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Erin F. DiMauro, Ph.D. - Publications

Affiliations: 
2003 University of Pennsylvania, Philadelphia, PA, United States 
Area:
asymmetric catalysts
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35 high-probability publications. We are testing a new system for linking publications to authors. You can help! If you notice any inaccuracies, please sign in and mark papers as correct or incorrect matches. If you identify any major omissions or other inaccuracies in the publication list, please let us know.

Year Citation  Score
2018 Boezio AA, Andrews K, Boezio C, Chu-Moyer M, Copeland KW, DiMauro EF, Foti RS, Fremeau RT, Gao H, Geuns-Meyer S, Graceffa RF, Gunaydin H, Huang H, La DS, Ligutti J, et al. 1,2,4-Triazolsulfone: A novel isosteric replacement of acylsulfonamides in the context of Na1.7 inhibition. Bioorganic & Medicinal Chemistry Letters. PMID 29709252 DOI: 10.1016/J.Bmcl.2018.04.035  0.326
2017 Sparling BA, DiMauro EF. Progress in the discovery of small molecule modulators of the Cys-loop superfamily receptors. Bioorganic & Medicinal Chemistry Letters. PMID 28606760 DOI: 10.1016/J.Bmcl.2017.04.073  0.311
2017 Graceffa RF, Boezio AA, Able J, Altmann S, Berry LM, Boezio CM, Butler JR, Chu-Moyer MY, Cooke M, DiMauro EF, Dineen TA, Feric Bojic E, Foti RS, Fremeau RT, Guzman-Perez A, et al. Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency, Pharmacokinetics, and Metabolic Properties to Obtain Atropisomeric Quinolinone (AM-0466) that Affords Robust In Vivo Activity. Journal of Medicinal Chemistry. PMID 28324649 DOI: 10.1021/Acs.Jmedchem.6B01850  0.321
2017 Weiss MM, Dineen TA, Marx IE, Altmann S, Boezio AA, Bregman H, Chu-Moyer MY, DiMauro EF, Feric Bojic E, Foti RS, Gao H, Graceffa RF, Gunaydin H, Guzman-Perez A, Huang H, et al. Sulfonamides as Selective NaV1.7 Inhibitors: Optimizing Potency and Pharmacokinetics While Mitigating Metabolic Liabilities. Journal of Medicinal Chemistry. PMID 28287723 DOI: 10.1021/Acs.Jmedchem.6B01851  0.307
2016 DiMauro EF, Altmann S, Berry LM, Bregman H, Chakka N, Chu-Moyer M, Feric Bojic E, Foti RS, Fremeau RT, Gao H, Gunaydin H, Guzman-Perez A, Hall BE, Huang H, Jarosh M, et al. Application of a Parallel Synthetic Strategy in the Discovery of Biaryl Acyl Sulfonamides as Efficient and Selective NaV1.7 Inhibitors. Journal of Medicinal Chemistry. PMID 27441383 DOI: 10.1021/Acs.Jmedchem.6B00425  0.376
2013 Huang H, Guzman-Perez A, Acquaviva L, Berry V, Bregman H, Dovey J, Gunaydin H, Huang X, Huang L, Saffran D, Serafino R, Schneider S, Wilson C, DiMauro EF. Structure-based design of 2-aminopyridine oxazolidinones as potent and selective tankyrase inhibitors. Acs Medicinal Chemistry Letters. 4: 1218-23. PMID 24900633 DOI: 10.1021/Ml4003315  0.317
2013 Hua Z, Bregman H, Buchanan JL, Chakka N, Guzman-Perez A, Gunaydin H, Huang X, Gu Y, Berry V, Liu J, Teffera Y, Huang L, Egge B, Emkey R, Mullady EL, ... ... Dimauro EF, et al. Development of novel dual binders as potent, selective, and orally bioavailable tankyrase inhibitors. Journal of Medicinal Chemistry. 56: 10003-15. PMID 24294969 DOI: 10.1021/Jm401317Z  0.307
2013 Bregman H, Chakka N, Guzman-Perez A, Gunaydin H, Gu Y, Huang X, Berry V, Liu J, Teffera Y, Huang L, Egge B, Mullady EL, Schneider S, Andrews PS, Mishra A, ... ... DiMauro EF, et al. Discovery of novel, induced-pocket binding oxazolidinones as potent, selective, and orally bioavailable tankyrase inhibitors. Journal of Medicinal Chemistry. 56: 4320-42. PMID 23701517 DOI: 10.1021/Jm4000038  0.309
2013 Bregman H, Gunaydin H, Gu Y, Schneider S, Wilson C, DiMauro EF, Huang X. Discovery of a class of novel tankyrase inhibitors that bind to both the nicotinamide pocket and the induced pocket. Journal of Medicinal Chemistry. 56: 1341-5. PMID 23316926 DOI: 10.1021/Jm301607V  0.306
2012 Huang H, Acquaviva L, Berry V, Bregman H, Chakka N, O'Connor A, DiMauro EF, Dovey J, Epstein O, Grubinska B, Goldstein J, Gunaydin H, Hua Z, Huang X, Huang L, et al. Structure-Based Design of Potent and Selective CK1γ Inhibitors. Acs Medicinal Chemistry Letters. 3: 1059-64. PMID 24900428 DOI: 10.1021/Ml300278F  0.314
2012 Bregman H, Nguyen HN, Feric E, Ligutti J, Liu D, McDermott JS, Wilenkin B, Zou A, Huang L, Li X, McDonough SI, Dimauro EF. The discovery of aminopyrazines as novel, potent Na(v)1.7 antagonists: hit-to-lead identification and SAR. Bioorganic & Medicinal Chemistry Letters. 22: 2033-42. PMID 22306122 DOI: 10.1016/J.Bmcl.2012.01.023  0.311
2009 Marx IE, DiMauro EF, Cheng A, Emkey R, Hitchcock SA, Huang L, Huang MY, Human J, Lee JH, Li X, Martin MW, White RD, Fremeau RT, Patel VF. Discovery of alpha-amidosulfones as potent and selective agonists of CB2: synthesis, SAR, and pharmacokinetic properties. Bioorganic & Medicinal Chemistry Letters. 19: 31-5. PMID 19062274 DOI: 10.1016/J.Bmcl.2008.11.026  0.342
2008 Cheng Y, Albrecht BK, Brown J, Buchanan JL, Buckner WH, DiMauro EF, Emkey R, Fremeau RT, Harmange JC, Hoffman BJ, Huang L, Huang M, Lee JH, Lin FF, Martin MW, et al. Discovery and optimization of a novel series of N-arylamide oxadiazoles as potent, highly selective and orally bioavailable cannabinoid receptor 2 (CB2) agonists. Journal of Medicinal Chemistry. 51: 5019-34. PMID 18680277 DOI: 10.1021/Jm800463F  0.307
2008 DiMauro EF, Buchanan JL, Cheng A, Emkey R, Hitchcock SA, Huang L, Huang MY, Janosky B, Lee JH, Li X, Martin MW, Tomlinson SA, White RD, Zheng XM, Patel VF, et al. Structural modifications of N-arylamide oxadiazoles: Identification of N-arylpiperidine oxadiazoles as potent and selective agonists of CB2. Bioorganic & Medicinal Chemistry Letters. 18: 4267-74. PMID 18640038 DOI: 10.1016/J.Bmcl.2008.06.096  0.31
2008 DiMauro EF, Newcomb J, Nunes JJ, Bemis JE, Boucher C, Chai L, Chaffee SC, Deak HL, Epstein LF, Faust T, Gallant P, Gore A, Gu Y, Henkle B, Hsieh F, et al. Structure-guided design of aminopyrimidine amides as potent, selective inhibitors of lymphocyte specific kinase: synthesis, structure-activity relationships, and inhibition of in vivo T cell activation. Journal of Medicinal Chemistry. 51: 1681-94. PMID 18321037 DOI: 10.1021/Jm7010996  0.307
2008 Deak HL, Newcomb JR, Nunes JJ, Boucher C, Cheng AC, DiMauro EF, Epstein LF, Gallant P, Hodous BL, Huang X, Lee JH, Patel VF, Schneider S, Turci SM, Zhu X. N-(3-(phenylcarbamoyl)arylpyrimidine)-5-carboxamides as potent and selective inhibitors of Lck: structure, synthesis and SAR. Bioorganic & Medicinal Chemistry Letters. 18: 1172-6. PMID 18083554 DOI: 10.1016/J.Bmcl.2007.11.123  0.342
2007 DiMauro EF, Newcomb J, Nunes JJ, Bemis JE, Boucher C, Buchanan JL, Buckner WH, Cheng A, Faust T, Hsieh F, Huang X, Lee JH, Marshall TL, Martin MW, McGowan DC, et al. Discovery of 4-amino-5,6-biaryl-furo[2,3-d]pyrimidines as inhibitors of Lck: development of an expedient and divergent synthetic route and preliminary SAR. Bioorganic & Medicinal Chemistry Letters. 17: 2305-9. PMID 17280833 DOI: 10.1016/J.Bmcl.2007.01.057  0.358
2007 Martin MW, Newcomb J, Nunes JJ, Bemis JE, McGowan DC, White RD, Buchanan JL, DiMauro EF, Boucher C, Faust T, Hsieh F, Huang X, Lee JH, Schneider S, Turci SM, et al. Discovery of novel 2,3-diarylfuro[2,3-b]pyridin-4-amines as potent and selective inhibitors of Lck: synthesis, SAR, and pharmacokinetic properties. Bioorganic & Medicinal Chemistry Letters. 17: 2299-304. PMID 17276681 DOI: 10.1016/J.Bmcl.2007.01.048  0.356
2007 Dimauro EF, Kennedy JM. Rapid synthesis of 3-amino-imidazopyridines by a microwave-assisted four-component coupling in one pot. The Journal of Organic Chemistry. 72: 1013-6. PMID 17253825 DOI: 10.1021/Jo0622072  0.417
2007 Martin MW, Newcomb J, Nunes JJ, Bemis JE, McGowan DC, White RD, Buchanan JL, DiMauro EF, Boucher C, Faust T, Hsieh F, Huang X, Lee JH, Schneider S, Turci SM, et al. Erratum to “Discovery of novel 2,3-diarylfuro[2,3-b]pyridin-4-amines as potent and selective inhibitors of Lck: Synthesis, SAR, and pharmacokinetic properties” [Bioorg. Med. Chem. Lett. 17 (2007) 2299–2304] Bioorganic & Medicinal Chemistry Letters. 17: 5279. DOI: 10.1016/J.Bmcl.2007.05.003  0.346
2007 DiMauro EF, Newcomb J, Nunes JJ, Bemis JE, Boucher C, Buchanan JL, Buckner WH, Cheng A, Faust T, Hsieh F, Huang X, Lee JH, Marshall TL, Martin MW, McGowan DC, et al. Erratum to “Discovery of 4-amino-5,6-biaryl-furo[2,3-d]pyrimidines as inhibitors of Lck: Development of an expedient and divergent synthetic route and preliminary SAR” [Bioorg. Med. Chem. Lett. 17 (2007) 2305–2309] Bioorganic & Medicinal Chemistry Letters. 17: 5280. DOI: 10.1016/J.Bmcl.2007.05.002  0.309
2006 DiMauro EF, Vitullo JR. Microwave-assisted preparation of fused bicyclic heteroaryl boronates: application in one-pot Suzuki couplings. The Journal of Organic Chemistry. 71: 3959-62. PMID 16674073 DOI: 10.1021/Jo060218P  0.349
2005 Fennie MW, DiMauro EF, O'Brien EM, Annamalai V, Kozlowski MC. Mechanism and scope of salen bifunctional catalysts in asymmetric aldehyde and α-ketoester alkylation Tetrahedron. 61: 6249-6265. DOI: 10.1016/J.Tet.2005.03.117  0.638
2003 Annamalai V, DiMauro EF, Carroll PJ, Kozlowski MC. Catalysis of the Michael addition reaction by late transition metal complexes of BINOL-derived salens. The Journal of Organic Chemistry. 68: 1973-81. PMID 12608819 DOI: 10.1021/Jo025993T  0.723
2003 DiMauro EF, Mamai A, Kozlowski MC. Synthesis, characterization, and metal complexes of a salen ligand containing a quinoline base Organometallics. 22: 850-855. DOI: 10.1021/Om0205795  0.601
2002 DiMauro EF, Kozlowski MC. The first catalytic asymmetric addition of dialkylzincs to alpha-ketoesters. Organic Letters. 4: 3781-4. PMID 12599457 DOI: 10.1021/Ol026315W  0.571
2002 DiMauro EF, Kozlowski MC. Development of bifunctional salen catalysts: rapid, chemoselective alkylations of alpha-ketoesters. Journal of the American Chemical Society. 124: 12668-9. PMID 12392407 DOI: 10.1021/Ja026498H  0.686
2002 DiMauro EF, Kozlowski MC. Phosphabenzenes as electron withdrawing phosphine ligands in catalysis Journal of the Chemical Society. Perkin Transactions 1. 439-444. DOI: 10.1039/B101454O  0.563
2002 DiMauro EF, Kozlowski MC. The First Catalytic Asymmetric Addition of Dialkylzincs to α-Ketoesters Organic Letters. 4: 3781-3784. DOI: 10.1021/ol026315w  0.561
2002 DiMauro EF, Kozlowski MC. Development of bifunctional salen catalysts: Rapid, chemoselective alkylations of α-ketoesters Journal of the American Chemical Society. 124: 12668-12669. DOI: 10.1021/ja026498h  0.634
2002 Li X, Xu Z, DiMauro EF, Kozlowski MC. Unusual oxidative rearrangement of 1,5-diazadecalin Tetrahedron Letters. 43: 3747-3750. DOI: 10.1016/S0040-4039(02)00559-2  0.564
2001 DiMauro EF, Kozlowski MC. Salen-derived catalysts containing secondary basic groups in the addition of diethylzinc to aldehydes. Organic Letters. 3: 3053-6. PMID 11554841 DOI: 10.1021/Ol016535U  0.651
2001 DiMauro EF, Kozlowski MC. BINOL-salen metal catalysts incorporating a bifunctional design. Organic Letters. 3: 1641-4. PMID 11405675 DOI: 10.1021/Ol0158213  0.688
2001 DiMauro EF, Kozlowski MC. BINOL - Salen Metal Catalysts Incorporating a Bifunctional Design Organic Letters. 3: 1641-1644. DOI: 10.1021/ol0158213  0.597
1999 DiMauro E, Fry AJ. Convenient synthesis of a reactive ester homoenolate Tetrahedron Letters. 40: 7945-7949. DOI: 10.1016/S0040-4039(99)01653-6  0.392
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