James John Crawford
Affiliations: | Genentech, Inc., San Francisco, CA, United States |
Area:
Medicinal Chemistry; Organic Chemistry; Drug DiscoveryGoogle:
"James Crawford"Parents
Sign in to add mentor| John A. Murphy | research assistant | 1999-1999 | University of Strathclyde |
| Kenneth W. Henderson | grad student | 2001-2004 | Notre Dame |
| William J. Kerr | grad student | 2001-2004 | University of Strathclyde |
| K. C. Nicolaou | post-doc | 2005-2006 | Scripps Institute |
Children
Sign in to add trainee| Catherine Laura Austin Salvini | grad student | ||
| Mark G. McLaughlin | grad student | 2012-2012 | Genentech, Inc. |
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Publications
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| Anderson M, Carton T, Salvini C, et al. (2024) Micelle-Promoted Reductive Amination of DNA-Conjugated Amines for DNA-Encoded Library Synthesis. Chemistry (Weinheim An Der Bergstrasse, Germany). e202400239 |
| Salvini CLA, Darlot B, Davison J, et al. (2023) Fragment expansion with NUDELs - poised DNA-encoded libraries. Chemical Science. 14: 8288-8294 |
| Hunter JH, Anderson MJ, Castan IFSF, et al. (2021) Highly efficient on-DNA amide couplings promoted by micelle forming surfactants for the synthesis of DNA encoded libraries. Chemical Science. 12: 9475-9484 |
| Crawford JJ, Lee W, Johnson AR, et al. (2020) Stereochemical Differences in Fluorocyclopropyl Amides Enable Tuning of Btk Inhibition and Off-Target Activity. Acs Medicinal Chemistry Letters. 11: 1588-1597 |
| Zhang C, Crawford JJ, Landry ML, et al. (2020) Strategies to Mitigate the Bioactivation of Aryl Amines. Chemical Research in Toxicology |
| Landry ML, Crawford JJ. (2020) Log Contributions of Substituents Commonly Used in Medicinal Chemistry. Acs Medicinal Chemistry Letters. 11: 72-76 |
| Crawford JJ, Liao D, Kolesnikov A, et al. (2020) Synthesis of an Azabicyclo[3.1.0]hexanone-Containing Inhibitor of NF-κΒ Inducing Kinase via Catalytic C–H Activation Synthesis |
| Bronner SM, Merrick KA, Murray J, et al. (2019) Design of a brain-penetrant CDK4/6 inhibitor for glioblastoma. Bioorganic & Medicinal Chemistry Letters |
| Crawford JJ, Bronner SM, Zbieg JR. (2018) Hippo pathway inhibition by blocking the YAP/TAZ-TEAD interface: a patent review. Expert Opinion On Therapeutic Patents |
| Blaquiere N, Castanedo G, Burch J, et al. (2018) A scaffold-hopping approach to discover potent, selective and efficacious inhibitors of NF-κB inducing kinase. Journal of Medicinal Chemistry |