaffari S, Abdel-Hamied Zahran M, Mostafa Osman A, Kumar Tiwari R, Parang K. Comparative Molecular Transporter Properties of Cyclic Peptides Containing Tryptophan and Arginine Residues Formed through Disulfide Cyclization. Molecules (Basel, Switzerland). 25. PMID 32498339 DOI: 10.3390/Molecules25112581 |
0.409 |
|
| 2020 |
Parang K, El-Sayed NS, Kazeminy AJ, Tiwari RK. Comparative Antiviral Activity of Remdesivir and Anti-HIV Nucleoside Analogs Against Human Coronavirus 229E (HCoV-229E). Molecules (Basel, Switzerland). 25. PMID 32429580 DOI: 10.3390/Molecules25102343 |
0.593 |
|
| 2020 |
Chhikara BS, Ashraf S, Mozaffari S, St Jeans N, Mandal D, Tiwari RK, Ul-Haq Z, Parang K. Phenylpyrazalopyrimidines as Tyrosine Kinase Inhibitors: Synthesis, Antiproliferative Activity, and Molecular Simulations. Molecules (Basel, Switzerland). 25. PMID 32370213 DOI: 10.3390/Molecules25092135 |
0.616 |
|
| 2020 |
Kumar S, Singh D, Kumari P, Malik RS, Poonam, Parang K, Tiwari RK. PEGylation and Cell-Penetrating Peptides: Glimpse from Past and Prospects in Future. Current Topics in Medicinal Chemistry. PMID 31994461 DOI: 10.2174/1568026620666200128142603 |
0.615 |
|
| 2019 |
Zoghebi KA, Bousoik E, Parang K, Elsaid KA. Design and Biological Evaluation of Colchicine-CD44-Targeted Peptide Conjugate in an In Vitro Model of Crystal Induced Inflammation. Molecules (Basel, Switzerland). 25. PMID 31877739 DOI: 10.3390/Molecules25010046 |
0.414 |
|
| 2019 |
Park SE, Sajid MI, Parang K, Tiwari RK. Cyclic Cell-Penetrating Peptides As Efficient Intracellular Drug Delivery Tools. Molecular Pharmaceutics. PMID 31329448 DOI: 10.1021/Acs.Molpharmaceut.9B00633 |
0.823 |
|
| 2019 |
Park SE, Shamloo K, Kristedja TA, Darwish S, Bisoffi M, Parang K, Tiwari RK. EDB-FN Targeted Peptide-Drug Conjugates for Use against Prostate Cancer. International Journal of Molecular Sciences. 20. PMID 31277465 DOI: 10.3390/Ijms20133291 |
0.799 |
|
| 2019 |
Mozaffari S, Bousoik E, Amirrad F, Lamboy R, Coyle M, Hall R, Alasmari A, Mahdipoor P, Parang K, Montazeri Aliabadi H. Amphiphilic Peptides for Efficient siRNA Delivery. Polymers. 11. PMID 30999603 DOI: 10.3390/Polym11040703 |
0.477 |
|
| 2019 |
El-Sayed NS, Shirazi AN, Sajid MI, Park SE, Parang K, Tiwari RK. Synthesis and Antiproliferative Activities of Conjugates of Paclitaxel and Camptothecin with a Cyclic Cell-Penetrating Peptide. Molecules (Basel, Switzerland). 24. PMID 30978971 DOI: 10.3390/Molecules24071427 |
0.836 |
|
| 2019 |
Yeong KY, Nor Azizi MIH, Berdigaliyev N, Chen WN, Lee WL, Shirazi AN, Parang K. Sirtuin inhibition and anti-cancer activities of ethyl 2-benzimidazole-5-carboxylate derivatives Medchemcomm. 10: 2140-2145. DOI: 10.1039/C9Md00323A |
0.318 |
|
| 2018 |
Hanna SE, Mozaffari S, Tiwari RK, Parang K. Comparative Molecular Transporter Efficiency of Cyclic Peptides Containing Tryptophan and Arginine Residues. Acs Omega. 3: 16281-16291. PMID 31458264 DOI: 10.1021/acsomega.8b02589 |
0.636 |
|
| 2018 |
David AA, Park SE, Parang K, Tiwari RK. Antibiotics-Peptide Conjugates Against Multidrug-Resistant Bacterial Pathogens. Current Topics in Medicinal Chemistry. PMID 30499392 DOI: 10.2174/1568026619666181129141524 |
0.793 |
|
| 2018 |
Darwish S, Sadeghiani N, Fong S, Mozaffari S, Hamidi P, Withana T, Yang S, Tiwari RK, Parang K. Synthesis and antiproliferative activities of doxorubicin thiol conjugates and doxorubicin-SS-cyclic peptide. European Journal of Medicinal Chemistry. 161: 594-606. PMID 30396106 DOI: 10.1016/J.Ejmech.2018.10.042 |
0.642 |
|
| 2018 |
Riahifard N, Mozaffari S, Aldakhil T, Nunez F, Alshammari Q, Alshammari S, Yamaki J, Parang K, Tiwari RK. Design, Synthesis, and Evaluation of Amphiphilic Cyclic and Linear Peptides Composed of Hydrophobic and Positively-Charged Amino Acids as Antibacterial Agents. Molecules (Basel, Switzerland). 23. PMID 30360400 DOI: 10.3390/Molecules23102722 |
0.655 |
|
| 2018 |
El-Sayed NS, Miyake T, Shirazi AN, Park SE, Clark J, Buchholz S, Parang K, Tiwari R. Design, Synthesis, and Evaluation of Homochiral Peptides Containing Arginine and Histidine as Molecular Transporters. Molecules (Basel, Switzerland). 23. PMID 29966296 DOI: 10.3390/Molecules23071590 |
0.831 |
|
| 2018 |
Shirazi AN, Mozaffari S, Sherpa RT, Tiwari R, Parang K. Efficient Intracellular Delivery of Cell-Impermeable Cargo Molecules by Peptides Containing Tryptophan and Histidine. Molecules (Basel, Switzerland). 23. PMID 29949881 DOI: 10.3390/Molecules23071536 |
0.684 |
|
| 2018 |
Singh A, Mehra V, Sadeghiani N, Mozaffari S, Parang K, Kumar V. Ferrocenylchalcone–uracil conjugates: synthesis and cytotoxic evaluation Medicinal Chemistry Research. 27: 1260-1268. DOI: 10.1007/S00044-018-2145-5 |
0.361 |
|
| 2017 |
Reddy Kotla SK, Vandavasi JK, Wang JJ, Parang K, Tiwari RK. Palladium-Catalyzed Intramolecular Cross-Dehydrogenative Coupling: Synthesis of Fused Imidazo[1,2-]pyrimidines and Pyrazolo[1,5-]pyrimidines. Acs Omega. 2: 11-19. PMID 31457205 DOI: 10.1021/acsomega.6b00417 |
0.507 |
|
| 2017 |
Do H, Sharma M, El-Sayed NS, Mahdipoor P, Bousoik E, Parang K, Montazeri Aliabadi H. Difatty Acyl-Conjugated Linear and Cyclic Peptides for siRNA Delivery. Acs Omega. 2: 6939-6957. PMID 30023535 DOI: 10.1021/acsomega.7b00741 |
0.344 |
|
| 2017 |
Marshall J, Szmydynger-Chodobska J, Rioult-Pedotti MS, Lau K, Chin AT, Kotla SKR, Tiwari RK, Parang K, Threlkeld SW, Chodobski A. TrkB-enhancer facilitates functional recovery after traumatic brain injury. Scientific Reports. 7: 10995. PMID 28887487 DOI: 10.1038/S41598-017-11316-8 |
0.54 |
|
| 2017 |
Darwish S, Parang K, Marshall J, Goebel DJ, Tiwari R. Efficient synthesis of CN2097 using in situ activation of sulfhydryl group. Tetrahedron Letters. 58: 3053-3056. PMID 28824209 DOI: 10.1016/J.Tetlet.2017.06.066 |
0.628 |
|
| 2017 |
Sharma M, El-Sayed NS, Do H, Parang K, Tiwari RK, Aliabadi HM. Tumor-targeted delivery of siRNA using fatty acyl-CGKRK peptide conjugates. Scientific Reports. 7: 6093. PMID 28733622 DOI: 10.1038/S41598-017-06381-Y |
0.672 |
|
| 2017 |
Riahifard N, Tavakoli K, Yamaki J, Parang K, Tiwari R. Synthesis and Evaluation of Antimicrobial Activity of [R₄W₄K]-Levofloxacin and [R₄W₄K]-Levofloxacin-Q Conjugates. Molecules (Basel, Switzerland). 22. PMID 28594345 DOI: 10.3390/Molecules22060957 |
0.613 |
|
| 2017 |
Agarwal HK, Chhikara BS, Doncel GF, Parang K. Synthesis and anti-HIV activities of unsymmetrical long chain dicarboxylate esters of dinucleoside reverse transcriptase inhibitors. Bioorganic & Medicinal Chemistry Letters. PMID 28351588 DOI: 10.1016/J.Bmcl.2017.03.031 |
0.657 |
|
| 2017 |
Manchanda P, Parshad B, Kumar A, Tiwari RK, Shirazi AN, Parang K, Sharma SK. Design, Synthesis, and Evaluation of the Kinase Inhibition Potential of Pyridylpyrimidinylaminophenyl Derivatives. Archiv Der Pharmazie. PMID 28317151 DOI: 10.1002/Ardp.201600390 |
0.614 |
|
| 2017 |
Darwish S, Mozaffari S, Parang K, Tiwari R. Cyclic peptide conjugate of curcumin and doxorubicin as an anticancer agent Tetrahedron Letters. 58: 4617-4622. DOI: 10.1016/J.Tetlet.2017.10.065 |
0.692 |
|
| 2016 |
Tiwari RK, Brown A, Shirazi AN, Bolton J, Tse A, Verkhivker G, Parang K, Sun G. Design, Synthesis, and Evaluation of Dasatinib-Amino Acid and Dasatinib-Fatty Acid Conjugates as Protein Tyrosine Kinase Inhibitors. Chemmedchem. PMID 27875633 DOI: 10.1002/Cmdc.201600387 |
0.609 |
|
| 2016 |
Oh D, Darwish SA, Shirazi AN, Tiwari RK, Parang K. Corrigendum: Amphiphilic Bicyclic Peptides as Cellular Delivery Agents. Chemmedchem. 11: 2095. PMID 27647739 DOI: 10.1002/Cmdc.201600431 |
0.657 |
|
| 2016 |
Weerakkody D, Moshnikova A, El-Sayed NS, Adochite RC, Slaybaugh G, Golijanin J, Tiwari RK, Andreev OA, Parang K, Reshetnyak YK. Novel pH-Sensitive Cyclic Peptides. Scientific Reports. 6: 31322. PMID 27515582 DOI: 10.1038/Srep31322 |
0.656 |
|
| 2016 |
El-Sayed NS, Shirazi AN, El-Meligy MG, El-Ziaty AK, Nagieb ZA, Parang K, Tiwari RK. Design, synthesis, and evaluation of chitosan conjugated GGRGDSK peptides as a cancer cell-targeting molecular transporter. International Journal of Biological Macromolecules. 87: 611-22. PMID 26976071 DOI: 10.1016/J.Ijbiomac.2016.03.020 |
0.625 |
|
| 2016 |
Banerjee A, Sayeh N, Shirazi AN, Tiwari R, Parang K, Yadav A. Arginine-rich cyclic peptides enhance cellular delivery of anticancer agents: Molecular insights Letters in Drug Design and Discovery. 13: 591-604. DOI: 10.2174/1570180813999160429113034 |
0.804 |
|
| 2016 |
Shirazi AN, El-Sayed NS, Tiwari RK, Tavakoli K, Parang K. Cyclic peptide containing hydrophobic and positively charged residues as a drug delivery system for curcumin Current Drug Delivery. 13: 409-417. |
0.389 |
|
| 2015 |
Shirazi AN, El-Sayed NS, Mandal D, Tiwari RK, Tavakoli K, Etesham M, Parang K. Cysteine and arginine-rich peptides as molecular carriers. Bioorganic & Medicinal Chemistry Letters. PMID 26631317 DOI: 10.1016/J.Bmcl.2015.11.052 |
0.669 |
|
| 2015 |
Nasrolahi Shirazi A, El-Sayed NS, Tiwari RK, Tavakoli K, Parang K. Cyclic Peptide Containing Hydrophobic and Positively Charged Residues as a Drug Delivery System for Curcumin. Current Drug Delivery. PMID 26511089 DOI: 10.2174/1567201812666151029101102 |
0.69 |
|
| 2015 |
Ramos-Molina B, Lick AN, Nasrolahi Shirazi A, Oh D, Tiwari R, El-Sayed NS, Parang K, Lindberg I. Cationic Cell-Penetrating Peptides Are Potent Furin Inhibitors. Plos One. 10: e0130417. PMID 26110264 DOI: 10.1371/Journal.Pone.0130417 |
0.837 |
|
| 2015 |
Marshall J, Wong KY, Rupasinghe CN, Tiwari R, Zhao X, Berberoglu ED, Sinkler C, Liu J, Lee I, Parang K, Spaller MR, Hüttemann M, Goebel DJ. Inhibition of N-Methyl-D-Aspartate-Induced Retinal Neuronal Death by Polyarginine Peptides is Linked to the Attenuation of Stress-Induced Hyperpolarization of the Inner Mitochondrial Membrane Potential. The Journal of Biological Chemistry. PMID 26100636 DOI: 10.1074/Jbc.M115.662791 |
0.579 |
|
| 2015 |
Pemmaraju BP, Malekar S, Agarwal HK, Tiwari RK, Oh D, Doncel GF, Worthen DR, Parang K. Design, synthesis, antiviral activity, and pre-formulation development of poly-L-arginine-fatty acyl derivatives of nucleoside reverse transcriptase inhibitors. Nucleosides, Nucleotides & Nucleic Acids. 34: 1-15. PMID 25513860 DOI: 10.1080/15257770.2014.945649 |
0.779 |
|
| 2015 |
Yoon YK, Ali MA, Wei AC, Choon TS, Shirazi AN, Parang K. Discovery of a potent and highly fluorescent sirtuin inhibitor Medchemcomm. 6: 1857-1863. DOI: 10.1039/C5Md00307E |
0.341 |
|
| 2015 |
Saunthwal RK, Patel M, Tiwari RK, Parang K, Verma AK. On water: Catalyst-free chemoselective synthesis of highly functionalized tetrahydroquinazolines from 2-aminophenylacrylate Green Chemistry. 17: 1434-1441. DOI: 10.1039/C4Gc02154A |
0.539 |
|
| 2015 |
Chand K, Tiwari RK, Kumar S, Shirazi AN, Sharma S, Van Der Eycken EV, Parmar VS, Parang K, Sharma SK. Synthesis, antiproliferative, and c-Src kinase inhibitory activities of 4-oxo-4H-1-benzopyran derivatives Journal of Heterocyclic Chemistry. 52: 562-572. DOI: 10.1002/Jhet.2106 |
0.618 |
|
| 2014 |
Fowler BJ, Gelfand BD, Kim Y, Kerur N, Tarallo V, Hirano Y, Amarnath S, Fowler DH, Radwan M, Young MT, Pittman K, Kubes P, Agarwal HK, Parang K, Hinton DR, et al. Nucleoside reverse transcriptase inhibitors possess intrinsic anti-inflammatory activity. Science (New York, N.Y.). 346: 1000-3. PMID 25414314 DOI: 10.1126/Science.1261754 |
0.638 |
|
| 2014 |
Nasrolahi Shirazi A, Tiwari RK, Oh D, Sullivan B, Kumar A, Beni YA, Parang K. Cyclic peptide-selenium nanoparticles as drug transporters. Molecular Pharmaceutics. 11: 3631-41. PMID 25184366 DOI: 10.1021/Mp500364A |
0.826 |
|
| 2014 |
Shirazi AN, Paquin KL, Howlett NG, Mandal D, Parang K. Cyclic peptide-capped gold nanoparticles for enhanced siRNA delivery Molecules. 19: 13319-13331. PMID 25170952 DOI: 10.3390/Molecules190913319 |
0.466 |
|
| 2014 |
Oh D, Sun J, Nasrolahi Shirazi A, LaPlante KL, Rowley DC, Parang K. Antibacterial activities of amphiphilic cyclic cell-penetrating peptides against multidrug-resistant pathogens. Molecular Pharmaceutics. 11: 3528-36. PMID 25157458 DOI: 10.1021/Mp5003027 |
0.804 |
|
| 2014 |
Oh D, Darwish SA, Shirazi AN, Tiwari RK, Parang K. Amphiphilic bicyclic peptides as cellular delivery agents. Chemmedchem. 9: 2449-53. PMID 25047914 DOI: 10.1002/Cmdc.201402230 |
0.678 |
|
| 2014 |
Almansour AI, Kumar RS, Beevi F, Shirazi AN, Osman H, Ismail R, Choon TS, Sullivan B, McCaffrey K, Nahhas A, Parang K, Ali MA. Facile, regio- and diastereoselective synthesis of spiro-pyrrolidine and pyrrolizine derivatives and evaluation of their antiproliferative activities. Molecules (Basel, Switzerland). 19: 10033-55. PMID 25014532 DOI: 10.3390/Molecules190710033 |
0.344 |
|
| 2014 |
Yoon YK, Ali MA, Wei AC, Shirazi AN, Parang K, Choon TS. Benzimidazoles as new scaffold of sirtuin inhibitors: green synthesis, in vitro studies, molecular docking analysis and evaluation of their anti-cancer properties. European Journal of Medicinal Chemistry. 83: 448-54. PMID 24992072 DOI: 10.1016/J.Ejmech.2014.06.060 |
0.35 |
|
| 2014 |
Oh D, Nasrolahi Shirazi A, Northup K, Sullivan B, Tiwari RK, Bisoffi M, Parang K. Enhanced cellular uptake of short polyarginine peptides through fatty acylation and cyclization. Molecular Pharmaceutics. 11: 2845-54. PMID 24978295 DOI: 10.1021/Mp500203E |
0.82 |
|
| 2014 |
Pemmaraju B, Agarwal HK, Oh D, Buckheit KW, Buckheit RW, Tiwari R, Parang K. Synthesis and Biological Evaluation of 5'-O-Dicarboxylic Fatty Acyl Monoester Derivatives of Anti-HIV Nucleoside Reverse Transcriptase Inhibitors. Tetrahedron Letters. 55: 1983-1986. PMID 24791029 DOI: 10.1016/J.Tetlet.2014.02.001 |
0.744 |
|
| 2014 |
Mandal D, Nasrolahi Shirazi A, Parang K. Self-assembly of peptides to nanostructures. Organic & Biomolecular Chemistry. 12: 3544-61. PMID 24756480 DOI: 10.1039/C4Ob00447G |
0.792 |
|
| 2014 |
El-Sayed NS, Shirazi AN, El-Meligy MG, El-Ziaty AK, Nagib ZA, Parang K. Synthesis of 4-aryl-6-indolylpyridine-3-carbonitriles and evaluation of their antiproliferative activity. Tetrahedron Letters. 55: 1154-1158. PMID 24678129 DOI: 10.1016/J.Tetlet.2013.12.081 |
0.351 |
|
| 2014 |
Chand K, Prasad S, Tiwari RK, Shirazi AN, Kumar S, Parang K, Sharma SK. Synthesis and evaluation of c-Src kinase inhibitory activity of pyridin-2(1H)-one derivatives. Bioorganic Chemistry. 53: 75-82. PMID 24632506 DOI: 10.1016/J.Bioorg.2014.02.001 |
0.605 |
|
| 2014 |
Motavallizadeh S, Fallah-Tafti A, Maleki S, Shirazi AN, Pordeli M, Safavi M, Ardestani SK, Asd S, Tiwari R, Oh D, Shafiee A, Foroumadi A, Parang K, Akbarzadeh T. Synthesis and evaluation of antiproliferative activity of substituted N-(9-oxo-9H-xanthen-4-yl)benzenesulfonamides. Tetrahedron Letters. 55: 373-375. PMID 24453382 DOI: 10.1016/J.Tetlet.2013.11.033 |
0.669 |
|
| 2014 |
Yoon YK, Ali MA, Wei AC, Choon TS, Osman H, Parang K, Shirazi AN. Synthesis and evaluation of novel benzimidazole derivatives as sirtuin inhibitors with antitumor activities. Bioorganic & Medicinal Chemistry. 22: 703-10. PMID 24387981 DOI: 10.1016/J.Bmc.2013.12.029 |
0.363 |
|
| 2014 |
Verma AK, Patel M, Joshi M, Likhar PR, Tiwari RK, Parang K. Base-mediated chemo- and stereoselective addition of 5-aminoindole/tryptamine and histamines onto alkynes. The Journal of Organic Chemistry. 79: 172-86. PMID 24215621 DOI: 10.1021/Jo402352V |
0.75 |
|
| 2014 |
Sayeh N, Shirazi AN, Oh D, Sun J, Rowley D, Banerjee A, Yadav A, Tiwari RK, Parang K. Amphiphilic triazolyl peptides: Synthesis and evaluation as nanostructures Current Organic Chemistry. 18: 2665-2671. DOI: 10.2174/138527281820141028110625 |
0.807 |
|
| 2014 |
Chhikara BS, Rao MS, Rao VK, Kumar A, Buckheit KW, Buckheit RW, Parang K. Carbocyclodipeptides as modified nucleosides: Synthesis and anti-HIV activities Canadian Journal of Chemistry. 92: 1145-1149. DOI: 10.1139/Cjc-2014-0356 |
0.391 |
|
| 2014 |
Mandal D, Nasrolahi Shirazi A, Parang K. Self-assembly of peptides to nanostructures Organic and Biomolecular Chemistry. 12: 3544-3561. DOI: 10.1039/c4ob00447g |
0.774 |
|
| 2013 |
Cao C, Rioult-Pedotti MS, Migani P, Yu CJ, Tiwari R, Parang K, Spaller MR, Goebel DJ, Marshall J. Correction: Impairment of TrkB-PSD-95 Signaling in Angelman Syndrome. Plos Biology. 11. PMID 29364881 DOI: 10.1371/Annotation/F32Bc670-C9Cf-4Bb0-9376-Cd8Cfd1053C1 |
0.51 |
|
| 2013 |
Nasrolahi Shirazi A, Oh D, Tiwari RK, Sullivan B, Gupta A, Bothun GD, Parang K. Peptide amphiphile containing arginine and fatty acyl chains as molecular transporters. Molecular Pharmaceutics. 10: 4717-27. PMID 24215132 DOI: 10.1021/Mp400539R |
0.806 |
|
| 2013 |
Mandal D, Tiwari RK, Shirazi AN, Oh D, Ye G, Banerjee A, Yadav A, Parang K. Self-Assembled Surfactant Cyclic Peptide Nanostructures as Stabilizing Agents. Soft Matter. 9. PMID 24187575 DOI: 10.1039/C3Sm50764E |
0.735 |
|
| 2013 |
Rao VK, Tiwari R, Chhikara BS, Shirazi AN, Parang K, Kumar A. Copper triflate-mediated synthesis of 1,3,5-triarylpyrazoles in [bmim][PF6] ionic liquid and evaluation of their anticancer activities. Rsc Advances. 3: 15396-15403. PMID 24163734 DOI: 10.1039/C3Ra41830H |
0.595 |
|
| 2013 |
Suresh N, Nagesh HN, Sekhar KV, Kumar A, Shirazi AN, Parang K. Synthesis of novel ciprofloxacin analogues and evaluation of their anti-proliferative effect on human cancer cell lines. Bioorganic & Medicinal Chemistry Letters. 23: 6292-5. PMID 24138941 DOI: 10.1016/J.Bmcl.2013.09.077 |
0.369 |
|
| 2013 |
Pericherla K, Shirazi AN, Rao VK, Tiwari RK, DaSilva N, McCaffrey KT, Beni YA, González-SarrÃas A, Seeram NP, Parang K, Kumar A. Synthesis and antiproliferative activities of quebecol and its analogs. Bioorganic & Medicinal Chemistry Letters. 23: 5329-31. PMID 23953195 DOI: 10.1016/J.Bmcl.2013.07.058 |
0.606 |
|
| 2013 |
Nasrolahi Shirazi A, Tiwari RK, Oh D, Sullivan B, McCaffrey K, Mandal D, Parang K. Surface decorated gold nanoparticles by linear and cyclic peptides as molecular transporters. Molecular Pharmaceutics. 10: 3137-51. PMID 23834324 DOI: 10.1021/Mp400199E |
0.831 |
|
| 2013 |
Nasrolahi Shirazi A, Tiwari RK, Brown A, Mandal D, Sun G, Parang K. Cyclic peptides containing tryptophan and arginine as Src kinase inhibitors. Bioorganic & Medicinal Chemistry Letters. 23: 3230-4. PMID 23602444 DOI: 10.1016/J.Bmcl.2013.03.124 |
0.816 |
|
| 2013 |
Rao VK, Shelke GM, Tiwari R, Parang K, Kumar A. A simple and efficient synthesis of 2,3-diarylnaphthofurans using sequential hydroarylation/Heck oxyarylation. Organic Letters. 15: 2190-3. PMID 23586966 DOI: 10.1021/Ol400738R |
0.56 |
|
| 2013 |
Nasrolahi Shirazi A, Tiwari RK, Oh D, Banerjee A, Yadav A, Parang K. Efficient delivery of cell impermeable phosphopeptides by a cyclic peptide amphiphile containing tryptophan and arginine. Molecular Pharmaceutics. 10: 2008-20. PMID 23537165 DOI: 10.1021/Mp400046U |
0.799 |
|
| 2013 |
Cao C, Rioult-Pedotti MS, Migani P, Yu CJ, Tiwari R, Parang K, Spaller MR, Goebel DJ, Marshall J. Impairment of TrkB-PSD-95 signaling in Angelman syndrome. Plos Biology. 11: e1001478. PMID 23424281 DOI: 10.1371/Journal.Pbio.1001478 |
0.551 |
|
| 2013 |
Nasrolahi Shirazi A, Tiwari R, Chhikara BS, Mandal D, Parang K. Design and biological evaluation of cell-penetrating peptide-doxorubicin conjugates as prodrugs. Molecular Pharmaceutics. 10: 488-99. PMID 23301519 DOI: 10.1021/Mp3004034 |
0.82 |
|
| 2013 |
Nasrolahi Shirazi A, Mandal D, Tiwari RK, Guo L, Lu W, Parang K. Cyclic peptide-capped gold nanoparticles as drug delivery systems. Molecular Pharmaceutics. 10: 500-11. PMID 22998473 DOI: 10.1021/Mp300448K |
0.823 |
|
| 2013 |
Agarwal HK, Chhikara BS, Bhavaraju S, Mandal D, Doncel GF, Parang K. Emtricitabine prodrugs with improved anti-HIV activity and cellular uptake. Molecular Pharmaceutics. 10: 467-76. PMID 22917277 DOI: 10.1021/Mp300361A |
0.673 |
|
| 2013 |
Cao C, Rioult-Pedotti MS, Migani P, Yu CJ, Tiwari R, Parang K, Spaller MR, Goebel DJ, Marshall J. Defective BDNF-mediated synaptic plasticity in AS mice is mitigated by CN2097. Plos Biology. DOI: 10.1371/Journal.Pbio.1001478.G001 |
0.502 |
|
| 2013 |
Shelke GM, Rao VK, Tiwari RK, Chhikara BS, Parang K, Kumar A. Bismuth triflate-catalyzed condensation of indoles with acetone Rsc Advances. 3: 22346-22352. DOI: 10.1039/C3Ra44693J |
0.544 |
|
| 2012 |
Rafinejad A, Fallah-Tafti A, Tiwari R, Shirazi AN, Mandal D, Shafiee A, Parang K, Foroumadi A, Akbarzadeh T. 4-Aryl-4H-naphthopyrans derivatives: one-pot synthesis, evaluation of Src kinase inhibitory and anti-proliferative activities. Daru : Journal of Faculty of Pharmacy, Tehran University of Medical Sciences. 20: 100. PMID 23351304 DOI: 10.1186/2008-2231-20-100 |
0.668 |
|
| 2012 |
Chhikara BS, Tiwari R, Parang K. N-Myristoylglutamic Acid Derivative of 3'-Fluoro-3'-Deoxythymidine as an Organogel. Tetrahedron Letters. 53: 5335-5337. PMID 23175585 DOI: 10.1016/J.Tetlet.2012.07.101 |
0.591 |
|
| 2012 |
Sharma RK, Singh S, Tiwari R, Mandal D, Olsen CE, Parmar VS, Parang K, Prasad AK. O-Aryl α,β-d-ribofuranosides: synthesis & highly efficient biocatalytic separation of anomers and evaluation of their Src kinase inhibitory activity. Bioorganic & Medicinal Chemistry. 20: 6821-30. PMID 23098606 DOI: 10.1016/J.Bmc.2012.09.057 |
0.557 |
|
| 2012 |
Kumar A, Muthyala MK, Choudhary S, Tiwari RK, Parang K. Ionic liquid as soluble support for synthesis of 1,2,3-thiadiazoles and 1,2,3-selenadiazoles. The Journal of Organic Chemistry. 77: 9391-6. PMID 23020655 DOI: 10.1021/Jo301607A |
0.532 |
|
| 2012 |
Agarwal HK, Buckheit KW, Buckheit RW, Parang K. Synthesis and anti-HIV activities of symmetrical dicarboxylate esters of dinucleoside reverse transcriptase inhibitors. Bioorganic & Medicinal Chemistry Letters. 22: 5451-4. PMID 22858097 DOI: 10.1016/J.Bmcl.2012.07.037 |
0.657 |
|
| 2012 |
Shaik IH, Agarwal HK, Parang K, Mehvar R. Hepatic immunosuppressive effects of systemically administered novel dextran-methylprednisolone prodrugs with peptide linkers in rats. Journal of Pharmaceutical Sciences. 101: 4003-12. PMID 22829462 DOI: 10.1002/Jps.23274 |
0.625 |
|
| 2012 |
Tiwari RK, Parang K. Conformationally constrained peptides as protein tyrosine kinase inhibitors. Current Pharmaceutical Design. 18: 2852-66. PMID 22571654 DOI: 10.2174/138161212800672714 |
0.639 |
|
| 2012 |
Agarwal HK, Chhikara BS, Hanley MJ, Ye G, Doncel GF, Parang K. Synthesis and biological evaluation of fatty acyl ester derivatives of (-)-2',3'-dideoxy-3'-thiacytidine. Journal of Medicinal Chemistry. 55: 4861-71. PMID 22533850 DOI: 10.1021/Jm300492Q |
0.741 |
|
| 2012 |
Agarwal HK, Doncel GF, Parang K. Synthesis and anti-HIV activities of suramin conjugates of 3'-fluoro- 2',3'-dideoxythymidine and 3'-azido-2',3'-dideoxythymidine. Medicinal Chemistry (ShāRiqah (United Arab Emirates)). 8: 193-7. PMID 22385137 DOI: 10.2174/157340612800493737 |
0.642 |
|
| 2012 |
Agarwal HK, Chhikara BS, Quiterio M, Doncel GF, Parang K. Synthesis and anti-HIV activities of glutamate and peptide conjugates of nucleoside reverse transcriptase inhibitors. Journal of Medicinal Chemistry. 55: 2672-87. PMID 22352809 DOI: 10.1021/Jm201551M |
0.695 |
|
| 2012 |
Chhikara BS, Mandal D, Parang K. Synthesis, anticancer activities, and cellular uptake studies of lipophilic derivatives of doxorubicin succinate. Journal of Medicinal Chemistry. 55: 1500-10. PMID 22276998 DOI: 10.1021/Jm201653U |
0.394 |
|
| 2012 |
Rao VK, Chhikara BS, Tiwari R, Shirazi AN, Parang K, Kumar A. One-pot regioselective synthesis of tetrahydroindazolones and evaluation of their antiproliferative and Src kinase inhibitory activities. Bioorganic & Medicinal Chemistry Letters. 22: 410-4. PMID 22119472 DOI: 10.1016/J.Bmcl.2011.10.124 |
0.608 |
|
| 2012 |
Rao MS, Chhikara BS, Tiwari R, Shirazi AN, Parang K, Kumar A. Microwave-assisted and scandium triflate catalyzed synthesis of tetrahydrobenzo[a]xanthen-11-ones Monatshefte Fur Chemie. 143: 263-268. DOI: 10.1007/S00706-011-0577-4 |
0.583 |
|
| 2011 |
Ahmadibeni Y, Tiwari R, Swepson C, Pandhare J, Dash C, Doncel GF, Parang K. Synthesis and anti-HIV activities of bis-(cycloSaligenyl) pronucleotides derivatives of 3'-fluoro-3'-deoxythymidine and 3'-azido-3'-deoxythymidine. Tetrahedron Letters. 52: 802-805. PMID 26661937 DOI: 10.1016/J.Tetlet.2010.12.038 |
0.601 |
|
| 2011 |
Mandal D, Nasrolahi Shirazi A, Parang K. Cell-penetrating homochiral cyclic peptides as nuclear-targeting molecular transporters. Angewandte Chemie (International Ed. in English). 50: 9633-7. PMID 21919161 DOI: 10.1002/Anie.201102572 |
0.801 |
|
| 2011 |
Fallah-Tafti A, Foroumadi A, Tiwari R, Shirazi AN, Hangauer DG, Bu Y, Akbarzadeh T, Parang K, Shafiee A. Thiazolyl N-benzyl-substituted acetamide derivatives: synthesis, Src kinase inhibitory and anticancer activities. European Journal of Medicinal Chemistry. 46: 4853-8. PMID 21852023 DOI: 10.1016/J.Ejmech.2011.07.050 |
0.678 |
|
| 2011 |
Fallah-Tafti A, Tiwari R, Shirazi AN, Akbarzadeh T, Mandal D, Shafiee A, Parang K, Foroumadi A. 4-Aryl-4H-chromene-3-carbonitrile derivatives: evaluation of Src kinase inhibitory and anticancer activities. Medicinal Chemistry (ShāRiqah (United Arab Emirates)). 7: 466-72. PMID 21801146 DOI: 10.2174/157340611796799258 |
0.669 |
|
| 2011 |
Rao VK, Chhikara BS, Shirazi AN, Tiwari R, Parang K, Kumar A. 3-substitued indoles: one-pot synthesis and evaluation of anticancer and Src kinase inhibitory activities. Bioorganic & Medicinal Chemistry Letters. 21: 3511-4. PMID 21612925 DOI: 10.1016/J.Bmcl.2011.05.010 |
0.618 |
|
| 2011 |
Dash C, Ahmadibeni Y, Hanley MJ, Pandhare J, Gotte M, Le Grice SF, Parang K. Inhibition of multi-drug resistant HIV-1 reverse transcriptase by nucleoside β-triphosphates. Bioorganic & Medicinal Chemistry Letters. 21: 3519-22. PMID 21605974 DOI: 10.1016/J.Bmcl.2011.05.005 |
0.303 |
|
| 2011 |
Chhikara BS, St Jean N, Mandal D, Kumar A, Parang K. Fatty acyl amide derivatives of doxorubicin: synthesis and in vitro anticancer activities. European Journal of Medicinal Chemistry. 46: 2037-42. PMID 21420207 DOI: 10.1016/J.Ejmech.2011.02.056 |
0.389 |
|
| 2011 |
Gupta A, Mandal D, Ahmadibeni Y, Parang K, Bothun G. Hydrophobicity drives the cellular uptake of short cationic peptide ligands. European Biophysics Journal : Ebj. 40: 727-36. PMID 21409455 DOI: 10.1007/S00249-011-0685-4 |
0.389 |
|
| 2011 |
Agarwal HK, Loethan K, Mandal D, Doncel GF, Parang K. Synthesis and biological evaluation of fatty acyl ester derivatives of 2',3'-didehydro-2',3'-dideoxythymidine. Bioorganic & Medicinal Chemistry Letters. 21: 1917-21. PMID 21382714 DOI: 10.1016/J.Bmcl.2011.02.070 |
0.686 |
|
| 2011 |
Kumar A, Ahmad I, Chhikara BS, Tiwari R, Mandal D, Parang K. Synthesis of 3-phenylpyrazolopyrimidine-1,2,3-triazole conjugates and evaluation of their Src kinase inhibitory and anticancer activities. Bioorganic & Medicinal Chemistry Letters. 21: 1342-6. PMID 21300544 DOI: 10.1016/J.Bmcl.2011.01.047 |
0.603 |
|
| 2011 |
Kumar D, Reddy VB, Kumar A, Mandal D, Tiwari R, Parang K. Click chemistry inspired one-pot synthesis of 1,4-disubstituted 1,2,3-triazoles and their Src kinase inhibitory activity. Bioorganic & Medicinal Chemistry Letters. 21: 449-52. PMID 21084189 DOI: 10.1016/J.Bmcl.2010.10.121 |
0.605 |
|
| 2010 |
Agarwal HK, Kumar A, Doncel GF, Parang K. Synthesis, antiviral and contraceptive activities of nucleoside-sodium cellulose sulfate acetate and succinate conjugates. Bioorganic & Medicinal Chemistry Letters. 20: 6993-7. PMID 20965725 DOI: 10.1016/J.Bmcl.2010.09.133 |
0.66 |
|
| 2010 |
Chhikara BS, Mandal D, Parang K. Synthesis and evaluation of fatty acyl ester derivatives of cytarabine as anti-leukemia agents. European Journal of Medicinal Chemistry. 45: 4601-8. PMID 20692740 DOI: 10.1016/J.Ejmech.2010.07.024 |
0.337 |
|
| 2010 |
Sharma D, Sharma RK, Bhatia S, Tiwari R, Mandal D, Lehmann J, Parang K, Olsen CE, Parmar VS, Prasad AK. Synthesis, Src kinase inhibitory and anticancer activities of 1-substituted 3-(N-alkyl-N-phenylamino)propane-2-ols. Biochimie. 92: 1164-72. PMID 20447438 DOI: 10.1016/J.Biochi.2010.04.022 |
0.59 |
|
| 2010 |
Ahmadibeni Y, Dash C, Hanley MJ, Le Grice SF, Agarwal HK, Parang K. Synthesis of nucleoside 5'-O-alpha,beta-methylene-beta-triphosphates and evaluation of their potency towards inhibition of HIV-1 reverse transcriptase. Organic & Biomolecular Chemistry. 8: 1271-4. PMID 20204192 DOI: 10.1039/B922846B |
0.608 |
|
| 2010 |
Tiwari R, Brown A, Narramaneni S, Sun G, Parang K. Synthesis and evaluation of conformationally constrained peptide analogues as the Src SH3 domain binding ligands. Biochimie. 92: 1153-63. PMID 20109515 DOI: 10.1016/J.Biochi.2010.01.017 |
0.646 |
|
| 2010 |
Ye G, Gupta A, DeLuca R, Parang K, Bothun GD. Bilayer disruption and liposome restructuring by a homologous series of small Arg-rich synthetic peptides. Colloids and Surfaces. B, Biointerfaces. 76: 76-81. PMID 19913394 DOI: 10.1016/J.Colsurfb.2009.10.016 |
0.603 |
|
| 2010 |
Penugonda S, Agarwal HK, Parang K, Mehvar R. Plasma pharmacokinetics and tissue disposition of novel dextran-methylprednisolone conjugates with peptide linkers in rats. Journal of Pharmaceutical Sciences. 99: 1626-37. PMID 19780131 DOI: 10.1002/Jps.21934 |
0.637 |
|
| 2009 |
Tiwari R, Parang K. Protein conjugates of SH3-domain ligands and ATP-competitive inhibitors as bivalent inhibitors of protein kinases. Chembiochem : a European Journal of Chemical Biology. 10: 2445-8. PMID 19731277 DOI: 10.1002/Cbic.200900462 |
0.56 |
|
| 2009 |
Ye G, Schuler AD, Ahmadibeni Y, Morgan JR, Faruqui A, Huang K, Sun G, Zebala JA, Parang K. Synthesis and evaluation of phosphopeptides containing iminodiacetate groups as binding ligands of the Src SH2 domain. Bioorganic Chemistry. 37: 133-42. PMID 19539345 DOI: 10.1016/J.Bioorg.2009.05.003 |
0.596 |
|
| 2009 |
Ahmadibeni Y, Tiwari RK, Sun G, Parang K. Synthesis of nucleoside mono-, di-, and triphosphoramidates from solid-phase cyclosaligenyl phosphitylating reagents. Organic Letters. 11: 2157-60. PMID 19364114 DOI: 10.1021/Ol900320R |
0.551 |
|
| 2008 |
Ahmadibeni Y, Parang K. Solid-supported diphosphitylating and triphosphitylating reagents for nucleoside modification. Current Protocols in Nucleic Acid Chemistry / Edited by Serge L. Beaucage ... [Et Al.]. Unit 13.8. PMID 18551427 DOI: 10.1002/0471142700.Nc1308S33 |
0.311 |
|
| 2008 |
Ye G, Tiwari R, Parang K. Development of Src tyrosine kinase substrate binding site inhibitors. Current Opinion in Investigational Drugs (London, England : 2000). 9: 605-13. PMID 18516760 |
0.652 |
|
| 2008 |
Penugonda S, Kumar A, Agarwal HK, Parang K, Mehvar R. Synthesis and in vitro characterization of novel dextran-methylprednisolone conjugates with peptide linkers: effects of linker length on hydrolytic and enzymatic release of methylprednisolone and its peptidyl intermediates. Journal of Pharmaceutical Sciences. 97: 2649-64. PMID 17853426 DOI: 10.1002/Jps.21161 |
0.694 |
|
| 2008 |
Agarwal HK, Doncel GF, Parang K. Synthesis and anti-HIV activities of phosphate triester derivatives of 3′-fluoro-2′,3′-dideoxythymidine and 3′-azido-2′,3′-dideoxythymidine Tetrahedron Letters. 49: 4905-4907. DOI: 10.1016/J.Tetlet.2008.05.149 |
0.624 |
|
| 2007 |
Chimalakonda KC, Agarwal HK, Kumar A, Parang K, Mehvar R. Synthesis, analysis, in vitro characterization, and in vivo disposition of a lamivudine-dextran conjugate for selective antiviral delivery to the liver. Bioconjugate Chemistry. 18: 2097-108. PMID 17922546 DOI: 10.1021/Bc700193D |
0.643 |
|
| 2007 |
Bhandari R, Saiardi A, Ahmadibeni Y, Snowman AM, Resnick AC, Kristiansen TZ, Molina H, Pandey A, Werner JK, Juluri KR, Xu Y, Prestwich GD, Parang K, Snyder SH. Protein pyrophosphorylation by inositol pyrophosphates is a posttranslational event. Proceedings of the National Academy of Sciences of the United States of America. 104: 15305-10. PMID 17873058 DOI: 10.1073/Pnas.0707338104 |
0.359 |
|
| 2007 |
Ahmadibeni Y, Hanley M, White M, Ayrapetov M, Lin X, Sun G, Parang K. Metal-binding properties of a dicysteine-containing motif in protein tyrosine kinases. Chembiochem : a European Journal of Chemical Biology. 8: 1592-605. PMID 17674392 DOI: 10.1002/Cbic.200700242 |
0.344 |
|
| 2007 |
Ye G, Nam NH, Kumar A, Saleh A, Shenoy DB, Amiji MM, Lin X, Sun G, Parang K. Synthesis and evaluation of tripodal peptide analogues for cellular delivery of phosphopeptides. Journal of Medicinal Chemistry. 50: 3604-17. PMID 17580848 DOI: 10.1021/Jm070416O |
0.636 |
|
| 2007 |
Kumar A, Wang Y, Lin X, Sun G, Parang K. Synthesis and evaluation of 3-phenylpyrazolo[3,4-d]pyrimidine-peptide conjugates as Src kinase inhibitors. Chemmedchem. 2: 1346-60. PMID 17530729 DOI: 10.1002/Cmdc.200700074 |
0.461 |
|
| 2007 |
Agarwal HK, Parang K. Application of solid-phase chemistry for the synthesis of 3'-fluoro-3'-deoxythymidine. Nucleosides, Nucleotides & Nucleic Acids. 26: 317-22. PMID 17454740 DOI: 10.1080/15257770701257608 |
0.634 |
|
| 2006 |
Gu X, Wang Y, Kumar A, Ye G, Parang K, Sun G. Design and evaluation of hydroxamate derivatives as metal-mediated inhibitors of a protein tyrosine kinase. Journal of Medicinal Chemistry. 49: 7532-9. PMID 17149882 DOI: 10.1021/Jm061058C |
0.56 |
|
| 2006 |
Kumar A, Ye G, Ahmadibeni Y, Parang K. Synthesis of polymer-bound 4-acetoxy-3-phenylbenzaldehyde derivatives: applications in solid-phase organic synthesis. The Journal of Organic Chemistry. 71: 7915-8. PMID 16995713 DOI: 10.1021/Jo061328Z |
0.545 |
|
| 2006 |
Kumar A, Ye G, Wang Y, Lin X, Sun G, Parang K. Synthesis and structure-activity relationships of linear and conformationally constrained peptide analogues of CIYKYY as Src tyrosine kinase inhibitors. Journal of Medicinal Chemistry. 49: 3395-401. PMID 16722659 DOI: 10.1021/Jm060334K |
0.66 |
|
| 2005 |
Ye G, Ayrapetov M, Nam NH, Sun G, Parang K. Solid-phase binding assays of peptides using EGFP-Src SH2 domain fusion protein and biotinylated Src SH2 domain. Bioorganic & Medicinal Chemistry Letters. 15: 4994-7. PMID 16169725 DOI: 10.1016/J.Bmcl.2005.08.005 |
0.599 |
|
| 2005 |
Hines AC, Parang K, Kohanski RA, Hubbard SR, Cole PA. Bisubstrate analog probes for the insulin receptor protein tyrosine kinase: molecular yardsticks for analyzing catalytic mechanism and inhibitor design. Bioorganic Chemistry. 33: 285-97. PMID 16023488 DOI: 10.1016/J.Bioorg.2005.02.002 |
0.809 |
|
| 2005 |
Carballeira NM, O'Neill R, Parang K. Racemic and optically active 2-methoxy-4-oxatetradecanoic acids: novel synthetic fatty acids with selective antifungal properties. Chemistry and Physics of Lipids. 136: 47-54. PMID 15899476 DOI: 10.1016/J.Chemphyslip.2005.03.002 |
0.317 |
|
| 2005 |
Ayrapetov MK, Nam NH, Ye G, Kumar A, Parang K, Sun G. Functional diversity of Csk, Chk, and Src SH2 domains due to a single residue variation. The Journal of Biological Chemistry. 280: 25780-7. PMID 15890649 DOI: 10.1074/Jbc.M504022200 |
0.533 |
|
| 2005 |
Parang K, Sun G. Recent advances in the discovery of Src kinase inhibitors Expert Opinion On Therapeutic Patents. 15: 1183-1207. DOI: 10.1517/13543776.15.9.1183 |
0.303 |
|
| 2004 |
Nam NH, Sardari S, Selecky M, Parang K. Carboxylic acid and phosphate ester derivatives of fluconazole: synthesis and antifungal activities. Bioorganic & Medicinal Chemistry. 12: 6255-69. PMID 15519168 DOI: 10.1016/J.Bmc.2004.08.049 |
0.341 |
|
| 2004 |
Nam NH, Lee S, Ye G, Sun G, Parang K. ATP-phosphopeptide conjugates as inhibitors of Src tyrosine kinases. Bioorganic & Medicinal Chemistry. 12: 5753-66. PMID 15498652 DOI: 10.1016/J.Bmc.2004.08.043 |
0.57 |
|
| 2004 |
Schmidt B, Jiricek J, Titz A, Ye G, Parang K. Copper dipicolinates as peptidomimetic ligands for the Src SH2 domain. Bioorganic & Medicinal Chemistry Letters. 14: 4203-6. PMID 15261270 DOI: 10.1016/J.Bmcl.2004.06.018 |
0.607 |
|
| 2004 |
Nam NH, Ye G, Sun G, Parang K. Conformationally constrained peptide analogues of pTyr-Glu-Glu-Ile as inhibitors of the Src SH2 domain binding. Journal of Medicinal Chemistry. 47: 3131-41. PMID 15163193 DOI: 10.1021/Jm040008+ |
0.638 |
|
| 2004 |
Carballeira NM, Ortiz D, Parang K, Sardari S. Total synthesis and in vitro-antifungal activity of (+/-)-2-methoxytetradecanoic Acid. Archiv Der Pharmazie. 337: 152-5. PMID 15038060 DOI: 10.1002/Ardp.200300824 |
0.316 |
|
| 2004 |
Nam NH, Pitts RL, Sun G, Sardari S, Tiemo A, Xie M, Yan B, Parang K. Design of tetrapeptide ligands as inhibitors of the Src SH2 domain. Bioorganic & Medicinal Chemistry. 12: 779-87. PMID 14759738 DOI: 10.1016/J.Bmc.2003.10.060 |
0.391 |
|
| 2003 |
Lee S, Lin X, Nam NH, Parang K, Sun G. Determination of the substrate-docking site of protein tyrosine kinase C-terminal Src kinase. Proceedings of the National Academy of Sciences of the United States of America. 100: 14707-12. PMID 14657361 DOI: 10.1073/Pnas.2534493100 |
0.3 |
|
| 2003 |
Nam NH, Parang K. Current targets for anticancer drug discovery. Current Drug Targets. 4: 159-79. PMID 12558068 DOI: 10.2174/1389450033346966 |
0.306 |
|
| 2002 |
Parang K, Cole PA. Designing bisubstrate analog inhibitors for protein kinases. Pharmacology & Therapeutics. 93: 145-57. PMID 12191607 DOI: 10.1016/S0163-7258(02)00184-5 |
0.498 |
|
| 2002 |
Parang K, Kohn JA, Saldanha SA, Cole PA. Development of photo-crosslinking reagents for protein kinase-substrate interactions. Febs Letters. 520: 156-60. PMID 12044889 DOI: 10.1016/S0014-5793(02)02778-3 |
0.487 |
|
| 2001 |
Parang K, Fournier EJ, Hindsgaul O. A solid phase reagent for the capture phosphorylation of carbohydrates and nucleosides. Organic Letters. 3: 307-9. PMID 11430061 DOI: 10.1021/Ol0069498 |
0.504 |
|
| 2001 |
Parang K, Till JH, Ablooglu AJ, Kohanski RA, Hubbard SR, Cole PA. Mechanism-based design of a protein kinase inhibitor. Nature Structural Biology. 8: 37-41. PMID 11135668 DOI: 10.1038/83028 |
0.527 |
|
| 2000 |
Parang K, Wiebe LI, Knaus EE. Novel approaches for designing 5'-O-ester prodrugs of 3'-Azido-2',3'-dideoxythymidine (AZT) Current Medicinal Chemistry. 7: 995-1039. PMID 10911016 DOI: 10.2174/0929867003374372 |
0.671 |
|
| 2000 |
Kim K, Parang K, Lau OD, Cole PA. Tyrosine analogues as alternative substrates for protein tyrosine kinase Csk: Insights into substrate selectivity and catalytic mechanism Bioorganic and Medicinal Chemistry. 8: 1263-1268. PMID 10896106 DOI: 10.1016/S0968-0896(00)00053-5 |
0.52 |
|
| 2000 |
Ablooglu AJ, Till JH, Kim K, Parang K, Cole PA, Hubbard SR, Kohanski RA. Probing the catalytic mechanism of the insulin receptor kinase with a tetrafluorotyrosine-containing peptide substrate. The Journal of Biological Chemistry. 275: 30394-8. PMID 10869355 DOI: 10.1074/Jbc.M003524200 |
0.509 |
|
| 1998 |
Parang K, Wiebe LI, Knaus EE. Synthesis, in vitro anti-human immunodeficiency virus structure-activity relationships and biological stability of 5'-O-myristoyl analogue derivatives of 3'-azido-2',3'-dideoxythymidine (AZT) as potential prodrugs Antiviral Chemistry and Chemotherapy. 9: 311-323. PMID 9875410 DOI: 10.1177/095632029800900403 |
0.658 |
|
| 1998 |
Parang K, Wiebe LI, Knaus EE. Pharmacokinetics and tissue distribution of (±)-3'-azido-2',3'-dideoxy-5'-O-(2-bromomyristoyl)thymidine, a prodrug of 3'-azido-2',3'-dideoxythymidine (AZT) in mice Journal of Pharmacy and Pharmacology. 50: 989-996. PMID 9811159 DOI: 10.1111/J.2042-7158.1998.Tb06913.X |
0.615 |
|
| 1998 |
Parang K, Knaus EE, Wiebe LI. Synthesis, in vitro anti-HIV activity, and biological stability of 5'- O-myristoyl analogue derivatives of 3'-fluoro-2',3'dideoxythymidine (FLT) as potential bifunctional prodrugs of FLT Nucleosides and Nucleotides. 17: 987-1008. PMID 9708320 DOI: 10.1080/07328319808004216 |
0.643 |
|
| 1997 |
Parang K, Wiebe LI, Knaus EE, Huang JS, Tyrrell DL, Csizmadia F. In vitro antiviral activities of myristic acid analogs against human immunodeficiency and hepatitis B viruses Antiviral Research. 34: 75-90. PMID 9191015 DOI: 10.1016/S0166-3542(96)01022-4 |
0.658 |
|
| 1997 |
Parang K, Wiebe LI, Knaus EE. Syntheses and biological evaluation of 5'-O-myristoyl derivatives of thymidine against human immunodeficiency virus Antiviral Chemistry and Chemotherapy. 8: 417-427. DOI: 10.1177/095632029700800504 |
0.648 |
|
| 1996 |
Parang K, Knaus EE, Wiebe LI, Sardari S, Daneshtalab M, Csizmadia F. Synthesis and antifungal activities of myristic acid analogs Archiv Der Pharmazie. 329: 475-482. PMID 8997896 DOI: 10.1002/Ardp.19963291102 |
0.64 |
|
| 1992 |
Shafiee A, Parang K, Khazan M, Ghasemian F. Nitroimidazoles X . Syntheses of substituted 2‐(1‐methyl‐5‐nitro‐2‐imidazolyl)quinolines Journal of Heterocyclic Chemistry. 29: 1859-1861. DOI: 10.1002/jhet.5570290732 |
0.354 |
|
| 1992 |
Shafiee A, Pirouzzadeh B, Ghasemian F, Parang K. Nitroimidazoles. IX. Synthesis of 2‐acetyl‐1‐methyl‐5‐nitroimidazole Journal of Heterocyclic Chemistry. 29: 1021-1023. DOI: 10.1002/jhet.5570290461 |
0.354 |
|
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