| Antonella Converso | | Chemistry | 2003 | 2005 | K. C. Nicolaou (post-doc) |
| Armando Cordova | | Chemistry Chemistry | | | Kim David Janda (post-doc), Carlos F. Barbas, III (research scientist) |
| Josep Cornella | Catalysis | Chemistry | 2015 | 2017 | Phil S. Baran (post-doc) |
| Joseph H Davis | Macromolecular complexes, biochemistry | Molecular Biology | 2012 | 2017 | James R. Williamson (post-doc) |
| Landon J Edgar | Immunology, Pharmacology, Chemical Biology, Glycobiology, Organic Chemistry | Molecular Medicine | 2016 | 2021 | James C. Paulson (post-doc) |
| Yu Tom Gao | Chemical Biology, Proteomics, Bioinformatics | | | | |
| Ritika Gautam | Bioinorganic, Bioorganic and Immunology | Chemistry | 2017 | 2018 | Kim David Janda (research scientist) |
| Nicolas Giuseppone | | | | | K. C. Nicolaou (post-doc) |
| Daniel Globisch | Organic Chemistry, Chemical Biology, Metabolomics | Department of Chemistry | 2011 | 2015 | Kim David Janda (post-doc) |
| Jason E. Hein | Catalysis, Kinetics, Crystallization, Robotics | | 2009 | 2011 | K. Barry Sharpless (post-doc), Valery V. Fokin (post-doc), Donna G. Blackmond (research scientist) |
| Andreas Hoenger | Parasitology Biology, Biochemistry | Cell Biology | 1993 | 1996 | Ronald Milligan (post-doc) |
| Rebekah Joy Karadeema | Biochemistry | | | | |
| Krish Krishnan | NMR Spectroscopy, Bio-statistics | Molecular Biology | 1991 | 1994 | Mark Rance (post-doc) |
| Ang Li | Total synthesis of structually and biologically interesting natural products | | 2004 | 2009 | K. C. Nicolaou (grad student) |
| Jeffrey J Liu | GPCR | Molecular Biology Molecular Biology | 2009 | 2013 | Raymond C. Stevens (grad student), Kurt Wüthrich (grad student) |
| Masanori Nagatomo | Organic Chemistry, Synthetic Chemistry, Natural Product Synthesis | | 2012 | 2012 | Phil S. Baran (post-doc) |
| John Nielsen | | Chemistry | | | Kim David Janda (grad student) |
| Louis Noodleman | quantum chemistry, inorganic chemistry, physical chemistry, spectroscopy, structural biology, bioenergetics, metalloenzymes | | | | |
| Corwin M. Nycholat | Glycoscience, Organic Chemistry | | | | |
| Heather L Osswald | Organic Chemistry, medicinal chemistry, chemical biology | | | | |
| Rainer Riedl | | | 1998 | 2000 | Peter G. Schultz (post-doc) |
| Litao Sun | Protein | | | | |
| Patrick H. Toy | Organic Chemistry | Chemistry | 1998 | 2000 | Kim David Janda (post-doc) |
| Fábio Cohen Tucci | Industrial Chemistry, Medicinal Chemistry, Pharmaceuticals | Department of Chemistry Departmento of Chemistry | 1998 | 1999 | Julius Rebek, Jr. (post-doc), Dmitry M. Rudkevich (post-doc) |
| Cody J. Wenthur | | | | | |
| guoqin xia | organometallic chemistry | | | | |
| Jari Yli-Kauhaluoma | | Chemistry | | | Kim David Janda (grad student) |
| Shuli You | | | 2001 | 2004 | Jeffery W. Kelly (post-doc) |
| Qinghai Zhang | Self-assembling membrane mimics | | | | Xiyan Lu (grad student) |